Contact

All Stories

  1. N-Arylsulfonylated C-Homoaporphines as a New Class of Antiplatelet and Antimicrobial Agents

    Article • ACS Medicinal Chemistry Letters, December 2024, American Chemical Society (ACS)

    Prof. Sandeep Chaudhary

  2. Emerging Trends in Quinoxaline‐Based Analogs as Protein Kinase Inhibitors: Structural Developments and SAR Insights

    Article • ChemMedChem, December 2024, Wiley

    Prof. Sandeep Chaudhary

  3. Targeting cancer using scaffold-hopping approaches: illuminating SAR to improve drug design

    Article • Drug Discovery Today, September 2024, Elsevier

    Prof. Sandeep Chaudhary

  4. Pyrazolo[1,5-a]pyrimidine as a Prominent Framework for Tropomyosin Receptor Kinase (Trk) Inhibitors—Synthetic Strategies and SAR Insights

    Article • Molecules, July 2024, MDPI AG

    Prof. Sandeep Chaudhary

  5. ‘Cephalandole A’ analogues as a new class of antioxidant agents: Design, microwave-assisted synthesis, bioevaluation, SAR and in silico studies

    Article • Journal of Molecular Structure, May 2024, Elsevier

    Prof. Sandeep Chaudhary

  6. 1,2,4,5‐Tetraoxane derivatives/hybrids as potent antimalarial endoperoxides: Chronological advancements, structure−activity relationship (SAR) studies and future perspectives

    Article • Medicinal Research Reviews, April 2024, Wiley

    Prof. Sandeep Chaudhary

  7. Transformation of PMMA from sunlight‐blocking to sunlight‐activated coupled with DNH photocatalytic platform for oxidative coupling of amines and generation/regeneration of LDC/NADH

    Article • Photochemistry and Photobiology, December 2023, Wiley

    Prof. Sandeep Chaudhary

  8. Chemo-/Regio-Selective Synthesis of Novel Functionalized Spiro[pyrrolidine-2,3′-oxindoles] under Microwave Irradiation and Their Anticancer Activity

    Article • Molecules, September 2023, MDPI AG

    Prof. Sandeep Chaudhary

  9. Artemisinin-inspired novel functionalized aryloxy-arylvinyl-1,2,4-trioxanes as potent anticancer agents: Design, synthesis, bioevaluation, SAR and in silico studies

    Article • Journal of Molecular Structure, September 2023, Elsevier

    Dr. Dharmendra Kumar Yadav, Prof. Sandeep Chaudhary

  10. Natural-Product-Inspired Microwave-Assisted Synthesis of Novel Spirooxindoles as Antileishmanial Agents: Synthesis, Stereochemical Assignment, Bioevaluation, SAR, and Molecular Docking Studies

    Article • Molecules, June 2023, MDPI AG

    Prof. Sandeep Chaudhary

  11. Discovering the role of N-heterocyclic carbene as hydrogen borrowing organocatalyst: metal-free, directN-alkylation of amines with benzyl alcohols

    Article • Organic Chemistry Frontiers, January 2023, Royal Society of Chemistry

    Prof. Sandeep Chaudhary

  12. Regiodivergent Cu-Promoted, AcOH-Switchable Distal Versus Proximal Direct Cyanation of 1-Aryl-1H-indazoles and 2-Aryl-2H-indazoles via Aerobic Oxidative C–H Bond Activation

    Article • The Journal of Organic Chemistry, November 2022, American Chemical Society (ACS)

    Prof. Sandeep Chaudhary

  13. Unprecedented TMEDA‐Catalyzed Regioselective Decarboalkoxy C‐N Bond Formation: A Unified Direct Access to Indolo[2,1‐a]isoquinoline and Dibenzopyrrocoline Alkaloids

