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  1. β-Sitosterol vs. synthetic steroid in anticancer treatment.

    Article • Drug Development Research, March 2025, Wiley

    Dr Marisa Cabeza

  2. Current Understanding of Androgen Signaling in Prostatitis and its Treatment: A Review

    Article • Current Medicinal Chemistry, August 2024, Bentham Science Publishers

    Dr Marisa Cabeza

  3. Sex hormone dose escalation for treating abnormal sleep in ovariectomized rats: in vitro GABA synthesis in sleep-related brain areas

    Article • Canadian Journal of Physiology and Pharmacology, October 2023, Canadian Science Publishing

    Dr Marisa Cabeza

  4. Novel compounds with the potential to block prostate cell cancer growth

    Article • Oriental Journal Of Chemistry, June 2023, Oriental Scientific Publishing Company

    Dr Marisa Cabeza

  5. New Nonsteroidal Molecules as Blockers of the Steroidogenic Pathway

    Article • Current Enzyme Inhibition, March 2022, Bentham Science Publishers

    Dr Marisa Cabeza

  6. Synthesis of novel andostane-N-cyclohexyl-17-carboxamides, and their effect on the 5α-reductase isoform 2, the androgen receptor, and androgen-dependent glands

    Article • Pharmaceutical Sciences, November 2021, MaadRayan Publishing Company

    Dr Marisa Cabeza

  7. In vitro and In vivo Effects of 17β-N-(4-phenylcarbamoyl) androst-4-en-3- one Derivatives as 5a-reductase Inhibitors on Androgen-dependent Glands

    Article • Current Enzyme Inhibition, March 2021, Bentham Science Publishers

    Dr Marisa Cabeza

  8. Effect of Pregnenolone Derivatives on the Selective Inhibition of 5α-Reductase 2 Activity

    Article • Current Enzyme Inhibition, March 2020, Bentham Science Publishers

    Dr Marisa Cabeza

  9. Molecular Interactions of Different Steroids Contributing to Sebum Production. Review

    Article • Current Drug Targets, October 2018, Bentham Science Publishers

    Dr Marisa Cabeza

  10. Activity of steroid 4 and derivatives 4a–4f as inhibitors of the enzyme 5α-reductase 1

    Article • Bioorganic & Medicinal Chemistry, August 2018, Elsevier

    Dr Marisa Cabeza

  11. 17β-N-arylcarbamoylandrost-4-en-3-one Derivatives as Inhibitors of the Enzymes 3α-Hydroxysteroid Dehydrogenase and 5α-Reductase

    Article • Current Enzyme Inhibition, March 2018, Bentham Science Publishers

    Dr Marisa Cabeza

  12. Synthesis of new derivatives of 21-imidazolyl-16-dehydropregnenolone as inhibitors of 5α-reductase 2 and with cytotoxic activity in cancer cells

    Article • Bioorganic & Medicinal Chemistry, March 2017, Elsevier

    Dr Marisa Cabeza

  13. Synthesis of 17β-N-arylcarbamoylandrost-4-en-3-one derivatives and their anti-proliferative effect on human androgen-sensitive LNCaP cell line

    Article • European Journal of Medicinal Chemistry, October 2016, Elsevier

    Dr Marisa Cabeza

  14. New Dehydroepiandrosterone-triazole Derivatives Identified as Inhibitors of 17β.-Hydroxysteroid Dehydrogenase Enzyme in the Prostate

    Article • Current Enzyme Inhibition, July 2016, Bentham Science Publishers

    Dr Marisa Cabeza

  15. Recent Advances in Drug Design and Drug Discovery for Androgen- Dependent Diseases

    Article • Current Medicinal Chemistry, March 2016, Bentham Science Publishers

    Dr Marisa Cabeza

  16. Synthesis and activity of novel 16-dehydropregnenolone acetate derivatives as inhibitors of type 1 5α-reductase and on cancer cell line SK-LU-1

    Article • Bioorganic & Medicinal Chemistry, December 2015, Elsevier

    Dr Marisa Cabeza

  17. Synthesis and biological evaluation of esters of 16-formyl-17-methoxy-dehydroepiandrosterone derivatives as inhibitors of 5α-reductase type 2

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, November 2015, Taylor & Francis

    Dr Marisa Cabeza

  18. Novel dehydroepiandrosterone benzimidazolyl derivatives as 5α-reductase isozymes inhibitors

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, September 2015, Taylor & Francis

    Dr Marisa Cabeza

  19. Synthesis and Identification of Pregnenolone Derivatives as Inhibitors of Isozymes of 5α-Reductase

    Article • Archiv der Pharmazie, September 2015, Wiley

    Dr Marisa Cabeza

  20. Biological activity of pyrazole and imidazole-dehydroepiandrosterone derivatives on the activity of 17β-hydroxysteroid dehydrogenase

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, September 2015, Taylor & Francis

    Dr Marisa Cabeza

  21. Effect of new hybrids based on 5,16-pregnadiene scaffold linked to an anti-inflammatory drug on the growth of a human astrocytoma cell line (U373)

    Article • European Journal of Medicinal Chemistry, March 2015, Elsevier

    Dr Marisa Cabeza

  22. Effect of dehydroepiandrosterone derivatives on the activity of 5α-reductase isoenzymes and on cancer cell line PC-3

    Article • Bioorganic & Medicinal Chemistry, November 2014, Elsevier

    Dr Marisa Cabeza

  23. Bioactive withanolides from Withania obtusifolia

    Article • Phytochemistry Letters, September 2014, Elsevier

    Dr Marisa Cabeza

  24. Recent advances in structure of progestins and their binding to progesterone receptors

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, March 2014, Taylor & Francis

