All Stories

  1. Engineering a bifunctional cellobiose 2-epimerase into an isomerase capable of selective lactulose production

    Article • Bioresource Technology, May 2026, Elsevier

    Professor Walter Cabri

  2. Water-enabled organometallic and enzymatic catalysis: Sustainable technologies supporting API manufacturing

    Article • Current Opinion in Green and Sustainable Chemistry, February 2026, Elsevier

    Professor Walter Cabri

  3. Eco-Friendly Catalyst Development: Bidentate Nitrogen Ligands in the Suzuki–Miyaura Reaction of Aryl Iodides and Bromides in Green Solvents

    Article • ACS Sustainable Chemistry & Engineering, October 2025, American Chemical Society (ACS)

    Professor Walter Cabri

  4. Comparing the performance of electrostatic repulsion-reversed phase chromatography approaches in the resolution of complex peptide mixture: Liraglutide as case study

    Article • European Journal of Pharmaceutical Sciences, August 2025, Elsevier

    Professor Walter Cabri

  5. Improving Solid-State Properties of the Side-Chain Peptide Building Blocks for the Synthesis of GLP-1 Analogs through Their Complexation with Metal Cations

    Article • Organic Process Research & Development, February 2025, American Chemical Society (ACS)

    Professor Walter Cabri

  6. Mastering palladium-catalyzed cross-coupling reactions: the critical role of in situ pre-catalyst reduction design

    Article • Organic Chemistry Frontiers, January 2025, Royal Society of Chemistry

    Professor Walter Cabri

  7. Electrochemical oxidative CF3 radical-induced lactonization and etherification of terminal and internal alkenes

    Article • RSC Advances, January 2025, Royal Society of Chemistry

    Professor Walter Cabri

  8. Replace, reduce, and reuse organic solvents in peptide downstream processing: the benefits of dimethyl carbonate over acetonitrile

    Article • Green Chemistry, January 2025, Royal Society of Chemistry

    Professor Walter Cabri

  9. A Sustainable Chemo-Enzymatic Approach to the Synthesis of Liraglutide

    Article • ACS Sustainable Chemistry & Engineering, November 2024, American Chemical Society (ACS)

    Professor Walter Cabri

  10. Rediscovery of an Old Named Reaction: From Micellar Catalysis to Unusual Schotten–Baumann Conditions

    Article • Organic Process Research & Development, August 2024, American Chemical Society (ACS)

    Professor Walter Cabri

  11. Understanding Glucagon Aggregation: In Silico Insights and Experimental Validation

    Article • Molecular Pharmaceutics, July 2024, American Chemical Society (ACS)

    Roberto Pisano, Professor Walter Cabri

  12. Assessing the performance of new chromatographic technologies for the separation of peptide epimeric impurities: the case of Icatibant

    Article • European Journal of Pharmaceutical Sciences, February 2024, Elsevier

    Professor Walter Cabri

  13. Solid phase peptide synthesis using side-chain unprotected arginine and histidine with Oxyma Pure/TBEC in green solvents

    Article • Green Chemistry, January 2024, Royal Society of Chemistry

    Professor Walter Cabri

  14. Dimethyl carbonate as a green alternative to acetonitrile in reversed-phase liquid chromatography. Part II: Purification of a therapeutic peptide

    Article • Journal of Chromatography A, January 2024, Elsevier

    Professor Walter Cabri

  15. Dimethyl carbonate as a green alternative to acetonitrile in reversed-phase liquid chromatography. Part I: Separation of small molecules

    Article • Journal of Chromatography A, December 2023, Elsevier

    Professor Walter Cabri

  16. Copper-Free Heck–Cassar–Sonogashira and Suzuki–Miyaura Reactions of Aryl Chlorides: A Sustainable Approach

    Article • ACS Sustainable Chemistry & Engineering, October 2023, American Chemical Society (ACS)

    Professor Walter Cabri

  17. Fast Solution-Phase and Liquid-Phase Peptide Syntheses (SolPSS and LPPS) Mediated by Biomimetic Cyclic Propylphosphonic Anhydride (T3P®)

    Article • Molecules, October 2023, MDPI AG

    Professor Walter Cabri

  18. New Mechanistic Insights into the Copper-Free Heck–Cassar–Sonogashira Cross-Coupling Reaction

    Article • ACS Catalysis, August 2023, American Chemical Society (ACS)

