All Stories

  1. 3D Histological Analysis of Soft Tissues by Contrast-Enhanced X-Ray Microfocus Computed Tomography: Screening and Staining Optimization of Contrast-Enhancing Staining Agents
  2. Enhanced decoupling of conductivity relaxation from structural relaxation in non-stoichiometric protic ionic liquids involving triflic acid and 2-aminoethyl hydrogen sulfate
  3. Novel Far-Red Fluorescent 1,4-Dihydropyridines for L-Type Calcium Channel Imaging
  4. Perfluorooxosulfate Salts as SOF4‐Gas‐Free Precursors to Multidimensional SuFEx Electrophiles
  5. Perfluorooxosulfate Salts as SOF4‐Gas‐Free Precursors to Multidimensional SuFEx Electrophiles
  6. Ex-situ ChloGen: A facile and straightforward entry to Aryl-IF4 compounds
  7. 1.10 The Pentafluorosulfanyl Group (SF5)
  8. An Extrusion Strategy for On-Demand SF5Cl Gas Generation from a Commercial Disulfide
  9. Solvent‐Free Hydrohalogenation and Deuteriohalogenation by Ex Situ Generation of HX and DX Gas
  10. Charge transport in highly acidic glass-forming protic ionic liquids tailored by zwitterionic precursors
  11. Polyketide Synthase‐Mediated O‐Methyloxime Formation in the Biosynthesis of the Oximidine Anticancer Agents
  12. Ex situ Generation of Thiazyl Trifluoride (NSF3) as a Gaseous SuFEx Hub**
  13. Ex situ Generation of Thiazyl Trifluoride (NSF3) as a Gaseous SuFEx Hub**
  14. Revealing the three-dimensional murine brain microstructure by contrast-enhanced computed tomography
  15. Does Supramolecular Gelation Require an External Trigger?
  16. De-risking S–F bond formation: A gas cylinder-free strategy to access S(IV) and S(VI) fluorinated compounds.
  17. Cryogenic contrast-enhanced microCT enables nondestructive 3D quantitative histopathology of soft biological tissues
  18. 3-Methyl 5-{3-[(4-Methylbenzenesulfonyl)oxy]propyl} 4-(2,3-Dichlorophenyl)-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate
  19. Chemistry of Pentafluorosulfanyl Derivatives and Related Analogs: From Synthesis to Applications
  20. From the North Sea to Drug Repurposing, the Antiseizure Activity of Halimide and Plinabulin
  21. Carbonylation Chemistry Applied to the Synthesis of Benzimidazo[2,1‐ b ]quinazolin‐12‐ones
  22. 1,3-Diazepines
  23. Penicillins
  24. SuFEx-enabled, chemoselective synthesis of triflates, triflamides and triflimidates
  25. Correction: SuFEx-enabled, chemoselective synthesis of triflates, triflamides and triflimidates
  26. Characterization of Microbial Degradation Products of Steviol Glycosides
  27. Can the Philicity of Radicals Be Influenced by Oriented External Electric Fields?
  28. LSA-50 paper: An alternative to P81 phosphocellulose paper for radiometric protein kinase assays
  29. Computational Tools to Rationalize and Predict the Self-Assembly Behavior of Supramolecular Gels
  30. Frontispiece: Lighting Up the Plasma Membrane: Development and Applications of Fluorescent Ligands for Transmembrane Proteins
  31. Bioassay-guided isolation of antibacterial compounds from the leaves of Tetradenia riparia with potential bactericidal effects on food-borne pathogens
  32. Lighting Up the Plasma Membrane: Development and Applications of Fluorescent Ligands for Transmembrane Proteins
  33. Developments in the Discovery and Design of Protein Kinase D Inhibitors
  34. Copper(0) nanoparticle catalyzed Z ‐Selective Transfer Semihydrogenation of Internal Alkynes
  35. The presence of benzophenone in sunscreens and cosmetics containing the organic UV filter octocrylene: A laboratory study
  36. Solvent-free N-Boc deprotection by ex situ generation of hydrogen chloride gas
  37. Ultrasmall iron oxide nanoparticles functionalized with BODIPY derivatives as potential bimodal probes for MRI and optical imaging
  38. Design, synthesis and biological evaluation of pyrazolo[3,4-d]pyrimidine-based protein kinase D inhibitors
  39. Concomitant positive patch test reactions in FreeStyle‐allergic patients sensitized to isobornyl acrylate
  40. Facile Method to Obtain Low DS β-ketoesters and Esters of Microfibrillated Cellulose
