Dr Fabrizio Machetti
Current affiliation: Consiglio Nazionale delle Ricerche
Subject: Chemistry
Primary location: Italy
Design, Synthesis, and Applications of 3-Aza-6,8-Dioxabicyclo[3.2.1]Octane-Based Scaffolds for Peptidomimetic Chemistry
Published in:Synlett
Publication date:2006-01-01
Enantiospecific synthesis of 3-aza-6,8-dioxa-bicyclo[3.2.1]octane carboxylic acids from erythrose
Published in:Tetrahedron
Publication date:2003-07-01
Identification of Inhibitors of Drug-Resistant Candida albicans Strains from a Library of Bicyclic Peptidomimetic Compounds
Published in:Journal of Medicinal Chemistry
Publication date:2010-03-25
Effect of C-ring modifications in benzo[c]quinolizin-3-ones, new selective inhibitors of human 5α-reductase 1
Published in:Bioorganic & Medicinal Chemistry
Publication date:2001-06-01
Synthesis of a new enantiopure bicyclic γ/δ-amino acid (BTKa) derived from tartaric acid and α-amino acetophenone
Published in:Tetrahedron
Publication date:2002-12-01
Synthesis and Reactivity of Bicycles Derived from Tartaric Acid and α-Amino Acids: A Novel Class of Conformationally Constrained Dipeptide Isoster...
Published in:The Journal of Organic Chemistry
Publication date:1999-10-01
Design and synthesis of a new bicyclic dipeptide isostere
Published in:Chemical Communications
Publication date:2001-01-01
Isoxazoline derivatives from activated primary nitrocompounds and tertiary diamines
Published in:Tetrahedron Letters
Publication date:2005-11-01
Isoxazoline Derivatives from Activated Primary Nitro Compounds and Tertiary Diamines.
Published in:ChemInform
Publication date:2006-02-07
Condensation of Primary Nitro Compounds to Isoxazole Derivatives: Stoichiometric To Catalytic
Published in:Methods and Applications of Cycloaddition Reactions in Organic Syntheses
Publication date:2014-01-10
ChemInform Abstract: 4,5-Dihydroisoxazoles by Copper(II)-Catalyzed Condensation of Primary Nitroalkanes with Dipolarophiles.
Published in:ChemInform
Publication date:2008-01-29
Five-Membered Heterocycles: 1,3-Azoles
Published in:Modern Heterocyclic Chemistry
Publication date:2011-07-27
ChemInform Abstract: Five-Membered Heterocycles: 1,3-Azoles
Published in:ChemInform
Publication date:2011-12-09
ChemInform Abstract: Design and Synthesis of a New Bicyclic Dipeptide Isostere.
Published in:ChemInform
Publication date:2010-05-23
Novel inhibitors of 5α-reductase
Published in:Expert Opinion on Therapeutic Patents
Publication date:2002-02-01
4,5-Dihydroisoxazoles by Copper(II)-Catalysed Condensation of Primary Nitroalkanes with Dipolarophiles
Published in:Synlett
Publication date:2007-09-01
Neat reaction of carboxylic acid methyl esters and amines for efficient parallel synthesis of scaffold amide libraries
Published in:Comptes Rendus Chimie
Publication date:2003-05-01
The Synthesis of 4-Hydroxypipecolic Acids by Stereoselective Cycloaddition of Configurationally Stable Nitrones
Published in:Liebigs Annalen der Chemie
Publication date:2006-07-01
Practical synthesis of both enantiomers of protected 4-oxopipecolic acid
Published in:Tetrahedron
Publication date:2001-06-01
ChemInform Abstract: Acid-Base-Catalyzed Condensation Reaction in Water: Isoxazolines and Isoxazoles from Nitroacetates and Dipolarophiles.
Published in:ChemInform
Publication date:2012-05-31
Conversion of a nitrosocarbonyl hetero Diels–Alder cycloadduct to useful isoxazoline-carbocyclic aminols
Published in:Tetrahedron
Publication date:2009-12-01
A new synthesis of (2S)-4-oxopipecolic acid by thermal rearrangement of enantiopure spirocyclopropaneisoxazolidine
Published in:Tetrahedron Letters
Publication date:1996-06-01
Synthesis of Taurine Analogues from Alkenes
Published in:Advances in Experimental Medicine and Biology
Publication date:2002-01-01
ChemInform Abstract: Conjugate Addition versus Cycloaddition/Condensation of Nitro Compounds in Water: Selectivity, Acid-Base Catalysis, and Induct...
Published in:ChemInform
Publication date:2013-06-06
ChemInform Abstract: Reactivity of [60]Fullerene with Primary Nitro Compounds: Addition or Catalyzed Condensation to Isoxazolo[60]fullerenes.