    Professor Walter Cabri

  19. Investigation of the GnRH antagonist degarelix isomerization in biological matrices

    Article • Pharmacology Research & Perspectives, July 2023, Wiley

    Professor Walter Cabri

  20. Speeding up sustainable solution-phase peptide synthesis using T3P® as a green coupling reagent: methods and challenges

    Article • Green Chemistry, January 2023, Royal Society of Chemistry

    Professor Walter Cabri

  21. From green innovations in oligopeptide to oligonucleotide sustainable synthesis: differences and synergies in TIDES chemistry

    Article • Green Chemistry, January 2023, Royal Society of Chemistry

    Professor Walter Cabri

  22. Characterizing the Interactions of Dimethyl Sulfoxide with Water: A Rotational Spectroscopy Study

    Article • The Journal of Physical Chemistry A, September 2022, American Chemical Society (ACS)

    Professor Walter Cabri

  23. Application of Af4-Multidetection to Liraglutide in Its Formulation: Preserving and Representing Native Aggregation

    Article • Molecules, August 2022, MDPI AG

    Professor Walter Cabri

  24. Fast MacMillan’s Imidazolidinone-Catalyzed Enantioselective Synthesis of Polyfunctionalized 4-Isoxazoline Scaffolds

    Article • ACS Omega, July 2022, American Chemical Society (ACS)

    Professor Walter Cabri

  25. Carbodiimide-Mediated Beckmann Rearrangement of Oxyma-B as a Side Reaction in Peptide Synthesis

    Article • Molecules, June 2022, MDPI AG

    Professor Walter Cabri

  26. Benefits of a Mixed-Mode Stationary Phase to Address the Challenging Purification of an Industrially Relevant Peptide: A Proof-of-Concept Study

    Article • Separations, May 2022, MDPI AG

    Professor Walter Cabri

  27. A New Approach to Supramolecular Structure Determination in Pharmaceutical Preparation of Self-Assembling Peptides: A Case Study of Lanreotide Autogel

    Article • Pharmaceutics, March 2022, MDPI AG

    Professor Walter Cabri

  28. Sustainability in peptide chemistry: current synth. & purification techn. and future challenges

    Article • Green Chemistry, January 2022, Royal Society of Chemistry

    Professor Walter Cabri

  29. A translation of the twelve principles of green chemistry to guide the development of cross-coupling reactions

    Article • Catalysis Today, September 2021, Elsevier

    Professor Walter Cabri

  30. Downstream Processing of Therapeutic Peptides by Means of Preparative Liquid Chromatography

    Article • Molecules, August 2021, MDPI AG

    Professor Walter Cabri

  31. Expanding the Use of Dynamic Electrostatic Repulsion Reversed-Phase Chromatography: An Effective Elution Mode for Peptides Control and Analysis

    Article • Molecules, July 2021, MDPI AG

    Professor Walter Cabri

  32. Copper(II) Lysinate and Pseudoproline Assistance in the Convergent Synthesis of the GLP-1 Receptor Agonists Liraglutide and Semaglutide

    Article • Organic Process Research & Development, June 2021, American Chemical Society (ACS)

    Professor Walter Cabri

  33. Therapeutic Peptides Targeting PPI in Clinical Development: Overview, Mechanism of Action and Perspectives

    Article • Frontiers in Molecular Biosciences, June 2021, Frontiers

    Professor Walter Cabri

  34. Palladium Catalyst Recycling for Heck‐Cassar‐Sonogashira Cross‐Coupling Reactions in Green Solvent/Base Blend

    Article • ChemSusChem, May 2021, Wiley

    Professor Walter Cabri

  35. Process Intensification for the Purification of Peptidomimetics: The Case of Icatibant through Multicolumn Countercurrent Solvent Gradient Purification (MCSGP)

    Article • Industrial & Engineering Chemistry Research, May 2021, American Chemical Society (ACS)

    Professor Walter Cabri

  36. Replacing piperidine in solid phase peptide synthesis: effective Fmoc removal by alternative bases

    Article • Green Chemistry, January 2021, Royal Society of Chemistry

    Professor Walter Cabri

  37. Steps towards sustainable solid phase peptide synthesis: use and recovery of N-octyl pyrrolidone

    Article • Green Chemistry, January 2021, Royal Society of Chemistry

    Professor Walter Cabri

  38. Ampicillin sodium: Isolation, identification and synthesis of the last unknown impurity after 60 years of clinical use

