Dr Anthony P Davenport
Current affiliation: University of Cambridge
Subject: Medicine And Medical Sciences
Primary location: United Kingdom
Functional and immunocytochemical evidence for a role of ghrelin and des-octanoyl ghrelin in the regulation of vascular tone in man
Published in:Cardiovascular Research
Publication date:2006-01-01
Expression and vasoconstrictor function of anorexigenic peptides neuromedin U-25 and S in the human cardiovascular system
Published in:Cardiovascular Research
Publication date:2008-12-01
Endothelin receptor antagonism in patients with chronic heart failure
Published in:Cardiovascular Research
Publication date:2000-07-01
The CCR5 chemokine receptor mediates vasoconstriction and stimulates intimal hyperplasia in human vessels in vitro
Published in:Cardiovascular Research
Publication date:2013-12-09
Presence of messenger ribonucleic acid for endothelin-1, endothelin-2, and endothelin-3 in human endometrium and a change in the ratio of ETA and E...
Published in:The Journal of Clinical Endocrinology & Metabolism
Publication date:1992-12-01
The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands
Published in:Nucleic Acids Research
Publication date:2015-10-12What's it about?Databases have become central to all the biomedical sciences. This one has a focus on pharmacology and indexes thousands of chemical strcutures, i...
The endothelin hormones, structure and function
Published in:Pharmacological Reviews
Publication date:2016-03-08What's it about?The is a review of endothelins, a family of three structurally similar 21-amino acid peptides. Endothelin-1 and -2 activate two G-protein coupled r...
Endothelins in reproduction
Published in:Reproductive Medicine Review
Publication date:1992-03-01
Chemokine receptor CCR5: from AIDS to atherosclerosis
Published in:British Journal of Pharmacology
Publication date:2011-03-04CCR5: from AIDS to atherosclerosis
Characterisation of Immunoreactive Endothelin in Human kidney by RP-HPLC and RIA
Published in:Clinical Science
Publication date:1993-03-01
Mitogenic Effects of Vasoactive Peptides on Rat Vascular Smooth Muscle Cells
Published in:Clinical Science
Publication date:1991-03-01
Emerging pharmacology and physiology of neuromedin U and the structurally related peptide neuromedin S
Published in:British Journal of Pharmacology
Publication date:2009-09-01
Validation of mRNA Quantification in Human Kidney by a Novel Fluorescent Nested RT-PCR Method
Published in:Clinical Science
Publication date:1994-01-01
The IUPHAR/BPS Guide to PHARMACOLOGY: an expert-driven knowledgebase of drug targets and their ligands
Published in:Nucleic Acids Research
Publication date:2013-11-14
GuideToPharmacology.org - an update
Published in:British Journal of Pharmacology
Publication date:2012-09-25Editorial
The Concise Guide to PHARMACOLOGY 2015/16: G protein-coupled receptors
Published in:British Journal of Pharmacology
Publication date:2015-12-01The Concise Guide to PHARMACOLOGY 2015/16: G protein-coupled receptors
Endothelin ETA receptors predominate in chronic thromboembolic pulmonary hypertension
Published in:Life Sciences
Publication date:2016-08-01
International Union of Pharmacology. LXXII. Recommendations for Trace Amine Receptor Nomenclature
Published in:Pharmacological Reviews
Publication date:2009-03-06
International Union of Basic and Clinical Pharmacology. LXXVII. Kisspeptin Receptor Nomenclature, Distribution, and Function
Published in:Pharmacological Reviews
Publication date:2010-11-15
International Union of Basic and Clinical Pharmacology. LXXIV. Apelin Receptor Nomenclature, Distribution, Pharmacology, and Function
Published in:Pharmacological Reviews
Publication date:2010-07-06
International Union of Basic and Clinical Pharmacology. LXXXVIII. G Protein-Coupled Receptor List: Recommendations for New Pairings with Cognate Li...
Published in:Pharmacological Reviews
Publication date:2013-05-17
International Union of Pharmacology. XLVI. G Protein-Coupled Receptor List
Published in:Pharmacological Reviews
Publication date:2005-06-01
International Union of Pharmacology. LVI. Ghrelin Receptor Nomenclature, Distribution, and Function
Published in:Pharmacological Reviews
Publication date:2005-12-01
Regional Hemodynamic Actions of Selective Corticotropin-Releasing Factor Type 2 Receptor Ligands in Conscious Rats
Published in:Journal of Pharmacology and Experimental Therapeutics
Publication date:2004-08-11
The dual endothelin converting enzyme/neutral endopeptidase inhibitor SLV-306 (daglutril), inhibits systemic conversion of big endothelin-1 in humans
Published in:Life Sciences
Publication date:2012-10-01
Preface
Published in:Journal of Cardiovascular Pharmacology
Publication date:2000-01-01
18 F-Fluoride and 18 F-Fluorodeoxyglucose Positron Emission Tomography After Transient Ischemic At...
Published in:Circulation Cardiovascular Imaging
Publication date:2017-03-01Case–Control Study
Smooth Muscle Endothelin B Receptors Regulate Blood Pressure but Not Vascular Function or Neointimal RemodelingNovelty and Significance
Published in:Hypertension
Publication date:2016-12-27
Elabela/Toddler Is an Endogenous Agonist of the Apelin APJ Receptor in the Adult Cardiovascular System, and Exogenous Administration of the Peptide...
