All Stories

  1. Water-based coupling of amino acids for sustainable solid-phase peptide synthesis
  2. Molecular Click Adventures — A Leap From the Shoulders of Giants
  3. Click‐Cyclized Cell Penetrating Peptides Containing Hydrophobic Proline Derivatives for Efficient Intracellular Delivery
  4. Click‐Cyclized Cell Penetrating Peptides Containing Hydrophobic Proline Derivatives for Efficient Intracellular Delivery
  5. Parthenolide disrupts mitosis by inhibiting ZNF207/BUGZ-promoted kinetochore-microtubule attachment
  6. Green Resins for All: Sustainable Preparation of PEGA Resin for Peptide and Protein Synthesis and Immobilization
  7. Hydrodynamic Control of Alzheimer Aβ Fibrillation with Glucosaminic Acid Containing Click-Cyclized β-Bodies
  8. Development of Selective ADAMTS-5 Peptide Substrates to Monitor Proteinase Activity
  9. Cascade autohydrolysis of Alzheimer's Aβ peptides
  10. British Society for Matrix Biology Spring 2021 Meeting: “Inflammation, Fibrosis, Resolution and the Matrix”
  11. Attachment of cyclodextrin acids to PEGA resin and study of binding with fluorescence microscopy
  12. C-Terminal lactamization of peptides
  13. Dihydroquinazolinones via A 3 ‐Type Reactions of N ‐Carbamoyliminium Ions
  14. Recent Fascinating Aspects of the CuAAC Click Reaction
  15. Design and Combinatorial Development of Shield-1 Peptide Mimetics Binding to Destabilized FKBP12
  16. Synthesis of Shld Derivatives, Their Binding to the Destabilizing Domain, and Influence on Protein Accumulation in Transgenic Plants
  17. Azotides as Modular Peptide-Based Ligands for Asymmetric Lewis Acid Catalysis
  18. Semisynthesis of an Active Enzyme by Quantitative Click Ligation
  19. Computational Evolution of Threonine-Rich β-Hairpin Peptides Mimicking Specificity and Affinity of Antibodies
  20. Metallo-Organozymes with Specific Proteolytic Activity
  21. Sustainable Flow Synthesis of Encoded Beads for Combinatorial Chemistry and Chemical Biology
  22. Innenrücktitelbild: Rational Tuning of Fluorobenzene Probes for Cysteine-Selective Protein Modification (Angew. Chem. 27/2018)
  23. Rational Tuning of Fluorobenzene Probes for Cysteine-Selective Protein Modification
  24. Rational Tuning of Fluorobenzene Probes for Cysteine-Selective Protein Modification
  25. MC4R Agonists: Structural Overview on Antiobesity Therapeutics
  26. Screening for selective aggrecanase substrates to detect early proteolytic events in cartilage degradation
  27. Catalytic Click Reactions
  28. Click-Chemistry-Mediated Synthesis of Selective Melanocortin Receptor 4 Agonists
  29. Diversity-Oriented Syntheses by Combining CuAAC and Stereoselective INCIC Reactions with Peptides
  30. Mechanism and Scope of Base-Controlled Catalyst-Free N-Arylation of Amines with Unactivated Fluorobenzenes
  31. Recent advances in covalent, site-specific protein immobilization
  32. Comparative studies of adhesion peptides based onl- ord-amino acids
  33. Faculty of 1000 evaluation for Click chemistry in complex mixtures: bioorthogonal bioconjugation.
  34. Faculty of 1000 evaluation for Enzymatic bioconjugation of nanoparticles: developing specificity and control.
  35. Faculty of 1000 evaluation for Enhanced enzyme stability through site-directed covalent immobilization.
  36. Faculty of 1000 evaluation for Site-specific protein immobilization using unnatural amino acids.
  37. Faculty of 1000 evaluation for Oriented immobilization of proteins on solid supports for use in biosensors and biochips: a review.
  38. Faculty of 1000 evaluation for Sortase A mediated site-specific immobilization for identification of protein interactions in affinity purification-mass spectrometry experiments.
  39. Faculty of 1000 evaluation for A chemoenzymatic approach to protein immobilization onto crystalline cellulose nanoscaffolds.
  40. Faculty of 1000 evaluation for Cellular incorporation of unnatural amino acids and bioorthogonal labeling of proteins.
  41. Faculty of 1000 evaluation for In situ regeneration of bioactive coatings enabled by an evolved Staphylococcus aureus sortase A.
  42. Faculty of 1000 evaluation for Biomolecular patterning of glass surfaces via strain-promoted cycloaddition of azides and cyclooctynes
  43. Faculty of 1000 evaluation for Continuous monitoring of enzymatic reactions on surfaces by real-time flow cytometry: sortase a catalyzed protein immobilization as a case study.
  44. Faculty of 1000 evaluation for Site-specific immobilization of protein layers on gold surfaces via orthogonal sortases.
  45. Faculty of 1000 evaluation for Chemoenzymatic reversible immobilization and labeling of proteins without prior purification.
  46. Faculty of 1000 evaluation for Bio-orthogonal Immobilization of Fibroblast Growth Factor 2 for Spatial Controlled Cell Proliferation
  47. Faculty of 1000 evaluation for Covalent Modification of Synthetic Hydrogels with Bioactive Proteins via Sortase-Mediated Ligation.
  48. Faculty of 1000 evaluation for Enzyme directed formation of un-natural side-chains for covalent surface attachment of proteins.
  49. Faculty of 1000 evaluation for Covalent and density-controlled surface immobilization of E-cadherin for adhesion force spectroscopy.
  50. Faculty of 1000 evaluation for An intein-mediated site-specific click conjugation strategy for improved tumor targeting of nanoparticle systems.
  51. Faculty of 1000 evaluation for Immobilization of actively thromboresistant assemblies on sterile blood-contacting surfaces.
  52. Faculty of 1000 evaluation for Site-specific protein labelling and immobilization mediated by microbial transglutaminase.
