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  1. Novel 4-(2-arylidenehydrazineyl)thienopyrimidine derivatives as anticancer EGFR inhibitors: Design, synthesis, biological evaluation, kinome selectivity and in silico insights

    Article • Bioorganic Chemistry, November 2023, Elsevier

    Dr. Moataz Ahmed Shaldam, Wagdy Eldehna

  2. Identification of 3‐(5‐cyano‐6‐oxo‐pyridin‐2‐yl)benzenesulfonamides as novel anticancer agents endowed with EGFR inhibitory activity

    Article • Archiv der Pharmazie, October 2023, Wiley

    Dr. Moataz Ahmed Shaldam, Wagdy Eldehna

  3. 1,5-Diaryl-1,2,4-triazole Ureas as New SLC-0111 Analogues Endowed with Dual Carbonic Anhydrase and VEGFR-2 Inhibitory Activities

    Article • Journal of Medicinal Chemistry, July 2023, American Chemical Society (ACS)

    Dr. Moataz Ahmed Shaldam

  4. Discovery of sulfonamide-tethered isatin derivatives as novel anticancer agents and VEGFR-2 inhibitors

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, April 2023, Taylor & Francis

    Dr. Moataz Ahmed Shaldam

  5. Protective Potential of Saussurea costus (Falc.) Lipsch. Roots against Cyclophosphamide-Induced Pulmonary Injury in Rats and Its In Vitro Antiviral Effect

    Article • Pharmaceuticals, February 2023, MDPI AG

    Dr. Moataz Ahmed Shaldam

  6. Synthesis, crystallographic, DNA binding, and molecular docking/dynamic studies of a privileged chalcone-sulfonamide hybrid scaffold as a promising anticancer agent

    Article • Journal of Biomolecular Structure and Dynamics, October 2022, Taylor & Francis

    Dr. Moataz Ahmed Shaldam

  7. Ketoprofen, piroxicam and indomethacin-suppressed quorum sensing and virulence factors in Acinetobacter baumannii

    Article • Journal of Applied Microbiology, October 2022, Oxford University Press (OUP)

    Dr. Moataz Ahmed Shaldam

  8. Bilosomes as Nanoplatform for Oral Delivery and Modulated In Vivo Antimicrobial Activity of Lycopene

    Article • Pharmaceuticals, August 2022, MDPI AG

    Dr. Moataz Ahmed Shaldam

  9. Anti-Biofilm and Antibacterial Activities of Cycas media R. Br Secondary Metabolites: In Silico, In Vitro, and In Vivo Approaches

    Article • Antibiotics, July 2022, MDPI AG

    Dr. Moataz Ahmed Shaldam

  10. Sodium Citrate Alleviates Virulence in Pseudomonas aeruginosa

    Article • Microorganisms, May 2022, MDPI AG

    Dr. Moataz Ahmed Shaldam

  11. Novel 3-(6-methylpyridin-2-yl)coumarin-based chalcones as selective inhibitors of cancer-related carbonic anhydrases IX and XII endowed with anti-proliferative activity

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, April 2022, Taylor & Francis

    Dr. Moataz Ahmed Shaldam, Wagdy Eldehna

  12. Multi-Spectroscopic, thermodynamic and molecular dynamic simulation studies for investigation of interaction of dapagliflozin with bovine serum albumin

    Article • Spectrochimica Acta Part A Molecular and Biomolecular Spectroscopy, January 2022, Elsevier

    Dr. Moataz Ahmed Shaldam

  13. Virtual Screening Attributes Male Biased COVID-19 Mortality to Predicted Antiviral Activity of Female Sex Hormones

    Article • Letters in Drug Design & Discovery, November 2021, Bentham Science Publishers

    PhD Basem Awad Mansour, Dr. Moataz Ahmed Shaldam, Kristina Keuper, Galal Metwally, Ahmed El-Baz

  14. A Novel Use of Allopurinol as A Quorum-Sensing Inhibitor in Pseudomonas aeruginosa

    Article • Antibiotics, November 2021, MDPI AG

    Dr. Moataz Ahmed Shaldam

  15. Secnidazole Is a Promising Imidazole Mitigator of Serratia marcescens Virulence

    Article • Microorganisms, November 2021, MDPI AG

    Dr. Moataz Ahmed Shaldam

  16. Development of Novel Quinoline-Based Sulfonamides as Selective Cancer-Associated Carbonic Anhydrase Isoform IX Inhibitors

