All Stories

  1. Identification, isolation, and synthesis of seven novel impurities of anti-diabetic drug Repaglinide
  2. Copper(ii)-catalyzed Chan–Lam cross-coupling: chemoselective N-arylation of aminophenols
  3. Ruthenium-catalyzed site-selective C–H arylation of 2-pyridones and 1-isoquinolinones
  4. ChemInform Abstract: Copper-Catalyzed N-Arylation of Tautomerizable Heterocycles with Boronic Acids and its Application to Synthesis of Oxygenated Carbazoles.
  5. Palladium/Silver Synergistic Catalysis in Direct Aerobic Carbonylation of C(sp2)−H Bonds Using DMF as a Carbon Source: Synthesis of Pyrido-Fused Quinazolinones and Phenanthridinones
  6. Copper-Catalyzed CNH2Arylation of 2-Aminobenzimidazoles and Related C-Amino-NH-azoles
  7. ChemInform Abstract: Site-Selective Intermolecular Oxidative C-3 Alkenylation of 7-Azaindoles at Room Temperature.
  8. Metal-Free Aminooxygenation of Alkynes: Efficient Synthesis of 3-Aroylimidazo[1,2-a]-N-Heterocycles
  9. Site-Selective Intermolecular Oxidative C-3 Alkenylation of 7-Azaindoles at Room Temperature
  10. Copper-CatalyzedN-Arylation of Tautomerizable Heterocycles with Boronic Acids and Its Application to Synthesis of Oxygenated Carbazoles
  11. ChemInform Abstract: Palladium-Catalyzed Arylation of 2H-Chromene: A New Entry to Pyrano[2,3-c]carbazoles.
  12. ChemInform Abstract: Copper-Catalyzed Inter- and Intramolecular C-N Bond Formation: Synthesis of Benzimidazole-Fused Heterocycles.
  13. ChemInform Abstract: Copper-Catalyzed Oxidative C-H Amination: Synthesis of Imidazo[1,2-a]-N-Heterocycles from N-Heteroaryl Enaminones.
  14. Copper-Catalyzed Inter- and Intramolecular C–N Bond Formation: Synthesis of Benzimidazole-Fused Heterocycles
  15. ChemInform Abstract: Divergent Synthesis of 4,6-Diarylated Pyridin-2(1H)-ones from Chalcones: Novel Access to 2,4,6-Triaryl Pyridines.
  16. ChemInform Abstract: Sulfuric Acid Immobilized on Silica Gel (H2SO4-SiO2) as an Eco-Friendly Catalyst for Transamidation.
  17. ChemInform Abstract: Cu-Catalyzed Arylation of the Amino Group in the Indazole Ring: Regioselective Synthesis of Pyrazolo-Carbazoles.
  18. Copper-Catalyzed Oxidative C−H Amination: Synthesis of Imidazo[1,2-a]-N-Heterocycles from N-Heteroaryl Enaminones
  19. ChemInform Abstract: Hypervalent Iodine(III) Catalyzed Oxidative C-N Bond Formation in Water: Synthesis of Benzimidazole-Fused Heterocycles.
  20. Sulphuric acid immobilized on silica gel (H2SO4–SiO2) as an eco-friendly catalyst for transamidation
  21. Cu-catalyzed arylation of the amino group in the indazole ring: regioselective synthesis of pyrazolo-carbazoles
  22. Divergent synthesis of 4,6-diarylated pyridin-2(1H)-ones from chalcones: novel access to 2,4,6-triaryl pyridines
  23. Palladium-catalyzed arylation of 2H-chromene: a new entry to pyrano[2,3-c]carbazoles
  24. ChemInform Abstract: C-N Bond Formation via Cu-Catalyzed Cross-Coupling with Boronic Acids Leading to Methyl Carbazole-3-carboxylate: Synthesis of Carbazole Alkaloids.
