All Stories

  1. Study of SQ109 analogs binding to mycobacterium MmpL3 transporter using MD simulations and alchemical relative binding free energy calculations
  2. Synthesis and Testing of Analogs of the Tuberculosis Drug Candidate SQ109 against Bacteria and Protozoa: Identification of Lead Compounds against Mycobacterium abscessus and Malaria Parasites
  3. Probing Adamantane Arylhydroxamic Acids against Trypanosoma brucei and Trypanosoma cruzi
  4. Mapping the Melatonin Receptor. 8. Selective MT2 Agonists Derived from 5,6‐Dihydroindolo[2,1‐ a ]isoquinolines and Related Systems
  5. Biophysical Evaluation and In Vitro Controlled Release of Two Isomeric Adamantane Phenylalkylamines with Antiproliferative/Anticancer and Analgesic Activity
  6. Evidence for spontaneous cannabinoid withdrawal in mice
  7. Improved cyclobutyl nabilone analogs as potent CB1 receptor agonists
  8. An Overview on Target-Based Drug Design against Kinetoplastid Protozoan Infections: Human African Trypanosomiasis, Chagas Disease and Leishmaniases
  9. Selective MT 2 Melatonin Receptor Antagonist Modulates Circadian Activity via Inhibition of the Endogenous Melatonin Signal in the East Bound Jet Lag Model
  10. Pineal hormone melatonin as an adjuvant treatment for COVID‑19 (Review)
  11. Chemical Probes for Blocking of Influenza A M2 Wild-type and S31N Channels
  12. Repurposing current therapeutic regimens against SARS-CoV-2 (Review)
  13. Multicomponent Reaction of Aldehydes, Amines and Oxalacetate Analogues Leading to Biologically Attractive Pyrrole Derivatives
  14. Synthetic Melatonin Receptor Agonists and Antagonists
  15. Synthesis and evaluation of novel 2,4-disubstituted arylthiazoles against T. brucei
  16. Design, Synthesis and in vitro Controlled Release of New Adamantanodiarylketone Antimycobacterials
  17. New antitubercular isoniazid-based adamantane derivatives
  18. Synthesis of New Indole and Adamantane Amido Derivatives with Pharmacological Interest
  19. Synthesis and evaluation of new nifurtimox‐adamantane adducts with trypanocidal activity
  20. Synthesis of diphenoxyadamantane alkylamines with pharmacological interest
  21. Fluorine substituted methoxyphenylalkyl amides as potent melatonin receptor agonists
  22. Synthesis of Pyrrole derivatives-Multicomponent reaction-Microwave assisted
  23. Insights in Organometallic Synthesis of Various Adamantane Derivatives with Sigma Receptor-Binding Affinity and Antiproliferative/Anticancer Activity
  24. Synthesis of Adamantane Aminoethers with Antitubercular Potential
  25. Sigma Receptor (σR) Ligands with Antiproliferative and Anticancer Activity
  26. In vitro Controlled Release from Solid Pharmaceutical Formulations
  27. In vitro Controlled Release from Solid Pharmaceutical Formulations of two new Adamantane Aminoethers with Antitubercular Activity (I).
  28. 4-(1-Adamantyl)phenylalkylamines with Potential Antiproliferative Activity
  29. New hydrazones of 5-nitro-2-furaldehyde with adamantanealkanohydrazides: synthesis and in vitro trypanocidal activity
  30. Synthesis and Cytotoxicity of 4-(2-Adamantyl)phenylalkylamines
  31. New aminoadamantane derivatives with antiproliferative activity
  32. Synthesis and trypanocidal action of new adamantane substituted imidazolines
  33. New Adamantane Phenylalkylamines with σ-Receptor Binding Affinity and Anticancer Activity, Associated with Putative Antagonism of Neuropathic Pain
  34. New Adamantane Derivatives with Sigma Affinity and Antiproliferative Activity
  35. Synthesis, σ1, σ2-receptors binding affinity and antiproliferative action of new C1-substituted adamantanes
  36. Novel 1′,1′-Chain Substituted Hexahydrocannabinols: 9β-Hydroxy-3-(1-hexyl-cyclobut-1-yl)-hexahydrocannabinol (AM2389) a Highly Potent Cannabinoid Receptor 1 (CB1) Agonist
  37. Design and synthesis of new adamantyl-substituted antileishmanial ether phospholipids
  38. ChemInform Abstract: Microwave-Assisted Synthesis of Sodium Sulfonates: Precursors of Sulfonyl Chlorides and Fluorides.
  39. Microwave-assisted synthesis of sodium sulfonates precursors of sulfonyl chlorides and fluorides
  40. Design and Synthesis ofTrypanosoma bruceiActive 1-Alkyloxy and 1-Benzyloxyadamantano 2-Guanylhydrazones
  41. ChemInform Abstract: Synthesis of Conformationally Constrained Adamantane Imidazolines with Trypanocidal Activity.
  42. ChemInform Abstract: Conformationally Constrained Adamantaneoxazolines of Pharmacological Interest.
  43. Synthesis of conformationally constrained adamantane imidazolines with trypanocidal activity
  44. ChemInform Abstract: An Intriguing, Regioselective Synthesis of Novel 2-(1-Adamantylmethyl)tetrahydropyridines.
  45. Design, Synthesis, and Trypanocidal Activity of New Aminoadamantane Derivatives
  46. Conformationally Constrained Adamantaneoxazolines of Pharmacological Interest
  47. An Intriguing, Regioselective Synthesis of Novel 2-(1-Adamantylmethyl) tetrahydropyridines
  48. Heterocyclic rimantadine analogues with antiviral activity
  49. The novel GABA adamantane derivative (AdGABA): design, synthesis, and activity relationship with gabapentin