  53. Specific Electrostatic Molecular Recognition in Water
  54. Click-chemistry of polymersomes on nanoporous polymeric surfaces
  55. Novel Application of Peptidyl-Lys Metallopeptidase as a C-Terminal Processing Protease
  56. Intramolecular N-Acyliminium Cascade (INAIC) Reactions in Cyclization of Peptide-Like Molecules
  57. C-Terminally modified peptides via cleavage of the HMBA linker by O-, N- or S-nucleophiles
  58. Click Chemistry Mediated Functionalization of Vertical Nanowires for Biological Applications
  59. Heterologous expression of peptidyl-Lys metallopeptidase ofArmillaria melleaand mutagenic analysis of the recombinant peptidase
  60. ChemInform Abstract: Fmox: A Base-Labile Aldehyde Protecting Group.
  61. Substrate Specificity Profiling of Peptidyl-Lys Metallopeptidase of Armillaria mellea by FRET Based Peptide Library
  62. A single-vector EYFP reporter gene assay for G protein-coupled receptors
  63. Faculty of 1000 evaluation for Biosynthesis of versipelostatin: identification of an enzyme-catalyzed [4+2]-cycloaddition required for macrocyclization of spirotetronate-containing polyketides.
  64. Covalent and Stable CuAAC Modification of Silicon Surfaces for Control of Cell Adhesion
  65. Fmox: A Base-Labile Aldehyde Protecting Group
  66. Advances in Merging Triazoles with Peptides and Proteins
  67. Alkyne-Azide Reactions
  68. In vivo imaging of MMP-13 activity in the murine destabilised medial meniscus surgical model of osteoarthritis
  69. In Vivo Imaging of Matrix Metalloproteinase 12 and Matrix Metalloproteinase 13 Activities in the Mouse Model of Collagen-Induced Arthritis
  70. Faculty of 1000 evaluation for Discovery of Chemoselective and Biocompatible Reactions Using a High-Throughput Immunoassay Screening.
  71. Organozymes: Molecular Engineering and Combinatorial Selection of Peptidic Organo- and Transition-Metal Catalysts
  72. Award Lectures
  73. Methods for the preparation of chlorophyllide a: An intermediate of the chlorophyll biosynthetic pathway
  74. Metabolically Stable Cellular Adhesion to Inert Surfaces
  75. Simultaneous “One Pot” Expressed Protein Ligation and CuI-Catalyzed Azide/Alkyne Cycloaddition for Protein Immobilization
  76. A comparative study of the physicochemical properties of iron isomaltoside 1000 (Monofer®), a new intravenous iron preparation and its clinical implications
  77. Lectin Domains of Polypeptide GalNAc Transferases Exhibit Glycopeptide Binding Specificity
  78. ChemInform Abstract: Dipolar Cycloaddition Reactions in Peptide Chemistry
  79. Maintaining Biological Activity by Using Triazoles as Disufide Bond Mimetics
  80. Maintaining Biological Activity by Using Triazoles as Disufide Bond Mimetics
  81. Faculty of 1000 evaluation for Activity Landscape Representations for Structure-Activity Relationship Analysis.
  82. ChemInform Abstract: A Facile One-Pot Synthesis of 3,4-Dihydro-3-hydroxy-4-oxo-1,2,3- benzotriazine and Derivatives.
  83. ChemInform Abstract: Multiple Column Solid Phase Glycopeptide Synthesis.
  84. ChemInform Abstract: Pentafluorophenyl Esters for Temporary Carboxyl Group Protection in Solid Phase Synthesis of N-Linked Glycopeptides.
  85. ChemInform Abstract: Multiple-Column Solid-Phase Glycopeptide Synthesis
  86. ChemInform Abstract: A New Strategy for Solid-Phase Synthesis of O-Glycopeptides.
  87. ChemInform Abstract: Synthesis and Immunological Properties of Glycopeptide T-Cell Determinants
  88. ChemInform Abstract: Protected-Mode Synthesis of N-Linked Glycopeptides: Single-Step Preparation of Building Blocks as Peracetyl Glycosylated NαFmoc Asparagine OPfp Esters
  89. ChemInform Abstract: Synthesis of Mannose 6-Phosphate-Containing Disaccharide Threonine Building Blocks and Their Use in Solid-Phase Glycopeptide Synthesis.
  90. ChemInform Abstract: Large-Scale Synthesis of D-Mannose 6-Phosphate and Other Hexose 6- Phosphates.
  91. ChemInform Abstract: Glycosylation of Phenols: Preparation of 1,2-cis and 1,2-trans Glycosylated Tyrosine Derivatives to be used in Solid-Phase Glycopeptide Synthesis.
  92. ChemInform Abstract: Glycopeptide Synthesis
  93. ChemInform Abstract: Recent Developments in Glycopeptide and Oligosaccharide Synthesis
  94. ChemInform Abstract: The Use of O-Glycosyl Trichloroacetimidates in the Synthesis of Unsymmetrical Trehalose Analogues.
  95. ChemInform Abstract: A PEGA Resin for Use in the Solid-Phase Chemical-Enzymatic Synthesis of Glycopeptides.
  96. ChemInform Abstract: Synthesis of 2′- and 2′′-O-Acylated Maltotriosides as Potential Fluorescence-Quenched Substrates for α-Amylase.
  97. ChemInform Abstract: Gram-Scale Synthesis of α,α-Trehalose 6-Monophosphate and . alpha.,α-Trehalose 6,6′-Diphosphate.
  98. ChemInform Abstract: Convenient Synthesis of O-(2-Acetamido-2-deoxy-β-D-glucopyranosyl) -serine and -threonine Building Blocks for Solid-Phase Glycopeptide Assembly.
  99. ChemInform Abstract: Synthesis and Application of a PEGA Polymeric Support for High Capacity Continuous Flow Solid-Phase Peptide Synthesis.
  100. ChemInform Abstract: 2′-Deoxypuromycin: Synthesis and Antiviral Evaluation.
  101. ChemInform Abstract: Dithiasuccinoyl (Dts) Amino-Protecting Group Used in Syntheses of 1,2- trans-Amino Sugar Glycosides.
  102. ChemInform Abstract: Synthesis of Aliphatic O-Dimannosyl Amino Acid Building Blocks for Solid-Phase Assembly of Glycopeptide Libraries.
  103. ChemInform Abstract: Solid-Phase Synthesis of a Fucosylated Glycopeptide of Human Factor IX with a Fucose-α-(1 → O)-serine Linkage.