    Article • Chemistry - An Asian Journal, May 2022, Wiley

    Dr. MOHIT K TIWARI, Prof. Sandeep Chaudhary

  14. Biological Evaluation in Resistant Cancer Cells and Study of Mechanism of Action of Arylvinyl-1,2,4-Trioxanes

    Article • Pharmaceuticals, March 2022, MDPI AG

    Dr. MOHIT K TIWARI, Dr. Dharmendra Kumar Yadav, Prof. Sandeep Chaudhary

  15. Discovery of Natural Product Inspired 3-Phenyl-1H-isochromen-1-ones as Highly Potent Antioxidant and Antiplatelet Agents: Design, Synthesis, Biological Evaluation, SAR and In Silico Studies

    Article • Current Pharmaceutical Design, March 2022, Bentham Science Publishers

    Prof. Sandeep Chaudhary, Dr. Dharmendra Kumar Yadav, Na'il Saleh

  16. Artemisinin Analogues as a Novel Class of Antimalarial Agents: Recent Developments, Current Scenario and Future Perspectives

    Article • February 2022, Bentham Science Publishers

    Dr. MOHIT K TIWARI, Prof. Sandeep Chaudhary

  17. Oxidant-Switched Palladium-Catalyzed Regioselective Mono- versus Bis-ortho-Aroylation of 1-Aryl-1H-indazoles with Aldehydes via C–H Bond Activation

    Article • The Journal of Organic Chemistry, February 2022, American Chemical Society (ACS)

    Prof. Sandeep Chaudhary

  18. Developments in Organocatalyzed C(Ar)- C(Ar) Bond formation Reactions Involving Single Electron Transfer Mechanism: An Overview

    Article • Current Organocatalysis, December 2021, Bentham Science Publishers

    Prof. Sandeep Chaudhary

  19. Reaction of Hetareno[e]pyrrole‐2,3‐diones with Thiols: An Approach to Two Distinct 5‐Thio‐Substituted Pyrrole‐2‐one Derivatives

    Article • ChemistrySelect, December 2021, Wiley

    Prof. Sandeep Chaudhary

  20. Novel halogenated Arylvinyl-1,2,4 trioxanes as potent antiplasmodial as well as anticancer agents: Synthesis, Bioevaluation, structure-activity relationship and in-silico studies

    Article • European Journal of Medicinal Chemistry, July 2021, Elsevier

    Dr. MOHIT K TIWARI, Dr. Dharmendra Kumar Yadav, Prof. Sandeep Chaudhary

  21. Recent Advancements in the Synthesis and Chemistry of Benzo-fused Nitrogen- and Oxygen-based Bioactive Heterocycles

    Article • Current Topics in Medicinal Chemistry, July 2021, Bentham Science Publishers

    Prof. Sandeep Chaudhary, Nawal Kishore Sahu

  22. Lewis Acid/Oxidant as Rapid Regioselective Halogenating Reagent System for Direct Halogenation of Fused Bi‐/Tri‐cyclic Hetero‐Aromatic Congeners via−H bond Functionalization

    Article • Asian Journal of Organic Chemistry, June 2021, Wiley

    Prof. Sandeep Chaudhary

  23. Organic Antifungal Drugs and Targets of Their Action

    Article • Current Topics in Medicinal Chemistry, March 2021, Bentham Science Publishers

    Prof. Sandeep Chaudhary

  24. A Novel Approach Towards Green Synthesis of Nanodiamonds as Biocompatible Agents

    Article • Journal of Nano- and Electronic Physics, January 2021, Sumy State University

    Prof. Sandeep Chaudhary

  25. Microwave-Irradiated Synthesis of Imidazo[1,2-a]pyridine Class of Bio-heterocycles: Green Avenues and Sustainable Developments

    Article • January 2021, Springer Science + Business Media

    Prof. Sandeep Chaudhary

  26. Oxidative cross-dehydrogenative coupling (CDC) via C(sp2)–H bond functionalization: tert-butyl peroxybenzoate (TBPB)-promoted regioselective direct C-3 acylation/benzoylation of 2H-indazoles with aldehydes/benzyl alcohol...