  41. Nematicidal Activity of Holigarna caustica (Dennst.) Oken Fruit Is Due to Linoleic Acid
  42. Tuning the Properties of Polyether Alkyl Urea Derivatives as Rheology Modifiers in Cosmetic Solvents
  43. Stereoselective Reductions of 3-Substituted Cyclobutanones: A Comparison between Experiment and Theory
  44. Biofilm inhibiting properties of compounds from the leaves of Warburgia ugandensis Sprague subsp ugandensis against Candida and staphylococcal biofilms
  45. Exploring polyoxometalates as non-destructive staining agents for contrast-enhanced microfocus computed tomography of biological tissues
  46. Ex situ gas generation for lab scale organic synthesis
  47. Molecular dynamics based descriptors for predicting supramolecular gelation
  48. Rationalising Supramolecular Hydrogelation of Bis‐Urea‐Based Gelators through a Multiscale Approach
  49. Rationalising Supramolecular Hydrogelation of Bis‐Urea‐Based Gelators through a Multiscale Approach
  50. Rationalising Supramolecular Hydrogelation of Bis‐Urea‐Based Gelators through a Multiscale Approach
  51. Introduction of Aryl Fluorosulfates into the Realm of Catellani Reaction Substrates
  52. Green approach for the activation and functionalization of jute fibers through ball milling
  53. Modeling of Nanomolecular and Reticular Architectures with 6-fold Grooved, Programmable Interlocking Disks
  54. Nanocarrier systems assembled from PEGylated hyperbranched poly(arylene oxindole)
  55. Acylated sulfonamide adenosines as potent inhibitors of the adenylate-forming enzyme superfamily
  56. An Effective and Reusable Hyperbranched Polymer Immobilized Rhodium Catalyst for the Hydroformylation of Olefins
  57. Electrochemistry and Photoredox Catalysis: A Comparative Evaluation in Organic Synthesis
  58. Ketone Synthesis by a Nickel-Catalyzed Dehydrogenative Cross-Coupling of Primary Alcohols
  59. Synthesis of N-Acyl Sulfamates from Fluorosulfates and Amides
  60. Ball milling: a green technology for the preparation and functionalisation of nanocellulose derivatives
  61. Robust scalable synthesis of a bis-urea derivative forming thixotropic and cytocompatible supramolecular hydrogels
  62. Chemical structure and biological properties of sulfated fucan from the sequential extraction of subAntarctic Lessonia sp (Phaeophyceae)
  63. Bioassay-guided isolation of active substances from Semen Torreyae identifies two new anthelmintic compounds with novel mechanism of action
  64. A Robust and Scalable Continuous Flow Process for Glycerol Carbonate
  65. Bioassay-guided isolation of three anthelmintic compounds from Warburgia ugandensis Sprague subspecies ugandensis, and the mechanism of action of polygodial
  66. Identification of fukinolic acid from Cimicifuga heracleifolia and its derivatives as novel antiviral compounds against enterovirus A71 infection
  67. Direct Access to Aryl Bis(trifluoromethyl)carbinols from Aryl Bromides or Fluorosulfates: Palladium-Catalyzed Carbonylation
  68. Direct Access to Aryl Bis(trifluoromethyl)carbinols from Aryl Bromides or Fluorosulfates: Palladium-Catalyzed Carbonylation
  69. Active principles of Tetradenia riparia . IV. Anthelmintic activity of 8(14),15-sandaracopimaradiene-7α,18-diol
  70. Non-innocent probes in direct sonication: Metal assistance in oxidative radical C H functionalization
  71. Methylated flavonoids as anti-seizure agents: Naringenin 4′,7-dimethyl ether attenuates epileptic seizures in zebrafish and mouse models
  72. Synthesis and peptide functionalization of hyperbranched poly(arylene oxindole) towards versatile biomaterials
  73. Synthesis of an IS and Steviol Glycoside Analysis by a Validated Internal Standard Method
  74. Flow-Assisted Synthesis of Heterocycles via Multicomponent Reactions
  75. Functionalization of Heteroarenes Under Continuous Flow
  76. Water Tolerant and Reusable Sulfonated Hyperbranched Poly(aryleneoxindole) Acid Catalyst for Solvent-Free Esterification
  77. Ex Situ Generation of Sulfuryl Fluoride for the Synthesis of Aryl Fluorosulfates