  104. ChemInform Abstract: Ralph F. Hirschmann Award Address 2009: Merger of Organic Chemistry with Peptide Diversity
  105. ChemInform Abstract: Recent Developments in Glycopeptide Synthesis
  106. ChemInform Abstract: Stereoselective Synthesis of the C-Analogue of β-D- Glucopyranosyl Serine.
  107. ChemInform Abstract: Properties of Solid Supports
  108. ChemInform Abstract: Synthetic Methods of Glycopeptide Assembly and Biological Analysis of Glycopeptide Products
  109. ChemInform Abstract: Novel Acylation Catalysts in Peptide Synthesis: Derivatives of N-Hydroxytriazoles and N-Hydroxytetrazoles.
  110. ChemInform Abstract: N-Acyliminium Intermediates in Solid-Phase Synthesis
  111. ChemInform Abstract: Novel Type of Rigid C-Linked Glycosylacetylene-Phenylalanine Building Blocks for Combinatorial Synthesis of C-Linked Glycopeptides.
  112. ChemInform Abstract: Evaluation of the Effect of Glycosylation on the Enzymic Hydrolysis of Peptides.
  113. ChemInform Abstract: Carbohydrate Chemistry: Synthetic and Structural Challenges Towards the End of the 20th Century
  114. ChemInform Abstract: Glycopeptide and Oligosaccharide Libraries
  115. ChemInform Abstract: Glycopeptide and Oligosaccharide Libraries
  116. ChemInform Abstract: Glycopeptides: A Link Between Complex Carbohydrates and Glycoproteins
  117. ChemInform Abstract: Preparation of Novel O-Sulfated Amino Acid Building Blocks with Improved Acid Stability for Fmoc-Based Solid-Phase Peptide Synthesis.
  118. ChemInform Abstract: Preparation and Screening of Glycopeptide Libraries
  119. ChemInform Abstract: Solid-Phase Synthesis of Complex and Pharmacologically Interesting Heterocycles
  120. Microparticle Matrix Encoding of Beads
  121. Microparticle Matrix Encoding of Beads
  122. Small-Molecule Affinity Ligands for Protein Purification: Combined Computational Enrichment and Automated In-line Screening of an Optically Encoded Library
  123. Faculty of 1000 evaluation for Proteome-derived, database-searchable peptide libraries for identifying protease cleavage sites.
  124. Amino acid derived 1,4-dialkyl substituted imidazolones
  125. N-acyliminium intermediates in solid-phase synthesis
  126. Ralph F. Hirschmann award address 2009: Merger of organic chemistry with peptide diversity
  127. Imidazolones in Diastereoselective Cyclization Reactions and CuII-Catalysed Cross-Coupling Reactions
  128. 9-Acridinylpeptides and 9-acridinyl-4-nitrophenylsulfonylpeptides
  129. Susceptibility of glycans to β-elimination in Fmoc-based O-glycopeptide synthesis
  130. Multiple column peptide synthesis, Part 2 (1, 2)
  131. Amidation of growth hormone releasing factor (1-29) by serine carboxypeptidase catalysed transpeptidation
  132. Faculty of 1000 evaluation for Highly efficient molybdenum-based catalysts for enantioselective alkene metathesis.
  133. ChemInform Abstract: Cu-Catalyzed Azide-Alkyne Cycloaddition
  134. Green Catalysts: Solid-Phase Peptide Carbene Ligands in Aqueous Transition-Metal Catalysis
  135. Expression and substrate specificity of a recombinant cysteine proteinase B of Leishmania braziliensis
  136. Faculty of 1000 evaluation for Switch-peptides: design and characterization of controllable super-amyloid-forming host-guest peptides as tools for identifying anti-amyloid agents.
  137. Cu-Catalyzed Azide−Alkyne Cycloaddition
  138. Polymer “Clicking” by CuAAC Reactions
  139. Divergent Pathway for the Solid-Phase Conversion of Aromatic Acetylenes to Carboxylic Acids, α-Ketocarboxylic Acids, and Methyl Ketones
  140. Optically Active (Peptido-carbene)palladium Complexes: Towards True Solid-Phase Combinatorial Libraries of Transition Metal Catalysts
  141. Solid-Phase Synthesis of Aryl-Substituted Thienoindolizines: Sequential Pictet−Spengler, Bromination and Suzuki Cross-Coupling Reactions of Thiophenes
  142. Scaffold Diversity through Intramolecular Cascade Reactions of Solid-Supported CyclicN-Acyliminium Intermediates
  143. Specific Recognition of Disaccharides in Water by an Artificial Bicyclic Carbohydrate Receptor
  144. Specific Recognition of Disaccharides in Water by an Artificial Bicyclic Carbohydrate Receptor (Eur. J. Org. Chem. 30/2007)
  145. Controlled Peptide Solvation in Portion-Mixing Libraries of FRET Peptides:  Improved Specificity Determination for Dengue 2 Virus NS2B-NS3 Protease and Human Cathepsin S
  146. Solid-Phase Synthesis of Carboxylic and Oxamic Acids via OsO4/NaIO4/HMTA-Mediated Oxidative Cleavage of Acetylenic Peptides
  147. Solid-Phase Synthesis of Tetrahydro-β-carbolines and Tetrahydroisoquinolines by Stereoselective IntramolecularN-Carbamyliminium Pictet–Spengler Reactions
  148. Faculty of 1000 evaluation for Development of O-acyl isopeptide method.
  149. Solid-Phase Synthesis of a Peptide-Based P,S-Ligand System Designed for Generation of Combinatorial Catalyst Libraries
  150. Faculty of 1000 evaluation for Construction and structural characterization of versatile lactosaminoglycan-related compound library for the synthesis of complex glycopeptides and glycosphingolipids.
  151. Faculty of 1000 evaluation for Evaluation of "credit card" libraries for inhibition of HIV-1 gp41 fusogenic core formation.
  152. Solid-Phase Synthesis of Tetrahydro-β-carbolines and Tetrahydroisoquinolines by Stereoselective IntramolecularN-Carbamyliminium Pictet–Spengler Reactions
  153. Faculty of 1000 evaluation for A differential array of metalated synthetic receptors for the analysis of tripeptide mixtures.