    Article • RSC Advances, January 2021, Royal Society of Chemistry

    Prof. Sandeep Chaudhary

  27. [2,3‐Bis‐(2‐pyridyl) pyrazine] as an Efficient Organocatalyst for the Direct C (sp 2 ) ‐H Arylation of Unactivated Arenes/Heteroarenes via C−H Bond Activation

    Article • ChemistrySelect, October 2020, Wiley

    Dr. MOHIT K TIWARI, Prof. Sandeep Chaudhary

  28. Metal‐Free, H2O2‐Mediated, Regioselective Direct C‐3 Hydroxylation of Imidazo[1,2‐a]pyridines via C(sp2)‐H Bond Functionalization

    Article • ChemistrySelect, August 2020, Wiley

    Prof. Sandeep Chaudhary

  29. Microwave-assisted modified synthesis of C8-analogues of naturally occurring methylxanthines: Synthesis, biological evaluation and their practical applications

    Article • Fitoterapia, June 2020, Elsevier

    Prof. Sandeep Chaudhary

  30. Organocatalyst in Direct C(sp2)–H Arylation of Unactivated Arenes: [1-(2-Hydroxyethyl)-piperazine]-catalyzed Inter- /Intra-molecular C–H bond activation

    Article • The Journal of Organic Chemistry, May 2020, American Chemical Society (ACS)

    Dr. MOHIT K TIWARI, Prof. Sandeep Chaudhary

  31. Advanced Properties and Applications of AIEgens-Inspired Smart Materials

    Article • Industrial & Engineering Chemistry Research, May 2020, American Chemical Society (ACS)

    Prof. Sandeep Chaudhary

  32. Design, Synthesis, Structure‐Activity Relationship and Docking Studies of Novel Functionalized Arylvinyl‐1,2,4‐Trioxanes as Potent Antiplasmodial as well as Anticancer Agents

    Article • ChemMedChem, May 2020, Wiley

    Dr. MOHIT K TIWARI, Prof. Sandeep Chaudhary

  33. Computational Modeling on Aquaporin-3 as Skin Cancer Target: A Virtual Screening Study

    Article • Frontiers in Chemistry, April 2020, Frontiers

    Dr. Dharmendra Kumar Yadav, Prof. Sandeep Chaudhary

  34. Reduction‐Triggered Doxorubicin Delivery by Self‐Assembled Nanospheres of Lipoylated Caffeine

    Article • ChemMedChem, April 2020, Wiley

    Prof. Sandeep Chaudhary

  35. Synthesis, Bioevaluation, Structure-Activity Relationship and Docking Studies of Natural Product Inspired (Z)-3-benzylideneisobenzofuran-1(3H)-ones as Highly Potent antioxidants and Antiplatelet agents

    Article • Scientific Reports, February 2020, Springer Science + Business Media

    Dr. MOHIT K TIWARI, Dr. Dharmendra Kumar Yadav, Prof. Sandeep Chaudhary

  36. AIEgen‐Based Fluorescent Nanomaterials for Bacterial Detection and its Inhibition

    Article • ChemistrySelect, January 2020, Wiley

    Prof. Sandeep Chaudhary

  37. Artemisinin‐derived antimalarial endoperoxides from bench‐side to bed‐side: Chronological advancements and future challenges

    Article • Medicinal Research Reviews, January 2020, Wiley

    Prof. Sandeep Chaudhary, Dr. MOHIT K TIWARI

  38. Bu4NI-catalyzed, oxidative C(sp2)–C(sp3) cross dehydrogenative coupling for the regioselective direct C-3 benzylation of 2H-indazoles

    Article • Organic & Biomolecular Chemistry, January 2020, Royal Society of Chemistry

