All Stories

  1. Increasing the Chemical Space of L-SIGN Specific Glycomimetics

    Article • Journal of Medicinal Chemistry, October 2025, American Chemical Society (ACS)

    Professor Anna Bernardi

  2. Expanding the Chemical Space of Sugar Frameworks by Quaternization of the Anomeric Carbon Atom

    Article • European Journal of Organic Chemistry, July 2025, Wiley

    Professor Anna Bernardi

  3. Increasing the chemical space of L-SIGN specific glycomimetics

    Article • June 2025, American Chemical Society (ACS)

    Professor Anna Bernardi

  4. Toward Dual-Target Glycomimetics against Two Bacterial Lectins to Fight Pseudomonas aeruginosa–Burkholderia cenocepacia Infections: A Biophysical Study

    Article • Journal of Medicinal Chemistry, April 2025, American Chemical Society (ACS)

    Professor Anna Bernardi

  5. Synthesis of α-arylglycosides by Ni-photoredox arylation of sugars with an organic photocatalyst

    Article • January 2025, American Chemical Society (ACS)

    Professor Anna Bernardi

  6. Achieving High Affinity for a Bacterial Lectin with Reversible Covalent Ligands

    Article • Journal of Medicinal Chemistry, October 2024, American Chemical Society (ACS)

    Professor Anna Bernardi

  7. Polyvalent Glycomimetic-Gold Nanoparticles Revealing Critical Roles of Glycan Display on Multivalent Lectin–Glycan Interaction Biophysics and Antiviral Properties

    Article • JACS Au, August 2024, American Chemical Society (ACS)

    Professor Anna Bernardi

  8. Polyvalent Glycomimetic-Gold Nanoparticle Conjugates reveal effects of glycan display on Multivalent Lectin-Glycan Interactions

    Article • January 2024, American Chemical Society (ACS)

    Professor Anna Bernardi

  9. Powerful Avidity with a Limited Valency for Virus-Attachment Blockers on DC-SIGN: Combining Chelation and Statistical Rebinding with Structural Plasticity of the Receptor

    Article • ACS Central Science, February 2023, American Chemical Society (ACS)

    Professor Anna Bernardi

  10. Identification of New L-Fucosyl and L-Galactosyl Amides as Glycomimetic Ligands of TNF Lectin Domain of BC2L-C from Burkholderia cenocepacia

    Article • Molecules, February 2023, MDPI AG

    Professor Anna Bernardi

  11. Scalemic natural products

    Article • Natural Product Reports, January 2023, Royal Society of Chemistry

    Professor Anna Bernardi

  12. Targeting a Multidrug-Resistant Pathogen: First Generation Antagonists of Burkholderia cenocepacia’s BC2L-C Lectin

    Article • ACS Chemical Biology, September 2022, American Chemical Society (ACS)

    Professor Anna Bernardi

  13. Front Cover: Precision Glycodendrimers for DC‐SIGN Targeting (Eur. J. Org. Chem. 29/2022)

    Article • European Journal of Organic Chemistry, July 2022, Wiley

    Professor Anna Bernardi

  14. Rhamnose-based glycomimetic for recruitment of endogenous anti-rhamnose antibodies

    Article • Tetrahedron Letters, June 2022, Elsevier

    Professor Anna Bernardi

  15. Precision Glycodendrimers for DC‐SIGN Targeting**

    Article • European Journal of Organic Chemistry, May 2022, Wiley

    Professor Anna Bernardi

  16. Glycomimetic ligands block the interaction of SARS-CoV-2 spike protein with C-type lectin co-receptors

    Article • Chemical Communications, January 2022, Royal Society of Chemistry

    Professor Anna Bernardi

  17. DC/L-SIGN recognition of spike glycoprotein promotes SARS-CoV-2 trans-infection and can be inhibited by a glycomimetic antagonist

    Article • PLoS Pathogens, May 2021, PLOS

    Professor Anna Bernardi

  18. One pot synthesis ofthio-glycosidesviaaziridine opening reactions

    Article • Organic & Biomolecular Chemistry, January 2021, Royal Society of Chemistry

    Professor Anna Bernardi

  19. Chemo‐Enzymatic Synthesis of S. mansoni O‐Glycans and Their Evaluation as Ligands for C‐Type Lectin Receptors MGL, DC‐SIGN, and DC‐SIGNR

    Article • Chemistry - A European Journal, September 2020, Wiley

    Professor Anna Bernardi

  20. Interfering with the Sugar Code: Ten Years Later

    Article • European Journal of Organic Chemistry, April 2020, Wiley

    Professor Anna Bernardi

  21. BC2L-C N-Terminal Lectin Domain Complexed with Histo Blood Group Oligosaccharides Provides New Structural Information

