All Stories

  1. D-galactose-conjugated thiazole-thiourea hybrids: Synthesis, in vitro inhibition against DPP-4 and PTP1B, their molecular docking, molecular dynamics simulations and DFT calculations
  2. Maltose-Conjugated Thiosemicarbazones from Substituted Benzaldehydes: Synthesis and Inhibitory Activity against Gram-(+) and Gram-(−) Bacteria
  3. Synthesis and Biological Activity for 1,3,4‐Thiadiazole–2‐Iminothiazolidin‐4‐Ones: Antidiabetic and Anti‐Alzheimer Activity
  4. Substituted D‐Galactose‐Conjugated Thiazole‐Thioureas Derivatives as Promising Antidiabetic Agents: Synthesis, In Vitro Inhibition, and Molecular Simulation for α‐Amylase, α‐Glucosidase, Protein Glycation, and Oxidative Stress
  5. d-Glucose-Conjugated Benzo[d]thiazole–thiazolidin-4-one Hybrids: Design and Synthesis as Multitarget Anti-Alzheimer Compounds
  6. D-glucose-conjugated thioureas containing 2-aminopyrimidine as potential multitarget inhibitors for type 2 diabetes mellitus: Synthesis and biological activity study
  7. Sulphonyl thiourea compounds containing pyrimidine as dual inhibitors of I, II, IX, and XII carbonic anhydrases and cancer cell lines: synthesis, characterization and in silico studies
  8. Synthesis, antiproliferative activity, ADMET, molecular docking, molecular dynamics simulation, and DFT study for coumarin-based 1,5-benzothiazepines
  9. Lactose-conjugated 2-iminothiazolidin-4-ones: synthesis, inhibitory activity and molecular simulations as potential inhibitors against enzymes responsible for type 2 diabetes
  10. Sulfonyl thiourea derivatives from 2‐aminodiarylpyrimidines: In vitro and in silico evaluation as potential carbonic anhydrase I, II, IX, and XII inhibitors
  11. Sulfonyl thioureas with a benzo[d]thiazole ring as dual acetylcholinesterase/butyrylcholinesterase and human monoamine oxidase A and B inhibitors: An in vitro and in silico study
  12. Design, synthesis, inhibitory activity, and molecular simulations study for d-glucose-conjugated thioureas containing pyrimidine ring as multitarget inhibitors against α-amylase, α-glucosidase, DDP-4, and PTP1B in Type 2 diabetes mellitus
  13. Synthesis, anticancer activity, and molecular simulation of N-(2,3,4,6-tetra-O-acetyl-β-d-glucopyranosyl)thioureas containing a pyrimidine ring
  14. Substituted isatin-thiosemicarbazones containing d-galactose moiety: Synthesis, antimicrobial inhibition assay and molecular simulation study
  15. Synthesis and Potential Dual Inhibitory Activity Against Acetylcholinesterase and Butyrylcholinesterase of Galactose‐Conjugated Isatin β‐Thiosemicarbazones
  16. Design, synthesis, molecular docking study and molecular dynamics simulation of new coumarin-pyrimidine hybrid compounds having anticancer and antidiabetic activity
  17. Glyco-conjugated thiosemicarbazones of substituted isatin containing D-galactose moiety: Synthesis, bacterial/fungal inhibition assay and molecular docking study
  18. Synthesis and in vitro anticancer activity of 4H-pyrano[2,3-d]pyrimidine−1H-1,2,3-triazole hybrid compounds bearing D-glucose moiety with dual EGFR/HER2 inhibitory activity and induced fit docking study
