Publication
Open-science discovery of DNDI-6510, a compound that addresses genotoxic and metabolic liabilities of the COVID Moonshot SARS-CoV-2 Mpro lead inhibitor
Ed J. Griffen, Daren Fearon, Briana L. McGovern, Lizbe Koekemoer, Blake H. Balcomb, Tamas Szommer, Gwendolyn Fate, Ralph P. Robinson, Bruce A. Lefker, Shirly Duberstein, Noa Lahav, Stephanie Braillard, Laura Vangeel, Manon Laporte, Fabienne Burgat Charvillon, A. Kenneth MacLeod, Andrew Wells, Pauline Garner, Richard Knight, Paul Rees, Anthony Simon, Dirk Jochmans, Johan Neyts, Kevin D. Read, Haim Barr, Matthew Robinson, Alpha Lee, Nir London, John Chodera, Frank von Delft, Kris M. White, Ben Perry, Peter Sjö, Annette von Delft
June 2025, Cold Spring Harbor Laboratory Press
DOI: 10.1101/2025.06.16.660018