    Article • Molecules, January 2020, MDPI AG

    Professor Anna Bernardi

  22. Development of C-type lectin-oriented surfaces for high avidity glycoconjugates: towards mimicking multivalent interactions on the cell surface

    Article • Organic & Biomolecular Chemistry, January 2020, Royal Society of Chemistry

    Professor Anna Bernardi

  23. Development of c-type lectin oriented surfaces for high avidity glycoconjugates: towards mimicking multivalent interactions on the cell surface

    Article • September 2019, Cold Spring Harbor Laboratory Press

    Professor Anna Bernardi

  24. Design and synthesis of glycomimetics: Recent advances

    Article • Medicinal Research Reviews, July 2019, Wiley

    Professor Anna Bernardi

  25. Design and synthesis of constrained bicyclic molecules as candidate inhibitors of influenza A neuraminidase

    Article • PLOS One, February 2018, PLOS

    Professor Anna Bernardi

  26. Rational-Differential Design of Highly Specific Glycomimetic Ligands: Targeting DC-SIGN and Excluding Langerin Recognition

    Article • ACS Chemical Biology, January 2018, American Chemical Society (ACS)

    Professor Anna Bernardi

  27. Glycodendron–rhenium complexes as luminescent probes for lectin sensing

    Article • Organic & Biomolecular Chemistry, January 2018, Royal Society of Chemistry

    Professor Anna Bernardi

  28. Observation of a Tricyclic[4.1.0.02,4]heptane During a Michael Addition-Ring Closure Reaction and a Computational Study on Its Mechanism of Formation

    Article • The Journal of Organic Chemistry, November 2017, American Chemical Society (ACS)

    Professor Anna Bernardi

  29. From optimized monovalent ligands to size-controlled dendrimers: an efficient strategy towards high-activity DC-SIGN antagonists

    Article • Canadian Journal of Chemistry, September 2017, Canadian Science Publishing

    Professor Anna Bernardi

  30. Towards new cholera prophylactics and treatment: Crystal structures of bacterial enterotoxins in complex with GM1 mimics

    Article • Scientific Reports, May 2017, Nature

    Professor Anna Bernardi

  31. Frontispiece: Design of Allosteric Stimulators of the Hsp90 ATPase as New Anticancer Leads

    Article • Chemistry - A European Journal, April 2017, Wiley

    Professor Anna Bernardi

  32. Design of Allosteric Stimulators of the Hsp90 ATPase as New Anticancer Leads

    Article • Chemistry - A European Journal, March 2017, Wiley

    Professor Anna Bernardi

  33. Glyco-functionalized dinuclear rhenium(i) complexes for cell imaging

    Article • Organic & Biomolecular Chemistry, January 2017, Royal Society of Chemistry

    Professor Anna Bernardi

  34. Clickable Polymeric Coating for Glycan Microarrays

    Article • November 2016, Springer Science + Business Media

    Professor Anna Bernardi

  35. Pseudo-Mannosylated DC-SIGN Ligands as Immunomodulants

    Article • Scientific Reports, October 2016, Nature

    Professor Anna Bernardi

  36. A relevant pharmacological target in TBI

    Article • Journal of Cerebral Blood Flow & Metabolism, July 2016, SAGE Publications

    Maria-Grazia De Simoni, Matteo Stravalaci, Professor Anna Bernardi

  37. A New Surface Plasmon Resonance Assay for In Vitro Screening of Mannose-Binding Lectin Inhibitors

    Article • SLAS DISCOVERY, July 2016, SAGE Publications

    Matteo Stravalaci, Dr. Marco Gobbi, Professor Anna Bernardi

  38. Synthesis of Functionalized 2-(4-Hydroxyphenyl)-3-methylbenzofuran Allosteric Modulators of Hsp90 Activity

    Article • European Journal of Organic Chemistry, June 2016, Wiley

    Professor Anna Bernardi

  39. Glycoconjugates and Glycomimetics as Microbial Anti-Adhesives

    Article • Trends in Biotechnology, June 2016, Elsevier

    Professor Anna Bernardi

  40. Molecular Dynamics Simulations Reveal the Mechanisms of Allosteric Activation of Hsp90 by Designed Ligands

    Article • Scientific Reports, April 2016, Nature

    Professor Anna Bernardi

  41. Solution Behavior of Amphiphilic Glycodendrimers with a Rod-Like Core

    Article • Macromolecular Bioscience, February 2016, Wiley

    Professor Anna Bernardi

  42. Scaffold Optimisation of Tetravalent Antagonists of the Mannose Binding Lectin

    Article • Chemistry - A European Journal, January 2016, Wiley

    Professor Anna Bernardi, Matteo Stravalaci

  43. Detection and quantitative analysis of two independent binding modes of a small ligand responsible for DC-SIGN clustering

    Article • Organic & Biomolecular Chemistry, January 2016, Royal Society of Chemistry