  154. Artificial Enzymes. Herausgegeben von Ronald Breslow.
  155. Artificial Enzymes. Edited by Ronald Breslow.
  156. Smart Assays in Combinatorial Chemistry
  157. Smart Combinatorial Assays for the Determination of Protease Activity and Inhibition
  158. Solid-phase synthesis of biarylalanines via Suzuki cross-coupling and intramolecular N-acyliminium Pictet–Spengler reactions
  159. GAG Mimetic Libraries: Sulphated Peptide as Heparin-like Glycosaminoglycan Mimics in Their Interaction with FGF-1
  160. Faculty of 1000 evaluation for Facile preparation of carbohydrate microarrays by site-specific, covalent immobilization of unmodified carbohydrates on hydrazide-coated glass slides.
  161. Faculty of 1000 evaluation for AFM-tip-integrated amperometric microbiosensors: high-resolution imaging of membrane transport.
  162. Faculty of 1000 evaluation for A topologically segregated one-bead-one-compound combinatorial glycopeptide library for identification of lectin ligands.
  163. Solid-Phase Synthesis of Bicyclic Dipeptide Mimetics by Intramolecular Cyclization of Alcohols, Thiols, Amines, and Amides withN-Acyliminium Intermediates
  164. Efficient Solid-Phase Synthesis of Peptide-Based Phosphine Ligands: Towards Combinatorial Libraries of Selective Transition Metal Catalysts
  165. Solid-Phase Synthesis of Pyrroloisoquinolines via the IntramolecularN-Acyliminium Pictet−Spengler Reaction
  166. Highly Efficient Solid-Phase Oxidative Cleavage of Olefins by OsO4−NaIO4in the IntramolecularN-Acyliminium Pictet−Spengler Reaction
  167. Application of a Photolabile Backbone Amide Linker for Cleavage of Internal Amides in the Synthesis towards Melanocortin Subtype-4 Agonists
  168. One Bead Two Compound Libraries for Detecting Chemical and Biochemical Conversions
  169. Reversible Dimerization of Acid-Denatured ACBP Controlled by Helix A4†
  170. Versatile Solid-Phase Synthesis of Peptide-Derived 2-Oxazolines. Application in the Synthesis of Ligands for Asymmetric Catalysis
  171. Complex of sialoadhesin with a glycopeptide ligand
  172. N-TERMINAL DOMAIN OF SIALOADHESIN (MOUSE) IN COMPLEX WITH GLYCOPEPTIDE
  173. High Capacity Poly(ethylene glycol) Based Amino Polymers for Peptide and Organic Synthesis
  174. ULTRAMINE: A High-Capacity Polyethylene-Imine-Based Polymer and Its Application as a Scavenger Resin
  175. Faculty of 1000 evaluation for Discovery and characterization of catalysts for azide-alkyne cycloaddition by fluorescence quenching.
  176. Differences in substrate specificities between cysteine protease CPB isoforms of Leishmania mexicana are mediated by a few amino acid changes
  177. The Pictet—Spengler Reaction in Solid-Phase Combinatorial Chemistry
  178. ‘One bead two compound libraries’ for detecting chemical and biochemical conversions
  179. Faculty of 1000 evaluation for Synthesis of monofunctionalized gold nanoparticles by fmoc solid-phase reactions.
  180. Solid-Phase IntramolecularN-Acyliminium Pictet−Spengler Reactions as Crossroads to Scaffold Diversity
  181. Combinatorial Library of Peptidotriazoles:  Identification of [1,2,3]-Triazole Inhibitors against a RecombinantLeishmaniamexicanaCysteine Protease
  182. Pyrazines on Solid Support from Peptides by Periodinane Oxidation of Threonine Side-Chains. A Quantitative Chemical Transformation (QCT) for Combinatorial Chemistry
  183. Bicyclic Organo-Peptides as Selective Carbohydrate Receptors: Design, Solid-phase Synthesis, and on-bead Binding Capability
  184. Synthesis of 3-Boc-(1,3)-oxazinane-Protected Amino Aldehydes from Amino Acids and Their Conversion into Urea Precursors. Novel Building Blocks for Combinatorial Synthesis
  185. Faculty of 1000 evaluation for Carboxydipeptidase activities of recombinant cysteine peptidases. Cruzain of Trypanosoma cruzi and CPB of Leishmania mexicana.
  186. Faculty of 1000 evaluation for Dyad beads and the combinatorial discovery of catalysts.
  187. α-Keto Amide Peptides:  A Synthetic Strategy to Resin-Bound Peptide Isosteres for Protease Inhibitor Screening on Solid Support
  188. Automated Sorting of Beads from a“One-Bead-Two-Compounds” Combinatorial Library of Metalloproteinase Inhibitors
  189. Solid Phase Combinatorial Library of 1,3-Azole Containing Peptides for the Discovery of Matrix Metallo Proteinase Inhibitors
  190. MUC1-derived glycopeptide libraries with improved MHC anchors are strong antigens and prime mouse T cells for proliferative responses to lysates of human breast cancer tissue
  191. Solid-Phase Combinatorial Library of Norstatine-Type Isosters by the Nitroaldol Reaction
  192. Solid-Phase Synthesis and Biological Activity of a Thioether Analogue of Conotoxin G1
  193. Glycopeptides as Oligosaccharide Mimics:  High Affinity Sialopeptide Ligands for Sialoadhesin from Combinatorial Libraries
  194. ChemInform Abstract: Physical Properties of Polyethylene Glycol (PEG)‐Based Resins for Solid‐Phase Organic Chemistry: A Comparison of PEG Crosslinked and PEG Grafted Resins.
  195. EXPO3000—a new expandable polymer for synthesis and enzymatic assays
  196. A Solid-Phase Approach to Mouse Melanocortin Receptor Agonists Derived from a Novel Thioether Cyclized Peptidomimetic Scaffold
  197. Faculty of 1000 evaluation for Synthesis and screening of libraries of synthetic tripodal receptor molecules with three different amino acid or peptide arms: identification of iron binders.
  198. SPOCC-194, a New High Functional Group Density PEG-Based Resin for Solid-Phase Organic Synthesis
  199. Processing of glycans on glycoprotein and glycopeptide antigens in antigen-presenting cells
  200. Combinatorial chemistry
  201. Optimizing Delays in the MBOB, Broadband HMBC, and Broadband XLOC NMR Pulse Sequences
  202. Faculty of 1000 evaluation for Amplification of screening sensitivity through selective destruction: theory and screening of a library of carbonic anhydrase inhibitors.