Published in:ChemInform
Publication date:2015-03-01
1,4-Diazabicyclo[2.2.2]octane (DABCO) as an Efficient Reagent for the Synthesis of Isoxazole Derivatives from Primary Nitro Compounds and Dipolarop...
Published in:ChemInform
Publication date:2007-02-20
ChemInform Abstract: Isoxazoles and Isoxazolines by 1,3-Dipolar Cycloaddition: Base-Catalyzed Condensation of Primary Nitro Compounds with Dipolaro...
Published in:ChemInform
Publication date:2008-01-01
Conjugate Addition versus Cycloaddition/Condensation of Nitro Compounds in Water: Selectivity, Acid-Base Catalysis, and Induction Period
Published in:Chemistry - A European Journal
Publication date:2012-11-14
Design, Synthesis, and Applications of 3-Aza-6,8-dioxabicyclo[3.2.1]octane-Based Scaffolds for Peptidomimetic Chemistry
Published in:ChemInform
Publication date:2006-05-16
1,2,5-Oxadiazole (Furazan) Derivatives from Benzoylnitromethane and Dipolarophiles in the Presence of DABCO: Structure and Intermediates
Published in:Liebigs Annalen der Chemie
Publication date:2006-07-01
Synthesis of 4,5-Dihydroisoxazoles by Condensation of Primary Nitro Compounds with Alkenes by Using a Copper/Base Catalytic System
Published in:Chemistry - A European Journal
Publication date:2008-09-08
ChemInform Abstract: Synthesis of 4,5-Dihydroisoxazoles by Condensation of Primary Nitro Compounds with Alkenes by Using a Copper/Base Catalytic Sy...
Published in:ChemInform
Publication date:2009-01-13
Synthesis of Benzo[c]quinolizin-3-ones: Discovery and Development of Novel Inhibitors of Human Steroid 5α-Reductase
Published in:ChemInform
Publication date:2006-08-01
Inhibition of rabbit brain 4-aminobutyrate transaminase by some taurine analogues: A kinetic analysis
Published in:Biochemical Pharmacology
Publication date:2006-05-01
Acid-Base-Catalysed Condensation Reaction in Water: Isoxazolines and Isoxazoles from Nitroacetates and Dipolarophiles
Published in:Chemistry - A European Journal
Publication date:2012-01-10
Michael Additions versus Cycloaddition Condensations with Ethyl Nitroacetate and Electron-Deficient Olefins
Published in:Chemistry - A European Journal
Publication date:2009-08-10
Isoxazoles and Isoxazolines by 1,3-Dipolar Cycloaddition: Base-Catalysed Condensation of Primary Nitro Compounds with Dipolarophiles
Published in:Liebigs Annalen der Chemie
Publication date:2007-09-01
ChemInform Abstract: Synthesis of Taurine Analogues. Part 2. Amino-Sulfonation of Alkenes in a Three-Component Reaction.
Published in:ChemInform
Publication date:2010-05-20
ChemInform Abstract: Practical Synthesis of Both Enantiomers of Protected 4-Oxopipecolic Acid.
Published in:ChemInform
Publication date:2010-05-24
ChemInform Abstract: Synthesis of Taurine Analogues. Part 1. 2-Aminosulfonic Acids from Alkene-Sulfur Monochloride Adducts.
Published in:ChemInform
Publication date:2001-02-27
Amino-Sulfonation of Alkenes in a Three-Component Reaction
Published in:Liebigs Annalen der Chemie
Publication date:2002-04-01
A New Bicyclic Dipeptide Isostere with Pyrrolizidinone Skeleton
Published in:The Journal of Organic Chemistry
Publication date:2005-02-01
Stereoselectivity in the TiCl4-catalysed reaction of Danishefsky's diene with a N-(acyloxy)iminium ion: Synthesis of 5α versus 5β Δ1(2)-19-Nor-10-a...
Published in:Tetrahedron
Publication date:1998-09-01
Effects of Taurine and some Structurally Related Analogues on the Central Mechanism of Thermoregulation
Published in:Advances in Experimental Medicine and Biology
Publication date:2002-01-01
Reactivity of [60]Fullerene with Primary Nitro Compounds: Addition or Catalysed Condensation to Isoxazolo[60]fullerenes
Published in:Liebigs Annalen der Chemie
Publication date:2014-10-29Reactivity of [60]Fullerene with Primary Nitro Compounds
A specific taurine recognition site in the rabbit brain is responsible for taurine effects on thermoregulation
Published in:British Journal of Pharmacology
Publication date:2003-06-01
Synthesis of bicyclic molecular scaffolds (BTAa): An investigation towards new selective MMP-12 inhibitors
Published in:Bioorganic & Medicinal Chemistry
Publication date:2006-11-01
Interactions of taurine and structurally related analogues with the GABAergic system and taurine binding sites of rabbit brain
Published in:British Journal of Pharmacology
Publication date:2003-03-01
1,4-Diazabicyclo[2.2.2]octane (DABCO) as an Efficient Reagent for the Synthesis of Isoxazole Derivatives from Primary Nitro Compounds and Dipolarop...