    Professor Anna Bernardi, Pedro M Nieto

  44. Stereoselective innovative synthesis and biological evaluation of new real carba analogues of minimal epitope Manα(1,2)Man as DC-SIGN inhibitors

    Article • RSC Advances, January 2016, Royal Society of Chemistry

    Professor Anna Bernardi

  45. Synthesis and evaluation of influenza A viral neuraminidase candidate inhibitors based on a bicyclo[3.1.0]hexane scaffold

    Article • Organic & Biomolecular Chemistry, January 2016, Royal Society of Chemistry

    Professor Anna Bernardi

  46. Critical Role and Therapeutic Control of the Lectin Pathway of Complement Activation in an Abortion-Prone Mouse Mating

    Article • The Journal of Immunology, November 2015, The American Association of Immunologists

    Professor Anna Bernardi

  47. Activation of Hsp90 Enzymatic Activity and Conformational Dynamics through Rationally Designed Allosteric Ligands

    Article • Chemistry - A European Journal, August 2015, Wiley

    Professor Anna Bernardi

  48. Carbohydrates: A phenol sandwich fights diabetes

    Article • Nature Chemical Biology, August 2015, Nature

    Professor Anna Bernardi

  49. New “clickable” polymeric coating for glycan microarrays

    Article • Sensors and Actuators B Chemical, August 2015, Elsevier

    Professor Anna Bernardi, Professor Marco Buscaglia

  50. Designing nanomolar antagonists of DC-SIGN-mediated HIV infection: ligand presentation using molecular rods

    Article • Chemical Communications, January 2015, Royal Society of Chemistry

    Professor Anna Bernardi

  51. Effective Targeting of DC-SIGN by α-Fucosylamide Functionalized Gold Nanoparticles

    Article • Bioconjugate Chemistry, December 2014, American Chemical Society (ACS)

    Professor Anna Bernardi

  52. Comprehensive analysis of blood group antigen binding to classical and El Tor cholera toxin B-pentamers by NMR

    Article • Glycobiology, May 2014, Oxford University Press (OUP)

    Professor Anna Bernardi

  53. Unique DC-SIGN Clustering Activity of a Small Glycomimetic: A Lesson for Ligand Design

    Article • ACS Chemical Biology, May 2014, American Chemical Society (ACS)

    Professor Anna Bernardi

  54. Synthesis of potential allosteric modulators of Hsp90 by chemical glycosylation of Eupomatenoid-6

    Article • Carbohydrate Research, May 2014, Elsevier

    Professor Anna Bernardi

  55. A multivalent inhibitor of the DC-SIGN dependent uptake of HIV-1 and Dengue virus

    Article • Biomaterials, April 2014, Elsevier

    Professor Anna Bernardi

  56. Pseudo-Mannosylated DC-SIGN Ligands as Potential Adjuvants for HIV Vaccines

    Article • Viruses, January 2014, MDPI AG

    Professor Anna Bernardi

  57. A Facile Synthesis of α-N-Ribosyl-Asparagine and α-N-Ribosyl-Glutamine Building Blocks

    Article • Molecules, July 2013, MDPI AG

    Professor Anna Bernardi

  58. Synthesis and Characterization of Linker-Armed Fucose-Based Glycomimetics

    Article • European Journal of Organic Chemistry, July 2013, Wiley

    Professor Anna Bernardi

  59. Selective Targeting of Dendritic Cell-Specific Intercellular Adhesion Molecule-3-Grabbing Nonintegrin (DC-SIGN) with Mannose-Based Glycomimetics: Synthesis and Interaction Studies of Bis(benzylamide) Derivatives of a Pseudomannobioside

    Article • Chemistry - A European Journal, February 2013, Wiley

    Professor Anna Bernardi, Dr Jesus Angulo

  60. Structure of a Glycomimetic Ligand in the Carbohydrate Recognition Domain of C-type Lectin DC-SIGN. Structural Requirements for Selectivity and Ligand Design

    Article • Journal of the American Chemical Society, February 2013, American Chemical Society (ACS)

    Professor Anna Bernardi, Dr Jesus Angulo

  61. Efficient synthesis of phenylene-ethynylene rods and their use as rigid spacers in divalent inhibitors

    Article • Beilstein Journal of Organic Chemistry, January 2013, Beilstein Institut

    Professor Anna Bernardi

  62. Multivalent glycoconjugates as anti-pathogenic agents

    Article • Chemical Society Reviews, January 2013, Royal Society of Chemistry

    Francesco Sansone, Professor Alessandro Casnati, Professor Anna Bernardi, Paul Murphy

  63. Targeting MBL in cerebral ischemia induces long lasting protection with a wide therapeutic window

    Article • Immunobiology, November 2012, Elsevier

    Professor Anna Bernardi

  64. Targeting Mannose-Binding Lectin Confers Long-Lasting Protection With a Surprisingly Wide Therapeutic Window in Cerebral Ischemia