    Article • Journal of Pharmaceutical and Biomedical Analysis, November 2020, Elsevier

    Professor Walter Cabri

  39. Ganoderma lucidum Ethanol Extracts Enhance Re-Epithelialization and Prevent Keratinocytes from Free-Radical Injury

    Article • Pharmaceuticals, August 2020, MDPI AG

    Professor Walter Cabri

  40. High–throughput enantioseparation of Nα–fluorenylmethoxycarbonyl proteinogenic amino acids through fast chiral chromatography on zwitterionic-teicoplanin stationary phases

    Article • Journal of Chromatography A, August 2020, Elsevier

    Professor Walter Cabri

  41. From batch to continuous chromatographic purification of a therapeutic peptide through multicolumn countercurrent solvent gradient purification

    Article • Journal of Chromatography A, August 2020, Elsevier

    Professor Walter Cabri

  42. Fast Heck–Cassar–Sonogashira (HCS) Reactions in Green Solvents

    Article • Organic Letters, April 2020, American Chemical Society (ACS)

    Professor Walter Cabri

  43. Modeling the nonlinear behavior of a bioactive peptide in reversed-phase gradient elution chromatography

    Article • Journal of Chromatography A, April 2020, Elsevier

    Professor Walter Cabri

  44. Overcoming Chemical Challenges in the Solid-Phase Synthesis of High-Purity GnRH Antagonist Degarelix. Part 2

    Article • Organic Process Research & Development, January 2020, American Chemical Society (ACS)

    Professor Walter Cabri

  45. Boosting basic-peptide separation through dynamic electrostatic-repulsion reversed-phase (d-ERRP) liquid chromatography

    Article • RSC Advances, January 2020, Royal Society of Chemistry

    Professor Walter Cabri

  46. Natural Occurring and Engineered Enzymes for Peptide Ligation and Cyclization

    Article • Frontiers in Chemistry, November 2019, Frontiers

    Professor Walter Cabri

  47. Overcoming Chemical Challenges in the Solid-Phase Synthesis of High-Purity GnRH Antagonist Degarelix. Part 1.

    Article • Organic Process Research & Development, November 2019, American Chemical Society (ACS)

    Professor Walter Cabri

  48. Novel insights into the chemistry of an old medicine: A general degradative pathway for penicillins from a piperacillin/tazobactam stability study

    Article • European Journal of Pharmaceutical Sciences, August 2019, Elsevier

    Professor Walter Cabri

  49. Green Solvent Mixtures for Solid-Phase Peptide Synthesis: A Dimethylformamide-Free Highly Efficient Synthesis of Pharmaceutical-Grade Peptides

    Article • ACS Sustainable Chemistry & Engineering, June 2019, American Chemical Society (ACS)

    Professor Walter Cabri

  50. Investigating the Neuroprotective Effects of Turmeric Extract: Structural Interactions of β-Amyloid Peptide with Single Curcuminoids

    Article • Scientific Reports, December 2016, Springer Science + Business Media

    Professor Walter Cabri

  51. Innovative chemical synthesis and conformational hints on the lipopeptide liraglutide

    Article • Journal of Peptide Science, May 2016, Wiley

    Dr Ivan Guryanov, Professor Walter Cabri

  52. Recovery of bioactive compounds from artichoke brines by nanofiltration

    Article • Food and Bioproducts Processing, April 2016, Elsevier

    Professor Walter Cabri

  53. Production of peptides as generic drugs: a patent landscape of octreotide

    Article • Expert Opinion on Therapeutic Patents, March 2016, Informa Healthcare

    Professor Walter Cabri

  54. Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2AReceptor Ligands

    Article • ChemMedChem, May 2015, Wiley

    Professor Walter Cabri

  55. Hypoglycemic effects of a standardized extract of salvia miltiorrhiza roots in rats

    Article • Pharmacognosy Magazine, January 2015, Medknow

    Professor Walter Cabri

  56. ST7612AA1, a Thioacetate-ω(γ-lactam carboxamide) Derivative Selected from a Novel Generation of Oral HDAC Inhibitors

    Article • Journal of Medicinal Chemistry, October 2014, American Chemical Society (ACS)

