All Stories

  1. An Approach Toward Radioiodination and Radiopharmacological Evaluation of a Carborane-Containing Analog of Indomethacin
  2. Nitrosoarenes as Versatile Precursors for 18 F-Fluorination
  3. Next-Gen 18F-Relay Reagent: Optimising [18F]Ethanesulfonyl Fluoride
  4. Diagnostic Twins: Exploring the Radiohybrid Concept with Iodine-123 and Lanthanum-133 for PSMA-Targeted SPECT and PET Imaging
  5. Radioiodination of Two Carborane‐Based Dual Cyclooxygenase‐2/5‐Lipoxygenase Inhibitors and Their In Vitro and In Vivo Evaluation
  6. Front Cover: Radioiodination of Two Carborane‐Based Dual Cyclooxygenase‐2/5‐Lipoxygenase Inhibitors and Their In Vitro and In Vivo Evaluation (ChemBioChem 7/2026)
  7. Sex determines the natural killer cell-mediated immunity against pancreatic cancer
  8. nido-carborane conjugates with ibuprofen, flurbiprofen and fenoprofen: synthesis, characterization, COX inhibition potential and anticancer activity
  9. Smart Delivery: Designing Peptides that Use Cancer Enzymes to Find Their Target
  10. Automatic Delineation of Tumor Spheroids in Microscopic Images Using Deep-Learning
  11. A biomaterial-based platform of pancreatic cancer reveals kallikrein-related peptidase 6 (KLK6) as a mediator of neutrophil recruitment and immunosuppression
  12. In Vitro Characterization of the Published Glypican-3-Targeting Peptide TJ12P2 Reveals a Lack of Specificity and Potency
  13. Novel Ruthenacarborane–NSAID Conjugates
  14. “Precision on Two Wheels”─Structural Refinement of 64 Cu- and 68 Ga-Labeled Bicyclic Peptides Targeting Nectin-4 for Improved Tumor Imaging: From Prec...
  15. Investigation of the Putative Relationship Between Copper Transport and the Anticancer Activity of Cisplatin in Ductal Pancreatic Adenocarcinoma
  16. Radioresistant mouse pheochromocytoma cell lines
  17. Exploring the Role of Peripheral Macrophages in Glioma Progression: The Metabolic Significance of Cyclooxygenase-2 (COX-2)
  18. It’s a match: use of the radionuclide theranostic pair 133La/225Ac for the radiopharmacological characterization of EGFR-targeted single-domain antibodies
  19. Front Cover: Carborane‐Based Analogs of Celecoxib and Flurbiprofen, their COX Inhibition Potential, and COX Selectivity Index (ChemMedChem 11/2025)
  20. Cover Feature: Advances in Diclofenac Derivatives: Exploring Carborane‐Substituted N‐Methyl and Nitrile Analogs for Anticancer Therapy (ChemMedChem 11/2025)
  21. Deciphering the Tumor Uptake of Heterobivalent (SST2/Albumin) [64Cu]Cu-NODAGA-cLAB-TATEs
  22. Development of [99mTc]TcO-ABX474: Design, Synthesis, and Biological Evaluation of PSMA-Binding Technetium-99m Radioligands for SPECT Imaging of Prostate Cancer
  23. Carborane‐based Analogues of Celecoxib and Flurbiprofen, their COX Inhibition Potential and COX Selectivity Index
  24. Advances in Diclofenac Derivatives: Exploring Carborane‐Substituted N‐Methyl and Nitrile Analogs for Anti‐Cancer Therapy
  25. Exploring a Nitric Oxide-Releasing Celecoxib Derivative as a Potential Modulator of Bone Healing: Insights from Ex Vivo and In Vivo Imaging Experiments
  26. Front Cover: Carborane Conjugates with Ibuprofen, Fenoprofen and Flurbiprofen: Synthesis, Characterization, COX Inhibition Potential and In Vitro Activity (ChemMedChem 1/2025)
  27. Re-design and evaluation of diclofenac-based carborane-substituted prodrugs and their anti-cancer potential
  28. Towards more reliable experimental models for pancreatic cancer
  29. Cyclohexanediamine Triazole (CHDT) Functionalization Enables Labeling of Target Molecules with Al18F/68Ga/111In
  30. Programmable Release of Chemotherapeutics from Ferrocene‐Based Injectable Hydrogels Slows Melanoma Growth
  31. Carborane Conjugates with Ibuprofen, Fenoprofen and Flurbiprofen: Synthesis, Characterization, COX Inhibition Potential and In Vitro Activity
  32. Cover Feature: 64Cu tumor labeling with hexadentate picolinic acid‐based bispidine immunoconjugates (Chem. Eur. J. 32/2024)
  33. 64 Cu tumor labeling with hexadentate picolinic acid‐based bispidine immunoconjugates
  34. Impact of Viscosity on Human Hepatoma Spheroids in Soft Core–Shell Microcapsules
  35. Correction to: Radiosynthesis and biological evaluation of [18F]AG-120 for PET imaging of the mutant isocitrate dehydrogenase 1 in glioma
  36. Preclinical evaluation of an 18F-labeled Nε-acryloyllysine piperazide for covalent targeting of transglutaminase 2
  37. Improving susceptibility of neuroendocrine tumors to radionuclide therapies: personalized approaches towards complementary treatments