    Article • Circulation, August 2012, Wolters Kluwer Health

    Professor Anna Bernardi, Matteo Stravalaci

  65. Stereoselective Synthesis of α- and β-Glycofuranosyl Amides by Traceless Ligation of Glycofuranosyl Azides

    Article • Chemistry - A European Journal, April 2012, Wiley

    Professor Anna Bernardi

  66. Both El Tor and classical cholera toxin bind blood group determinants

    Article • Biochemical and Biophysical Research Communications, February 2012, Elsevier

    Professor Anna Bernardi

  67. A glycomimetic compound inhibits DC-SIGN-mediated HIV infection in cellular and cervical explant models

    Article • AIDS, January 2012, Wolters Kluwer Health

    Javier Rojo, Professor Anna Bernardi

  68. α-N-Linked glycopeptides: conformational analysis and bioactivity as lectin ligands

    Article • Organic & Biomolecular Chemistry, January 2012, Royal Society of Chemistry

    Professor Anna Bernardi

  69. Mannose binding lectin as a target for cerebral ischemic injury

    Article • Molecular Immunology, August 2011, Elsevier

    Professor Anna Bernardi

  70. 2-Azidoethoxy derivatives of 2-aminocyclohexanecarboxylic acids (ACHC): interesting building blocks for the synthesis of cyclic β-peptide conjugates

    Article • Tetrahedron, August 2011, Elsevier

    Professor Anna Bernardi

  71. Pseudosaccharide Functionalized Dendrimers as Potent Inhibitors of DC-SIGN Dependent Ebola Pseudotyped Viral Infection

    Article • Bioconjugate Chemistry, June 2011, American Chemical Society (ACS)

    Javier Rojo, Professor Anna Bernardi

  72. Synthesis of α-N-Linked Glycopeptides

    Article • European Journal of Organic Chemistry, May 2011, Wiley

    Professor Anna Bernardi

  73. Stereoselective synthesis of N-galactofuranosyl amides

    Article • Carbohydrate Research, March 2011, Elsevier

    Professor Anna Bernardi

  74. Insights into molecular recognition of LewisX mimics by DC-SIGN using NMR and molecular modelling

    Article • Organic & Biomolecular Chemistry, January 2011, Royal Society of Chemistry

    Professor Anna Bernardi, Dr Jesus Angulo

  75. Second generation of fucose-based DC-SIGN ligands : affinity improvement and specificity versus Langerin

    Article • Organic & Biomolecular Chemistry, January 2011, Royal Society of Chemistry

    Javier Rojo, Professor Anna Bernardi

  76. Design, synthesis and activity evaluation of mannose-based DC-SIGN antagonists

    Article • Molecular Diversity, November 2010, Springer Science + Business Media

    Professor Anna Bernardi

  77. DFG-in and DFG-out homology models of TrkB kinase receptor: Induced-fit and ensemble docking

    Article • Journal of Molecular Graphics and Modelling, November 2010, Elsevier

    Professor Anna Bernardi

  78. An assay for functional dendritic cell-specific ICAM-3-grabbing nonintegrin (DC–SIGN) inhibitors of human dendritic cell adhesion

    Article • Analytical Biochemistry, November 2010, Elsevier

    Professor Anna Bernardi

  79. Synthesis of non glycosidic nucleobase-sugar mimetics

    Article • Comptes Rendus Chimie, October 2010, Elsevier

    Professor Anna Bernardi

  80. HIV microbicides: state-of-the-art and new perspectives on the development of entry inhibitors

    Article • Future Medicinal Chemistry, July 2010, Future Science

    Javier Rojo, Professor Anna Bernardi

  81. Monovalent and bivalent N-fucosyl amides as high affinity ligands for Pseudomonas aeruginosa PA-IIL lectin

    Article • Carbohydrate Research, July 2010, Elsevier

    Professor Anna Bernardi

  82. Synthesis and Affinity Evaluation of a Small Library of Bidentate Cholera Toxin Ligands: Towards Nonhydrolyzable Ganglioside Mimics

    Article • Chemistry - A European Journal, February 2010, Wiley

    Professor Anna Bernardi

  83. Inhibition of DC-SIGN-Mediated HIV Infection by a Linear Trimannoside Mimic in a Tetravalent Presentation

    Article • ACS Chemical Biology, January 2010, American Chemical Society (ACS)