Published in:Circulation
Publication date:2017-01-30
[Pyr1]Apelin-13(1–12) Is a Biologically Active ACE2 Metabolite of the Endogenous Cardiovascular Peptide [Pyr1]Apelin-13
Published in:Frontiers in Neuroscience
Publication date:2017-02-28
Cardiac action of the first G protein biased small molecule apelin agonist
Published in:Biochemical Pharmacology
Publication date:2016-09-01
The Prodomain-bound Form of Bone Morphogenetic Protein 10 Is Biologically Active on Endothelial Cells
Published in:Journal of Biological Chemistry
Publication date:2015-12-02
Apelin, Elabela/Toddler, and biased agonists as novel therapeutic agents in the cardiovascular system
Published in:Trends in Pharmacological Sciences
Publication date:2015-09-01
LGR5 Activates Noncanonical Wnt Signaling and Inhibits Aldosterone Production in the Human Adrenal
Published in:The Journal of Clinical Endocrinology & Metabolism
Publication date:2015-06-01
Design, Characterization, and First-In-Human Study of the Vascular Actions of a Novel Biased Apelin Receptor Agonist
Published in:Hypertension
Publication date:2015-02-23
Endothelin Receptors and Their Antagonists
Published in:Seminars in Nephrology
Publication date:2015-03-01
Identifying active vascular microcalcification by 18F-sodium fluoride positron emission tomography
Published in:Nature Communications
Publication date:2015-07-07
Endothelin@25 - new agonists, antagonists, inhibitors and emerging research frontiers: IUPHAR Review 12
Published in:British Journal of Pharmacology
Publication date:2014-11-24Endothelin@25
Changes in biomechanical properties of the coronary artery wall contribute to maintained contractile responses to endothelin-1 in atherosclerosis
Published in:Life Sciences
Publication date:2014-11-01
Modulation of endothelin receptors in the failing right ventricle of the heart and vasculature of the lung in human pulmonary arterial hypertension
Published in:Life Sciences
Publication date:2014-11-01
Characterization of [125I]GLP-1(9-36), a novel radiolabeled analog of the major metabolite of glucagon-like peptide 1 to a receptor distinct from G...
Published in:Life Sciences
Publication date:2014-05-01
The Concise Guide to PHARMACOLOGY 2013/14: Overview
Published in:British Journal of Pharmacology
Publication date:2013-12-01Overview
Evolving pharmacology of orphan GPCRs: IUPHAR Commentary
Published in:British Journal of Pharmacology
Publication date:2013-10-01Evolving pharmacology of GPCRs
Somatic mutations in ATP1A1 and CACNA1D underlie a common subtype of adrenal hypertension
Published in:Nature Genetics
Publication date:2013-08-04
Screening β-Arrestin Recruitment for the Identification of Natural Ligands for Orphan G-Protein–Coupled Receptors
Published in:Journal of Biomolecular Screening
Publication date:2013-06-01
Endothelin-2, the forgotten isoform: emerging role in the cardiovascular system, ovarian development, immunology and cancer
Published in:British Journal of Pharmacology
Publication date:2012-12-20Emerging role of ET-2
IUPHAR-DB: updated database content and new features
Published in:Nucleic Acids Research
Publication date:2012-10-18
Themed section: endothelin
Published in:British Journal of Pharmacology
Publication date:2012-12-20Themed section. Endothelin
No evidence for a local renin-angiotensin system in liver mitochondria
Published in:Scientific Reports
Publication date:2013-08-20
Comparison of endothelin receptors in normal versus cirrhotic human liver and in the liver from endothelial cell-specific ETB knockout mice
Published in:Life Sciences
Publication date:2012-10-01
Comparison of human ETA and ETB receptor signalling via G-protein and β-arrestin pathways
Published in:Life Sciences
Publication date:2012-10-01
Defining the affinity and receptor sub-type selectivity of four classes of endothelin antagonists in clinically relevant human cardiovascular tissues
Published in:Life Sciences
Publication date:2012-10-01
The Twelfth International Conference on Endothelin (ET-12), Cambridge 2011
Published in:Life Sciences
Publication date:2012-10-01
Cellular Localization of Receptors Using Antibodies Visualized by Light and Dual Labeling Confocal Microscopy
Published in:Receptor Binding Techniques
Publication date:2012-01-01
Dynamic In Vivo Imaging of Receptors in Small Animals Using Positron Emission Tomography
Published in:Receptor Binding Techniques
Publication date:2012-01-01
How to Use the IUPHAR Receptor Database to Navigate Pharmacological Data
Published in:Receptor Binding Techniques
Publication date:2012-01-01
Quantitative Phosphor Imaging Autoradiography of Radioligands for Positron Emission Tomography
Published in:Receptor Binding Techniques
Publication date:2012-01-01
Radioligand Binding Assays and Their Analysis
Published in:Receptor Binding Techniques
Publication date:2012-01-01
Discovery of a Competitive Apelin Receptor (APJ) Antagonist
Published in:ChemMedChem
Publication date:2011-05-10
Inotropic Action of the Puberty Hormone Kisspeptin in Rat, Mouse and Human: Cardiovascular Distribution and Characteristics of the Kisspeptin Receptor
Published in:PLoS ONE
Publication date:2011-11-22
Pharmacology of Renal Endothelin Receptors
Published in:Contributions to Nephrology
Publication date:2011-01-01
Evidence for a novel vasospastic transmitter system, neuromedin U, in the equine digital circulation
Published in:The Veterinary Journal
Publication date:2010-10-01
Modulation of the apelin/APJ system in heart failure and atherosclerosis in man
Published in:British Journal of Pharmacology
Publication date:2010-04-26Apelin/APJ system in human cardiovascular disease
Endothelial cell-specific ETBreceptor knockout: autoradiographic and histological characterisation and crucial role in the clearance of endothelin-...