  203. Peptidotriazoles on Solid Phase:  [1,2,3]-Triazoles by Regiospecific Copper(I)-Catalyzed 1,3-Dipolar Cycloadditions of Terminal Alkynes to Azides
  204. Solid-Phase Library Synthesis, Screening, and Selection of Tight-Binding Reduced Peptide Bond Inhibitors of a RecombinantLeishmaniamexicanaCysteine Protease B
  205. SULFATED PEPTIDES AS HEPARIN MIMICS DESIGNED FOR FGF RECEPTOR INTERACTIONS
  206. Preparation of novel O-sulfated amino acid building blocks with improved acid stability for Fmoc-based solid-phase peptide synthesis
  207. Faculty of 1000 evaluation for Solid phase synthesis of mixture-based acyclic and heterocyclic small molecule combinatorial libraries from resin-bound polyamides.
  208. The one-bead two-compound assay for solid phase screening of combinatorial libraries
  209. Analysis of O-and N-linked glycopeptide libraries by MALDI-TOF MS: Application in solid phase assays of carbohydrate-binding-proteins
  210. Palladium on Carbon Encapsulated in POEPOP1500:  A Resin-Supported Catalyst for Hydrogenation Reactions
  211. Faculty of 1000 evaluation for Monitoring of solid-phase organic synthesis on macroscopic supports by high-resolution magic angle spinning NMR.
  212. Peptido-organic Diels–Alder reactions on hydrophilic resin: scope for combinatorial chemistry
  213. Radically altered T cell receptor signaling in glycopeptide-specific T cell hybridoma induced by antigen with minimal differences in the glycan group
  214. Faculty of 1000 evaluation for From Split-Pool Libraries to Spatially Addressable Microarrays and Its Application to Functional Proteomic Profiling.
  215. Titelbild
  216. Cover Picture
  217. Unichemo Protection: A Concept for Chemical Synthesis
  218. Titelbild
  219. Unichemo Protection: A Concept for Chemical Synthesis This work was supported by the Danish National Research Foundation.
  220. Combinatorial Library of Peptide Isosters Based on Diels−Alder Reactions:  Identification of Novel Inhibitors against a Recombinant Cysteine Protease fromLeishmania mexicana
  221. Solid-Phase Glycosylation of Peptide Templates and On-Bead MAS-NMR Analysis: Perspectives for Glycopeptide Libraries
  222. Diffusion of Reagents in Macrobeads
  223. Substrate specificity of recombinant cysteine proteinase, CPB, of Leishmania mexicana
  224. Phosphinic Peptide Inhibitors of Macrophage Metalloelastase (MMP-12). Selectivity and Mechanism of Binding
  225. Identification of peptides inhibitory to recombinant cysteine proteinase, CPB, of Leishmania mexicana
  226. α-Ketocarbonyl Peptides:  A General Approach to Reactive Resin-Bound Intermediates in the Synthesis of Peptide Isosteres for Protease Inhibitor Screening on Solid Support
  227. UniChemo Protection (UCP)
  228. Peptidotriazoles: Copper(I)-Catalyzed 1,3-Dipolar Cycloadditions on Solid-Phase
  229. A Novel Solid Phase Approach to Thioether Cyclized Peptides: Discovery of Mouse Melanocortin-1 Receptor Agonists
  230. Determining the Fate of Glycopeptides During Antigen Processing in Antigen Presenting Cells
  231. Oxidation of Threonine and Serine Residues on Solid-Phase: Pyrazine Formation by Dess-Martin Periodinane Oxidation
  232. Solid-Phase Synthesis Utilizing Azido-α-Amino Acids: Reduction of Azido-Protected Proline
  233. Synthesis of Aldehyde Building Blocks Protected as Acid LabileN-BocN,O-Acetals:  Toward Combinatorial Solid Phase Synthesis of Novel Peptide Isosteres1,†
  234. ChemInform Abstract: Identification of Protease Inhibitors Using Biocompatible Resins and Library Synthesis
  235. Synthesis of tumor associated sialyl-T-glycopeptides and their immunogenicity
  236. Surfactant Mediated Cationic and Anionic Suspension Polymerization of PEG-Based Resins in Silicon Oil:  Beaded SPOCC 1500 and POEPOP 1500
  237. ChemInform Abstract: Synthesis and Application of Sialic Acid Containing Building Blocks for Glycopeptide Libraries. Establishing Glycosylation Conditions.
  238. N-Terminal Peptide Aldehydes as Electrophiles in Combinatorial Solid Phase Synthesis of Novel Peptide Isosteres
  239. Internally quenched fluorescent peptide substrates disclose the subsite preferences of human caspases 1, 3, 6, 7 and 8
  240. Internally quenched fluorescent peptide substrates disclose the subsite preferences of human caspases 1, 3, 6, 7 and 8
  241. Epitope affinity for MHC class I determines helper requirement for CTL priming
  242. Solid-phase Synthesis of Chemotactic Peptides Using α-Azido Acids
  243. Hydrolysis by Cathepsin B of Fluorescent Peptides Derived From Human Prorenin
  244. Expression and characterization of a recombinant cysteine proteinase of Leishmania mexicana
  245. Expression and characterization of a recombinant cysteine proteinase of Leishmania mexicana
  246. Glycopeptid- und Oligosaccharidbibliotheken
  247. Glycopeptide and Oligosaccharide Libraries
  248. Enzymatic and chiral HPLC resolution of α-azido acids and amides
  249. Physical Properties of Poly(ethylene glycol) (PEG)-Based Resins for Combinatorial Solid Phase Organic Chemistry:  A Comparison of PEG-Cross-Linked and PEG-Grafted Resins
  250. Towards peptide isostere libraries: aqueous aldol reactions on hydrophilic solid supports
  251. HYDRA: A novel hydroxy and amine functionalised resin synthesised by reductive amination of PEG aldehyde and a polyamine
  252. Single-bead structure elucidation. Requirements for analysis of combinatorial solid-phase libraries by Nanoprobe MAS-NMR spectroscopy
  253. Novel methodology for the solid-phase synthesis of phosphinic peptides †
  254. Synthesis and application of sialic acid-containing building blocks for glycopeptide libraries. Establishing glycosylation conditions
  255. ?-Azido acids for direct use in solid-phase peptide synthesis
  256. Synthesis of tumor associated sialyl-T-glycopeptides and their immunogenicity
  257. Solid-phase Synthesis of Chemotactic Peptides Using ?-Azido Acids
  258. Glycopeptide and Oligosaccharide Libraries