  25. ChemInform Abstract: Direct C‐2 Arylation of 7‐Azaindoles: Chemoselective Access to Multiarylated Derivatives.
  26. C–N bond formation via Cu-catalyzed cross-coupling with boronic acids leading to methyl carbazole-3-carboxylate: synthesis of carbazole alkaloids
  27. Hypervalent iodine(iii) catalyzed oxidative C–N bond formation in water: synthesis of benzimidazole-fused heterocycles
  28. Copper-catalyzed sequential N-arylation of C-amino-NH-azoles
  29. Direct C-2 Arylation of 7-Azaindoles: Chemoselective Access to Multiarylated Derivatives
  30. ChemInform Abstract: Synthesis and Characterization of 5‐(6‐Substituted phenyl‐2H‐chromen‐3‐yl) Oxazole Derivatives.
  31. Base and ligand free copper-catalyzed N-arylation of 2-amino-N-heterocycles with boronic acids in air
  32. Synthesis and Characterisation of 5-(6-substituted phenyl -2H-chromen-3- yl) Oxazole Derivatives
  33. ChemInform Abstract: Synthesis and Characterization of 9‐Methyl‐2‐morpholin‐4‐yl‐8‐substituted Phenyl‐1H‐purine Derivatives Using Polyphosphoric Acid (PPA) as an Efficient Catalyst.
  34. Synthesis and characterization of 9-methyl-2-morpholin-4-yl-8-substituted phenyl-1H-purine derivatives using polyphosphoric acid (PPA) as an efficient catalyst
  35. ChemInform Abstract: Direct Synthesis of N‐Aryl Derivatives of Quinazolin‐4(3H)‐ones Employing Arylboronic Acids in the Presence of Cu(OAc)2.
  36. ChemInform Abstract: Dithiocarbamate‐ and DBU‐Promoted Amide Bond Formation under Microwave Condition.
  37. Direct Synthesis of N-Aryl Derivatives of Quinazolin-4(3H)-ones Employing Arylboronic Acids in the Presence of Cu(OAc)2
  38. Dithiocarbamate and DBU-promoted amide bond formation under microwave condition
  39. An efficient synthesis of varenicline
  40. Total Synthesis of (±)-Petasitolone and (±)-Fukinone
  41. Total Synthesis of (±)-Petasitolone and (±)-Fukinone
  42. Studies toward a Total Synthesis of Rhizoxin D: Stereoselective Preparation of the C11-C19 Fragment¹
  43. Stereoselective Preparation of C1-C10 and C11-O14 Fragments of Narbonolide: Exploiting the Versatility of Thiazolidinethione Chiral Auxiliary¹
  44. ChemInform Abstract: A New Route to Eremophilanes: Synthesis of (.+‐.)‐Eremophilenolide (VII), (.+‐.)‐Eremophiledinone (VI), and (.+‐.)‐Deoxyeremopetasidione (X).
  45. A new route to eremophilanes: synthesis of (±)-eremophilenolide, (±)-eremophiledinone, and (±)-deoxyeremopetasidione
  46. A Cross-Metathesis Approach to the Synthesis of Key Precursor of the Macrolide Core of Rhizoxin D
  47. ChemInform Abstract: Dithiocarbamate‐ and CuO‐Promoted One‐Pot Synthesis of 2‐(N‐Substituted)‐aminobenzimidazoles and Related Heterocycles.
  48. Studies towards the total synthesis of narbonolide: stereoselective preparation of the C1–C10 fragment
  49. A Stereoselective Synthesis of the Macrolide Core of Migrastatin
  50. Dithiocarbamate and CuO promoted one-pot synthesis of 2-(N-substituted)-aminobenzimidazoles and related heterocycles
  51. ChemInform Abstract: Studies Toward the Total Synthesis of (—)‐Dictyostatin (I): Stereoselective Preparation of the C1—C10 Fragment.