    Prof. Sandeep Chaudhary

  39. Weak Bases‐Mediated Modified Favorskii Reaction‐Type Direct Alkynylation/(E)‐Alkenylation

    Article • Asian Journal of Organic Chemistry, November 2019, Wiley

    Dr. MOHIT K TIWARI, Prof. Sandeep Chaudhary

  40. Computational Modeling on Aquaporin-3 as Skin Cancer Target: A Virtual Screening and Molecular Dynamic Simulation Study

    Article • October 2019, MDPI AG

    Prof. Sandeep Chaudhary, Dr. Dharmendra Kumar Yadav

  41. Efficacious Doxorubicin Delivery Using Glutathione‐Responsive Hollow Non‐phospholipid Vesicles Bearing Lipoyl Cholesterols

    Article • ChemMedChem, September 2019, Wiley

    Prof. Sandeep Chaudhary

  42. Recent Developments in Natural Product Inspired Synthetic 1,2,4- Trioxolanes (Ozonides)

    Article • Current Topics in Medicinal Chemistry, July 2019, Bentham Science Publishers

    Dr. Dharmendra Kumar Yadav, Dr. MOHIT K TIWARI, Prof. Sandeep Chaudhary

  43. Molecular Targets for Malarial Chemotherapy: A Review

    Article • Current Topics in Medicinal Chemistry, July 2019, Bentham Science Publishers

    Surendra Kumar, Dr. Dharmendra Kumar Yadav, Prof. Sandeep Chaudhary

  44. Molecular dynamic simulations of oxidized skin lipid bilayer and permeability of reactive oxygen species

    Article • Scientific Reports, March 2019, Springer Science + Business Media

    Prof. Sandeep Chaudhary, Dr. Dharmendra Kumar Yadav

  45. Efficient Antibacterial and Low Cytotoxic Potential of Silver Nanoparticles Produced Instantaneously Using Dimeric Gallate

    Article • ChemistrySelect, December 2018, Wiley

    Prof. Sandeep Chaudhary

  46. Efficacious fungicidal potential of composite derived from nano-aggregates of Cu-Diclofenac complexes and ZnO nanoparticles

    Article • Composites Communications, December 2018, Elsevier

    Prof. Sandeep Chaudhary

  47. Correction to Organocatalytic Modified Guareschi–Thorpe Type Regioselective Synthesis: A Unified Direct Access to 5,6,7,8-Tetrahydroquinolines and Other Alicyclic[b]-Fused Pyridines

    Article • Organic Letters, November 2018, American Chemical Society (ACS)

    Prof. Sandeep Chaudhary

  48. Organocatalytic Modified Guareschi–Thorpe Type Regioselective Synthesis: A Unified Direct Access to 5,6,7,8-Tetrahydroquinolines and Other Alicyclic[b]-Fused Pyridines

    Article • Organic Letters, September 2018, American Chemical Society (ACS)

    Prof. Sandeep Chaudhary

  49. An efficient synthesis and biological evaluation of novel analogues of natural product Cephalandole A: A new class of antimicrobial and antiplatelet agents

    Article • Fitoterapia, September 2018, Elsevier

    Prof. Sandeep Chaudhary

  50. Discovery of Aporphine Analogues as Potential Antiplatelet and Antioxidant Agents: Design, Synthesis, Structure-Activity Relationships, Biological Evaluations, and in silico Molecular Docking Studies

    Article • ChemMedChem, August 2018, Wiley

    Dr. Dharmendra Kumar Yadav, Prof. Sandeep Chaudhary

  51. Inverse docking based screening and identification of protein targets for Cassiarin alkaloids against Plasmodium falciparum

    Article • Saudi Pharmaceutical Journal, May 2018, Elsevier

    Prof. Sandeep Chaudhary

  52. Discovery of C-3 Tethered 2-oxo-benzo[1,4]oxazines as Potent Antioxidants: Bio-Inspired Based Design, Synthesis, Biological Evaluation, Cytotoxic, and in Silico Molecular Docking Studies