  38. Towards an advanced clinical use of radiocopper in cancer theranostics
  39. Radiosynthesis and biological evaluation of [18F]AG-120 for PET imaging of the mutant isocitrate dehydrogenase 1 in glioma
  40. Lysyl Oxidases as Targets for Cancer Therapy and Diagnostic Imaging
  41. Correction to Impedimetric Nanobiosensor for the Detection of SARS-CoV-2 Antigens and Antibodies
  42. Anti-Cancer Prodrug Cyclophosphamide Exerts Thrombogenic Effects on Human Venous Endothelial Cells Independent of CYP450 Activation—Relevance to Thrombosis
  43. Comparative Saturation Binding Analysis of 64Cu-Labeled Somatostatin Analogues Using Cell Homogenates and Intact Cells
  44. Synthesis and In Vitro Biological Evaluation of p-Carborane-Based Di-tert-butylphenol Analogs
  45. Outside Back Cover: (Biotechnology Journal 6/2023)
  46. Reactivating damaged motor neurons using magnetic fields
  47. Preclinical Characterization of the 177Lu-Labeled Prostate Stem Cell Antigen (PSCA)-Specific Monoclonal Antibody 7F5
  48. Isonimesulide and Its Carborane Analogues as Isoform‐Selective COX Inhibitors and Antitumor Agents
  49. Carborane‐based Tebufelone Analogs and their Biological Evaluation In Vitro
  50. Specific and safe targeting of glioblastoma using switchable and logic-gated RevCAR T cells
  51. Metastatic pheochromocytoma and paraganglioma: Somatostatin receptor 2 expression, genetics and therapeutic responses
  52. Shell engineering in soft alginate‐based capsules for culturing liver spheroids
  53. Dipeptide-Derived Alkynes as Potent and Selective Irreversible Inhibitors of Cysteine Cathepsins
  54. A self-assembled dynamic extracellular matrix-like hydrogel system with multi-scale structures for cell bioengineering applications
  55. Front Cover: Carborane Analogues of Fenoprofen Exhibit Improved Antitumor Activity (ChemMedChem 5/2023)
  56. Impedimetric Nanobiosensor for the Detection of SARS-CoV-2 Antigens and Antibodies
  57. Microdialysis Reveals Anti-Inflammatory Effects of Sulfated Glycosaminoglycanes in the Early Phase of Bone Healing
  58. Solid-Phase Parallel Synthesis of Dual Histone Deacetylase-Cyclooxygenase Inhibitors
  59. Prostaglandins and the Lung
  60. The Impact of Nε-Acryloyllysine Piperazides on the Conformational Dynamics of Transglutaminase 2
  61. Modulating the Renal Clearance of Targeted Radiopharmaceuticals
  62. Carborane-based Compounds in Dual Inhibitor Design
  63. Pheochromocytoma radionuclide theranostics and radiation transcriptomics
  64. Carborane Analogues of Fenoprofen Exhibit Improved Antitumor Activity
  65. Impact of Sulfated Hyaluronan on Bone Metabolism in Diabetic Charcot Neuroarthropathy and Degenerative Arthritis
  66. Toward Personalized Medicine: One Chelator for Imaging and Therapy with Lutetium-177 and Actinium-225
  67. Targeting neuropeptide receptors for cancer imaging
  68. New link between dietary phosphate and coronary heart disease
  69. NO• donors in cancer therapy
  70. Case report: Incidentally discovered case of pheochromocytoma as a cause of long COVID-19 syndrome
  71. Better understanding the metabolic stability of radiotracers
  72. Shell engineering in soft alginate-based capsules for culturing liver tumoroids
  73. Carboranyl Analogues of Mefenamic Acid and Their Biological Evaluation
  74. Application of a Fluorescence Anisotropy-Based Assay to Quantify Transglutaminase 2 Activity in Cell Lysates
  75. The Role of Transglutaminase 2 in the Radioresistance of Melanoma Cells
  76. Acceleration to the next level
  77. Personalized drug testing in human pheochromocytoma/paraganglioma primary cultures
  78. CRISPR/Cas9 Mediated Knockout of Cyclooxygenase-2 Gene Inhibits Invasiveness in A2058 Melanoma Cells
  79. A Self‐Assembled Matrix System for Cell‐Bioengineering Applications in Different Dimensions, Scales, and Geometries
  80. Targeting estrogen receptors in melanoma
  81. Targeting bone with copper radionuclides
  82. “Clickable” Albumin Binders for Modulating the Tumor Uptake of Targeted Radiopharmaceuticals
  83. Solid-Phase Synthesis of Selectively Mono-Fluorobenz(o)ylated Polyamines as a Basis for the Development of 18F-Labeled Radiotracers
  84. Hybrid agents for multimodal imaging
  85. Men who stare at bone: multimodal monitoring of bone healing
  86. Radiolabelled Cyclic Bisarylmercury: High Chemical and in vivo Stability for Theranostics
  87. Modulation of γ-Secretase Activity by a Carborane-Based Flurbiprofen Analogue
  88. Conductive Hydrogels with Dynamic Reversible Networks for Biomedical Applications