  19. Synthesis and inhibitory activity against MurA and MurZ enzymes of 4H-pyrano[2,3-d]pyrimidine–1H-1,2,3-triazole hybrid compounds having piperidine and morpholine rings
  20. Thiourea derivatives containing 4-arylthiazoles and d-glucose moiety: design, synthesis, antimicrobial activity evaluation, and molecular docking/dynamics simulations
  21. Synthesis, antimicrobial activity and molecular simulation of thiourea derivatives containing 6-carboalkoxybenzo[d]thiazole andd-glucose moieties
  22. Synthesis, biological and molecular modelling for 1,3,4-thiadiazole sulfonyl thioureas: bacterial and fungal activity
  23. Design, Synthesis, α‐Amylase/α‐Glucosidase Inhibition Assay, Induced Fit Docking Study of New Hybrid Compounds Containing 4H‐Pyrano[2,3‐d]pyrimidine, 1H‐1,2,3‐Triazole and D‐Glucose Components
  24. 1H‐1,2,3‐Triazole−4H‐chromene−D‐glucose hybrid compounds: Synthesis and inhibitory activity against Mycobacterium tuberculosis protein tyrosine phosphatase B
  25. Synthesis, bacterial and fungal inhibition assay, molecular docking study of substituted isatin (N-substituted 1,2,3,4-tetra-O-acetyl-β-glucopyranosyl)thiosemicarbazones
  26. Synthesis, Cytotoxicity, ADMET and Molecular Docking Studies of Some Quinoline-Pyrimidine Hybrid Compounds: 3-(2-Amino-6-arylpyrimidin-4- yl)-4-hydroxy-1-methylquinolin-2(1H)-ones
  27. Synthesis and antiproliferative activity of 1H-1,2,3-triazole-4H-chromene-d-glucose hybrid compounds with dual inhibitory activity against EGFR/VEGFR-2 and molecular docking studies
  28. Synthesis, biological evaluation and induced fit docking simulation study of d-glucose-conjugated 1H-1,2,3-triazoles having 4H-pyrano[2,3-d]pyrimidine ring as potential agents against bacteria and fungi
  29. Synthesis and antiproliferative activity of hybrid thiosemicarbazone derivatives bearing coumarin and d-galactose moieties with EGFR inhibitory activity and molecular docking study
  30. Study on synthesis of some substituted N-propargyl isatins by propargylation reaction of corresponding isatins using potassium carbonate as base under ultrasound- and microwave-assisted conditions
  31. N-(2,3,4,6-tetra-O-acetyl-β-d-glucopyranosyl)thiosemicarbazones of 6-alkoxy-2-oxo-2H-chromene-4-carbaldehydes: synthesis, evaluation of their antibacterial, anti-MRSA, antifungal activity, and docking study
  32. Novel thiazoline–coumarin hybrid compounds containing sugar moieties: synthesis, biological evaluation and molecular docking study as antiproliferative agents
  33. Substituted 4-Formyl-2H-chromen-2-ones: Their Reaction with N-(2,3,4,6-Tetra-Oacetyl- β-D-galactopyranosyl)thiosemicarbazide, Antibacterial and Antifungal Activity of Their Thiosemicarbazone Products
  34. Synthesis of 6- and 7-alkoxy-4-methylcoumarins from corresponding hydroxy coumarins and their conversion into 6- and 7-alkoxy-4-formylcoumarin derivatives
  35. Synthesis of some 1H-1,5-benzodiazepine Series Containing Chromene Ring from α,β-Unsaturated Ketones of 6-Acetyl-5-Hydroxy-4-Methylcoumarin
  36. Synthesis, cytotoxic activity, ADMET and molecular docking study of quinoline-based hybrid compounds of 1,5-benzothiazepines