    Article • Frontiers in Chemistry, March 2018, Frontiers

    Dr. Dharmendra Kumar Yadav, Prof. Sandeep Chaudhary

  53. Molecular Insights into the Interaction of RONS and Thieno[3,2-c]pyran Analogs with SIRT6/COX-2: A Molecular Dynamics Study

    Article • Scientific Reports, March 2018, Nature

    Dr. Dharmendra Kumar Yadav, Prof. Sandeep Chaudhary

  54. Non-peptide-based new class of platelet aggregation inhibitors: Design, synthesis, bioevaluation, SAR, and in silico studies

    Article • Archiv der Pharmazie, March 2018, Wiley

    Dr. Dharmendra Kumar Yadav, Prof. Sandeep Chaudhary

  55. A Tandem Approach towards Diastereoselective Synthesis of Quinoline C-3 Tethered γ-Lactones

    Article • ChemistrySelect, January 2018, Wiley

    Prof. Sandeep Chaudhary

  56. Ag2O nanoparticle-catalyzed substrate-controlled regioselectivities: direct access to 3-ylidenephthalides and isocoumarins

    Article • RSC Advances, January 2018, Royal Society of Chemistry

    Prof. Sandeep Chaudhary, Dr. MOHIT K TIWARI

  57. Microwave-assisted One-pot Efficient Synthesis of Functionalized 2-Oxo-2-phenylethylidenes-linked 2-Oxobenzo[1,4]oxazines and 2-Oxoquino[1,4]oxalines: Synthetic Applications, Antioxidant Activity, SAR and Cytotoxic Studies

    Article • December 2017, Slovenian Chemical Society

    Dr. Dharmendra Kumar Yadav, Prof. Sandeep Chaudhary

  58. Efficacious cellular codelivery of doxorubicin and EGFP siRNA mediated by the composition of PLGA and PEI protected gold nanoparticles

    Article • Bioorganic & Medicinal Chemistry Letters, September 2017, Elsevier

    Prof. Sandeep Chaudhary

  59. Synthesis, antimicrobial activity, structure-activity relationship and cytotoxic studies of a new series of functionalized (Z)-3-(2-oxo-2-substituted ethylidene)-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-ones

    Article • Bioorganic & Medicinal Chemistry Letters, September 2017, Elsevier

    Prof. Sandeep Chaudhary

  60. “On water” ultrasound-assisted one pot efficient synthesis of functionalized 2-oxo-benzo[1,4]oxazines: First application to the synthesis of anticancer indole alkaloid, Cephalandole A

    Article • Tetrahedron Letters, May 2017, Elsevier

    Prof. Sandeep Chaudhary

  61. Influence of ceramic waste on the fresh properties and compressive strength of concrete

    Article • European Journal of Environmental and Civil engineering, January 2017, Taylor & Francis

    Prof. Sandeep Chaudhary

  62. Synthesis of arylated and aminated naphthalenes and their synthetic applications for aza-heterocycles

    Article • Tetrahedron, October 2016, Elsevier

    Prof. Sandeep Chaudhary

  63. New orally active diphenylmethyl-based ester analogues of dihydroartemisinin: Synthesis and antimalarial assessment against multidrug-resistant Plasmodium yoelii nigeriensis in mice

    Article • Bioorganic & Medicinal Chemistry Letters, March 2016, Elsevier

    Prof. Sandeep Chaudhary, Dr. MOHIT K TIWARI

  64. In(OTf)3catalysed an expeditious synthesis of β-carboline–imidazo[1,2-a]pyridine and imidazo[1,2-a]pyrazine conjugates

    Article • RSC Advances, January 2016, Royal Society of Chemistry

    Prof. Sandeep Chaudhary

  65. Synthesis and antimalarial activity of novel bicyclic and tricyclic aza-peroxides

    Article • RSC Advances, January 2016, Royal Society of Chemistry

    Prof. Sandeep Chaudhary, Dr. MOHIT K TIWARI

  66. Stable Tricyclic Antitubercular Ozonides Derived from Artemisinin

    Article • Organic Letters, October 2015, American Chemical Society (ACS)