  89. Immunocompatibility and non-thrombogenicity of gelatin-based hydrogels
  90. Convergent synthesis of diversified reversible network leads to liquid metal-containing conductive hydrogel adhesives
  91. Development of an 18F-Labeled Irreversible Inhibitor of Transglutaminase 2 as Radiometric Tool for Quantitative Expression Profiling in Cells and Tissues
  92. Development of a ghrelin receptor inverse agonist for positron emission tomography
  93. The transCampus Metabolic Training Programme Explores the Link of SARS-CoV-2 Virus to Metabolic Disease
  94. Response of Endothelial Cells to Gelatin-Based Hydrogels
  95. Pseudohypoxia causes radioresistance
  96. Screening Arrays of Laminin Peptides on Modified Cellulose for Promotion of Adhesion of Primary Endothelial and Neural Precursor Cells
  97. A modular, injectable, non-covalently assembled hydrogel system features widescale tunable degradability for controlled release and tissue integration
  98. The Pyrazolo[3,4-d]pyrimidine-Based Kinase Inhibitor NVP-BHG712: Effects of Regioisomers on Tumor Growth, Perfusion, and Hypoxia in EphB4-Positive A375 Melanoma Xenografts
  99. The influence of different artificial extracellular matrix implant coatings on the regeneration of a critical size femur defect in rats
  100. Pseudohypoxia promotes metastasis
  101. Recent Insights in Barium-131 as a Diagnostic Match for Radium-223: Cyclotron Production, Separation, Radiolabeling, and Imaging
  102. Radiopharmaceutical Cancer Research goes 3D
  103. Metabolomics, machine learning and immunohistochemistry to predict succinate dehydrogenase mutational status in phaeochromocytomas and paragangliomas
  104. Fighting Cancer: Targeting the Eph Receptor Tyrosine Kinase Subfamily
  105. Comparison of manual and automated ventricle segmentation in the maternal immune stimulation rat model of schizophrenia
  106. The sigma-1 receptor: Potential role in the modulation of cellular radiation sensitivity
  107. Adjuvant Drug-Assisted Bone Healing: Advances and Challenges in Drug Delivery Approaches
  108. Carboranyl Derivatives of Rofecoxib with Cytostatic Activity against Human Melanoma and Colon Cancer Cells
  109. Regulation of bone regeneration
  110. Adjuvant drug-assisted bone healing: Part I – Modulation of inflammation
  111. Adjuvant drug-assisted bone healing: Part II – Modulation of angiogenesis
  112. Adjuvant drug-assisted bone healing: Part III – Further strategies for local and systemic modulation
  113. Synthesis, radiolabelling and initial biological characterisation of 18F-labelled xanthine derivatives for PET imaging of Eph receptors
  114. Deuteration versus ethylation – strategies to improve the metabolic fate of an 18F-labeled celecoxib derivative
  115. Fluorescent mouse pheochromocytoma spheroids expressing hypoxia-inducible factor 2 alpha: Morphologic and radiopharmacologic characterization
  116. Active Targeting of Dendritic Polyglycerols for Diagnostic Cancer Imaging
  117. Bone healing made visible
  118. Synthesis and Cyclooxygenase Inhibition of Sulfonamide-Substituted (Dihydro)Pyrrolo[3,2,1-hi]indoles and Their Potential Prodrugs
  119. Pheochromocytoma/Paraganglioma: A Guide for the Practicing Clinician
  120. Characterization of Tissue Transglutaminase as a Potential Biomarker for Tissue Response toward Biomaterials
  121. A theranostic PSMA ligand for PET imaging and retargeting of T cells expressing the universal chimeric antigen receptor UniCAR
  122. Radiochemical and radiopharmacological characterization of a 64 Cu-labeled α-MSH analog conjugated with different chelators
  123. Targeting Cyclooxygenase-2 in Pheochromocytoma and Paraganglioma: Focus on Genetic Background
  124. Cytocompatible, Injectable, and Electroconductive Soft Adhesives with Hybrid Covalent/Noncovalent Dynamic Network
  125. Instant kit preparation of 68Ga-radiopharmaceuticals via the hybrid chelator DATA: clinical translation of [68Ga]Ga-DATA-TOC
  126. Carboranyl Analogues of Ketoprofen with Cytostatic Activity against Human Melanoma and Colon Cancer Cell Lines
  127. Nitric Oxide-Releasing Selective Estrogen Receptor Modulators: A Bifunctional Approach to Improve the Therapeutic Index
  128. Synthesis and preliminary radiopharmacological characterisation of an 11 C-labelled azadipeptide nitrile as potential PET tracer for imaging of cysteine cathepsins
  129. Impact of Extrinsic and Intrinsic Hypoxia on Catecholamine Biosynthesis in Absence or Presence of Hif2α in Pheochromocytoma Cells