    Javier Rojo, Professor Anna Bernardi

  84. Stereoselective Synthesis ofN-Glycosyl Amino Acids by Traceless Staudinger Ligation of Unprotected Glycosyl Azides

    Article • European Journal of Organic Chemistry, November 2009, Wiley

    Professor Anna Bernardi

  85. Interfering with the Sugar Code: Design and Synthesis of Oligosaccharide Mimics

    Article • Chemistry - A European Journal, August 2008, Wiley

    Professor Anna Bernardi

  86. Synthesis of Novel DC‐SIGN Ligands with an α‐Fucosylamide Anchor

    Article • ChemBioChem, August 2008, Wiley

    Javier Rojo, Professor Anna Bernardi

  87. Stereoselective synthesis of glycosyl amides by traceless Staudinger ligation of unprotected glycosyl azides

    Article • Carbohydrate Research, July 2008, Elsevier

    Professor Anna Bernardi

  88. Effect of structural modifications of ganglioside GM2 on intra-molecular carbohydrate-to-carbohydrate interaction and enzymatic susceptibility

    Article • Biochimica et Biophysica Acta (BBA) - General Subjects, March 2008, Elsevier

    Professor Anna Bernardi

  89. Synthesis and conformational analysis of an α-d-mannopyranosyl-(1→2)-α-d-mannopyranosyl-(1→6)-α-d-mannopyranose mimic

    Article • Carbohydrate Research, September 2007, Elsevier

    Professor Anna Bernardi

  90. First round of a focused library of cholera toxin inhibitors

    Article • Carbohydrate Research, September 2007, Elsevier

    Professor Anna Bernardi

  91. 1,2‐Mannobioside Mimic: Synthesis, DC‐SIGN Interaction by NMR and Docking, and Antiviral Activity

    Article • ChemMedChem, June 2007, Wiley

    Javier Rojo, Professor Anna Bernardi

  92. A Simple Model System for the Study of Carbohydrate−Aromatic Interactions

    Article • Journal of the American Chemical Society, March 2007, American Chemical Society (ACS)

    Professor Anna Bernardi

  93. Solid phase immunoadsorption for therapeutic and analytical studies on neuropathy-associated anti-GM1 antibodies

    Article • Glycobiology, December 2006, Oxford University Press (OUP)

    Professor Anna Bernardi

  94. Synthesis and Conformational Analysis of Galactose-Derived Bicyclic Scaffolds

    Article • European Journal of Organic Chemistry, July 2006, Wiley

    Professor Anna Bernardi

  95. A facile stereoselective synthesis of α-glycosyl ureas

    Article • Carbohydrate Research, July 2006, Elsevier

    Professor Anna Bernardi

  96. Traceless Staudinger Ligation of Glycosyl Azides with Triaryl Phosphines:  Stereoselective Synthesis of Glycosyl Amides †

    Article • The Journal of Organic Chemistry, June 2006, American Chemical Society (ACS)

    Professor Anna Bernardi

  97. Targeting integrins: Insights into structure and activity of cyclic RGD pentapeptide mimics containing azabicycloalkane amino acids

    Article • Bioorganic & Medicinal Chemistry, January 2006, Elsevier

    Professor Anna Bernardi, Dr Leonardo Manzoni

  98. A Synthetic Divalent Cholera Toxin Glycocalix[4]arene Ligand Having Higher Affinity than Natural GM1 Oligosaccharide

    Article • Journal of the American Chemical Society, February 2005, American Chemical Society (ACS)

    Professor Alessandro Casnati, Professor Anna Bernardi

  99. Neo-glycoconjugates: stereoselective synthesis of α-glycosyl amides via Staudinger ligation reactions

    Article • Tetrahedron Asymmetry, January 2005, Elsevier

    Professor Anna Bernardi

  100. Synthesis, Conformational Studies and Mannosidase Stability of a Mimic of 1,2-Mannobioside

    Article • European Journal of Organic Chemistry, December 2004, Wiley

    Professor Anna Bernardi

  101. Intramolecular Carbohydrate-Aromatic Interactions and Intermolecular van der Waals Interactions Enhance the Molecular Recognition Ability of GM1 Glycomimetics for Cholera Toxin

    Article • Chemistry - A European Journal, July 2004, Wiley

    Professor Anna Bernardi

  102. Conformational analysis and dynamics of mannobiosides and mannotriosides using Monte Carlo/stochastic dynamics simulations

    Article • Carbohydrate Research, April 2004, Elsevier

    Professor Anna Bernardi

  103. Selective synthesis of anomeric α-glycosyl acetamides via intramolecular Staudinger ligation of the α-azides

    Article • Tetrahedron Letters, March 2004, Elsevier

    Professor Anna Bernardi

  104. Synthesis and cholera toxin binding properties of multivalent GM1 mimicsElectronic supplementary information (ESI) available: characterization of the polyvalent compounds ? imide by-products. See http://www.rsc.org/suppdata/ob/b4/b405344c/

    Article • Organic & Biomolecular Chemistry, January 2004, Royal Society of Chemistry

    Professor Anna Bernardi

  105. Ganglioside GM1 mimics: lipophilic substituents improve affinity for cholera toxin

    Article • Bioorganic & Medicinal Chemistry Letters, November 2003, Elsevier

    Professor Anna Bernardi

  106. Mimics of ganglioside GM1 as cholera toxin ligands: replacement of the GalNAc residueElectronic supplementary information (ESI) available: synthetic details, product characterisations and full NOE contact list. See http://www.rsc.org/suppdata/ob/b2/b21...