    Professor Walter Cabri

  57. Reducing effect of the Chinese medicinal herb, Salvia miltiorrhiza, on alcohol self-administration in Sardinian alcohol-preferring rats

    Article • Alcohol, September 2014, Elsevier

    Professor Walter Cabri

  58. Towards the development of 5-HT7 ligands combining serotonin-like and arylpiperazine moieties

    Article • European Journal of Medicinal Chemistry, June 2014, Elsevier

    Professor Walter Cabri

  59. Protective effect of Panax ginseng in cisplatin-induced cachexia in rats

    Article • Future Oncology, May 2014, Future Medicine

    Professor Walter Cabri

  60. 4,5,6,7-Tetrahydro-isoxazolo-[4,5-c]-pyridines as a new class of cytotoxic Hsp90 inhibitors

    Article • European Journal of Medicinal Chemistry, April 2014, Elsevier

    Professor Walter Cabri

  61. Synthesis and Evaluation of New Hsp90 Inhibitors Based on a 1,4,5-Trisubstituted 1,2,3-Triazole Scaffold

    Article • Journal of Medicinal Chemistry, March 2014, American Chemical Society (ACS)

    Professor Walter Cabri

  62. Biotransformation of Colchicinoids into Their Corresponding 3-O-Glucosyl Derivatives by Selected Strains of Bacillus megaterium

    Article • Molecular Biotechnology, February 2014, Springer Science + Business Media

    Professor Walter Cabri

  63. Development of a practical and sustainable strategy for the synthesis of ST1535 by an iron-catalyzed Kumada cross-coupling reaction

    Article • Tetrahedron Letters, February 2014, Elsevier

    Professor Walter Cabri

  64. Thermodynamic and kinetic investigation of monoketo-aldehyde-peroxyhemiacetal (MKA), a stereolabile degradation product of dihydroartemisinin

    Article • RSC Advances, January 2014, Royal Society of Chemistry

    Professor Marco Pierini, Claudio Villani, Professor Walter Cabri

  65. Lactam based 7-amino suberoylamide hydroxamic acids as potent HDAC inhibitors

    Article • Bioorganic & Medicinal Chemistry Letters, January 2014, Elsevier

    Professor Walter Cabri

  66. Effect of SAMITAL® in the treatment of chemotherapy-induced mucositis in adult oncohematological patients

    Article • Future Oncology, November 2013, Future Medicine

    Professor Walter Cabri

  67. SAMITAL®: a new botanical drug for the treatment of mucositis induced by oncological therapies

    Article • Future Oncology, November 2013, Future Medicine

    Professor Walter Cabri

  68. Synthesis and Biological Evaluation of Metabolites of 2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), A Potent Antagonist of the A2A Adenosine Receptor for the Treatment of Parkinson’s Disease

    Article • Journal of Medicinal Chemistry, June 2013, American Chemical Society (ACS)

    Professor Walter Cabri

  69. Synthesis of (E)-8-(3-Chlorostyryl)caffeine Analogues Leading to 9-Deazaxanthine Derivatives as Dual A2A Antagonists/MAO-B Inhibitors

    Article • Journal of Medicinal Chemistry, January 2013, American Chemical Society (ACS)

    Professor Walter Cabri

  70. Identification of a novel arylpiperazine scaffold for fatty acid amide hydrolase inhibition with improved drug disposition properties

    Article • Bioorganic & Medicinal Chemistry Letters, January 2013, Elsevier

    Dr sandra gemma, Dr Stefania Butini, Professor Walter Cabri

  71. Camptothecins in tumor homing via an RGD sequence mimetic

    Article • Bioorganic & Medicinal Chemistry Letters, October 2012, Elsevier

    Professor Walter Cabri

  72. Discovery of Potent Inhibitors of Human and Mouse Fatty Acid Amide Hydrolases

    Article • Journal of Medicinal Chemistry, August 2012, American Chemical Society (ACS)