  130. Limited importance of EphrinA1–ligand, Src kinase, and focal adhesion kinase in EphA2-mediated regulation of metastasis in Mel-Juso and A375 human melanoma cells
  131. Regulation of A375 melanoma cell adhesion and migration by EphB4 and EphrinB2 – insights from co-culture experiments
  132. Cover Feature: Carboranyl Analogues of Celecoxib with Potent Cytostatic Activity against Human Melanoma and Colon Cancer Cell Lines (ChemMedChem 3/2019)
  133. Carboranyl Analogues of Celecoxib with Potent Cytostatic Activity against Human Melanoma and Colon Cancer Cell Lines
  134. Fluorine-18 Labeling of S100 Proteins for Small Animal Positron Emission Tomography
  135. One-Pot Cascade Synthesis of Pyrazole Based Isosteres of Valdecoxib by a [3+2] Cycloaddition Sequence and Evaluation of Their Cox Inhibitory Activity
  136. Strain-specific metastatic phenotypes in pheochromocytoma allograft mice
  137. Diverse effects of phospholipase A2 receptor expression on LNCaP and PC-3 prostate cancer cell growth in vitro and in vivo
  138. Synthesis, 18F-labelling and radiopharmacological characterisation of the C-terminal 30mer of Clostridium perfringens enterotoxin as a potential claudin-targeting peptide
  139. Development of a novel target module redirecting UniCAR T cells to Sialyl Tn-expressing tumor cells
  140. Exploring pitfalls of 64Cu-labeled EGFR-targeting peptide GE11 as a potential PET tracer
  141. Causative treatment of acid aspiration induced acute lung injury – Recent trends from animal experiments and critical perspective
  142. From mono- to bivalent: improving theranostic properties of target modules for redirection of UniCAR T cells against EGFR-expressing tumor cells in vitro and in vivo
  143. Evaluation of Fluorine-18-Labeled α1(I)-N-Telopeptide Analogs as Substrate-Based Radiotracers for PET Imaging of Melanoma-Associated Lysyl Oxidase
  144. Synthesis, Characterization, and Initial Biological Evaluation of [99m Tc]Tc-Tricarbonyl-labeled DPA-α-MSH Peptide Derivatives for Potential Melanoma Imaging
  145. Nε-Acryloyllysine Piperazides as Irreversible Inhibitors of Transglutaminase 2: Synthesis, Structure–Activity Relationships, and Pharmacokinetic Profiling
  146. Bridging from Brain to Tumor Imaging: (S)-(−)- and (R)-(+)-[18F]Fluspidine for Investigation of Sigma-1 Receptors in Tumor-Bearing Mice
  147. Engrafting human regulatory T cells with a flexible modular chimeric antigen receptor technology
  148. Overexpression of Receptor Tyrosine Kinase EphB4 Triggers Tumor Growth and Hypoxia in A375 Melanoma Xenografts: Insights from Multitracer Small Animal Imaging Experiments
  149. Novel valdecoxib derivatives by ruthenium(ii)-promoted 1,3-dipolar cycloaddition of nitrile oxides with alkynes – synthesis and COX-2 inhibition activity
  150. Retargeting of UniCAR T cells with an in vivo synthesized target module directed against CD19 positive tumor cells
  151. An orthotopic xenograft model for high-risk non-muscle invasive bladder cancer in mice: influence of mouse strain, tumor cell count, dwell time and bladder pretreatment
  152. Development of novel target modules for retargeting of UniCAR T cells to GD2 positive tumor cells
  153. Preparation of a novel radiotracer targeting the EphB4 receptor via radiofluorination using spiro azetidinium salts as precursor
  154. Biological characterization of novel nitroimidazole-peptide conjugates in vitr o and in vivo
  155. Novel Tumor Pretargeting System Based on Complementaryl-Configured Oligonucleotides
  156. In Vivo Examination of an Injectable Hydrogel System Crosslinked by Peptide-Oligosaccharide Interaction in Immunocompetent Nude Mice
  157. Human Endothelial Cell Models in Biomaterial Research
  158. Retargeting of T lymphocytes to PSCA- or PSMA positive prostate cancer cells using the novel modular chimeric antigen receptor platform technology “UniCAR”
  159. Cryogel-supported stem cell factory for customized sustained release of bispecific antibodies for cancer immunotherapy
  160. A novel nanobody-based target module for retargeting of T lymphocytes to EGFR-expressing cancer cells via the modular UniCAR platform
  161. Surface charge and particle size determine the metabolic fate of dendritic polyglycerols
  162. The why and how of amino acid analytics in cancer diagnostics and therapy
  163. Technetium-99m based small molecule radiopharmaceuticals and radiotracers targeting inflammation and infection
  164. Development of a18F-labeled Diaryl-Substituted Dihydropyrrolo[3,2,1-hi]indole as Potential Probe for Functional Imaging of Cyclooxygenase-2 with PET