Published in:Canadian Journal of Physiology and Pharmacology
Publication date:2010-06-01
Evaluation of translocator protein quantification as a tool for characterising macrophage burden in human carotid atherosclerosis
Published in:Atherosclerosis
Publication date:2010-06-01
Introduction
Published in:Canadian Journal of Physiology and Pharmacology
Publication date:2010-06-01
Positron emission tomography of [18F]-big endothelin-1 reveals renal excretion but tissue-specific conversion to [18F]-endothelin-1 in lung and liver
Published in:British Journal of Pharmacology
Publication date:2010-02-01PET imaging of tissue conversion of [18F]-big ET-1
EDITORIAL
Published in:British Journal of Pharmacology
Publication date:2010-02-01Editorial
FDG–PET can distinguish inflamed from non-inflamed plaque in an animal model of atherosclerosis
Published in:The International Journal of Cardiovascular Imaging
Publication date:2009-09-22
[Pyr1]Apelin-13 Identified as the Predominant Apelin Isoform in the Human Heart: Vasoactive Mechanisms and Inotropic Action in Disease
Published in:Hypertension
Publication date:2009-07-13
IUPHAR-DB: the IUPHAR database of G protein-coupled receptors and ion channels
Published in:Nucleic Acids Research
Publication date:2008-10-23
Automated synthesis of the generic peptide labelling agent N-succinimidyl 4-[18F]fluorobenzoate and application to 18F-label the vasoactive transmi...
Published in:Nuclear Medicine and Biology
Publication date:2008-08-01
Chronic Apoptosis of Vascular Smooth Muscle Cells Accelerates Atherosclerosis and Promotes Calcification and Medial Degeneration
Published in:Circulation Research
Publication date:2008-05-15
Immunocytochemical localization of the urotensin-II receptor, UT, to rat and human tissues: Relevance to function
Published in:Peptides
Publication date:2008-05-01
Haemodynamic and renal effects of endothelin receptor antagonism in patients with chronic kidney disease
Published in:Nephrology Dialysis Transplantation
Publication date:2007-06-05
Kisspeptins: a multifunctional peptide system with a role in reproduction, cancer and the cardiovascular system
Published in:British Journal of Pharmacology
Publication date:2009-01-29Kisspeptins are multifunctional peptides
Strategy for improved [11C]DAA1106 radiosynthesis and in vivo peripheral benzodiazepine receptor imaging using microPET, evaluation of [11C]DAA1106
Published in:Nuclear Medicine and Biology
Publication date:2007-05-01
Kisspeptins Are Novel Potent Vasoconstrictors in Humans, with a Discrete Localization of Their Receptor, G Protein-Coupled Receptor 54, to Atherosc...
Published in:Endocrinology
Publication date:2007-01-01
Characterization of the snake venom ligand [125I]-DNP binding to natriuretic peptide receptor-A in human artery and potent DNP mediated vasodilatation
Published in:British Journal of Pharmacology
Publication date:2006-12-01
Apoptosis of vascular smooth muscle cells induces features of plaque vulnerability in atherosclerosis
Published in:news nature com
Publication date:2006-08-06
Deletion of Endothelial Cell Endothelin B Receptors Does Not Affect Blood Pressure or Sensitivity to Salt
Published in:Hypertension
Publication date:2006-06-26
Neuropeptide B and W: neurotransmitters in an emerging G-protein-coupled receptor system
Published in:British Journal of Pharmacology
Publication date:2006-08-01
Novel Snake Venom Ligand Dendroaspis Natriuretic Peptide Is Selective for Natriuretic Peptide Receptor-A in Human Heart: Downregulation of Natriure...
Published in:Circulation Research
Publication date:2006-07-21
Regional heterogeneity in the haemodynamic responses to urotensin II infusion in relation to UT receptor localisation
Published in:British Journal of Pharmacology
Publication date:2009-01-30Urotensin II receptors and haemodynamics
Regulation of vascular reactivity by established and emerging GPCRs
Published in:Trends in Pharmacological Sciences
Publication date:2005-07-27
Emerging roles of apelin in biology and medicine
Published in:Pharmacology & Therapeutics
Publication date:2005-08-01
Immunocytochemical localisation of the apelin receptor, APJ, to human cardiomyocytes, vascular smooth muscle and endothelial cells
Published in:Regulatory Peptides
Publication date:2005-03-01
Positron emission tomography using 18F-labelled endothelin-1 reveals prevention of binding to cardiac receptors owing to tissue-specific clearance ...
