Dr Shailesh Natvarbhai Mistry
University of Nottingham
Professor, Pharmacy
United Kingdom
My co-authors include
Dr Kwok Ho Christopher Choy
Dr Sebastian George Barton Furness
Gopal Jadhav
Find me at
My Publications
27th Annual GP2A Medicinal Chemistry Conference
Pharmaceuticals
December 2019
Structure–Kinetic Profiling of Haloperidol Analogues at the Human Dopamine D2 Receptor
Journal of Medicinal Chemistry
October 2019
A Thieno[2,3-d]pyrimidine Scaffold Is a Novel Negative Allosteric Modulator of the Dopa...
Journal of Medicinal Chemistry
May 2018
Novel selective β1-adrenoceptor antagonists for concomitant cardiovascular and respirat...
The FASEB Journal
July 2017
New strategy to improve the current antipsychotics for treating symptoms of schizophrenia
Journal of Pharmacology and Experimental Therapeutics
September 2016
GPCRs through the keyhole: the role of protein flexibility in ligand binding to β-adren...
Journal of Biomolecular Structure and Dynamics
September 2016
Novel Fused Arylpyrimidinone Based Allosteric Modulators of the M1 Muscarinic Acetylcho...
ACS Chemical Neuroscience
March 2016
Potent dual inhibitors of Plasmodium falciparum M1 and M17 aminopeptidases through opti...
European Journal of Medicinal Chemistry
March 2016
4-Phenylpyridin-2-one Derivatives: A Novel Class of Positive Allosteric Modulator of th...
Journal of Medicinal Chemistry
December 2015
Discovery of a Novel Class of Negative Allosteric Modulator of the Dopamine D2 Receptor...
Journal of Medicinal Chemistry
August 2015
Structure–Activity Study of N-((trans)-4-(2-(7-Cyano-3,4-dihydroisoquinolin-2(1H)-yl)et...
Journal of Medicinal Chemistry
June 2015
Screening the Medicines for Malaria Venture "Malaria Box" against the Plasmodium falcip...
PLoS ONE
February 2015
Biased allosteric modulation at the CaS receptor engendered by structurally diverse cal...
British Journal of Pharmacology
December 2014
Two-Pronged Attack: Dual Inhibition of Plasmodium falciparum M1 and M17 Metalloaminopep...
Journal of Medicinal Chemistry
October 2014
Mechanistic Insights into Allosteric Structure-Function Relationships at the M1Muscarin...
Journal of Biological Chemistry
October 2014
Triphenylphosphonium Anhydride Trifluoromethanesulfonate
May 2014
Molecular Determinants of Allosteric Modulation at the M1Muscarinic Acetylcholine Receptor
Journal of Biological Chemistry
January 2014
Synthesis and Pharmacological Profiling of Analogues of Benzyl Quinolone Carboxylic Aci...
Journal of Medicinal Chemistry
June 2013
Synthesis and in Vitro and in Vivo Characterization of Highly β1-Selective β-Adrenocept...
Journal of Medicinal Chemistry
May 2013
4,5-Dihydro-1-[(1S)-1-(hydroxymethyl)-2,2-dimethylpropyl]-3-(2,4,6-trimethylphenyl)-1H-...
September 2012
Synthesis and Characterization of High-Affinity 4,4-Difluoro-4-bora-3a,4a-diaza-s-indac...
Journal of Medicinal Chemistry
October 2011
Triphenylphosphonium Anhydride Trifluoromethanesulfonate
September 2011