  78. A Convenient Multigram Synthesis of DABSO Using Sodium Sulfite as SO2 Source
  79. Crystal structure of 5-benzyl-8-bromo-2-methyl-1,3-oxazolo[4,5-c][1,8]naphthyridin-4(5H)-one
  80. Towards New Tricyclic Motifs: Intramolecular C-H Arylation as the Key Step in a Formal [3+3] Cyclocondensation Strategy
  81. Intramolecular Carbonylative C-H Functionalization of 1,2,3- Triazoles for the Synthesis of Triazolo[1,5-a]indolones
  82. Discovery of a potent protein kinase D inhibitor: insights in the binding mode of pyrazolo[3,4-d]pyrimidine analogues
  83. Carbonylation as a novel method for the assembly of pyrazine based oligoamide alpha-helix mimetics
  84. Nanocellulosic materials as bioinks for 3D bioprinting
  85. The orthorhombic pseudopolymorph of tacrine hydrochloride
  86. Low-cost instant CO generation at room temperature using formic acid, mesyl chloride and triethylamine
  87. Gadolinium(III)-DOTA Complex Functionalized with BODIPY as a Potential Bimodal Contrast Agent for MRI and Optical Imaging
  88. Luminescence and Relaxometric Properties of Heteropolymetallic Metallostar Complexes with Selectively Incorporated Lanthanide(III) Ions
  89. Improved detection of β-N-methylamino-l-alanine using N-hydroxysuccinimide ester of N-butylnicotinic acid for the localization of BMAA in blue mussels (Mytilus edulis)
  90. Synthesis of N -Hydroxypyrazin-2(1 H )-ones via Selective O -Debenzylation of 1-Benzyloxypyrazin-2(1 H )-ones Using Flow Methodology
  91. First Example of Alkyl–Aryl Negishi Cross-Coupling in Flow: Mild, Efficient and Clean Introduction of Functionalized Alkyl Groups
  92. Facile azide formation via diazotransfer reaction in a copper tube flow reactor
  93. The Zeamine Antibiotics Affect the Integrity of Bacterial Membranes
  94. First Example of a Continuous-Flow Carbonylation Reaction Using Aryl Formates as CO Precursors
  95. Synthesis of 1-benzyloxypyrazin-2(1H)-one derivatives
  96. Synthesis of 11-aza-artemisinin derivatives using the Ugi reaction and an evaluation of their antimalarial activity
  97. Synthesis of triterpenoid triazine derivatives from allobetulone and betulonic acid with biological activities
  98. Synthetic Protocol toward Fused Pyrazolone Derivatives via a Michael Addition and Reductive Ring Closing Strategy
  99. 8-HaloBODIPYs and Their 8-(C, N, O, S) Substituted Analogues: Solvent Dependent UV–Vis Spectroscopy, Variable Temperature NMR, Crystal Structure Determination, and Quantum Chemical Calculations
  100. Formation of amides when other approaches have failed
  101. Tanshinone IIA Exhibits Anticonvulsant Activity in Zebrafish and Mouse Seizure Models
  102. Diterpene glycosides from Stevia phlebophylla A. Gray
  103. Alpha-Helical Destabilization of the Bcl-2-BH4-Domain Peptide Abolishes Its Ability to Inhibit the IP3 Receptor
  104. Synthesis and in vitro evaluation of a PDT active BODIPY–NLS conjugate
  105. Asymmetric Synthesis of 1-Aza-4-deoxypicropodophyllotoxin
  106. Scaffold Hoppingviaa Transannular Rearrangement–Encompassing Cascade
  107. Absolute configuration of 3-acetylbetulinic acid
  108. Preparation and characterization of hydrogels based on homopolymeric fractions of sodium alginate and PNIPAAm
  109. Total Synthesis of Septocylindrin B and C-Terminus Modified Analogues
  110. Fused derivatives of (iso)steviol via pericyclic reactions
  111. Stevioside and Steviol as Starting Materials in Organic Synthesis
  112. Tetranuclear d-f Metallostars: Synthesis, Relaxometric, and Luminescent Properties
  113. A Tripodal Ruthenium–Gadolinium Metallostar as a Potential αvβ3Integrin Specific Bimodal Imaging Contrast Agent
  114. Anticonvulsant activity of bisabolene sesquiterpenoids of Curcuma longa in zebrafish and mouse seizure models
  115. Selective LC-MS/MS method for the identification of BMAA from its isomers in biological samples
  116. Identification of a Small Molecule That Modulates Platelet Glycoprotein Ib-von Willebrand Factor Interaction