Published in:British Journal of Pharmacology
Publication date:2009-01-29Dynamic PET imaging of endothelin receptors
Dynamic In Vivo Imaging of Receptors in Small Animals Using Positron Emission Tomography
Published in:Receptor Binding Techniques
Publication date:Not available
Imaging and Characterization of Radioligands for Positron Emission Tomography Using Quantitative Phosphor Imaging Autoradiography
Published in:Receptor Binding Techniques
Publication date:Not available
Immunocytochemical Localization of Receptors Using Light and Confocal Microscopy With Application to the Phenotypic Characterization of Knock-Out Mice
Published in:Receptor Binding Techniques
Publication date:Not available
Radioligand-Binding and Molecular-Imaging Techniques for the Quantitative Analysis of Established and Emerging Orphan Receptor Systems
Published in:Receptor Binding Techniques
Publication date:Not available
Alternative Pathway to Endothelin-Converting Enzyme for the Synthesis of Endothelin in Human Blood Vessels
Published in:Journal of Cardiovascular Pharmacology
Publication date:2004-11-01
Comparison of Endothelin-A and Endothelin-B Receptor Distribution Visualized by Radioligand Binding versus Immunocytochemical Localization using Su...
Published in:Journal of Cardiovascular Pharmacology
Publication date:2004-11-01
Down-regulation of ETA Receptors in ETB Receptor-deficient Mice
Published in:Journal of Cardiovascular Pharmacology
Publication date:2004-11-01
Endothelin Receptor Pharmacology and Function in the Mouse: Comparison with Rat and Man
Published in:Journal of Cardiovascular Pharmacology
Publication date:2004-11-01
In Vivo Imaging of Cardiovascular Endothelin Receptors Using the Novel Radiolabelled Antagonist [18F]-SB209670 and Positron Emission Tomography (mi...
Published in:Journal of Cardiovascular Pharmacology
Publication date:2004-11-01
CRF2receptors are highly expressed in the human cardiovascular system and their cognate ligands urocortins 2 and 3 are potent vasodilators
Published in:British Journal of Pharmacology
Publication date:2004-10-01
Cellular distribution of immunoreactive urotensin-II in human tissues with evidence of increased expression in atherosclerosis and a greater constr...
Published in:Peptides
Publication date:2004-10-01
Identification and cellular localisation of NPW1 (GPR7) receptors for the novel neuropeptide W-23 by [125I]-NPW radioligand binding and immunocytoc...
Published in:Brain Research
Publication date:2004-08-01
Immunocytochemical localization of the endogenous vasoactive peptide apelin to human vascular and endocardial endothelial cells
Published in:Regulatory Peptides
Publication date:2004-05-01
Maternal Dexamethasone Increases Endothelin-1 Sensitivity and Endothelin A Receptor Expression in Ovine Foetal Placental Arteries
Published in:Placenta
Publication date:2003-04-01
Peptide and trace amine orphan receptors: prospects for new therapeutic targets
Published in:Current Opinion in Pharmacology
Publication date:2003-04-01
Translating the human genome: renaissance of cardiovascular receptor pharmacology
Published in:Current Opinion in Pharmacology
Publication date:2003-04-01
Is urotensin-II the new endothelin?
Published in:British Journal of Pharmacology
Publication date:2002-11-01
Comparison of vasodilators in human internal mammary artery: ghrelin is a potent physiological antagonist of endothelin-1
Published in:British Journal of Pharmacology
Publication date:2002-08-01
Imaging Atherosclerotic Plaque Inflammation With [18F]-Fluorodeoxyglucose Positron Emission Tomography
Published in:Circulation
Publication date:2002-05-20
International Union of Pharmacology. XXIX. Update on Endothelin Receptor Nomenclature
Published in:Pharmacological Reviews
Publication date:2002-06-01
Discovery of recently adopted orphan receptors for apelin, urotensin II, and ghrelin identified using novel radioligands and functional role in the...
Published in:Canadian Journal of Physiology and Pharmacology
Publication date:2002-05-01
Of mice and men: advances in endothelin research and first antagonist gains FDA approval
Published in:Trends in Pharmacological Sciences
Publication date:2002-04-01
Radioligand binding reveals chymase as the predominant enzyme for mediating tissue conversion of angiotensin I in the normal human heart
Published in:Clinical Science
Publication date:2002-01-01
Thromboxane receptor density is increased in human cardiovascular disease with evidence for inhibition at therapeutic concentrations by the AT1rece...
Published in:British Journal of Pharmacology
Publication date:2001-12-01
Vasoconstrictor activity of novel endothelin peptide, ET-1(1 - 31), in human mammary and coronary arteriesin vitro
Published in:British Journal of Pharmacology
Publication date:2001-11-01
[125I-His9]-Ghrelin, a novel radioligand for localizing GHS orphan receptors in human and rat tissue; up-regulation of receptors with atherosclerosis
Published in:British Journal of Pharmacology
Publication date:2001-09-01
Physiological antagonism of endothelin-1 in human conductance and resistance coronary artery
Published in:British Journal of Pharmacology
Publication date:2001-06-01
Depressor and regionally-selective vasodilator effects of human and rat urotensin II in conscious rats
Published in:British Journal of Pharmacology
Publication date:2001-04-01
The endothelin system in human saphenous vein graft disease
Published in:Current Opinion in Pharmacology
Publication date:2001-04-01
[125I]-(Pyr1)Apelin-13 is a novel radioligand for localizing the APJ orphan receptor in human and rat tissues with evidence for a vasoconstrictor r...
