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  1. Synthesis and Biological Evaluation of Amino Acid and Peptide Conjugates of 5-Bromovaleric Acid

    Article • Medicinal Chemistry, December 2024, Bentham Science Publishers

    Dr. Rajesh K. Singh, Nitin Verma

  2. A Recent Advance on Phytochemicals, Nutraceutical and Pharmacological Activities of Buckwheat

    Article • Combinatorial Chemistry & High Throughput Screening, November 2024, Bentham Science Publishers

    Shweta Sharma, Dr. Rajesh K. Singh

  3. Natural flavonoid pectolinarin computationally targeted as a promising drug candidate against SARS-CoV-2

    Article • Current Research in Structural Biology, January 2024, Elsevier

    Dr. Rajesh K. Singh

  4. Synthesis, Drug-Likeness Evaluation of Some Heterocyclic Moieties Fused Indole Derivatives as Potential Antioxidants

    Article • Combinatorial Chemistry & High Throughput Screening, September 2023, Bentham Science Publishers

    Dr. Rajesh K. Singh

  5. Synthesis, Molecular Docking and ADME Prediction of 1H-indole/5- substituted Indole Derivatives as Potential Antioxidant and Anti- Inflammatory Agents

    Article • Medicinal Chemistry, February 2023, Bentham Science Publishers

    Dr. Rajesh K. Singh

  6. Pyrazoline Scaffold: Hit Identification to Lead Synthesis and Biological Evaluation As Antidiabetic Agents

    Article • Future Medicinal Chemistry, January 2023, Taylor & Francis

    Dr. Shakir Ali, Dr. Rajesh K. Singh

  7. Synthesis, Characterization and ADME Prediction Study of Heterocyclic Moieties-linked Indole Derivatives as Potential Antimicrobial Agents

    Article • Letters in Drug Design & Discovery, January 2023, Elsevier

    Dr. Rajesh K. Singh

  8. Morpholine: Pharmacophore Modulating Pharmacokinetic Properties of Anticancer Leads

    Article • September 2022, Bentham Science Publishers

    Dr. Rajesh K. Singh

  9. Progress in Nitrogen and Sulphur-based Heterocyclic Compounds for their Anticancer Activity

    Article • September 2022, Bentham Science Publishers

    Dr. Rajesh K. Singh

  10. Understanding Promising Anticancer Targets for Heterocyclic Leads: An Introduction

    Article • September 2022, Bentham Science Publishers

    Dr. Rajesh K. Singh, Shweta Sharma

  11. Key Heterocyclic Cores for Smart Anticancer Drug–Design Part II

    Article • September 2022, Bentham Science Publishers

    Dr. Rajesh K. Singh

  12. Progress in Nitrogen and Oxygen-based Heterocyclic Compounds for their Anticancer Activity: An Updates (2017-2020)

    Article • July 2022, Bentham Science Publishers

    Dr. Rajesh K. Singh, Sakshi Choudhary

  13. Recent Advances in Synthesis and the Anticancer Activity of Benzothiazole Hybrids as Anticancer Agents

    Article • July 2022, Bentham Science Publishers

    Dr. Rajesh K. Singh

  14. Key Heterocyclic Cores for Smart Anticancer Drug–Design Part I

    Article • July 2022, Bentham Science Publishers

    Dr. Rajesh K. Singh

  15. Target-based anticancer indole derivatives and insight into structure‒activity relationship: A mechanistic review update (2018–2021)

    Article • Acta Pharmaceutica Sinica B, July 2022, Elsevier

    Dr. Rajesh K. Singh

  16. Ethnobotany, Pharmacological Activities and Bioavailability Studies on “King of Bitters” (Kalmegh): A Review (2010-2020)

    Article • Combinatorial Chemistry & High Throughput Screening, April 2022, Bentham Science Publishers

    Dr. Rajesh K. Singh

  17. Mayapuri Radiological Catastrophe: Good Practices and the Lessons Learnt

    Article • Current Radiopharmaceuticals, March 2022, Bentham Science Publishers

    Dr. Rajesh K. Singh

  18. Advances in Ethnobotany, Synthetic Phytochemistry and Pharmacology of Endangered Herb Picrorhiza kurroa (Kutki): A Comprehensive Review (2010-2020)

    Article • Mini-Reviews in Medicinal Chemistry, November 2021, Bentham Science Publishers