Published in:Liebigs Annalen der Chemie
Publication date:2006-11-01
Base- and Copper-Catalysed Condensation of Primary Activated Nitro Compounds with Enolisable Compounds
Published in:Liebigs Annalen der Chemie
Publication date:2009-12-01
Synthesis of taurine analogues. Part 1: 2-aminosulfonic acids from alkene-sulfur monochloride adducts
Published in:Journal of Chemical Research
Publication date:2000-03-01
Synthesis of Free andNα-Fmoc-/Nγ-Boc-Protected (2S,4S)- and (2S,4R)-4-Aminopipecolic Acids
Published in:Liebigs Annalen der Chemie
Publication date:2004-07-01
Bicyclic Compounds Derived from Tartaric Acid and α-Amino Acids (BTAas): Synthesis of New Molecular Scaffolds Derived from the Combination of (R,R)...
Published in:Liebigs Annalen der Chemie
Publication date:2002-03-01
ChemInform Abstract: Modification of the Aza-Robinson Annulation for the Synthesis of 4-Methyl-benzo[c]quinolizin-3-ones, Potent Inhibitors of Ster...
Published in:ChemInform
Publication date:2001-04-03
ChemInform Abstract: Benzo[c]quinolizin-3-ones: A Novel Class of Potent and Selective Nonsteroidal Inhibitors of Human Steroid 5α-Reductase 1.
Published in:ChemInform
Publication date:2001-03-06
ChemInform Abstract: Oligomers of Enantiopure Bicyclic γ/δ-Amino Acids (BTAa). Part 1. Synthesis and Conformational Analysis of 3-Aza-6,8-dioxabicy...
Published in:ChemInform
Publication date:2001-02-27
Synthesis and X-ray study of hexahydro- and tetrahydrophospholo-[2,3-d]isoxazoles, a new class of heterocycles of potential fungicidal activity
Published in:Journal of Heterocyclic Chemistry
Publication date:1996-07-01
Modification of the Aza-Robinson Annulation for the Synthesis of 4-Methyl-Benzo[ c ]quinolizin-3-ones, Potent Inhibitors of Steroid 5α-Reductase 1
Published in:The Journal of Organic Chemistry
Publication date:2000-11-01
Parallel Synthesis of an Amide Library Based on the 6,8-Dioxa-3-azabicyclo[3.2.1]octane Scaffold by Direct Aminolysis of Methyl Esters
Published in:Journal of Combinatorial Chemistry
Publication date:2007-05-01
Benzo[ c ]quinolizin-3-ones: A Novel Class of Potent and Selective Nonsteroidal Inhibitors of Human Steroid 5α-Reductase 1
Published in:Journal of Medicinal Chemistry
Publication date:2000-10-01
Oligomers of Enantiopure Bicyclic γ/δ-Amino Acids (BTAa). 1. Synthesis and Conformational Analysis of 3-Aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxy...
Published in:Organic Letters
Publication date:2000-12-01
19-Nor-10-azasteroids: A Novel Class of Inhibitors for Human Steroid 5α-Reductases 1 and 2
Published in:Journal of Medicinal Chemistry
Publication date:1997-03-01
Isoxazoles
Published in:Comprehensive Heterocyclic Chemistry III
Publication date:2008-01-01
From nitro compounds to isoxazoles
Published in:Liebigs Annalen der Chemie
Publication date:2016-08-26Competitive Copper Catalysis in the Condensation of Primary Nitro Compounds with Terminal Alkynes: Synthesis of Isoxazoles
Synthesis and Reactivity of Bicycles Derived from Tartaric Acid and α-Amino Acids: A Novel Class of Conformationally Constrained Dipeptide Isoster...
Published in:The Journal of Organic Chemistry
Publication date:2000-07-01
A Concise Route to 19-Nor-10-azasteroids, a New Class of Steroid 5α-Reductase Inhibitors. 3. 1 Synthesis of (+)-19-Nor-10-azatestosterone and (+)-...
Published in:The Journal of Organic Chemistry
Publication date:1998-06-01
19-Nor-10-azasteroids. 5. 1 A Synthetic Strategy for the Preparation of (+)-17-(3-Pyridyl)-(5β)-10-azaestra-1,16- dien-3-one, a Novel Potential In...
Published in:The Journal of Organic Chemistry
Publication date:1999-06-01
19-Nor-10-azasteroids, a New Class of Steroid 5α-Reductase Inhibitors. 2. 1 X-ray Structure, Molecular Modeling, Conformational Analysis of 19-Nor...
Published in:Journal of Medicinal Chemistry
Publication date:1997-10-01
Copper-Catalyzed Synthesis of Isoxazoles
Published in:Synfacts
Publication date:2010-01-21