Published in:British Journal of Pharmacology
Publication date:2001-03-01
Nitric oxide-mediated modulation of the endothelin-1 signalling pathway in the human cardiovascular system
Published in:British Journal of Pharmacology
Publication date:2001-01-01
Cellular Expression of Isoforms of Endothelin-Converting Enzyme-1 (ECE-1c, ECE-1b and ECE-1a) and Endothelin-Converting Enzyme-2
Published in:Journal of Cardiovascular Pharmacology
Publication date:2000-01-01
Changes in ETA-, AT1- and AT2-Receptors in the Phenotypically Transformed Intimal Smooth Muscle Layer of Human Atherosclerotic Coronary Arteries
Published in:Journal of Cardiovascular Pharmacology
Publication date:2000-01-01
Endothelin-A-Receptors in Human Aorta and Pulmonary Arteries are Downregulated in Patients With Cardiovascular Disease
Published in:Journal of Cardiovascular Pharmacology
Publication date:2000-01-01An Adaptive Response to Increased Levels of Endothelin-1?
Expression and Characterization of the Human Endothelin-A-Receptor in Pichia pastoris
Published in:Journal of Cardiovascular Pharmacology
Publication date:2000-01-01Influence of N-Terminal Epitope Tags
No Alteration in Vasoconstrictor Endothelin-B-Receptor Density or Function in Human Coronary Artery Disease
Published in:Journal of Cardiovascular Pharmacology
Publication date:2000-01-01
Novel Nitric Oxide Donors Reverse Endothelin-1-Mediated Constriction in Human Blood Vessels
Published in:Journal of Cardiovascular Pharmacology
Publication date:2000-01-01
Syntheses of the First Endothelin-A- and -B-Selective Radioligands for Positron Emission Tomography
Published in:Journal of Cardiovascular Pharmacology
Publication date:2000-01-01
Tissue-Specific Modulation of Endothelin Receptors in a Rat Model of Hypertension
Published in:Journal of Cardiovascular Pharmacology
Publication date:2000-01-01
Orphan-receptor ligand human urotensin II: receptor localization in human tissues and comparison of vasoconstrictor responses with endothelin-1
Published in:British Journal of Pharmacology
Publication date:2000-10-01
Urotensin II: fish neuropeptide catches orphan receptor
Published in:Trends in Pharmacological Sciences
Publication date:2000-03-01
Evidence for Intracellular Endothelin-Converting Enzyme-2 Expression in Cultured Human Vascular Endothelial Cells
Published in:Circulation Research
Publication date:1999-04-30
Blockade and Reversal of Endothelin-Induced Constriction in Pial Arteries From Human Brain Editorial Comment
Published in:Stroke
Publication date:1999-03-01
Endothelin receptor expression and pharmacology in human saphenous vein graft
Published in:British Journal of Pharmacology
Publication date:1999-01-01
Secretory pathways in endothelin synthesis
Published in:British Journal of Pharmacology
Publication date:1999-01-01
The therapeutic potential of PD156707 and related butenolide endothelin antagonists
Published in:Expert Opinion on Investigational Drugs
Publication date:1999-01-01
Comparison of the vasoconstrictor effects of rizatriptan and sumatriptan in human isolated cranial arteries: immunohistological demonstration of th...
Published in:British Journal of Clinical Pharmacology
Publication date:2002-01-045-HT1B/1D-receptor agonists and vasoconstriction in human isolated arteries
The haemodynamic effects of iodinated water soluble radiographic contrast media: a review
Published in:European Journal of Radiology
Publication date:1998-11-01
Expression of EndothelinA Receptors in Human Gliomas and Meningiomas, with High Affinity for the Selective Antagonist PD156707
Published in:Neurosurgery
Publication date:1998-10-01
Increased response to big endothelin-1 in atherosclerotic human coronary artery: functional evidence for up-regulation of endothelin-converting enz...
Published in:British Journal of Pharmacology
Publication date:1998-09-01
Human Endothelial Cell Storage Granules : A Novel Intracellular Site for Isoforms of the Endothelin-Converting Enzyme
Published in:Circulation Research
Publication date:1998-08-10
Endothelin receptor subtypes and their functional relevance in human small coronary arteries
Published in:British Journal of Pharmacology
Publication date:1998-06-01
Evidence Using Immunoelectron Microscopy for Regulated and Constitutive Pathways in the Transport and Release of Endothelin
Published in:Journal of Cardiovascular Pharmacology
Publication date:1998-03-01
In vitro enzymatic processing of radiolabelled big ET-1 in human kidney
Published in:Biochemical Pharmacology
Publication date:1998-03-01
Characterization of [125I]-PD164333, an ETAselective non-peptide radiolabelled antagonist, in normal and diseased human tissues
Published in:British Journal of Pharmacology
Publication date:1998-01-01
Characterization of Site-Directed Antisera Against Endothelin-Converting Enzymes
Published in:Journal of Cardiovascular Pharmacology
Publication date:1998-01-01
Endothelin Peptide and Converting Enzymes in Human Endothelium
Published in:Journal of Cardiovascular Pharmacology
Publication date:1998-01-01
Endothelin-Converting Enzyme in the Human Vasculature: Evidence for Differential Conversion of Big Endothelin-3 by Endothelial and Smooth-Muscle Cells
Published in:Journal of Cardiovascular Pharmacology
Publication date:1998-01-01
PD156707: A Potent Antagonist of Endothelin-1 in Human Diseased Coronary Arteries and Vein Grafts
Published in:Journal of Cardiovascular Pharmacology
Publication date:1998-01-01
Relative Contribution of Endothelin A and Endothelin B Receptors to Vasoconstriction in Small Arteries from Human Heart and Brain
Published in:Journal of Cardiovascular Pharmacology
Publication date:1998-01-01
Endothelin converting enzyme (ECE) activity in human vascular smooth muscle
Published in:British Journal of Pharmacology
Publication date:1997-12-01
Detection of Endothelin Receptors in Human Coronary Artery Vascular Smooth Muscle Cells But Not Endothelial Cells by Using Electron Microscope Auto...