  165. S100 proteins and scavenger receptors: what's going on?
  166. Zwitterionic Polymer-Coated Ultrasmall Superparamagnetic Iron Oxide Nanoparticles with Low Protein Interaction and High Biocompatibility
  167. Extracellular S100A4 affects endothelial cell integrity and stimulates transmigration of A375 melanoma cells
  168. Corrigendum: Synthesis and Kinetic Characterisation of Water-Soluble Fluorogenic Acyl Donors for Transglutaminase 2
  169. Synthesis and Kinetic Characterisation of Water-Soluble Fluorogenic Acyl Donors for Transglutaminase 2
  170. Development of Antioxidant COX-2 Inhibitors as Radioprotective Agents for Radiation Therapy—A Hypothesis-Driven Review
  171. Interaction of extracellular S100A4 with RAGE prompts prometastatic activation of A375 melanoma cells
  172. 177Lu-labelled macrocyclic bisphosphonates for targeting bone metastasis in cancer treatment
  173. Protective effects of 2,3-diaryl-substituted indole-based cyclooxygenase-2 inhibitors on oxidative modification of human low density lipoproteins in vitro
  174. Controlled immobilization of His-tagged proteins for protein-ligand interaction experiments using Ni2+-NTA layer on glass surfaces
  175. Gelatin-based Hydrogel Degradation and Tissue Interactionin vivo: Insights from Multimodal Preclinical Imaging in Immunocompetent Nude Mice
  176. Multimodal Somatostatin Receptor Theranostics Using [64Cu]Cu-/[177Lu]Lu-DOTA-(Tyr3)octreotate and AN-238 in a Mouse Pheochromocytoma Model
  177. Radiopharmacological characterization of 64Cu-labeled α-MSH analogs for potential use in imaging of malignant melanoma
  178. 68Ga- und 177Lu-markierte Bisphosphonate als Knochenmetastasen-Theranostika
  179. Influence of irradiation on release of endothelial microparticles (EMP) in vitro
  180. Development of indazolylpyrimidine derivatives as high-affine EphB4 receptor ligands and potential PET radiotracers
  181. Novel (pyrazolyl)benzenesulfonamides with a nitric oxide-releasing moiety as selective cyclooxygenase-2 inhibitors
  182. Copper(II) Cyclam Complexes withN-­Propionic Acid Pendant Arms
  183. Effects of pulmonary acid aspiration on the regional pulmonary blood flow within the first hour after injury: An observational study in rats1
  184. 18F-Labeled 1,4-Dioxa-8-azaspiro[4.5]decane Derivative: Synthesis and Biological Evaluation of a σ1Receptor Radioligand with Low Lipophilicity as Potent Tumor Imaging Agent
  185. Cysteine cathepsins: their role in tumor progression and recent trends in the development of imaging probes
  186. Synthesis and Biodistribution Studies of 3 H- and 64 Cu-Labeled Dendritic Polyglycerol and Dendritic Polyglycerol Sulfate
  187. Diaryl-Substituted (Dihydro)pyrrolo[3,2,1-hi]indoles, a Class of Potent COX-2 Inhibitors with Tricyclic Core Structure
  188. Reduced pulmonary blood flow in regions of injury 2 hours after acid aspiration in rats
  189. Optical imaging of COX-2: Studies on an autofluorescent 2,3-diaryl-substituted indole-based cyclooxygenase-2 inhibitor
  190. Cyclopeptides containing the DEKS motif as conformationally restricted collagen telopeptide analogues: synthesis and conformational analysis
  191. Novel indole-based sigma-2 receptor ligands: synthesis, structure–affinity relationship and antiproliferative activity
  192. Biocompatibility and inflammatory response in vitro and in vivo to gelatin-based biomaterials with tailorable elastic properties
  193. In Vivo Fluorescence Imaging and Urinary Monoamines as Surrogate Biomarkers of Disease Progression in a Mouse Model of Pheochromocytoma
  194. Radiofluorination and first radiopharmacological characterization of a SWLAY peptide-based ligand targeting EphA2
  195. Binding properties of radiolabeled cetuximab conjugates
  196. Bispidine Dioxotetraaza Macrocycles: A New Class of Bispidines for 64Cu PET Imaging
  197. Radiolabeled Cetuximab Conjugates for EGFR Targeted Cancer Diagnostics and Therapy
  198. Metastatic potential of B16-F10 melanoma cells is enhanced by extracellular S100A4 derived from RAW264.7 macrophages
  199. ChemInform Abstract: Tissue Transglutaminase: An Emerging Target for Therapy and Imaging