    Article • Organic & Biomolecular Chemistry, February 2003, Royal Society of Chemistry

    Professor Anna Bernardi, Dr Leonardo Manzoni

  107. Solid-phase synthesis of combinatorial libraries based on enatiomerically pure (1S,2S,4R,5S)-4,5-dihydroxycyclohexan-1,2-dicarboxylic acid scaffolds

    Article • Il Farmaco, September 2002, Elsevier

    Professor Anna Bernardi

  108. Article • Neurochemical Research, January 2002, Springer Science + Business Media

    Professor Anna Bernardi

  109. Stereoselective Synthesis of Conformationally Constrained Cyclohexanediols:  A Set of Molecular Scaffolds for the Synthesis of Glycomimetics

    Article • The Journal of Organic Chemistry, September 2001, American Chemical Society (ACS)

    Dr Leonardo Manzoni, Professor Anna Bernardi

  110. Article • Organic Letters, April 2001, CrossRef Test Account

    Professor Anna Bernardi

  111. Article • Journal of Computer-Aided Molecular Design, January 2001, Springer Science + Business Media

    Professor Anna Bernardi

  112. Second generation mimics of ganglioside GM1 as artificial receptors for cholera toxin: replacement of the sialic acid moiety

    Article • Bioorganic & Medicinal Chemistry Letters, October 2000, Elsevier

    Professor Anna Bernardi

  113. Article • Glycoconjugate Journal, January 2000, Springer Science + Business Media

    Professor Anna Bernardi

  114. Improved synthesis of both enantiomers of trans-cyclohex-4-ene-1,2-dicarboxylic acid

    Article • Tetrahedron Asymmetry, August 1999, Elsevier

    Professor Anna Bernardi

  115. Structural Basis for the Resistance of Tay-Sachs Ganglioside GM2 to Enzymatic Degradation

    Article • Journal of Biological Chemistry, April 1999, American Society for Biochemistry & Molecular Biology (ASBMB)

    Professor Anna Bernardi

  116. Sugar Mimics:  An Artificial Receptor for Cholera Toxin

    Article • Journal of the American Chemical Society, March 1999, American Chemical Society (ACS)

    Professor Anna Bernardi

  117. Article • Bioscience Reports, January 1999, Portland Press Ltd.

    Professor Anna Bernardi

  118. A comparison and chemometric analysis of several molecular mechanics force fields and parameter sets applied to carbohydrates

    Article • Carbohydrate Research, December 1998, Elsevier

    Professor Anna Bernardi

  119. Application of structure-based thermodynamic calculations to the rationalization of the enantioselectivity of subtilisin in organic solvents

    Article • Tetrahedron Asymmetry, April 1998, Elsevier

    Professor Anna Bernardi

  120. Enantioselective conjugate additions of silylketene acetals to 2-carboxycyclopentenones promoted by chiral Ti complexes

    Article • Tetrahedron, September 1997, Elsevier

    Professor Anna Bernardi

  121. Simulation of Protein−Sugar Interactions:  A Computational Model of the Complex between Ganglioside GM1 and the Heat-Labile Enterotoxin of Escherichia coli †

    Article • Journal of Medicinal Chemistry, June 1997, American Chemical Society (ACS)

    Professor Anna Bernardi

  122. Computational studies on the aldol-type addition of boron enolates to imines: An ab-initio approach

    Article • Tetrahedron, June 1997, Elsevier

    Professor Anna Bernardi

  123. Conformational analysis of saccharides with Monte Carlo/stochastic dynamics simulations

    Article • Journal of Molecular Structure THEOCHEM, May 1997, Elsevier

    Professor Anna Bernardi

  124. Enantioselective mukaiyama-michael reactions of 2-carbomethoxy cyclopentenone catalyzed by chiral bis(Oxazoline)-Cu(II) complexes

    Article • Tetrahedron Letters, December 1996, Elsevier

    Professor Anna Bernardi

  125. Stereoselective conjugate addition of lithium and titanium enolates to γ - alkoxy enones

    Article • Tetrahedron, March 1996, Elsevier

    Professor Anna Bernardi

  126. The rational design and systematic analysis of asymmetric aldol reactions using enol borinates: Applications of transition state computer modelling

    Article • Tetrahedron Asymmetry, November 1995, Elsevier

    Professor Anna Bernardi

  127. Conformational Analysis of GM1 Oligosaccharide in Water Solution with a New Set of Parameters for the Neu5Ac Moiety

    Article • The Journal of Organic Chemistry, June 1995, American Chemical Society (ACS)