  117. An integrated fragment based screening approach for the discovery of small molecule modulators of the VWF–GPIbα interaction
  118. The C Terminus of Bax Inhibitor-1 Forms a Ca2+-permeable Channel Pore
  119. A Heterobimetallic Ruthenium–Gadolinium Complex as a Potential Agent for Bimodal Imaging
  120. Rational Design, Synthesis, and Spectroscopic and Photophysical Properties of a Visible-Light-Excitable, Ratiometric, Fluorescent Near-Neutral pH Indicator Based on BODIPY
  121. Isosteviol as a Starting Material in Organic Synthesis
  122. A Modular Approach towards the Synthesis of Target-Specific MRI Contrast Agents
  123. Synthesis of the orthogonally protected amino alcohol Phaol and analogs
  124. 2-(4-Methoxybenzyl)-4,6-diphenyl-2,5-diazabicyclo[2.2.2]oct-5-en-3-one
  125. Comparison of distance information in [TOAC1, Glu(OMe)7, 18, 19] alamethicin F50/5 from paramagnetic relaxation enhancement measurements with data obtained from an X-ray diffraction-based model
  126. Measuring cooperative Rev protein-protein interactions on Rev responsive RNA by fluorescence resonance energy transfer
  127. ChemInform Abstract: Synthesis of Pyridodiazepinediones by Using the Ugi Multicomponent Reaction.
  128. Triple Hyp→Pro replacement in integramide A, a peptaib inhibitor of HIV‐1 integrase: Effect on conformation and bioactivity
  129. Synthesis of Pyridodiazepinediones by Using the Ugi Multicomponent Reaction
  130. Generalized solvent scales as a tool for investigating solvent dependence of spectroscopic and kinetic parameters. Application to fluorescent BODIPY dyes
  131. Influence of Reducing Carbohydrates on (6S)-5-Methyltetrahydrofolic Acid Degradation during Thermal Treatments
  132. Direct functionalization of BODIPY dyes by oxidative nucleophilic hydrogen substitution at the 3- or 3,5-positions
  133. Synthesis and Substitution of 8-(4,6-Dichloropyrimidin-5-yl)-BODIPY
  134. Synthesis and Biological Evaluation of Bridged Analogues of the Platelet Aggregation Inhibitor Trifenagrel
  135. Flavonoids from Senecio viscosus
  136. Mechanism and Related Kinetics of 5-Methyltetrahydrofolic Acid Degradation during Combined High Hydrostatic Pressure−Thermal Treatments
  137. Photophysics and stability of cyano-substituted boradiazaindacene dyes
  138. Synthesis and modifications of a small library of 1,4-benzodiazepin-3-ones toward potential inhibitors of the collagen—von Willebrand Factor interaction
  139. Synthesis of 5,5′-Dialkyl-6,6′-dichloro-2, 2′-bipyridines
  140. ChemInform Abstract: Synthesis of Pyrazino[1,2‐a]benzimidazol‐1(2H)ones via a Microwave‐Assisted Buchwald—Hartwig Type Reaction.
  141. Structural property investigations of 1-[2-(2-methoxyphenyl)ethyl]piperidinium chloride: An experimental and computational study
  142. Synthesis of Highly Functionalized 2(1H)-Pyrazinone 3-Carboxamide Scaffolds
  143. Synthesis of pyrazino[1,2-a]benzimidazol-1(2H)ones via a microwave assisted Buchwald–Hartwig type reaction
  144. Ratiometric, Fluorescent BODIPY Dye with Aza Crown Ether Functionality: Synthesis, Solvatochromism, and Metal Ion Complex Formation
  145. Matrix-isolation FT-IR and theoretical investigation of the competitive intramolecular hydrogen bonding in 5-methyl-3-nitro-2-hydroxyacetophenone
  146. Spirocyclic Pyridoazepine Analogues of Galanthamine: Synthesis, Modelling Studies and Evaluation as Inhibitors of Acetylcholinesterase
  147. ATR-IR spectroscopic study of the structural changes in the hydrophobic region of ICPAN/DPPC bilayers
  148. Synthesis and Biological Evaluation of Methylene-Bridged Analogs of the Potent Cannabinoid Receptor Antagonist Rimonabant
  149. trans-Chlorido[6-chloro-4-(4-methoxybenzyl)-3-oxo-3,4-dihydropyrazin-2-yl]bis(triphenylphosphine)palladium(II)
  150. Matrix-isolation FT-IR and theoretical investigation of the vibrational properties of the sterically hindered ortho-hydroxy acylaromatic Schiff bases
  151. Synthesis of Spirocyclic Pyridoazepines as Analogues of Galanthamine by Nucleophilic Aromatic Substitution of 3‐Substituted 2‐Chloropyridines