Published in:Journal of Cardiovascular Pharmacology
Publication date:1997-06-01
Differential distribution of endothelin receptor subtypes in placentae from normal and growth-restricted pregnancies
Published in:Placenta
Publication date:1997-03-01
Differential distribution of endothelin peptides and receptors in human adrenal gland
Published in:The Histochemical Journal
Publication date:1996-11-01
Characterization of the binding of endothelin ETB selective ligands in human and rat heart
Published in:British Journal of Pharmacology
Publication date:1996-10-01
Endothelin Peptide and Receptors in Human Atherosclerotic Coronary Artery and Aorta
Published in:Circulation Research
Publication date:1996-10-01
Selective downregulation of ETA receptor mRNA in renal transplant recipients on cyclosporin A revealed by quantitative RT-PCR
Published in:Nephrology Dialysis Transplantation
Publication date:1996-10-01
The increase in human plasma immunoreactive endothelin but not big endothelin-1 or its C-terminal fragment induced by systemic administration of th...
Published in:British Journal of Pharmacology
Publication date:1996-09-01
Endocrinology and paracrinology
Published in:MHR Basic science of reproductive medicine
Publication date:1996-01-01Localization of endothelin receptors in human uterus throughout the menstrual cycle
Failure of BQ123, a more potent antagonist of sarafotoxin 6b than of endothelin-1, to distinguish between these agonists in binding experiments
Published in:British Journal of Pharmacology
Publication date:1996-05-01
Endothelin receptors in human coronary artery and aorta
Published in:British Journal of Pharmacology
Publication date:1996-03-01
Characterization of the endothelin receptor selective agonist, BQ3020 and antagonists BQ123, FR139317, BQ788, 50235, Ro462005 and bosentan in the h...
Published in:British Journal of Pharmacology
Publication date:1996-02-01
Localization of endothelin peptides in human kidney
Published in:Kidney International
Publication date:1996-02-01
Endothelin ETA receptor expression in human cerebrovascular smooth muscle cells
Published in:British Journal of Pharmacology
Publication date:1995-11-01
Phosphoramidon inhibition of the in vivo conversion of big endothelin-1 to endothelin-1 in the human forearm
Published in:British Journal of Pharmacology
Publication date:1995-09-01
Endothelin expression in the uterus
Published in:The Journal of Steroid Biochemistry and Molecular Biology
Publication date:1995-06-01
ETA receptor-mediated constrictor responses to endothelin peptides in human blood vessels in vitro
Published in:British Journal of Pharmacology
Publication date:1995-05-01
Endothelin ETA and ETB mRNA and receptors expressed by smooth muscle in the human vasculature: majority of the ETA sub-type
Published in:British Journal of Pharmacology
Publication date:1995-03-01
ETA and ETB endothelin receptors in human myometrium characterized by the subtype selective ligands BQ123, BQ3020, FR139317 and PD151242
Published in:Journal of Endocrinology
Publication date:1995-01-01
Secretion of endothelin-1 and endothelin-3 by human cultured vascular smooth muscle cells
Published in:British Journal of Pharmacology
Publication date:1995-01-01
Selectivity of [125I]-PD 151242 for human, rat and porcine endothelin ETA receptors in the heart
Published in:British Journal of Pharmacology
Publication date:1995-01-01
[125I]-PD151242: a selective ligand for endothelin ETA receptors in human kidney which localizes to renal vasculature
Published in:British Journal of Pharmacology
Publication date:1994-12-01
Vasoconstrictor endothelin receptors characterized in human renal artery and vein in vitro
Published in:British Journal of Pharmacology
Publication date:1994-09-01
Quantification of mRNA in Human Tissue Using Fluorescent Nested Reverse-Transcriptase Polymerase Chain Reaction
Published in:Analytical Biochemistry
Publication date:1994-08-01
Effects of an ET1-receptor antagonist, FR139317, on regional haemodynamic responses to endothelin-1 and [Ala11,15]Ac-endothelin-1 (6-21) in conscio...
Published in:British Journal of Pharmacology
Publication date:1994-06-01
Is endothelin-induced vasoconstriction mediated only by ETA receptors in humans?