    Article • International Journal of Molecular Sciences, October 2021, MDPI AG

    Dr. Moataz Ahmed Shaldam, Wagdy Eldehna

  17. Could the analgesic drugs, paracetamol and indomethacin, function as quorum sensing inhibitors?

    Article • Microbial Pathogenesis, September 2021, Elsevier

    Dr. Moataz Ahmed Shaldam

  18. Tackling Virulence of Pseudomonas aeruginosa by the Natural Furanone Sotolon

    Article • Antibiotics, July 2021, MDPI AG

    Dr. Moataz Ahmed Shaldam

  19. Xylitol Inhibits Growth and Blocks Virulence in Serratia marcescens

    Article • Microorganisms, May 2021, MDPI AG

    Dr. Moataz Ahmed Shaldam

  20. In silico screening of potent bioactive compounds from honeybee products against COVID-19 target enzymes

    Article • Environmental Science and Pollution Research, May 2021, Springer Science + Business Media

    Dr. Moataz Ahmed Shaldam

  21. Development of novel benzofuran-based SLC-0111 analogs as selective cancer-associated carbonic anhydrase isoform IX inhibitors

    Article • European Journal of Medicinal Chemistry, April 2021, Elsevier

    Dr. Moataz Ahmed Shaldam, Wagdy Eldehna

  22. New thiazolopyrimidine as anticancer agents: Synthesis, biological evaluation, DNA binding, molecular modeling and ADMET study

    Article • Bioorganic & Medicinal Chemistry Letters, December 2020, Elsevier

    Dr. Moataz Ahmed Shaldam

  23. In Silico Screening of Potent Bioactive Compounds from Honey Bee Products Against COVID-19 Target Enzymes

    Article • July 2020, American Chemical Society (ACS)

    Dr. Moataz Ahmed Shaldam

  24. Drugs with new lease of life as quorum sensing inhibitors: for combating MDR Acinetobacter baumannii infections

    Article • European Journal of Clinical Microbiology & Infectious Diseases, April 2020, Springer Science + Business Media

    Dr. Moataz Ahmed Shaldam

  25. Novel Pyruvate Kinase (PK) Inhibitors: New Target to Overcome Bacterial Resistance

    Article • ChemistrySelect, March 2020, Wiley

    Dr. Moataz Ahmed Shaldam

  26. Synthesis of imidazolidine‐2,4‐dione and 2‐thioxoimidazolidin‐4‐one derivatives as inhibitors of virulence factors production in Pseudomonas aeruginosa

    Article • Archiv der Pharmazie, March 2020, Wiley

    Hisham Abbas, Dr. Moataz Ahmed Shaldam

  27. Curtailing Quorum Sensing in Pseudomonas aeruginosa by Sitagliptin

    Article • Current Microbiology, February 2020, Springer Science + Business Media

    Dr. Moataz Ahmed Shaldam

  28. Synthesis and Antibacterial Evaluation of New2‐Phenylbenzimidazole Derivatives

    Article • ChemistrySelect, September 2019, Wiley

    Dr. Moataz Ahmed Shaldam

  29. Glyceryl trinitrate blocks staphyloxanthin and biofilm formation in Staphylococcus aureus

    Article • African Health Sciences, April 2019, African Journals Online (AJOL)

    Dr. Moataz Ahmed Shaldam

  30. Perturbation of Quorum Sensing in <i>Pseudomonas aeruginosa</i> by Febuxostat

    Article • Advances in Microbiology, January 2018, Scientific Research Publishing, Inc,

    Dr. Moataz Ahmed Shaldam

  31. Repurposing metformin as a quorum sensing inhibitor in <i>Pseudomonas aeruginosa</i>

    Article • African Health Sciences, September 2017, African Journals Online (AJOL)

    Dr. Moataz Ahmed Shaldam

  32. Simultaneous Determination of Formoterol Fumarate and Budesonide Epimers in Metered Dose Inhaler Using Ion-Pair Chromatography

    Article • Journal of Chromatographic Science, August 2017, Oxford University Press (OUP)

    Dr. Moataz Ahmed Shaldam

  33. Glyceryl trinitrate is a novel inhibitor of quorum sensing in <i>Pseudomonas aeruginosa</i>

    Article • African Health Sciences, March 2017, African Journals Online (AJOL)

    Dr. Moataz Ahmed Shaldam

  34. Synthesis, Evaluation of Pharmacological Activity, and Molecular Docking of 1,4-Dihydropyridines as Calcium Antagonists

    Article • Chemical and Pharmaceutical Bulletin, January 2016, Pharmaceutical Society of Japan

    Dr. Moataz Ahmed Shaldam

  35. Applying green analytical chemistry (GAC) for development of stability indicating HPLC method for determining clonazepam and its related substances in pharmaceutical formulations and calculating uncertainty

    Article • Arabian Journal of Chemistry, November 2014, Elsevier

    Dr. Moataz Ahmed Shaldam

  36. 1,4-Dihydropyridine Calcium Channel Blockers: Homology Modeling of the Receptor and Assessment of Structure Activity Relationship

    Article • ISRN Medicinal Chemistry, February 2014, Hindawi Publishing Corporation

    Dr. Moataz Ahmed Shaldam