  200. Radiolabeled anti-EGFR-antibody improves local tumor control after external beam radiotherapy and offers theragnostic potential
  201. 2,3-Diaryl-substituted indole based COX-2 inhibitors as leads for imaging tracer development
  202. Organotypical vascular model for characterization of radioprotective compounds: Studies on antioxidant 2,3-diaryl-substituted indole-based cyclooxygenase-2 inhibitors
  203. Synthesis and radiopharmacological evaluation of 64Cu-labeled bombesin analogs featuring a bis(2-pyridylmethyl)-1,4,7-triazacyclononane chelator
  204. Tissue transglutaminase: An emerging target for therapy and imaging
  205. Pulmonary Blood Flow Increases in Damaged Regions Directly after Acid Aspiration in Rats
  206. Optimization of Pentadentate Bispidines as Bifunctional Chelators for64Cu Positron Emission Tomography (PET)
  207. Synthesis and Radiopharmacological Characterisation of a Fluorine-18-Labelled Azadipeptide Nitrile as a Potential PET Tracer for in vivo Imaging of Cysteine Cathepsins
  208. Radiolabeled COX-2 Inhibitors for Non-Invasive Visualization of COX-2 Expression and Activity — A Critical Update
  209. Anti-tumor effects of peptide analogs targeting neuropeptide hormone receptors on mouse pheochromocytoma cells
  210. An Efficient Bioorthogonal Strategy Using CuAAC Click Chemistry for Radiofluorinations of SNEW Peptides and the Role of Copper Depletion
  211. Experimental hypoxia does not influence gene expression and protein synthesis of Eph receptors and ephrin ligands in human melanoma cells in vitro
  212. 2-Carbaborane-3-phenyl-1H-indoles-Synthesis via McMurry Reaction and Cyclooxygenase (COX) Inhibition Activity
  213. Copper(ii) chemistry of the functionalized macrocycle cyclam tetrapropionic acid
  214. Visualization of cyclooxygenase-2 using a 2,3-diarylsubstituted indole-based inhibitor and confocal laser induced cryofluorescence microscopy at 20K in melanoma cells in vitro
  215. 18F-Labeled phosphopeptide-cell-penetrating peptide dimers with enhanced cell uptake properties in human cancer cells
  216. Protein and non-protein biomarkers in melanoma: a critical update
  217. Fluorine-18 Radiolabeling and Radiopharmacological Characterization of a Benzodioxolylpyrimidine-based Radiotracer Targeting the Receptor Tyrosine Kinase EphB4
  218. Radiosynthesis of a 18F-labeled 2,3-diarylsubstituted indole via McMurry coupling for functional characterization of cyclooxygenase-2 (COX-2) in vitro and in vivo
  219. Design, Evaluation, and Comparison of Ghrelin Receptor Agonists and Inverse Agonists as Suitable Radiotracers for PET Imaging
  220. Irradiation affects cellular properties and Eph receptor expression in human melanoma cells
  221. Site-selective radiolabeling of peptides by 18F-fluorobenzoylation with [18F]SFB in solution and on solid phase: a comparative study
  222. Cyclin-Dependent Kinases (Cdk) as Targets for Cancer Therapy and Imaging
  223. Specific Targeting of Hypoxic Tumor Tissue with Nitroimidazole-Peptide Conjugates
  224. Synthesis of an 18F-labeled cyclin-dependent kinase-2 inhibitor
  225. Automated radiosynthesis of the thiol-reactive labeling agent N-[6-(4-[18F]fluorobenzylidene)aminooxyhexyl]maleimide ([18F]FBAM)
  226. Copper-mediated cross-linking of S100A4, but not of S100A2, results in proinflammatory effects in melanoma cells
  227. Phosphopeptides with improved cellular uptake properties as ligands for the polo-box domain of polo-like kinase 1
  228. ChemInform Abstract: Synthesis and Evaluation of 1,5‐Diaryl‐Substituted Tetrazoles (IV) as Novel Selective Cyclooxygenase‐2 (COX‐2) Inhibitors.
  229. A novel tetrabranched neurotensin(8–13) cyclam derivative: Synthesis, 64Cu-labeling and biological evaluation
  230. Synthesis, characterization and biological evaluation of [188Re(N)(cys∼)(PNP)]+/0 mixed-ligand complexes as prototypes for the development of 188Re(N)-based target-specific radiopharmaceuticals
  231. Synthesis and evaluation of 1,5-diaryl-substituted tetrazoles as novel selective cyclooxygenase-2 (COX-2) inhibitors
  232. Expression, purification and fluorine-18 radiolabeling of recombinant S100A4: a potential probe for molecular imaging of receptor for advanced glycation endproducts in vivo?
