Dr Fabrizio Machetti
Consiglio Nazionale delle Ricerche
Professor, Chemistry
Italy
My co-authors include
Dr Giuliano Giambastiani
Paolo Paoli
Prof Andrea Trabocchi
My Publications
Transesterification of activated esters
European Journal of Organic Chemistry
March 2020
Multiwalled carbon nanotubes for combination therapy: a biodistribution and efficacy pi...
Journal of Materials Chemistry B
January 2019
The role of molecular structure in determining the acidity of nitroacetoamides in water.
Molecules
December 2018
From nitro compounds to isoxazoles
European Journal of Organic Chemistry
August 2016
ChemInform Abstract: Reactivity of [60]Fullerene with Primary Nitro Compounds: Addition...
ChemInform
March 2015
Reactivity of [60]Fullerene with Primary Nitro Compounds: Addition or Catalysed Condens...
European Journal of Organic Chemistry
October 2014
Condensation of Primary Nitro Compounds to Isoxazole Derivatives: Stoichiometric To Cat...
January 2014
ChemInform Abstract: Conjugate Addition versus Cycloaddition/Condensation of Nitro Comp...
ChemInform
June 2013
Conjugate Addition versus Cycloaddition/Condensation of Nitro Compounds in Water: Selec...
Chemistry - A European Journal
November 2012
ChemInform Abstract: Acid-Base-Catalyzed Condensation Reaction in Water: Isoxazolines a...
ChemInform
May 2012
Acid-Base-Catalysed Condensation Reaction in Water: Isoxazolines and Isoxazoles from Ni...
Chemistry - A European Journal
January 2012
ChemInform Abstract: Five-Membered Heterocycles: 1,3-Azoles
ChemInform
December 2011
Five-Membered Heterocycles: 1,3-Azoles
July 2011
ChemInform Abstract: Practical Synthesis of Both Enantiomers of Protected 4-Oxopipecoli...
ChemInform
May 2010
ChemInform Abstract: Design and Synthesis of a New Bicyclic Dipeptide Isostere.
ChemInform
May 2010
ChemInform Abstract: Synthesis of Taurine Analogues. Part 2. Amino-Sulfonation of Alken...
ChemInform
May 2010
Identification of Inhibitors of Drug-Resistant <i>Candida albicans</i> Strains from a L...
Journal of Medicinal Chemistry
February 2010
Copper-Catalyzed Synthesis of Isoxazoles
Synfacts
January 2010
Conversion of a nitrosocarbonyl hetero Diels–Alder cycloadduct to useful isoxazoline-ca...
Tetrahedron
December 2009
Base- and Copper-Catalysed Condensation of Primary Activated Nitro Compounds with Enoli...
European Journal of Organic Chemistry
December 2009
Michael Additions versus Cycloaddition Condensations with Ethyl Nitroacetate and Electr...
Chemistry - A European Journal
August 2009
ChemInform Abstract: Synthesis of 4,5-Dihydroisoxazoles by Condensation of Primary Nitr...
ChemInform
January 2009
Synthesis of 4,5-Dihydroisoxazoles by Condensation of Primary Nitro Compounds with Alke...
Chemistry - A European Journal
September 2008
ChemInform Abstract: 4,5-Dihydroisoxazoles by Copper(II)-Catalyzed Condensation of Prim...
ChemInform
January 2008
ChemInform Abstract: Isoxazoles and Isoxazolines by 1,3-Dipolar Cycloaddition: Base-Cat...
ChemInform
January 2008
Isoxazoles
January 2008
4,5-Dihydroisoxazoles by Copper(II)-Catalysed Condensation of Primary Nitroalkanes with...
Synlett
September 2007
Isoxazoles and Isoxazolines by 1,3-Dipolar Cycloaddition: Base-Catalysed Condensation o...
European Journal of Organic Chemistry
September 2007
Parallel Synthesis of an Amide Library Based on the 6,8-Dioxa-3-azabicyclo[3.2.1]octane...
Journal of Combinatorial Chemistry
May 2007
1,4-Diazabicyclo[2.2.2]octane (DABCO) as an Efficient Reagent for the Synthesis of Isox...
ChemInform
February 2007
Synthesis of bicyclic molecular scaffolds (BTAa): An investigation towards new selectiv...
Bioorganic & Medicinal Chemistry
November 2006
1,4-Diazabicyclo[2.2.2]octane (DABCO) as an Efficient Reagent for the Synthesis of Isox...
European Journal of Organic Chemistry
November 2006
Synthesis of Benzo[c]quinolizin-3-ones: Discovery and Development of Novel Inhibitors o...
ChemInform
August 2006
The Synthesis of 4-Hydroxypipecolic Acids by Stereoselective Cycloaddition of Configura...
European Journal of Organic Chemistry
July 2006
1,2,5-Oxadiazole (Furazan) Derivatives from Benzoylnitromethane and Dipolarophiles in t...
European Journal of Organic Chemistry
July 2006
Design, Synthesis, and Applications of 3-Aza-6,8-dioxabicyclo[3.2.1]octane-Based Scaffo...