  52. Studies toward the Total Synthesis of (-)-Dictyostatin: Stereoselective Preparation­ of the C1-C10 Fragment
  53. A cross metathesis approach to the synthesis of the C11–C23 fragment of (−)-16-normethyldictyostatin
  54. A convergent synthesis of the macrolide core of migrastatin
  55. Direct Observation of ESR Spectra of Bicyclic Nine-Membered Enediynes at Ambient Temperature
  56. Spin Trapping of 13C‐Labeled p‐Benzynes Generated by Masamune–Bergman Cyclization of Bicyclic Nine‐Membered Enediynes
  57. Spin Trapping of 13C‐Labeled p‐Benzynes Generated by Masamune–Bergman Cyclization of Bicyclic Nine‐Membered Enediynes
  58. Asymmetric Synthesis of Cycloalkenyl and Alkenyloxiranes from Allylic Sulfoximines and Aldehydes and Application to Solid‐Phase Synthesis.
  59. Asymmetric Synthesis of Cycloalkenyl and Alkenyloxiranes From Allylic Sulfoximines and Aldehydes and Application to Solid-Phase Synthesis
  60. Asymmetric Synthesis of Protected β‐Substituted and β,β‐Disubstituted β‐Amino Acids Bearing Branched Hydroxyalkyl Side Chains and of Protected 1,3‐Amino Alcohols with Three Contiguous Stereogenic Centers from Allylic Sulfoximines and Aldehydes
  61. Synthesis of 13C‐Labeled, Bicyclic Mimetics of Natural Enediynes.
  62. Synthesis of 13C-labelled, bicyclic mimetics of natural enediynes
  63. ChemInform Abstract: Diastereoselective Additions of Ethynyl Grignard Reagent to Erythrulose Derivatives.
  64. Diastereoselective Additions of Ethynyl Grignard Reagent to Erythrulose Derivatives
  65. N-Methylsulfonimidoyl-Substituted (2-Alkenyl)titanium Complexes: Application to the Synthesis of β- and δ-Sulfonimidoyl-Substituted Chiral Homoallylic Alcohols, X-ray Crystal Structure Analysis, and Fluxional Behavior
  66. ChemInform Abstract: Diastereoselective Amination of Vinylic Sulfoximines: Application to the Asymmetric Synthesis of Functionalized β‐Substituted and β,β‐Disubstituted β‐Amino Acids, and of γ‐Amino Alcohols.
  67. ChemInform Abstract: Photoinduced Electron Transfer (PET) Promoted Oxidative Activation of 1‐(N‐Benzyl‐N‐methylglycyl)‐(S)‐prolinol: Development of Novel Strategies Towards Enantioselective Syntheses of α‐Amino Acids, Their N‐Methyl Derivatives, and α‐...
  68. Diastereoselective amination of vinylic sulfoximines: application to the asymmetric synthesis of functionalized β-substituted and β,β-disubstituted β-amino acids, and of γ-amino alcohols
  69. Photoinduced Electron Transfer (PET) Promoted Oxidative Activation of 1-(N-Benzyl-N-methylglycyl)-(S)-prolinol: Development of Novel Strategies Towards Enantioselective Syntheses of α-Amino Acids, TheirN-Methyl Derivatives and α-Hydroxy Acids Employing...
  70. ChemInform Abstract: Synthesis and Utilization of Chiral 3‐N‐Benzyl‐N‐methylaminoperhydropyrrolo[2,1‐c][1,4]oxazin‐4‐one as a Novel Precursor for the Enantioselective Synthesis of α‐Amino Acids and Their N‐Methyl Derivatives.
  71. Synthesis and utilisation of chiral 3-hydroxy perhydropyrrolo [2,1-c] [1,4] oxazin-4-one as a novel precursor for the enantioselective synthesis of α-hydroxy carboxylic acids
  72. Enantioselective α-alkylation of piperidine via chiral perhydropyrido [2,1-b] [1,3,4]-oxadiazinone: An easy route for the synthesis of both enantiomers of coniine
  73. Synthesis and utilization of a novel glycine derived chiral precursor, based on a recyclable L-Prolinol auxiliary, for the enantioselective preparation of α-amino acids and their N-methyl derivatives