  233. S100 proteins in health and disease
  234. Modulation of Adrenal Aldosterone Release by Oxidative Modification of Low-Density Lipoprotein
  235. S100A2 in cancerogenesis: a friend or a foe?
  236. Cyclin-Dependent Kinase 4/6 (Cdk4/6) Inhibitors: Perspectives in Cancer Therapy and Imaging
  237. Synthesis of neurotensin(8–13)–phosphopeptide heterodimers via click chemistry
  238. Scavenger receptors are associated with cellular interactions of S100A12 in vitro and in vivo
  239. Improved multimodality imaging using alginate molding in xenograft tumor models
  240. Effects of posture on regional pulmonary blood flow in rats as measured by PET
  241. Radiosynthesis and radiopharmacological evaluation of cyclin-dependent kinase 4 (Cdk4) inhibitors
  242. Eph receptors and ephrins: bloody players
  243. Influence of irradiation on metabolism and metastatic potential of B16-F10 melanoma cells
  244. Validation of 99mTc-labeled “4+1” fatty acids for myocardial metabolism and flow imaging
  245. Validation of 99mTc-labeled “4+1” fatty acids for myocardial metabolism and flow imaging
  246. Radiosynthesis and radiopharmacological evaluation of [N-methyl-11C]Org 34850 as a glucocorticoid receptor (GR)-binding radiotracer
  247. Synthesis and cyclooxygenase inhibition of various (aryl-1,2,3-triazole-1-yl)-methanesulfonylphenyl derivatives
  248. Cell Cycle Regulating Kinase Cdk4 as a Potential Target for Tumor Cell Treatment and Tumor Imaging
  249. Erratum
  250. Fluorine-18 labeling of phosphopeptides: A potential approach for the evaluation of phosphopeptide metabolism in vivo
  251. Reduction of Arteriosclerotic Nanoplaque Formation and Size by n-3 Fatty Acids in Patients after Valvular Defect Operation
  252. Effects of pioglitazone and/or simvastatin on low density lipoprotein subfractions in non-diabetic patients with high cardiovascular risk: A sub-analysis from the PIOSTAT study
  253. Prediabetic and diabetic in vivo modification of circulating low-density lipoprotein attenuates its stimulatory effect on adrenal aldosterone and cortisol secretion
  254. Synthesis and evaluation in vitro and in vivo of a 11C-labeled cyclooxygenase-2 (COX-2) inhibitor
  255. Radiolabeled Glucocorticoids as Molecular Probes for Imaging Brain Glucocorticoid Receptors by Means of Positron Emission Tomography (PET)
  256. Synthesis and Application of [18F]FDG-Maleimidehexyloxime ([18F]FDG-MHO): A [18F]FDG-Based Prosthetic Group for the Chemoselective18F-Labeling of Peptides and Proteins†
  257. Human S100A12: a novel key player in inflammation?
  258. Systematic comparison of two novel, thiol-reactive prosthetic groups for 18F labeling of peptides and proteins with the acylation agent succinimidyl-4-[18F]fluorobenzoate ([18F]SFB)
  259. Expression, purification and fluorine-18 radiolabeling of recombinant S100 proteins—potential probes for molecular imaging of receptor for advanced glycation endproducts (RAGE) in vivo
  260. Glycoxidation of Low Density Lipoprotein in Impaired Glucose Tolerance: Implications for the Pathogenesis of Diabetic Vascular Disease
  261. Yttrium-86-labelled human serum albumin microspheres: relation of surface structure with in vivo stability
  262. Modified “4 + 1” Mixed Ligand Technetium-Labeled Fatty Acids for Myocardial Imaging: Evaluation of Myocardial Uptake and Biodistribution
  263. L-Type Amino Acid Transporters LAT1 and LAT4 in Cancer: Uptake of 3-O-Methyl-6- 18F-Fluoro-L-Dopa in Human Adenocarcinoma and Squamous Cell Carcinoma In Vitro and In Vivo
  264. Localized proton magnetic resonance spectroscopy of lipids in adipose tissue at high spatial resolution in mice in vivo
  265. Factors influencing the formation of small dense low-density lipoprotein particles in dependence on the presence of the metabolic syndrome and on the degree of glucose intolerance
  266. Experimental hypoxia is a potent stimulus for radiotracer uptake in vitro: Comparison of different tumor cells and primary endothelial cells
  267. Myocardial uptake and biodistribution of newly designed technetium-labelled fatty acid analogues
  268. Synthesis and radiopharmacological characterization of [11C]AL-438 as a nonsteroidal ligand for imaging brain glucocorticoid receptors
  269. Glycoxidised LDL isolated from subjects with impaired glucose tolerance increases CD36 and peroxisome proliferator–activator receptor γ gene expression in macrophages
  270. Labeling of low-density lipoproteins using the 18F-labeled thiol-reactive reagent N-[6-(4-[18F]fluorobenzylidene)aminooxyhexyl]maleimide
  271. Lipid transfer protein activities in subjects with impaired glucose tolerance
  272. Synthesis and Biological Evaluation of a New Type of99mTechnetium-Labeled Fatty Acid for Myocardial Metabolism Imaging
  273. Biodistribution and catabolism of 18F-labeled N-ε-fructoselysine as a model of Amadori products
  274. Positron emission tomography in food sciences
  275. Glucose-Induced Enhancement of Hemin-Catalyzed LDL Oxidation In Vitro and In Vivo
  276. Small animal positron emission tomography in food sciences