    Dr sandra gemma, Dr Stefania Butini, Professor Walter Cabri

  73. Histone deacetylase inhibitors in the treatment of cancer: overview and perspectives

    Article • Future Medicinal Chemistry, July 2012, Future Science

    Professor Walter Cabri

  74. Isoxazolo(aza)naphthoquinones: A new class of cytotoxic Hsp90 inhibitors

    Article • European Journal of Medicinal Chemistry, July 2012, Elsevier

    Professor Walter Cabri

  75. New retinoid derivatives as back-ups of Adarotene

    Article • Bioorganic & Medicinal Chemistry, April 2012, Elsevier

    Professor Walter Cabri

  76. Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions

    Article • Organic & Biomolecular Chemistry, January 2012, Royal Society of Chemistry

    Professor Walter Cabri

  77. Novel 3,4-Isoxazolediamides as Potent Inhibitors of Chaperone Heat Shock Protein 90

    Article • Journal of Medicinal Chemistry, December 2011, American Chemical Society (ACS)

    Professor Walter Cabri

  78. Erratum to “Efficient organic monoliths prepared by γ-radiation induced polymerization in the evaluation of histone deacetylase inhibitors by capillary(nano)-high performance liquid chromatography and ion trap mass spectrometry” [J. Chromatogr. A 1218 ...

    Article • Journal of Chromatography A, December 2011, Elsevier

    Professor Marco Pierini, Claudio Villani, Professor Walter Cabri

  79. Identification of impurities in artemisinin, their behavior in high performance liquid chromatography and implications for the quality of derived anti-malarial drugs

    Article • Journal of Chromatography A, September 2011, Elsevier

    Professor Walter Cabri

  80. Derivatives of R-Aminocarnitine without Ammonium Moiety as Liver Carnitine Palmitoyltransferase I (L-CPT I) Inhibitors

    Article • ChemMedChem, August 2011, Wiley

    Professor Walter Cabri

  81. Efficient organic monoliths prepared by γ-radiation induced polymerization in the evaluation of histone deacetylase inhibitors by capillary(nano)-high performance liquid chromatography and ion trap mass spectrometry

    Article • Journal of Chromatography A, June 2011, Elsevier

    Professor Marco Pierini, Claudio Villani, Professor Walter Cabri

  82. Stereolability of Dihydroartemisinin, an Antimalarial Drug: A Comprehensive Kinetic Investigation. Part 2

    Article • The Journal of Organic Chemistry, May 2011, American Chemical Society (ACS)

    Professor Marco Pierini, Claudio Villani, Professor Walter Cabri

  83. Oxime Amides as a Novel Zinc Binding Group in Histone Deacetylase Inhibitors: Synthesis, Biological Activity, and Computational Evaluation

    Article • Journal of Medicinal Chemistry, March 2011, American Chemical Society (ACS)

    Professor Walter Cabri

  84. Stereolability of Dihydroartemisinin, an Antimalarial Drug: A Comprehensive Thermodynamic Investigation. Part 1

    Article • The Journal of Organic Chemistry, February 2011, American Chemical Society (ACS)

    Professor Marco Pierini, Claudio Villani, Professor Walter Cabri

  85. Non-Natural Macrocyclic Inhibitors of Histone Deacetylases: Design, Synthesis, and Activity

    Article • Journal of Medicinal Chemistry, December 2010, American Chemical Society (ACS)

    Professor Walter Cabri

  86. A new group of oxime carbamates as reversible inhibitors of fatty acid amide hydrolase

    Article • Bioorganic & Medicinal Chemistry Letters, August 2010, Elsevier

    Professor Walter Cabri

  87. Direct B-Alkyl Suzuki−Miyaura Cross-Coupling of 2-Halopurines. Practical Synthesis of ST1535, a Potent Adenosine A2A Receptor Antagonist

    Article • The Journal of Organic Chemistry, July 2010, American Chemical Society (ACS)

    Professor Walter Cabri

  88. Aminocarnitine Ureidic Derivatives as Inhibitors of Carnitine Palmitoyltransferase I

    Article • ChemMedChem, March 2010, Wiley

    Professor Walter Cabri

  89. Stereodynamic Investigation of Labile Stereogenic Centres in Dihydroartemisinin

    Article • Molecules, March 2010, MDPI AG

    Professor Marco Pierini, Claudio Villani, Professor Walter Cabri

  90. Enol Carbamates as Inhibitors of Fatty Acid Amide Hydrolase (FAAH) Endowed with High Selectivity for FAAH over the Other Targets of the Endocannabinoid System