    Professor Anna Bernardi

  128. Mechanistic insights from ab initio calculations on a nitrogen analogue of the boron-mediated aldol reaction

    Article • Tetrahedron, April 1995, Elsevier

    Professor Anna Bernardi

  129. Enantioselective michael-mukaiyama additions of silylketene acetals to 2-carboxycyclopentenones promoted by chiral Ti complexes

    Article • Tetrahedron Letters, February 1995, Elsevier

    Professor Anna Bernardi

  130. Stereoselective conjugate addition of propionate Ti ate enolate to unsaturated chiral ketones: A new insight in the reaction mechanism

    Article • Tetrahedron Letters, August 1994, Elsevier

    Professor Anna Bernardi

  131. Titanium Ate Enolate Complexes: An NMR Study

    Article • The Journal of Organic Chemistry, July 1994, American Chemical Society (ACS)

    Professor Anna Bernardi

  132. Origins of stereoselectivity in the addition of allyl- and crotylboronates to aldehydes : the development and application of a force field model of the transition state

    Article • Tetrahedron, January 1994, Elsevier

    Professor Anna Bernardi

  133. Computer-assisted design of chiral boron enolates: The role of ate complexes in determining aldol stereoselectivity.

    Article • Tetrahedron, January 1994, Elsevier

    Professor Anna Bernardi

  134. Origins of stereoselectivity in the addition of chiral allyl- and crotylboranes to aldehydes: the development and application of a force field model of the transition state

    Article • The Journal of Organic Chemistry, March 1993, American Chemical Society (ACS)

    Professor Anna Bernardi

  135. Origins of π-face selectivity in the aldol reactions of chiral E-enol borinates: a computational study using transition state modelling.

    Article • Tetrahedron, January 1993, Elsevier

    Professor Anna Bernardi

  136. Acceleration of the conjugate addition of Ti “ate” enolates via lewis acid catalysis.

    Article • Tetrahedron, January 1993, Elsevier

    Professor Anna Bernardi

  137. A computational study of the 1,4-addition of lithium enolates to conjugated carbonyl compounds

    Article • The Journal of Organic Chemistry, December 1992, American Chemical Society (ACS)

    Professor Anna Bernardi

  138. The rational design of highly stereoselective boron enolates using transition-state computer modeling: a novel, asymmetric anti aldol reaction for ketones

    Article • The Journal of Organic Chemistry, September 1992, American Chemical Society (ACS)

    Professor Anna Bernardi

  139. Stereoselective Michael additions of titanium “ate” complexes of ketone and ester enolates

    Article • Tetrahedron, July 1992, Elsevier

    Professor Anna Bernardi

  140. Norephedrine derived oxazolidines as chiral acylating agents: An NMR study of the intermediate cations.

    Article • Tetrahedron, January 1992, Elsevier

    Professor Anna Bernardi

  141. Developing a force field for the transition state of the aldol reaction of enolborinates: Evaluation of the use of fixed point charges.

    Article • Tetrahedron, January 1992, Elsevier

    Professor Anna Bernardi

  142. Addition of racemic alkoxyallylstannanes to an enantiomerically pure 2-methoxyoxazolidine: an example of combined mutual diastereoface selection and kinetic resolution

    Article • The Journal of Organic Chemistry, December 1991, American Chemical Society (ACS)

    Professor Anna Bernardi

  143. Highly stereoselective acetylations via norephedrine derived oxazolidines.

    Article • Tetrahedron, September 1991, Elsevier

    Professor Anna Bernardi

  144. Asymmetric hydrogenation of 3-methyl-fumaric and maleic ester monoaldehydes protected as neph-derived oxazolidines

    Article • Tetrahedron, August 1991, Elsevier

    Professor Anna Bernardi

  145. Highly selective binding of simple peptides by a C3 macrotricyclic receptor

    Article • Journal of the American Chemical Society, June 1991, American Chemical Society (ACS)

    Professor Anna Bernardi

  146. A computational study of the 1,4-addition of lithium enolates to conjugated carbonyl compounds.

    Article • Tetrahedron Letters, February 1991, Elsevier

    Professor Anna Bernardi

  147. Origins of stereoselectivity in chiral boron enolate aldol reactions: A computational study using transition state modellings

    Article • Tetrahedron, January 1991, Elsevier

    Professor Anna Bernardi

  148. Transition-state modeling of the aldol reaction of boron enolates: a force field approach

    Article • The Journal of Organic Chemistry, May 1990, American Chemical Society (ACS)

    Professor Anna Bernardi

  149. Stereoselective synthesis of statin analogues.

    Article • Tetrahedron Letters, January 1990, Elsevier

    Professor Anna Bernardi

  150. Norephedrine derived 2-methoxy oxazolidines as chiral formyl cation equivalents

    Article • Tetrahedron Letters, January 1990, Elsevier

    Professor Anna Bernardi

  151. Asymmetric synthesis of malic acid-type synthons VIA chiral norephedrine-derived oxazolidines

    Article • Tetrahedron, January 1990, Elsevier

    Professor Anna Bernardi

  152. 1,4-addition to α,β-unsaturated carbonyl compounds bearing a γ-stereocenter: A molecular mechanics model for steric interactions in the transition state.