Published in:Trends in Pharmacological Sciences
Publication date:1994-01-01
[125I]-PD 151242: a selective radioligand for human ETA receptors
Published in:British Journal of Pharmacology
Publication date:1994-01-01
Novel ligands BQ123 and BQ3020 characterize endothelin receptor subtypes ETA and ETB in human kidney
Published in:Kidney International
Publication date:1993-07-01
Alternatively Spliced mRNAs for Human Endothelin-2 and Their Tissue Distribution
Published in:Biochemical and Biophysical Research Communications
Publication date:1993-06-01
Endothelin: progress in pharmacology and physiology
Published in:Trends in Pharmacological Sciences
Publication date:1993-06-01
Identification of endothelin-1, endothelin-2 and endothelin-3 in human endometrium
Published in:Reproduction
Publication date:1993-05-01
Characterization and localization of endothelin receptor subtypes in the human atrioventricular conducting system and myocardium
Published in:Circulation Research
Publication date:1993-03-01
Presence of messenger ribonucleic acid for endothelin-1, endothelin-2, and endothelin-3 in human endometrium and a change in the ratio of ETA and E...
Published in:The Journal of Clinical Endocrinology & Metabolism
Publication date:1992-12-01
Characterization of two new ETB selective radioligands, [125I]-BQ3020 and [125I]-[Ala1,3,11,15]ET-1 in human heart
Published in:British Journal of Pharmacology
Publication date:1992-11-01
Localization of immunoreactive endothelin and proendothelin in the human lung
Published in:Pulmonary Pharmacology
Publication date:1992-09-01
Endothelin-like immunoreactivity in human endometrium
Published in:Reproduction
Publication date:1992-07-01
Cerebellar neurons and glia respond differentially to endothelins and sarafotoxin S6b
Published in:Brain Research
Publication date:1992-05-01
Localization and endogenous concentration of endothelin-like immunoreactivity in human placenta
Published in:Journal of Endocrinology
Publication date:1991-12-01
Binding sites for125I ET-1, ET-2, ET-3 and vasoactive intestinal contractor are present in adult rat brain and neurone-enriched primary cultures of...
Published in:Brain Research
Publication date:1991-07-01
Binding sites for iodinated endothelin-1, endothelin-2 and endothelin-3 demonstrated on human uterine glandular epithelial cells by quantitative hi...
Published in:Journal of Endocrinology
Publication date:1991-04-01
Endothelin-1 stimulates prostaglandin F2α release from human endometrium
Published in:Prostaglandins Leukotrienes and Essential Fatty Acids
Publication date:1991-03-01
The endothelin peptides ET-1, ET-2, ET-3 and sarafotoxin S6b are co-mitogenic with platelet-derived growth factor for vascular smooth muscle cells
Published in:Atherosclerosis
Publication date:1990-12-01
Endothelin-1 mRNA is widely expressed in porcine and human tissues.
Published in:Journal of Clinical Investigation
Publication date:1990-05-01
Experimental hemiparkinsonism in the rat following chronic unilateral infusion of MPP+ into the nigrostriatal dopamine pathway—II. Differential loc...
Published in:Neuroscience
Publication date:1988-10-01
Comparison between brain paste and polymer [125I]standards for quantitative receptor autoradiography
Published in:Journal of Neuroscience Methods
Publication date:1988-08-01
Effect of the formamidine insecticide chordimeform on feeding and reproduction in the noctuid moth, Spodoptera littoralis (Boisduval)
Published in:Crop Protection
Publication date:1987-02-01
Sex-related differences in the concentration of Met-enkephalin-like immunoreactivity in the nervous system of an insect,Schistocerca gregaria, reve...
Published in:Brain Research
Publication date:1986-09-01
Biogenic amines in the brain of the honeybee, Apis mellifera
Published in:Cell and Tissue Research
Publication date:1983-12-01
Receptor Binding Techniques
Published in:Not available
Publication date:2005-03-25
Endothelin Receptors
Published in:xPharm: The Comprehensive Pharmacology Reference
Publication date:2007-01-01
Urotensin-II Receptor
Published in:xPharm: The Comprehensive Pharmacology Reference
Publication date:2007-01-01
Receptor Binding Techniques
Published in:Methods in Molecular Biology™
Publication date:2012-01-01
Peptide Research Protocols
Published in:Not available
Publication date:2002-06-25
ET-B Endothelin Receptor
Published in:xPharm: The Comprehensive Pharmacology Reference
Publication date:2007-01-01
ET-A Endothelin Receptor
Published in:xPharm: The Comprehensive Pharmacology Reference
Publication date:2007-01-01
Apelins and the Apelin Receptor
Published in:Encyclopedia of Molecular Pharmacology
Publication date:Not available
Radioligand Binding Assays and Quantitative Autoradiography of Endothelin Receptors
Published in:Peptide Research Protocols
Publication date:Not available
Analysis of Endothelins by Enzyme-Linked Immunosorbent Assay and Radioimmunoassay
Published in:Peptide Research Protocols
Publication date:Not available
Radioligand Binding Assays: Theory and Practice
Published in:Current Directions in Radiopharmaceutical Research and Development
Publication date:1996-01-01
Importance of Subtype Selectivity for Endothelin Receptor Antagonists in the Human Vasculature
Published in:Translational Vascular Medicine
Publication date:2011-10-06
International Union of Basic and Clinical Pharmacology CIII: Chemerin Receptors CMKLR1 (Chemerin1) and GPR1 (Chemerin2) Nomenclature, Pharmacology,...