    Article • ChemMedChem, February 2010, Wiley

    Professor Walter Cabri

  91. Extending the use of “Inverted Chirality Columns Approach” for enantiomeric excess determination in absence of reference samples: Application to a water-soluble camptothecin derivative

    Article • Journal of Chromatography A, February 2010, Elsevier

    Claudio Villani, Professor Walter Cabri

  92. 2-Azetidinones: synthesis of new bis(indolyl)butyl-β-lactams

    Article • New Journal of Chemistry, January 2010, Royal Society of Chemistry

    Professor Walter Cabri

  93. Azetidinones as Zinc-Binding Groups to Design Selective HDAC8 Inhibitors

    Article • ChemMedChem, October 2009, Wiley

    Professor Walter Cabri

  94. Corrigendum to “N-Hydroxy-(4-oxime)-cinnamide: A versatile scaffold for the synthesis of novel histone deacetilase (HDAC) inhibitors” [Bioorg. Med. Chem. Lett. 19 (2009) 2346]

    Article • Bioorganic & Medicinal Chemistry Letters, July 2009, Elsevier

    Professor Walter Cabri

  95. Exploring bis-(indolyl)methane moiety as an alternative and innovative CAP group in the design of histone deacetylase (HDAC) inhibitors

    Article • Bioorganic & Medicinal Chemistry Letters, May 2009, Elsevier

    Professor Walter Cabri

  96. N-Hydroxy-(4-oxime)-cinnamide: A versatile scaffold for the synthesis of novel histone deacetilase (HDAC) inhibitors

    Article • Bioorganic & Medicinal Chemistry Letters, April 2009, Elsevier

    Professor Walter Cabri

  97. Catalysis: The pharmaceutical perspective

    Article • Catalysis Today, February 2009, Elsevier

    Professor Walter Cabri

  98. On-column epimerization of dihydroartemisinin: An effective analytical approach to overcome the shortcomings of the International Pharmacopoeia monograph☆

    Article • Journal of Chromatography B, November 2008, Elsevier

    Professor Walter Cabri

  99. Novel Substituted Aminoalkylguanidines as Potential Antihyperglycemic and Food Intake-Reducing Agents

    Article • Journal of Medicinal Chemistry, May 2008, American Chemical Society (ACS)

    Professor Walter Cabri

  100. E-ring-modified 7-oxyiminomethyl camptothecins: Synthesis and preliminary in vitro and in vivo biological evaluation

    Article • Bioorganic & Medicinal Chemistry Letters, May 2008, Elsevier

    Professor Walter Cabri

  101. Synthesis and Biological Activity of Fluorinated Combretastatin Analogues

    Article • Journal of Medicinal Chemistry, April 2008, American Chemical Society (ACS)

    Professor Walter Cabri

  102. Catalysis: A key technology for a green approach to pharmaceutical production

    Article • RENDICONTI LINCEI, December 2007, Springer Science + Business Media

    Professor Walter Cabri

  103. ω-Alkoxy analogues of SAHA (vorinostat) as inhibitors of HDAC: A study of chain-length and stereochemical dependence

    Article • Bioorganic & Medicinal Chemistry Letters, November 2007, Elsevier

    Professor Walter Cabri

  104. Combination of HPLC “Inverted Chirality Columns Approach” and MS/MS Detection for Extreme Enantiomeric Excess Determination Even in Absence of Reference Samples. Application to Camptothecin Derivatives

    Article • Analytical Chemistry, August 2007, American Chemical Society (ACS)

    Claudio Villani, Professor Walter Cabri

  105. Polymorphisms and Patent, Market, and Legal Battles:  Cefdinir Case Study

    Article • Organic Process Research & Development, December 2006, American Chemical Society (ACS)

    Professor Walter Cabri

  106. Cefdinir: A comparative study of anhydrous vs. monohydrate formMicrostructure and tabletting behaviour

    Article • European Journal of Pharmaceutics and Biopharmaceutics, October 2006, Elsevier

    Professor Walter Cabri

  107. Development of a Practical High-Yield Industrial Synthesis of Pergolide Mesylate

    Article • Organic Process Research & Development, February 2006, American Chemical Society (ACS)

