Publication
Preliminary investigation of 6,7-dihydropyrazolo[1,5-a]pyrazin-4-one derivatives as a novel series of mGlu5 receptor positive allosteric modulators with efficacy in preclinical models of schizophrenia
Susana Conde-Ceide, Jesús Alcázar, Sergio A. Alonso de Diego, Silvia López, María Luz Martín-Martín, Carlos M. Martínez-Viturro, Miguel-Angel Pena, Han Min Tong, Hilde Lavreysen, Claire Mackie, Thomas M. Bridges, J. Scott Daniels, Colleen M. Niswender, Carrie K. Jones, Gregor J. Macdonald, Thomas Steckler, P. Jeffrey Conn, Shaun R. Stauffer, Craig W. Lindsley, José Manuel Bartolomé-Nebreda
Bioorganic & Medicinal Chemistry Letters, January 2016, Elsevier
DOI: 10.1016/j.bmcl.2015.11.098