    Dr. Rajesh K. Singh

  19. Pharmacological activities and molecular mechanisms of pure and crude extract of Andrographis paniculata: An update

    Article • Phytomedicine Plus, November 2021, Elsevier

    Dr. Rajesh K. Singh

  20. Drug Repurposing Using Similarity-based Target Prediction, Docking Studies and Scaffold Hopping of Lefamulin

    Article • Letters in Drug Design & Discovery, September 2021, Bentham Science Publishers

    Shweta Sharma, Dr. Rajesh K. Singh

  21. Therapeutic Journey of Andrographis paniculata (Burm.f.) Nees from Natural to Synthetic and Nanoformulations

    Article • Mini-Reviews in Medicinal Chemistry, March 2021, Bentham Science Publishers

    Dr. Rajesh K. Singh

  22. Design, Synthesis and Studies on Novel Polymeric Prodrugs of Erlotinib for Colon Drug Delivery

    Article • Anti-Cancer Agents in Medicinal Chemistry, February 2021, Bentham Science Publishers

    Dr. Rajesh K. Singh

  23. Method validation for the simultaneous estimation of three-bioactive components in combined extracts of three hepatoprotective plants using RP-HPLC method

    Article • Journal of Applied Biology & Biotechnology, July 2020, Journal of Applied Pharmaceutical Science

    Dr. Rajesh K. Singh

  24. Multicomponent Catalytic Synthesis of 1,5-Benzodiazepines: An Update

    Article • Mini-Reviews in Organic Chemistry, June 2020, Bentham Science Publishers

    Sadhna SHARDA, Dr. Rajesh K. Singh

  25. Current Progress in the Multicomponent Catalytic Synthesis of Amidoalkyl- Naphthols: An Update

    Article • Current Organic Chemistry, May 2020, Bentham Science Publishers

    Ashima Dhiman, Dr. Rajesh K. Singh

  26. Synthesis, Anticancer and Antibacterial Studies of Benzylidene Bearing 5-substituted and 3,5-disubstituted-2,4-Thiazolidinedione Derivatives

    Article • Medicinal Chemistry, May 2020, Bentham Science Publishers

    Dr. Rajesh K. Singh

  27. Clinical Benefits of Switching from Original Infliximab to its Biosimilar (CT-P13) as a Potential TNF-α Inhibitor

    Article • Journal of Exploratory Research in Pharmacology, April 2020, Xia & He Publishing

    Dr. Rajesh K. Singh

  28. An Insight into the Synthesis and SAR of 2,4-Thiazolidinediones (2,4-TZD) as Multifunctional Scaffold: A Review

    Article • Mini-Reviews in Medicinal Chemistry, April 2020, Bentham Science Publishers

    Dr. Rajesh K. Singh

  29. Morpholine as ubiquitous pharmacophore in medicinal chemistry: Deep insight into the structure-activity relationship (SAR)

    Article • Bioorganic Chemistry, March 2020, Elsevier

    Dr. Rajesh K. Singh

  30. Medicinal chemistry of indole derivatives: Current to future therapeutic prospectives

    Article • Bioorganic Chemistry, August 2019, Elsevier

    Dr. Rajesh K. Singh

  31. Recent Advances in Vaccine Development for the Treatment of Emerging Infectious Diseases

    Article • Indian Journal of Pharmaceutical Education and Research, July 2019, EManuscript Services

    Dr. Rajesh K. Singh

  32. Novel ketoprofen–antioxidants mutual codrugs as safer nonsteroidal anti‐inflammatory drugs: Synthesis, kinetic and pharmacological evaluation

    Article • Archiv der Pharmazie, June 2019, Wiley

    Dr. Rajesh K. Singh

  33. Recent Advances in the Development of Polymeric Nanocarrier Formulations for the Treatment of Colon Cancer

    Article • Drug Delivery Letters, February 2019, Bentham Science Publishers

    Dr. Rajesh K. Singh

  34. Intricacies in the Approval of Radiopharmaceuticals – Regulatory Perspectives and the Way Forward

    Article • Current Science, January 2019, Current Science Association

    Dr. Rajesh K. Singh, Professor Ashish Baldi

  35. Drafting of comprehensive harmonized regulatory guideline for storage and disposal of radiopharmaceuticals

    Article • Journal of Drug Delivery and Therapeutics, December 2018, Society of Pharmaceutical Tecnocrats