Published in:Pharmacological Reviews
Publication date:2017-12-26
THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: G protein-coupled receptors
Published in:British Journal of Pharmacology
Publication date:2017-10-21THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: G protein-coupled receptors
THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Overview
Published in:British Journal of Pharmacology
Publication date:2017-10-21THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Overview
OUP accepted manuscript
Published in:Nucleic Acids Research
Publication date:2017-01-01
In Vivo Mapping of Vascular Inflammation Using the Translocator Protein Tracer 18 F-FEDAA1106
Published in:Molecular Imaging
Publication date:2014-08-01
Detection of Atherosclerotic Inflammation by 68 Ga-DOTATATE PET Compared to [ 18 F]FDG PET Imaging
Published in:Journal of the American College of Cardiology
Publication date:2017-04-01
Pharmacological targeting of apelin impairs glioblastoma growth
Published in:Brain
Publication date:2017-10-03
Vascular Imaging With 18 F-Fluorodeoxyglucose Positron Emission Tomography Is Influenced by Hypoxia
Published in:Journal of the American College of Cardiology
Publication date:2017-04-01
Chemerin Elicits Potent Constrictor Actions via Chemokine‐Like Receptor 1 (CMKLR1), not G‐Protein‐Coupled Receptor 1 (GPR1), in Human and Rat Vascu...
Published in:Journal of the American Heart Association
Publication date:2016-10-01
The Concise Guide to PHARMACOLOGY 2015/16: Overview
Published in:British Journal of Pharmacology
Publication date:2015-12-01The Concise Guide to PHARMACOLOGY 2015/16: Overview
The endothelin system in pulmonary and renal vasculopathy: les liaisons dangereuses
Published in:European Respiratory Review
Publication date:2009-11-30
Triptan-induced contractile (5-HT1Breceptor) responses in human cerebral and coronary arteries: relationship to clinical effect
Published in:Clinical Science
Publication date:2005-09-01
Emerging roles for orphan G-protein-coupled receptors in the cardiovascular system
Published in:Trends in Pharmacological Sciences
Publication date:2003-01-01
Life before birth: effects of cortisol on future cardiovascular and metabolic function*
Published in:Acta Paediatrica
Publication date:2003-01-01
Expression of Endothelin Peptides and Mrna in the Human Heart
Published in:Clinical Science
Publication date:1996-01-01
The endothelin system in the kidney
Published in:Nephrology
Publication date:1996-04-01
Davenport and Maguire reply
Published in:Trends in Pharmacological Sciences
Publication date:1994-05-01
Effects of Phosphoramidon and Pepstatin a on the Secretion of Endothelin-I and Big Endothelin-I by Human Umbilical Vein Endothelial Cells: Measurem...
Published in:Clinical Science
Publication date:1994-08-01
Isolation of Human Cardiac Endothelin Receptors by a Peptide-Receptor Mobility Shift Assay
Published in:Clinical Science
Publication date:1993-08-01
Quantitative autoradiography reveals higher densities of specific calcitonin-gene-related peptide receptors in small intramyocardial compared with ...
Published in:Clinical Science
Publication date:1993-01-01
Anatomical localization and pharmacological activity of mature endothelins and their precursors in human vascular tissue
Published in:Journal of Hypertension
Publication date:1992-11-01
Epidermal growth factor in human endometrium: proliferative effects in culture and immunocytochemical localization in normal and endometriotic tissues
Published in:Human Reproduction
Publication date:1991-10-01
A sensitive radioimmunoassay measuring endothelin-like immunoreactivity in human plasma: Comparison of levels in patients with essential hypertensi...
Published in:Clinical Science
Publication date:1990-03-01
Atrial natriuretic factor mRNA and binding sites in the adrenal gland
Published in:Biochemical Journal
Publication date:1990-10-15
Localisation off binding sites for iodinated endothelin and saraffotoxin peptides in mammalian tissues using quantitative receptor autoradiography
Published in:European Journal of Pharmacology
Publication date:1990-07-01
Binding Sites for125I-Labelled Endothelin-1 in the Kidneys: Differential Distribution in Rat, Pig and Man Demonstrated by Using Quantitative Autora...
Published in:Clinical Science
Publication date:1989-08-01
Octopamine distribution in the larvae and adults of two species of moth, Spodoptera littoralis and Manduca sexta
Published in:Journal of Insect Physiology
Publication date:1986-01-01
Quantitative receptor autoradiography
Published in:Nature
Publication date:1986-12-01
The action of formamidines on octopamine receptors in the locust
Published in:Pesticide Biochemistry and Physiology
Publication date:1985-08-01
Toxicity of chlordimeform and amitraz to the egyptian cotton leafworm (Spodoptera littoralis) and the tobacco budworm (Heliothis virescens)
Published in:Pesticide Science
Publication date:1985-02-01
Changes in haemolymph octopamine levels associated with food deprivation in the locust, Schistocerca gregaria
Published in:Physiological Entomology
Publication date:1984-09-01
Stress-induced changes in the octopamine levels of insect haemolymph
Published in:Insect Biochemistry
Publication date:1984-01-01