  277. Catabolism of native and oxidized low density lipoproteins: in vivo insights from small animal positron emission tomography studies
  278. Synthesis and biodistribution of an 18F-labelled resveratrol derivative for small animal positron emission tomography
  279. Biodistribution and catabolism of 18F-labelled isopeptide Nɛ-(γ-glutamyl)-L-lysine
  280. Fluorine-18 radiolabeling of low-density lipoproteins: a potential approach for characterization and differentiation of metabolism of native and oxidized low-density lipoproteins in vivo
  281. Oxidativ modifizierte Lipoproteine und deren Antik�rper bei Patienten mit Antiphospholipidsyndrom und Systemischem Lupus erythematodes
  282. The pivotal role of scavenger receptor CD36 and phagocyte-derived oxidants in oxidized low density lipoprotein-induced adhesion to endothelial cells
  283. The protective effects of HDL and its constitutents against neutrophil respiratory burst activation by hypochlorite-oxidized LDL
  284. The effect of garlic on arteriosclerotic nanoplaque formation and size
  285. Analysis of non-protein amino acids as specific markers of low density lipoprotein apolipoprotein B-100 oxidation in human atherosclerotic lesions: the use ofN(O)-ethoxycarbonyl trifluoroethyl ester derivatives and GC-MS1
  286. Analysis of 6-hydroxy-2-aminocaproic acid (HACA) as a specific marker of protein oxidation: The use of N(O,S)-ethoxycarbonyl trifluoroethyl ester derivatives and gas chromatography/mass spectrometry
  287. Measurement of 5-hydroxy-2-aminovaleric acid as a specific marker of metal catalysed oxidation of proline and arginine residues of low density lipoprotein apolipoprotein B-100 in human atherosclerotic lesions
  288. Lack of Association between Serum Paraoxonase 1 Activities and Increased Oxidized Low-Density Lipoprotein Levels in Impaired Glucose Tolerance and Newly Diagnosed Diabetes Mellitus
  289. Analysis of 3-chlorotyrosine as a specific marker of protein oxidation: the use ofN(O,S)-ethoxycarbonyltrifluoroethyl ester derivatives and gas chromatography/mass spectrometry
  290. Validation of different chemilumigenic substrates for detecting extracellular generation of reactive oxygen species by phagocytes and endothelial cells
  291. In Vivo Evidence for Increased Oxidation of Circulating LDL in Impaired Glucose Tolerance
  292. Protective Effects of Native But Not Oxidized High-Density Lipoprotein against Proinflammatory Respiratory Burst Activities of Polymorphonuclear Leukocytes Induced by Hypochlorite-Oxidized Low-Density Lipoprotein
  293. UVB-Induced Conversion of 7-Dehydrocholesterol to 1α,25-Dihydroxyvitamin D3 in an In Vitro Human Skin Equivalent Model
  294. Homocysteine levels in patients treated with lipid apheresis: effect of a vitamin therapy
  295. Different susceptibility to oxidation of proline and arginine residues of apolipoprotein B-100 among subspecies of low density lipoproteins
  296. Oxidation of Apolipoprotein B-100 in Circulating LDL Is Related to LDL Residence Time
  297. Impaired glucose tolerance (IGT) is not associated with disturbed homocysteine metabolism
  298. Conversion of vitamin D3 to 1alpha,25-dihydroxyvitamin D3 in human skin equivalents
  299. Measurement of 5-Hydroxy-2-aminovaleric Acid as a Specific Marker of Iron-Mediated Oxidation of Proline and Arginine Side-Chain Residues of Low-Density Lipoprotein Apolipoprotein B-100
  300. Urate modifies lipoprotein oxidation
  301. Human secretory group IIA phospholipase A2 is associated with lipid metabolism
  302. Störungen des Lipid- und Lipoproteinstoffwechsels
  303. Metabolic Basis of Low High Density Lipoprotein in Subjects with Impaired Glucose Tolerance
  304. Very Low Density Lipoprotein Overproduction Is Maximally Expressed in Early Insulin Resistant States
  305. In vivo evidence for increased apolipoprotein A-I catabolism in subjects with impaired glucose tolerance
  306. Human keratinocyte line HaCaT metabolizes 1α-hydroxyvitamin D3 and vitamin D3 to 1α,25-dihydroxyvitamin D3 (calcitriol)
  307. Determination of Total Homocysteine
  308. Hypochlorite-modified low-density lipoprotein stimulates human polymorphonuclear leukocytes for enhanced production of reactive oxygen metabolites, enzyme secretion, and adhesion to endothelial cells
  309. Stable isotope ratio analysis of amino acids: the use ofN(O,S)-ethoxycarbonyl trifluoroethyl ester derivatives and gas chromatography/mass spectrometry
  310. Stable isotope ratio analysis of amino acids: the use of N(O,S)-ethoxycarbonyl trifluoroethyl ester derivatives and gas chromatography/mass spectrometry
  311. Rapid Determination of Total Homocysteine in Human Plasma by Using N(O,S)-Ethoxycarbonyl Ethyl Ester Derivatives and Gas Chromatography–Mass Spectrometry,
  312. Very fast ultracentrifugation of serum lipoproteins: influence on lipoprotein separation and composition
  313. Recovery of Cholesterol and Triacylglycerol in Very-Fast Ultracentrifugation of Human Lipoproteins in a Large Range of Concentrations
  314. Very-fast ultracentrifugation of human plasma lipoproteins: influence of the centrifugal field on lipoprotein composition