    Professor Walter Cabri

  108. Evolution of an acylase active on cephalosporin C

    Article • Protein Science, December 2005, Wiley

    Professor Walter Cabri

  109. Blakeslea trispora Genes for Carotene Biosynthesis

    Article • Applied and Environmental Microbiology, September 2004, ASM Journals

    Professor Walter Cabri

  110. Biotechnological lycopene production by mated fermentation of Blakeslea trispora

    Article • Applied Microbiology and Biotechnology, July 2004, Springer Science + Business Media

    Professor Walter Cabri

  111. Natural lycopene from Blakeslea trispora: all-trans lycopene thermochemical and structural properties

    Article • Thermochimica Acta, July 2004, Elsevier

    Professor Walter Cabri

  112. A New Carbanionic One-Carbon Ring Enlargement—Alkylation of Lactams.

    Article • ChemInform, February 2004, Wiley

    Professor Walter Cabri

  113. A New Carbanionic One-Carbon Ring Enlargement-Alkylation of Lactams

    Article • Synlett, January 2003, Thieme Publishing Group

    Professor Walter Cabri

  114. Walter Cabri and Romano Di Fabio, From Bench to Market: The Evolution of Chemical Synthesis

    Article • Journal of Pharmacy and Pharmacology, December 2001, Oxford University Press (OUP)

    Professor Walter Cabri

  115. Palladium-catalysed reduction of 3-substituted cephems. A high yield approach to ceftizoxime synthetic intermediates

    Article • Tetrahedron Letters, May 1997, Elsevier

    Professor Walter Cabri

  116. Solid-phase synthesis of indoles using the palladium-catalysed coupling of alkynes with iodoaniline derivatives

    Article • Tetrahedron Letters, March 1997, Elsevier

    Professor Walter Cabri

  117. Preparation of diphenylmethyl esters by oxone® oxidation of benzophenone hydrazone

    Article • Tetrahedron Letters, February 1997, Elsevier

    Professor Walter Cabri

  118. Synthesis and cytotoxic activity of alkylidene- and alkyl-substituted camptothecins

    Article • Bioorganic & Medicinal Chemistry Letters, January 1997, Elsevier

    Professor Walter Cabri

  119. A high yield semisynthetic approach to 2′-epi-Taxol

    Article • Tetrahedron Letters, July 1996, Elsevier

    Professor Walter Cabri

  120. Synthesis and antitumor activity of a new class of water soluble camptothecin derivatives

    Article • Bioorganic & Medicinal Chemistry Letters, March 1996, Elsevier

    Professor Walter Cabri

  121. A new high yield semisynthetic approach to (20s)-9-NH2-camptothecin based on a sequence of palladium-catalysed reductions

    Article • Tetrahedron Letters, December 1995, Elsevier

    Professor Walter Cabri

  122. The Ligand Effect in Copper(I)-Catalyzed Chemoselective Amide Carbamoylation in Cabergoline Synthesis

    Article • Synlett, June 1995, Thieme Publishing Group

    Professor Walter Cabri

  123. Non-toxic ligands in samarium diiodide-mediated cyclizations

    Article • Tetrahedron Letters, February 1995, Elsevier

    Professor Walter Cabri

  124. Recent Developments and New Perspectives in the Heck Reaction

    Article • Accounts of Chemical Research, January 1995, American Chemical Society (ACS)

    Professor Walter Cabri

  125. Zinc halides-mediated nucleophilic attack of thioacid salts in non protic media. A key step in the total synthesis of penems

    Article • Tetrahedron Letters, May 1994, Elsevier

    Professor Walter Cabri

  126. Iron(III)–copper(II) and manganese(III)–copper(II) promoted cyclizations: a new stereoselective approach towards α-methyl substituted penicillin derivatives

    Article • Journal of the Chemical Society Chemical Communications, January 1994, Royal Society of Chemistry

    Professor Walter Cabri

  127. 1,10-Phenanthroline derivatives: a new ligand class in the Heck reaction. Mechanistic aspects

    Article • The Journal of Organic Chemistry, December 1993, American Chemical Society (ACS)

    Professor Walter Cabri

  128. Synthesis and β-lactamase inhibitory activity of 6-hydroxyethyl thiaclavulanic acid.

    Article • Bioorganic & Medicinal Chemistry Letters, November 1993, Elsevier

    Professor Walter Cabri

  129. Samarium diiodide mediated reduction of allyl halides. A new reductive approach to exomethylene cephams.

    Article • Tetrahedron Letters, October 1993, Elsevier

    Professor Walter Cabri

  130. Metal-catalyzed and -promoted cyclizations for the synthesis of cephalosporins: a possible DAOC/DAC synthetase biomimetic process.