    Article • Tetrahedron Asymmetry, January 1990, Elsevier

    Professor Anna Bernardi

  153. Allylic stereocentre directed cyclopropanation. A new highly enantioselective synthesis of hemicaronic aldehyde

    Article • Tetrahedron Letters, January 1989, Elsevier

    Professor Anna Bernardi

  154. Norephedrine-derived 2-alkenyloxazolidines: stereochemistry of cyclization and allylic stereocenter directed asymmetric conjugate addition

    Article • The Journal of Organic Chemistry, April 1988, American Chemical Society (ACS)

    Professor Anna Bernardi

  155. Catalytic osmylation of electron poor allylic alcohols and ethers.

    Article • Tetrahedron, January 1988, Elsevier

    Professor Anna Bernardi

  156. Asymmetric synthesis of functionalized α -amino-β-hydroxy acids via chiral norephedrine-derived oxazolidines

    Article • Tetrahedron, January 1988, Elsevier

    Professor Anna Bernardi

  157. Magnesium bromide-promoted addition of heterosubstituted methylketene silyl acetals to alkoxy aldehydes. Diastereoselective synthesis of 3,4-syn-2-methylene- and 2-(alkoxymethyl)-3-hydroxy-4-alkoxy esters

    Article • The Journal of Organic Chemistry, March 1987, American Chemical Society (ACS)

    Professor Anna Bernardi

  158. Conformational analysis of oxazolidines by molecular and quantum mechanics and NMR spectroscopy

    Article • Chemical Physics Letters, February 1987, Elsevier

    Professor Anna Bernardi

  159. Allylic stereocenter directed asymmetric conjugate addition. Enantioselective synthesis of 3-alkylsuccinaldehydic acid methyl esters

    Article • The Journal of Organic Chemistry, December 1986, American Chemical Society (ACS)

    Professor Anna Bernardi

  160. Lewis acid mediated aldol condensations using thioester silyl ketene acetals

    Article • Tetrahedron, January 1986, Elsevier

    Honorary Professor Roberto Todeschini, Professor Anna Bernardi

  161. Synthetic opportunities offered by anti .alpha.-methylene-.beta.-hydroxy-.gamma.-alkoxy esters: stereoselective reactions at the double bond

    Article • The Journal of Organic Chemistry, November 1985, American Chemical Society (ACS)

    Professor Anna Bernardi

  162. Enantioselective synthesis of anti-.alpha.-methyl-.beta.-hydroxy esters through titanium tetrachloride-mediated aldol condensation

    Article • Journal of the American Chemical Society, October 1985, American Chemical Society (ACS)

    Professor Anna Bernardi

  163. Stereoselective aldol reactions using ticl4 as stereochemical template

    Article • Tetrahedron Letters, January 1985, Elsevier

    Professor Anna Bernardi

  164. Stereoselective aldol additions to α-alkoxy aldehydes using thioester silyl ketene acetals,

    Article • Tetrahedron Letters, January 1985, Elsevier

    Professor Anna Bernardi

  165. Lewis acid promoted aldol additions of α-thiosilylketeneacetals to α-alkoxy aldehydes: diastereoselective synthesis of -α-methylene-β-hydroxy-∂-alkoxy esters.

    Article • Tetrahedron Letters, January 1985, Elsevier

    Professor Anna Bernardi

  166. High diastereoselectivity in lewis acid mediated aldol condensations using thioester silyl ketene acetals.

    Article • Tetrahedron Letters, January 1985, Elsevier

    Professor Anna Bernardi

  167. High diastereoface selection in an ester enolate addition to .alpha.-alkoxy aldehydes: stereoselective synthesis of .alpha.-methylene-.beta.-hydroxy-.gamma.-alkoxy esters

    Article • The Journal of Organic Chemistry, October 1984, American Chemical Society (ACS)

    Professor Anna Bernardi

  168. Ethyl-(r)-(4-methylphenylsulfinyl)-n-methoxy acetimidate a useful chiral acetate equivalent in aldol type condensations

    Article • Tetrahedron, January 1984, Elsevier

    Professor Anna Bernardi

  169. Stereoselective aldol condensations via alkenyloxy dialkoxyboranes: synthetic applications using thioesters

    Article • Tetrahedron, January 1984, Elsevier

    Professor Anna Bernardi

  170. Design and synthesis of glycomimetics

    Article • Royal Society of Chemistry

    Professor Anna Bernardi