    Prof. Sandeep Chaudhary

  67. Base mediated regioselective synthesis of highly functionalized conjugated enones

    Article • Tetrahedron Letters, September 2015, Elsevier

    Prof. Sandeep Chaudhary

  68. Streamlined Catalytic Asymmetric Synthesis of Atorvastatin

    Article • Chemistry - A European Journal, February 2013, Wiley

    Prof. Sandeep Chaudhary

  69. Linker-Based Hemisuccinate Derivatives of Artemisinin: Synthesis and Antimalarial Assessment against Multidrug-Resistant Plasmodium yoelii nigeriensis in Mice

    Article • Journal of Medicinal Chemistry, January 2012, American Chemical Society (ACS)

    Prof. Sandeep Chaudhary

  70. New aporphinoid 5-HT2A and α1A antagonists via structural manipulations of nantenine

    Article • Bioorganic & Medicinal Chemistry, October 2011, Elsevier

    Prof. Sandeep Chaudhary

  71. A probabilistic capacity spectrum strategy for the reliability analysis of bridge pile shafts considering soil structure interaction

    Article • Latin American Journal of Solids and Structures, September 2011, FapUNIFESP (SciELO)

    Prof. Sandeep Chaudhary

  72. Cytotoxicity of aporphines in human colon cancer cell lines HCT-116 and Caco-2: An SAR study

    Article • Bioorganic & Medicinal Chemistry Letters, August 2011, Elsevier

    Prof. Sandeep Chaudhary

  73. Synthesis of C-homoaporphines via microwave-assisted direct arylation

    Article • Tetrahedron, January 2011, Elsevier

    Prof. Sandeep Chaudhary

  74. Affinity of aporphines for the human 5-HT2A receptor: Insights from homology modeling and molecular docking studies

    Article • Bioorganic & Medicinal Chemistry, August 2010, Elsevier

    Prof. Sandeep Chaudhary

  75. Synthetic studies and pharmacological evaluations on the MDMA (‘Ecstasy’) antagonist nantenine

    Article • Bioorganic & Medicinal Chemistry Letters, January 2010, Elsevier

    Prof. Sandeep Chaudhary

  76. (±)-Nantenine analogs as antagonists at human 5-HT2A receptors: C1 and flexible congeners

    Article • Bioorganic & Medicinal Chemistry Letters, May 2009, Elsevier

    Prof. Sandeep Chaudhary

  77. Microwave-assisted direct biaryl coupling: first application to the synthesis of aporphines

    Article • Tetrahedron Letters, May 2009, Elsevier

    Prof. Sandeep Chaudhary

  78. New Drimane Sesquiterpenoids from Tidestromia Oblongifolia

    Article • Natural Product Communications, November 2008, SAGE Publications

    Prof. Sandeep Chaudhary

  79. Orally active esters of dihydroartemisinin: Synthesis and antimalarial activity against multidrug-resistant Plasmodium yoelii in mice

    Article • Bioorganic & Medicinal Chemistry Letters, February 2008, Elsevier

    Prof. Sandeep Chaudhary

  80. Conversion of Antimalarial Drug Artemisinin to a New Series of Tricyclic 1,2,4-Trioxanes1

    Article • Organic Letters, October 2007, American Chemical Society (ACS)

    Prof. Sandeep Chaudhary

  81. New Orally Active Derivatives of Artemisinin with High Efficacy against Multidrug-Resistant Malaria in Mice1

    Article • Journal of Medicinal Chemistry, November 2006, American Chemical Society (ACS)

    Prof. Sandeep Chaudhary

  82. Poster Session II Abstracts

    Article • Medicinal Chemistry Research, April 2006, Springer Science + Business Media

    Prof. Sandeep Chaudhary