  259. Phosphinic Peptide Matrix Metalloproteinase-9 Inhibitors by Solid-Phase Synthesis Using a Building Block Approach
  260. Shared structural motifs in TCR of glycopeptide-recognizing T cell hybridomas
  261. Carbohydrate chemistry: synthetic and structural challenges towards the end of the 20th century
  262. SPOCC:  A Resin for Solid-Phase Organic Chemistry and Enzymatic Reactions on Solid Phase
  263. Solid-Phase Synthesis of Peptide Isosters by Nucleophilic Reactions with N-Terminal Peptide Aldehydes on a Polar Support Tailored for Solid-Phase Organic Chemistry
  264. Solid-Phase Synthesis of Peptide Isosters by Nucleophilic Reactions withN-Terminal Peptide Aldehydes on a Polar Support Tailored for Solid-Phase Organic Chemistry
  265. Identification of Protease Inhibitors Using Biocompatible Resins and Library Synthesis
  266. Novel Type of Rigid C-Linked Glycosylacetylene−Phenylalanine Building Blocks for Combinatorial Synthesis of C-linked Glycopeptides
  267. Oligosaccharide Mimetics Obtained by Novel, Rapid Screening of Carboxylic Acid Encoded Glycopeptide Libraries
  268. A chemically inert hydrophilic resin for solid phase organic synthesis
  269. Analysis of organic reactions by thin layer chromatography combined with matrix‐assisted laser desorption/ionization time‐of‐flight mass spectrometry
  270. Kinetic Analysis of the Mechanism and Specificity of Protein-disulfide Isomerase Using Fluorescence-quenched Peptides
  271. Synthesis and characterization of polyethylene glycol polyacrylamide copolymer (PEGA) resins containing carbohydrate ligands. Evaluation as supports for affinity chromatography
  272. Fluorescence Energy-Transfer Probes of Conformation in Peptides:  The 2-Aminobenzamide/Nitrotyrosine Pair
  273. The extracellular polysaccharide of Pichia (Hansenula) holstii NRRL Y-2448: the phosphorylated side chains
  274. PEGA supports for combinatorial peptide synthesis and solid-phase enzymatic library assays
  275. PEGA supports for combinatorial peptide synthesis and solid-phase enzymatic library assays
  276. Inhibition of cruzipain visualized in a fluorescence quenched solid-phase inhibitor library assay.D-Amino Acid Inhibitors for cruzipain, cathepsin B and cathepsin L
  277. Preparation of fluorescence quenched libraries containing interchain disulphide bonds for studies of protein disulphide isomerases
  278. C-Linked glycosyl azido acid in novel solid-phase C-glycopeptide synthesis
  279. Fluorescent properties of amino acids labeled with ortho‐aminobenzoic acid
  280. Fluorescent properties of amino acids labeled withortho-aminobenzoic acid
  281. Synthesis and characterization of polyethylene glycol polyacrylamide copolymer (PEGA) resins containing carbohydrate ligands. Evaluation as supports for affinity chromatography
  282. Solid Phase Libraries of Glycopeptide Templates in the Study of Complex Oligosaccharide-Receptor Interactions
  283. Synthetic methods of glycopeptide assembly, and biological analysis of glycopeptide products
  284. Synthetic hFSH peptide constructs in the evaluation of previous studies on the hFSH receptor interaction
  285. Synthetic hFSH peptide constructs in the evaluation of previous studies on the hFSH receptor interaction
  286. Direkte Festphasen-Glycosylierung von Peptiden an einem neuartigen Polyethylenglycol-Harz
  287. Azido Acids in a Novel Method of Solid-Phase Peptide Synthesis.
  288. Synthesis and characterisation of highly glycosylated glycopeptides with Tn-antigenic structures corresponding to human glycophorin AN
  289. Stereoselective synthesis of the C-analogue of β-d-glucopyranosyl serine
  290. New solid-phase oligosaccharide synthesis on glycopeptides bound to a solid phase
  291. Internally quenched fluorogenic, α-helical dimeric peptides and glycopeptides for the evaluation of the effect of glycosylation on the conformation of peptides
  292. Synthesis of glycopeptide sequences of repeating units of the mucins MUC 2 and MUC 3 containing oligosaccharide side-chains with core 1, core 2, core 3, core 4 and core 6 structure
  293. [6] Properties of solid supports
  294. Constrained glycopeptide ligands for MPRs. Limitations of unprotected phosphorylated building blocks
  295. Glycopeptide mimics of mammalian Man9GlcNAc2. Ligand binding to mannan-binding proteins (MBPs)
  296. Specificity of O-glycosylation by bovine colostrum UDP-GalNAc: polypeptide ?-N-acetylgalactosaminyltransferase using synthetic glycopeptide substrates
  297. The extracellular polysaccharide of Pichia (Hansenula) holstii NRRL Y-2448: The structure of the phosphomannan backbone
  298. POEPOP and POEPS: Inert polyethylene glycol crosslinked polymeric supports for solid synthesis
  299. Multiple Column Synthesis of a Library of T-Cell Stimulating Tn-Antigenic Glycopeptide Analogues for the Molecular Characterization of T-Cell–Glycan Specificity
  300. Multiple Column Synthesis of a Library of T‐Cell Stimulating Tn-Antigenic Glycopeptide Analogues for the Molecular Characterization of T‐Cell–Glycan Specificity
  301. T cell recognition of Tn-glycosylated peptide antigens
  302. Studies of Binding Sites in the Subtilisin from Bacillus Lentus by Means of Site Directed Mutagenesis and Kinetic Investigations
  303. Spectroscopic and Protein Chemical Analyses Demonstrate the Presence of C-Mannosylated Tryptophan in Intact Human RNase 2 and Its Isoforms†
  304. Efficient synthesis of O-(2-acetamido-2-deoxy-β-d-glucopyranosyl)-ser/thr building blocks for spps of o-glcnac glycopeptides
  305. Additions and corrections
  306. Synthesis and application of a PEGA polymeric support for high capacity continuous flow solid-phase peptide synthesis
  307. 2’-Deoxypuromycin: Synthesis and Antiviral Evaluation
  308. Synthesis of the glycosyl amino acids Nα-Fmoc-Ser[Ac4-β-d-Gal p-(1 → 3)-Ac2-α-d-GalN3 p]-OPfp and Nα-Fmoc-Thr[Ac4-β-d-Gal p-(1 → 3)-Ac2-α-d-GalN3 p]-OPfp and the application in the solid-phase peptide synthesis of multiply glycosylated mucin peptides w...