    Article • Tetrahedron, July 1993, Elsevier

    Professor Walter Cabri

  131. Cobalt-catalyzed methoxycarbonylation of naphthalene mono- and di-sulfonates to naphthalene mono- and di-esters

    Article • Journal of Organometallic Chemistry, June 1993, Elsevier

    Professor Walter Cabri

  132. The total synthesis of ritipenems. Construction of penem thiazoline ring by incorporation of two 2C units of glycolic acid.

    Article • Tetrahedron Letters, May 1993, Elsevier

    Professor Walter Cabri

  133. A Facile One-Pot Synthesis of Polyfunctionalized 2-Unsubstituted Benzo[b]furans

    Article • Synlett, January 1993, Thieme Publishing Group

    Professor Walter Cabri

  134. Metal-promoted thiyl radical cyclizations in β-lactam antibiotics

    Article • Tetrahedron Letters, August 1992, Elsevier

    Professor Walter Cabri

  135. Palladium-catalyzed arylation of unsymmetrical olefins. Bidentate phosphine ligand controlled regioselectivity

    Article • The Journal of Organic Chemistry, June 1992, American Chemical Society (ACS)

    Professor Walter Cabri

  136. .alpha.-Regioselectivity in palladium-catalyzed arylation of acyclic enol ethers

    Article • The Journal of Organic Chemistry, February 1992, American Chemical Society (ACS)

    Professor Walter Cabri

  137. Bidentate Nitrogen Ligands in Heck Type Reactions

    Article • Synlett, January 1992, Thieme Publishing Group

    Professor Walter Cabri

  138. Synthesis of 5-Alkyl Substituted Uracil Derivatives from Barbituric Acid

    Article • Heterocycles, January 1992, Japan Institute of Heterocyclic Chemistry

    Professor Walter Cabri

  139. Heck reaction on anthraquinone derivatives: ligand, solvent and salt effects

    Article • The Journal of Organic Chemistry, September 1991, American Chemical Society (ACS)

    Professor Walter Cabri

  140. Palladium-catalyzed α-arylation of vinyl butyl ether with aryl halides

    Article • Tetrahedron Letters, April 1991, Elsevier

    Professor Walter Cabri

  141. The stereocontrolled formation of cyclic vicinal cis-diols via a samarium diiodide pinacol coupling of dialdehydes

    Article • Tetrahedron Letters, February 1991, Elsevier

    Dr Jose Luis Chiara, Professor Walter Cabri

  142. Ligand-controlled .alpha.-regioselectivity in palladium-catalyzed arylation of butyl vinyl ether

    Article • The Journal of Organic Chemistry, May 1990, American Chemical Society (ACS)

    Professor Walter Cabri

  143. A novel synthesis of (+)-4-demethoxydaunomycinone

    Article • Journal of the Chemical Society Perkin Transactions 1, January 1990, Royal Society of Chemistry

    Professor Walter Cabri

  144. Palladium-catalyzed reduction of aryl sulfonates. Reduction versus hydrolysis selectivity control

    Article • The Journal of Organic Chemistry, January 1990, American Chemical Society (ACS)

    Professor Walter Cabri

  145. Enzymic hydrolysis of alkyl 3,4-epoxybutyrates. A new route to (R)-(-)-carnitine chloride

    Article • The Journal of Organic Chemistry, January 1988, American Chemical Society (ACS)

    Professor Walter Cabri

  146. Enzymatic resolution of 2,3-epoxyalcohols, intermediates in the synthesis of the gypsy moth sex pheromone

    Article • Tetrahedron Letters, January 1988, Elsevier

    Professor Walter Cabri

  147. Lipase-catalyzed resolution of chiral 2-amino 1-alcohols

    Article • The Journal of Organic Chemistry, November 1987, American Chemical Society (ACS)

    Professor Walter Cabri