    Dr. Rajesh K. Singh

  36. An atom-economic efficient synthesis of 1-amidoalkyl-2-naphthols mediated By hexachlorocyclotriphosphazene (HCCP) as a novel catalyst

    Article • Letters in Organic Chemistry, December 2018, Bentham Science Publishers

    Dr. Rajesh K. Singh

  37. Drug targets for resistant malaria: Historic to future perspectives

    Article • Biomedicine & Pharmacotherapy, August 2018, Elsevier

    Dr. Rajesh K. Singh

  38. Prodrugs of Non-steroidal Anti-inflammatory Drugs (NSAIDs): A Long March Towards Synthesis of Safer NSAIDs

    Article • Mini-Reviews in Medicinal Chemistry, July 2018, Bentham Science Publishers

    Dr. Rajesh K. Singh

  39. Recent advances in colony stimulating factor-1 receptor/c-FMS as an emerging target for various therapeutic implications

    Article • Biomedicine & Pharmacotherapy, July 2018, Elsevier

    Dr. Rajesh K. Singh

  40. Therapeutic journery of nitrogen mustard as alkylating anticancer agents: Historic to future perspectives

    Article • European Journal of Medicinal Chemistry, May 2018, Elsevier

    Dr. Rajesh K. Singh

  41. Environment-friendly green chemistry approaches for an efficient synthesis of 1-amidoalkyl-2-naphthols catalyzed by tannic acid

    Article • Arabian Journal of Chemistry, January 2018, Elsevier

    Dr. Rajesh K. Singh

  42. Hexachlorocyclotriphosphazene Catalyzed One-Pot Multicomponent Synthesis of 2,3-Dihydro-1H-1,5-benzodiazepines

    Article • Asian Journal of Organic & Medicinal Chemistry, January 2018, Asian Journal of Chemistry

    Dr. Rajesh K. Singh

  43. Synthesis and Evaluation of Prodrugs of Ketoprofen with Antioxidants as Gastroprotective NSAIDs

    Article • Asian Journal of Chemistry, January 2018, Asian Journal of Chemistry

    Dr. Rajesh K. Singh

  44. Synthetic Methodologies and Pharmacological Significance of 2-Aminobenzophenones as Versatile Building Block

    Article • Asian Journal of Organic & Medicinal Chemistry, January 2018, Asian Journal of Chemistry

    Dr. Rajesh K. Singh

  45. Synthesis and in vitro degradation studies of substituted poly(organophosphazenes) for drug delivery applications

    Article • Journal of Drug Delivery Science and Technology, April 2017, Elsevier

    Dr. Rajesh K. Singh

  46. Design, synthesis, chemical and biological evaluation of brain targeted alkylating agent using reversible redox prodrug approach

    Article • Arabian Journal of Chemistry, March 2017, Elsevier

    Dr. Rajesh K. Singh

  47. Design, synthesis and in vitro cytotoxicity study of benzodiazepine-mustard conjugates as potential brain anticancer agents

    Article • Journal of Saudi Chemical Society, January 2017, Elsevier

    Dr. Rajesh K. Singh

  48. Therapeutic role of nitric oxide as emerging molecule

    Article • Biomedicine & Pharmacotherapy, January 2017, Elsevier

    Dr. Rajesh K. Singh

  49. Synthesis, physicochemical and biological evaluation of 2-amino-5-chlorobenzophenone derivatives as potent skeletal muscle relaxants

    Article • Arabian Journal of Chemistry, May 2015, Elsevier

    Dr. Rajesh K. Singh

  50. Synthesis, physicochemical and kinetic studies of redox derivative of bis(2-chloroethylamine) as alkylating cytotoxic agent for brain delivery

    Article • Arabian Journal of Chemistry, May 2015, Elsevier

    Dr. Rajesh K. Singh

  51. Synthesis and Evaluation of Substituted Poly(organophosphazenes) as a Novel Nanocarrier System for Combined Antimalarial Therapy of Primaquine and Dihydroartemisinin

    Article • Pharmaceutical Research, March 2015, Springer Science + Business Media

    Dr. Rajesh K. Singh

  52. Recent advances in novel heterocyclic scaffolds for the treatment of drug-resistant malaria

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, March 2015, Taylor & Francis