  309. Synthesis of Unsymmetrical Trehalose Analogues by Silver Trifluoromethanesulphonate Promoted Glycosylations
  310. Dithiasuccinoyl (Dts) amino-protecting group used in syntheses of 1,2-trans-amino sugar glycosides
  311. Synthesis of the building blocks Nα-Fmoc-O-[α-D-Ac3GalN3p-(1→3)-α-D-Ac2GalN3p]-Thr-OPfp and Nα-Fmoc-O-[α-D-Ac3GalN3p-(1→<...
  312. Synthesis, characterization and biocompatibility of PEGA resins
  313. Synthesis of an IgA1 hinge region glycopeptide
  314. Phosphorylated glycopeptide templates as high affinity ligands for the Man-6-P receptor
  315. Multiple Column Synthesis of Quenched Solid-Phase Bound Fluorogenic Substrates for Characterization of Endoprotease Specificity
  316. The use of O-glycosyl trichloroacetimidates in the synthesis of unsymmetrical trehalose analogues
  317. Silyl protection in the solid-phase synthesis of N-linked glycopeptides. Preparation of glycosylated fluorogenic substrates for subtilisins
  318. Recent developments in glycopeptide and oligosaccharide synthesis
  319. Gram-scale synthesis of α,α-trehalose 6-monophosphate and α,α-trehalose 6,6′-diphosphate
  320. Molecular Recognition of a Salmonella Trisaccharide Epitope by Monoclonal Antibody Se155-4
  321. UDPgalactose:glycoprotein-N-acetyl-d-galactosamine 3-beta-d-galactosyltransferase activity synthesizing O-glycan core 1 is controlled by the amino acid sequence and glycosylation of glycopeptide substrates
  322. Eine neue Strategie zur Festphasensynthese vonO-Glycopeptiden über 2-Azidoglycopeptide
  323. A general approach to the synthesis ofO- andN-linked glycopeptides
  324. Synthesis of glycosyltyrosine building blocks for solid-phase glycopeptide assembly: use of aryl tert-butyl ethers as glycosyl acceptors in aromatic glycosylations
  325. Convenient synthesis of O-(2-acitamido-2-deoxy-β-D-glucopyranosyl)-serine and -threonine building blocks for solid-phase glycopeptide assembly
  326. Synthesis of 2′- and 2″-O-acylated maltotriosides as potential fluorescence-quenched substrates for α-amylase
  327. A PEGA resin for use in the solid-phase chemical–enzymatic synthesis of glycopeptides
  328. Glycopeptide Synthesis
  329. Synthesis of glycopeptides containing 6'-O-phosphorylated disaccharides as ligands for the mannose 6-phosphate receptors
  330. Synthesis and Immunological Properties of Glycopeptide T-Cell Determinants
  331. Mutational replacements of the amino acid residues forming the hydrophobic S4 binding pocket of subtilisin 309 from Bacillus lentus
  332. S17.2 Solid phase synthesis of di-N-Glycosylated RGD-Analogues
  333. S12.4 Glycopeptides as T lymphocyte antigens. Influence on binding to MHC class II and immunogenicity
  334. Silyl protection in the solid-phase synthesis of N-linked neoglycopeptides. One-step deprotection of fully protected neoglycopeptides.
  335. Multiple column peptide synthesis: Development and application
  336. Solid phase peptide synthesis of a di-N-glycosylated RGD analog
  337. Large-scale synthesis of d-mannose 6-phosphate and other hexose 6-phosphates
  338. Solid phase peptide synthesis of mucin glycopeptides
  339. Synthesis of the 1-Amino-Alditols Derived from Cellobiose, Lactose and Maltose. A Comprehensive NMR Study of Some Alditols and Amino-Alditols
  340. Eine neue Strategie zur Festphasensynthese vonO-Glycopeptiden
  341. A New Strategy for Solid-Phase Synthesis ofO-Glycopeptides
  342. Extensive comparison of the substrate preferences of two subtilisins as determined with peptide substrates which are based on the principle of intramolecular quenching
  343. Pega: a flow stable polyethylene glycol dimethyl acrylamide copolymer for solid phase synthesis.
  344. Substrate preferences of glutamic-acid-specific endopeptidases assessed by synthetic Peptide Substrates based on intramolecular fluorescence quenching
  345. Multiple-column solid-phase glycopeptide synthesis
  346. Glycosylation of tyrosine derivatives and their application for solid phase synthesis
  347. Proline-specific endopeptidases from microbial sources: isolation of an enzyme from a Xanthomonas sp.
  348. Controlled reduction of acarbose: conformational analysis of acarbose and the resulting saturated products
  349. T-Helper-Cell Determinants in Protein Antigens are Preferentially Located in Cysteine-Rich Antigen Segments Resistant to Proteolytic Cleavage by Cathepsin B, L, and D
  350. Multiple column solid phase glycopeptide synthesis
  351. Anthranilamide and nitrotyrosine as a donor-acceptor pair in internally quenched fluorescent substrates for endopeptidases: Multicolumn peptide synthesis of enzyme substrates for subtilisin carlsberg and pepsin
  352. Solid phase synthesis of internally quenched protease substrates
  353. New self-indicating, activated esters for solid phase peptide synthesis
  354. ChemInform Abstract: Pentafluorophenyl Esters for the Temporary Protection of the α-Carboxy Group in Solid Phase Glycopeptide Synthesis.
  355. Pentafluorophenyl esters for the temporary protection of the α-carboxy group in solid phase glycopeptide synthesis
  356. Pentafluorophenyl esters for temporary carboxyl group protection in solid phase synthesis of N-linked glycopeptides.
  357. A Facile One-Pot Synthesis of 3,4-Dihydro-3-hydroxy-4-oxo-1,2,3-benzotriazine and Derivatives
  358. The active ester N-fmoc-3-O-[Ac4-α-D-Manp-(1→2)-Ac3-α-D-Manp-1-]=thre-O-Pfp as a building block in solid-phase synthesis of an o-linked dimannosyl glycopeptide.