  152. Photophysics of 3,5-diphenoxy substituted BODIPY dyes in solution
  153. Synthesis of Methylene‐Bridged Analogues of Biologically Active Pteridine Derivatives.
  154. Synthesis of Methylene‐Bridged Analogues of Biologically Active Pteridine Derivatives
  155. Conformational Analysis of TOAC‐Labelled Alamethicin F50/5 Analogues
  156. Design, Synthesis and Evaluation of Serine Protease Inhibitor Analogues
  157. Synthesis of 2(1H)‐Pyrazinone Phosphonates via an Arbuzov‐Type Reaction.
  158. Diastereoselective Diels—Alder Additions of Ethene to Substituted Homochiral 2(1H)‐Pyrazinones.
  159. Diastereoselective Diels–Alder Additions of Ethene to Substituted Homochiral 2(1H)-Pyrazinones
  160. Synthesis of 2(1H)-Pyrazinone Phosphonates via an Arbuzov-type Reaction
  161. 3,5‐Dihalo‐2(1H)‐pyrazinones: Versatile Scaffolds in Organic Synthesis
  162. 3,5-Dihalo-2(1 H )-pyrazinones: Versatile Scaffolds in Organic Synthesis
  163. Photophysical properties of an on/off fluorescent pH indicator excitable with visible light based on a borondipyrromethene-linked phenol
  164. Synthesis of 1,5-disubstituted 4-haloimidazoles from α-aminonitriles
  165. Solvent and pH Dependent Fluorescent Properties of a Dimethylaminostyryl Borondipyrromethene Dye in Solution
  166. Design, Synthesis, and Preferred Conformation of Peptides Based on a Highly Constrained, β,β′-Diphenyl Substituted Cyclopropane α-Amino Acid
  167. Preferred 3D-Structure of Peptides Rich in a Severely Conformationally Restricted Cyclopropane Analogue of Phenylalanine
  168. Structure based design of simplified analogues of insect kinins
  169. Development of New Amino(oxo)piperidinecarboxylate Scaffolds and Their Evaluation as -Turn Mimics
  170. BODIPY-Based Hydroxyaryl Derivatives as Fluorescent pH Probes
  171. Expanding the substitution pattern of 2(1H)-pyrazinones via Suzuki and Heck reactions
  172. Synthesis of sidechain adapted β-turn mimics for modifying the C-terminus of substance P
  173. Turn and Helical Peptide Handedness Governed Exclusively by Side-Chain Chiral Centers
  174. Synthesis of Novel Functionalised Symmetric Bi-2(1 H )-pyrazinones
  175. Design and synthesis of novel type VI-like β-turn mimetics. Diversity at the i+1 and the i+2 position
  176. New Routes for the Synthesis of 3‐ and 5‐Substituted 2(1H)‐Pyrazinones.
  177. Acid catalysed methanolysis of 2,5-diazabicyclo[2.2.2]octane-3,6-diones: scope and limitations
  178. New routes for the synthesis of 3- and 5-substituted 2(1H)-pyrazinones
  179. Stereoselective transformation of pyrazinones into substituted analogues of cis-5-amino-6-oxo-2-piperidinemethanol and cis-5-amino-2-piperidinemethanol
  180. Development of a Functionalizable External β-Turn Mimic Based on a cis-Fused 1,7-Naphthyridine Scaffold
  181. High-Speed Microwave-Promoted Hetero-Diels−Alder Reactions of 2(1H)-Pyrazinones in Ionic Liquid Doped Solvents
  182. Stereoselective intramolecular Diels–Alder reactions of 3-alkenyl(oxy)-2(1H)-pyrazinones
  183. Intramolecular Diels–Alder reactions of N-alkenyl-2(1H)-pyrazinones: generation of a novel type of cis-1,7-naphthyridine
  184. Synthesis of a conformationally restricted dipeptide analogue and its evaluation as a β-turn mimic
  185. Divergent pathways in the intramolecular diels-alder reaction of 2(1H)-pyrazinones substituted at the 3-position with a phenylalkyne containing side chain