ChemInform
May 2006
Inhibition of rabbit brain 4-aminobutyrate transaminase by some taurine analogues: A ki...
Biochemical Pharmacology
May 2006
Isoxazoline Derivatives from Activated Primary Nitro Compounds and Tertiary Diamines.
ChemInform
February 2006
Design, Synthesis, and Applications of 3-Aza-6,8-Dioxabicyclo[3.2.1]Octane-Based Scaffo...
Synlett
January 2006
Isoxazoline derivatives from activated primary nitrocompounds and tertiary diamines
Tetrahedron Letters
November 2005
A New Bicyclic Dipeptide Isostere with Pyrrolizidinone Skeleton
The Journal of Organic Chemistry
February 2005
Synthesis of Free andNα-Fmoc-/Nγ-Boc-Protected (2S,4S)- and (2S,4R)-4-Aminopipecolic Acids
European Journal of Organic Chemistry
July 2004
Enantiospecific synthesis of 3-aza-6,8-dioxa-bicyclo[3.2.1]octane carboxylic acids from...
Tetrahedron
July 2003
A specific taurine recognition site in the rabbit brain is responsible for taurine effe...
British Journal of Pharmacology
June 2003
Neat reaction of carboxylic acid methyl esters and amines for efficient parallel synthe...
Comptes Rendus Chimie
May 2003
Interactions of taurine and structurally related analogues with the GABAergic system an...
British Journal of Pharmacology
March 2003
Synthesis of a new enantiopure bicyclic γ/δ-amino acid (BTKa) derived from tartaric aci...
Tetrahedron
December 2002
Synthesis of analogues of taurine: 2-aminoalkanesulfonic acids
European Journal of Organic Chemistry
April 2002
Bicyclic Compounds Derived from Tartaric Acid and α-Amino Acids (BTAas): Synthesis of N...
European Journal of Organic Chemistry
March 2002
Novel inhibitors of 5α-reductase
Expert Opinion on Therapeutic Patents
February 2002
Synthesis of Taurine Analogues from Alkenes
January 2002
Effects of Taurine and some Structurally Related Analogues on the Central Mechanism of ...
January 2002
Effect of C-ring modifications in benzo[c]quinolizin-3-ones, new selective inhibitors o...
Bioorganic & Medicinal Chemistry
June 2001
Practical synthesis of both enantiomers of protected 4-oxopipecolic acid
Tetrahedron
June 2001
ChemInform Abstract: Modification of the Aza-Robinson Annulation for the Synthesis of 4...
ChemInform
April 2001
ChemInform Abstract: Benzo[c]quinolizin-3-ones: A Novel Class of Potent and Selective N...
ChemInform
March 2001
ChemInform Abstract: Synthesis of Taurine Analogues. Part 1. 2-Aminosulfonic Acids from...
ChemInform
February 2001
ChemInform Abstract: Oligomers of Enantiopure Bicyclic γ/δ-Amino Acids (BTAa). Part 1. ...
ChemInform
February 2001
Design and synthesis of a new bicyclic dipeptide isostere
Chemical Communications
January 2001
Oligomers of Enantiopure Bicyclic γ/δ-Amino Acids (BTAa). 1. Synthesis and Conformation...
Organic Letters
December 2000
Modification of the Aza-Robinson Annulation for the Synthesis of 4-Methyl-Benzo[ c ]qu...
The Journal of Organic Chemistry
November 2000
Benzo[ c ]quinolizin-3-ones: A Novel Class of Potent and Selective Nonsteroidal Inhib...
Journal of Medicinal Chemistry
October 2000
Synthesis and Reactivity of Bicycles Derived from Tartaric Acid and α-Amino Acids: A N...
The Journal of Organic Chemistry
July 2000
Synthesis of taurine analogues. Part 1: 2-aminosulfonic acids from alkene-sulfur monoch...
Journal of Chemical Research
March 2000
Synthesis and Reactivity of Bicycles Derived from Tartaric Acid and α-Amino Acids: A N...
The Journal of Organic Chemistry
September 1999
19-Nor-10-azasteroids. 5. 1 A Synthetic Strategy for the Preparation of (+)-17-(3-Pyri...
The Journal of Organic Chemistry
June 1999
Stereoselectivity in the TiCl4-catalysed reaction of Danishefsky's diene with a N-(acyl...
Tetrahedron
September 1998
A Concise Route to 19-Nor-10-azasteroids, a New Class of Steroid 5α-Reductase Inhibito...
The Journal of Organic Chemistry
June 1998
19-Nor-10-azasteroids, a New Class of Steroid 5α-Reductase Inhibitors. 2. 1 X-ray Stru...
Journal of Medicinal Chemistry
October 1997
19-Nor-10-azasteroids: A Novel Class of Inhibitors for Human Steroid 5α-Reductases 1 a...
Journal of Medicinal Chemistry
March 1997
Synthesis and X-ray study of hexahydro- and tetrahydrophospholo-[2,3-d]isoxazoles, a ne...
Journal of Heterocyclic Chemistry
July 1996
A new synthesis of (2S)-4-oxopipecolic acid by thermal rearrangement of enantiopure spi...
Tetrahedron Letters
June 1996