  359. The T-Lymphocyte Proliferative Response to Synthetic Peptide Antigens of Defined Secondary Structure
  360. ChemInform Abstract: Peptide Synthesis. Part 13. Feedback Control in Solid Phase Synthesis. Use of Fluorenylmethoxycarbonyl Amino Acid 3,4-Dihydro-4-oxo-1,2,3-benzotriazin-3-yl Esters in a Fully Automated System.
  361. ChemInform Abstract: Peptide Synthesis. Part 12. 3,4-Dihydro-4-oxo-1,2,3-benzotriazin-3-yl Esters of Fluorenylmethoxycarbonyl Amino Acids as Self-Indicating Reagents for Solid Phase Peptide Synthesis.
  362. Photonucleases
  363. Peptide synthesis. Part 12. 3,4-Dihydro-4-oxo-1,2,3-benzotriazin-3-yl esters of fluorenylmethoxycarbonyl amino acids as self-indicating reagents for solid phase peptide synthesis
  364. Peptide synthesis. Part 13. Feedback control in solid phase synthesis. Use of fluorenylmethoxycarbonyl amino acid 3,4-dihydro-4-oxo-1,2,3-benzotriazin-3-yl esters in a fully automated system
  365. ChemInform Abstract: Feedback Control in Organic Synthesis. A System for Solid Phase Peptide Synthesis with True Automation.
  366. ChemInform Abstract: Self-Indicating Activated Esters for Use in Solid Phase Peptide Synthesis. Fluorenylmethoxycarbonylamino Acid Derivatives of 3-Hydroxy-4-oxodihydrobenzotriazine.
  367. K88 fimbrial antigens: identification of antigenic determinants by the use of synthetic peptides
  368. Feedback control in organic synthesis. A system for solid phase peptide synthesis with true automation
  369. ChemInform Abstract: Synthesis of a Putative Antigenic Heptapeptide from Escherichia coli K88 ab Protein Fimbriae.
  370. ChemInform Abstract: Synthesis of a Putative Subtype Specific Antigenic Heptapeptide from Escherichia coli K88 ad Protein Fimbriae.
  371. ChemInform Abstract: Synthesis of a Proposed Antigenic Hexapeptide from Escherichia coli K88 Protein Fimbriae.
  372. Self-indicating activated esters for use in solid phase peptide synthesis. Fluorenylmethoxycarbonylamino acid derivatives of 3-hydroxy-4-oxodihydrobenzotriazine
  373. Synthesis of a Putative Antigenic Heptapeptide from Escherichia Coli K88 ab Protein Fimbriae.
  374. Synthesis of a Proposed Antigenic Hexapeptide from Escherichia Coli K88 Protein Fimbriae.
  375. Synthesis of a Putative Subtype Specific Antigenic Heptapeptide from Escherichia Coli K88 ad Protein Fimbriae.
  376. Immunochemistry ofSalmonellaO-antigens: Studies ofSalmonellaBO antigen epitopes by enzyme-linked immunosorbent inhibition assays
  377. ChemInform Abstract: SYNTHESIS OF TETRASACCHARIDES RELATED TO THE O-SPECIFIC DETERMINANTS OF SALMONELLA SEROGROUPS A, B AND D1
  378. ChemInform Abstract: SYNTHESIS OF THE BRANCHPOINT TETRASACCHARIDE OF THE O-SPECIFIC DETERMINANT OF SALMONELLA SEROGROUP B
  379. The conformation of Salmonella O-antigenic polysaccharide chains of serogroups A, B, and D1 predicted by semi-empirical, hard-sphere (HSEA) calculations
  380. The conformation of Salmonella O-antigenic oligosaccharides of serogroups A, B, and D1 inferred from 1H- and 13C-nuclear magnetic resonance spectroscopy
  381. ChemInform Abstract: MERCURY IODIDE AS A CATALYST IN OLIGOSACCHARIDE SYNTHESIS
  382. ChemInform Abstract: SYNTHESIS OF DISACCHARIDES RELATED TO THE O-SPECIFIC POLYSACCHARIDE OF SALMONELLA TYPHIMURIUM
  383. Synthesis of Tetrasaccharides Related to the O-Specific Determinants of Salmonella Serogroups A, B and D1.
  384. Synthesis of the Branchpoint Tetrasaccharide of the O-Specific Determinant of Salmonella Serogroup B.
  385. ChemInform Abstract: ISOMERIZATION OF D-GLUCOSE WITH GLUCOSE ISOMERASE. A MECHANISTIC STUDY
  386. Isomerization of D-Glucose with Glucose-isomerase. A Mechanistic Study.
  387. Synthesis of Disaccharides Related to the O-Specific Polysaccharide of Salmonella typhimurium.
  388. Mercury Iodide as a Catalyst in Oligosaccharide Synthesis.
  389. ChemInform Abstract: A FACILE ROUTE TO 2-SUBSTITUTED INDOLES
  390. A Facile Route to 2-Substituted Indoles.
  391. SPOCC resins: Polar and chemically inert resins for organic synthesis and library enzyme assays
  392. Investigation of enzyme activity and inhibition in the interior of novel solid supports
  393. Preparation of Biocompatible Resins for Library Syntheses
  394. Intramolecular Fluorescence-Quenched Substrate Libraries
  395. The Solid-Phase Enzyme Inhibitor Library Assay
  396. Dipolar Cycloaddition Reactions in Peptide Chemistry
  397. Introduction to Combinatorial Solid-Phase Assays for Enzyme Activity and Inhibition
  398. Preparation and Screening of Glycopeptide Libraries
  399. Backbone amide protection in solid-phase synthesis of peptide isosters derived from N-terminal γ-aldehydes
  400. Combinatorial library of phosphinic peptides for discovery of MMP inhibitors on solid-phase
  401. A combinatorial approach to the identification of cysteine protease substrates and inhibitors by application of a solid-phase fluorescence quenching assay
  402. Fluorescent quenched libraries for monitoring chemical and enzymatic disulfide bond formation and cleavage
  403. Fluorescent quenched substrates for protein disulfide isomerase (PDI) defined by the use of disulfide bridge containing libraries