    Dr. Rajesh K. Singh

  53. Design, synthesis and evaluation of antimalarial potential of polyphosphazene linked combination therapy of primaquine and dihydroartemisinin

    Article • European Journal of Pharmaceutical Sciences, January 2015, Elsevier

    Dr. Rajesh K. Singh

  54. Morphoanatomic, physicochemical, and phytochemical standardization with HPTLC fingerprinting of aerial parts of Aerva lanata (Linn) Juss ex Schult

    Article • Journal of Traditional Chinese Medical Sciences, January 2015, Elsevier

    Dr. Rajesh K. Singh

  55. Microwave-Assisted Synthesis, in silico ADME Prediction and Antibacterial Study of 2-(Substituted acetamido)-5-Nitrobenzophenone Derivatives

    Article • Asian Journal of Chemistry, January 2015, Asian Journal of Chemistry

    Dr. Rajesh K. Singh

  56. Hybrid pharmacophore-based drug design, synthesis, and antiproliferative activity of 1,4-dihydropyridines-linked alkylating anticancer agents

    Article • Medicinal Chemistry Research, August 2014, Springer Science + Business Media

    Dr. Rajesh K. Singh

  57. Sulfanilic acid: a versatile and efficient catalyst among various organoacids screened for the synthesis of 1-amidoalkyl-2-naphthols under solvent-free condition

    Article • Research on Chemical Intermediates, January 2014, Springer Science + Business Media

    Dr. Rajesh K. Singh

  58. Highly Efficient Zinc Oxide Nanoparticles Catalyzed Green Synthesis of 1,5-Benzodiazepines under Solvent-Free Path

    Article • Asian Journal of Chemistry, January 2014, Asian Journal of Chemistry

    Dr. Rajesh K. Singh

  59. Investigation of Various Organocatalysts for Improved and Efficient One Pot Synthesis of 2,3-Dihydro-1H-1,5-benzodiazepines Under Solvent-Free Condition

    Article • Asian Journal of Chemistry, January 2014, Asian Journal of Chemistry

    Dr. Rajesh K. Singh

  60. Multicomponent One-pot Green Synthesis of 1-Amidoalkyl-2-naphthols Promoted by p-Nitrobenzoic Acid Under Solvent-free Condition

    Article • Asian Journal of Chemistry, January 2014, Asian Journal of Chemistry

    Dr. Rajesh K. Singh

  61. Synthesis and Antimicrobial Evaluation of 2-Aminobenzophenone Linked 1,4-Dihydropyridine Derivatives

    Article • Asian Journal of Chemistry, January 2014, Asian Journal of Chemistry

    Dr. Rajesh K. Singh

  62. Reversible redox system-based drug design, synthesis, and evaluation for targeting nitrogen mustard across brain

    Article • Medicinal Chemistry Research, October 2013, Springer Science + Business Media

    Dr. Rajesh K. Singh

  63. Investigation of Various Green Chemistry Approaches for the Efficient Synthesis of Dialkyl-1, 4-dihydro-4-(substituted phenyl)-2, 6-dimethylpyridine-3, 5-dicarboxylate

    Article • Chemical Science Transactions, May 2013, Chemical Science Transactions

    Dr. Rajesh K. Singh

  64. Design, synthesis and evaluation of aminobenzophenone derivatives containing nitrogen mustard moiety as potential central nervous system antitumor agent

    Article • Medicinal Chemistry Research, March 2013, Springer Science + Business Media

    Dr. Rajesh K. Singh

  65. Synthesis in vitro/in vivo evaluation and in silico physicochemical study of prodrug approach for brain targeting of alkylating agent

    Article • Medicinal Chemistry Research, February 2013, Springer Science + Business Media

    Dr. Rajesh K. Singh

  66. Rapid and Efficient Synthesis of 2,3-Dihydro-1H-1,5-Benzodiazepines Catalyzed by Chloroacetic Acid Screened among Various Aliphatic Acids

    Article • Chemical Science Transactions, November 2012, Chemical Science Transactions

    Dr. Rajesh K. Singh

  67. Efficient p-Amino Benzoic Acid Catalyzed Eco-friendly Synthesis of 1,5-benzodiazepines among Various Amino Acids under Solvent Free Conditions

    Article • Current Research in Chemistry, June 2012, Science Alert

    Dr. Rajesh K. Singh