  37. Efficient click chemistry towards novel 1H-1,2,3-triazole-tethered 4H-chromene−d-glucose conjugates: Design, synthesis and evaluation of in vitro antibacterial, MRSA and antifungal activities
  38. Synthesis and structure of some substituted 2-amino-4-aryl-7-propargyloxy-4H-chromene-3-carbonitriles
  39. Synthesis, biological evaluation and molecular docking study of 1,2,3-1H-triazoles having 4H-pyrano[2,3-d]pyrimidine as potential Mycobacterium tuberculosis protein tyrosine phosphatase B inhibitors
  40. Reaction of Some Substituted 3-Aryl-4-formylsydnones with Tetra-Oacetyl- β-D-galactopyranosyl)thiosemicarbazide
  41. Synthesis and evaluation of in vivo antioxidant, in vitro antibacterial, MRSA and antifungal activity of novel substituted isatin N- (2,3,4,6-tetra- O -acetyl-β -d- glucopyranosyl)thiosemicarbazones
  42. Ionic Liquids as Catalyst for Synthesis of Some Aromatic Peracetylated N-(β-DGlucopyranosyl) Thiosemicarbazones
  43. Synthesis of Some Novel Substituted Benzaldehyde N-(2,3,6,2´,3´,4´,6´ - Hepta-O-Acetyl-β-D-Lactosyl)thiosemicarbazones
  44. Synthesis and Characterization of Some Novel Thiosemicarbazones of Substituted Benzaldehydes and N-(Hepta-O-Acetyl-β-d-Lactosyl)Thiosemicarbazide
  45. <strong>SYNTHESIS OF SOME (HEPTA-O-ACETYL-</strong><strong>b</strong><strong>-LACTOSYL)THIOSEMICARBAZONES CONTAINING AROMATIC NUCLEUS WITH IONIC LIQUID AS CATALYST</strong>
  46. SYNTHESIS OF 2-AMINOTHIAZOLIDIN-4-ONES FROM (HEPTA<em>-O-</em>ACETYL-b-MALTOSYL)THIOSEMICARBAZONES OF SUBSTITUTED ACETOPHENONES
  47. Synthesis and antibacterial and antifungal activities of N-(tetra-O-acetyl-β-d-glucopyranosyl)thiosemicarbazones of substituted 4-formylsydnones
  48. ChemInform Abstract: Study on Synthesis of 2‐(Substituted benzylidene) amino‐2‐deoxy‐1,3,4,6‐tetra‐O‐acetyl‐β‐D‐glucopyranones from D‐Glucosamine.
  49. Study on Synthesis of 2-(Substituted Benzylidene)amino-2-Deoxy-1,3,4,6- Tetra-O-Acetyl-β-D-Glucopyranoses from D-Glucosamine
  50. Antioxidant activities of thiosemicarbazones from substituted benzaldehydes and N-(tetra-O-acetyl-β-d-galactopyranosyl)thiosemicarbazide
  51. Reaction ofN-alkylisatins with 4-(2,3,4,6-tetra-O-acetyl-β-D-glucopyranosyl)thiosemicarbazide
  52. Synthesis of Some Peracetylated Glucopyranosyl Thiosemicarbazones of Substituted 4-Formylcoumarins
  53. ChemInform Abstract: Microwave‐Assisted Synthesis of Novel Tetra‐O‐acetyl‐β‐D‐glucopyranosyl Thiosemicarbazones of Substituted Isatins.
  54. Synthesis of Peracetylatedβ-D-Glucopyranosyl Thioureas from Substituted 2-Aminobenzo-1ʹ, 3ʹ-thiazoles
  55. Synthesis, structure and antioxidant activity of (tetra-O-acetyl-β-D-galactopyranosyl)thiosemicarbazones of substituted benzaldehydes
  56. Microwave-Assisted Synthesis of Novel Tetra-O-acetyl-β-D-glucopyranosyl Thiosemicarbazones of Substituted Isatins
  57. Reaction ofN-(Per-O-acetyl-β-D-glucopyranosyl)-Nʼ-(4ʼ,6ʼ-diarylpyrimidine-2ʼ-yl)thioureas with Ethyl Bromoacetate
  58. Microwave-Assisted Synthesis of Acetophenone (per-O-acetylated-β-D-glucopyranosyl)thiosemicarbazones
  59. Synthesis of N-tetra-O-acetyl-β-d-glucopyranosyl-N′-(4′,6′-diarylpyrimidin-2′-yl)thioureas