    Dr Marisa Cabeza

  25. Effect of Carbamates on mRNA Encoding Lipid Enzymes in Hamster Flank Organs

    Article • Archiv der Pharmazie, February 2014, Wiley

    Dr Marisa Cabeza

  26. Cytotoxic effect of novel dehydroepiandrosterone derivatives on different cancer cell lines

    Article • European Journal of Medicinal Chemistry, October 2013, Elsevier

    Dr Marisa Cabeza

  27. Biological Evaluation of Androstene Derivatives

    Article • Archiv der Pharmazie, December 2012, Wiley

    Dr Marisa Cabeza

  28. In vivoandin vitroeffect of androstene derivatives as 5α-reductase type 1 enzyme inhibitors

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, October 2012, Taylor & Francis

    Dr Marisa Cabeza

  29. Molecular interactions of natural and synthetic steroids in female hamsters’ flank organs

    Article • Journal of Dermatological Science, May 2012, Elsevier

    Dr Marisa Cabeza

  30. New ester derivatives of dehydroepiandrosterone as 5α-reductase inhibitors

    Article • Steroids, November 2011, Elsevier

    Dr Marisa Cabeza

  31. New steroidal lactones as 5α-reductase inhibitors and antagonists for the androgen receptor

    Article • The Journal of Steroid Biochemistry and Molecular Biology, November 2011, Elsevier

    Dr Marisa Cabeza

  32. Steroidal 5α-reductase inhibitors using 4-androstenedione as substrate

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, February 2011, Taylor & Francis

    Dr Marisa Cabeza

  33. Molecular interactions of progesterone derivatives with 5α-reductase types 1 and 2 and androgen receptors

    Article • Steroids, July 2010, Elsevier

    Dr Marisa Cabeza

  34. Crystal Structure and Synthesis of Three New Steroidal Derivatives as Antiandrogens

    Article • Journal of Chemical Crystallography, June 2010, Springer Science + Business Media

    Dr Marisa Cabeza

  35. Crystal Structure and Synthesis of 17α-Acetoxy-pregn-4,6-diene-3,20-dione

    Article • Journal of Chemical Crystallography, June 2010, Springer Science + Business Media

    Dr Marisa Cabeza

  36. Comparison Between Two Different Hamster Models used for the Determination of Testosterone and Finasteride Activity

    Article • Asian Journal of Animal and Veterinary Advances, April 2010, Science Alert

    Dr Marisa Cabeza

  37. New-D-homoandrost-4,6-diene derivatives as potent progesterone receptor antagonist

    Article • Steroids, January 2010, Elsevier

    Dr Marisa Cabeza

  38. Synthesis and biological activity of progesterone derivatives as 5α-reductase inhibitors, and their effect on hamster prostate weight

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, October 2009, Taylor & Francis

    Dr Marisa Cabeza

  39. Novel C-6 substituted and unsubstituted pregnane derivatives as 5α-reductase inhibitors and their effect on hamster flank organs diameter size

    Article • Steroids, October 2009, Elsevier

    Dr Marisa Cabeza

  40. Aromatic esters of progesterone as 5α-reductase and prostate growth inhibitors

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, June 2009, Taylor & Francis

    Dr Marisa Cabeza

  41. Biological activity of novel progesterone derivatives having a bulky ester side chains at C-3

    Article • Steroids, September 2008, Elsevier

    Dr Marisa Cabeza

  42. In vivo and in vitro effect of novel 4,16-pregnadiene-6,20-dione derivatives, as 5α-reductase inhibitors

    Article • The Journal of Steroid Biochemistry and Molecular Biology, September 2008, Elsevier

    Dr Marisa Cabeza

  43. Synthesis and biological effect of halogen substituted phenyl acetic acid derivatives of progesterone as potent progesterone receptor antagonists

    Article • The Journal of Steroid Biochemistry and Molecular Biology, September 2008, Elsevier

    Dr Marisa Cabeza

  44. Steroids with a carbamate function at C-17, a novel class of inhibitors for human and hamster steroid 5α-reductase

    Article • The Journal of Steroid Biochemistry and Molecular Biology, October 2007, Elsevier

    Dr Marisa Cabeza

  45. Antiandrogenic and apoptotic effects of RU-486 on animal prostate

    Article • The Journal of Steroid Biochemistry and Molecular Biology, May 2007, Elsevier

    Dr Marisa Cabeza

  46. New progesterone derivatives as inhibitors of 5α-reductase enzyme and prostate cancer cell growth

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, January 2006, Taylor & Francis

    Dr Marisa Cabeza

  47. Recent Advances in the Chemistry and Pharmacological Activity of New Steroidal Antiandrogens and 5α-Reductase Inhibitors

    Article • Current Medicinal Chemistry, April 2005, Bentham Science Publishers

    Dr Marisa Cabeza

  48. New 5?-reductase inhibitors: In vitro and in vivo effects

    Article • Steroids, March 2005, Elsevier

    Dr Marisa Cabeza

  49. Relative binding affinity of novel steroids to androgen receptors in hamster prostate

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, January 2005, Taylor & Francis

    Dr Marisa Cabeza

  50. Intracellular Ca2+ stimulates the binding to androgen receptors in platelets

    Article • Steroids, October 2004, Elsevier

    Dr Marisa Cabeza

  51. Steroid 5α-Reductase Inhibitors

    Article • Mini-Reviews in Medicinal Chemistry, May 2003, Bentham Science Publishers

    Dr Marisa Cabeza

  52. 5.ALPHA.-Reductase Inhibitory and Antiandrogenic Activities of Novel Steroids in Hamster Seminal Vesicles.

    Article • Chemical and Pharmaceutical Bulletin, January 2002, Pharmaceutical Society of Japan

    Dr Marisa Cabeza

  53. New Progesterone Esters as 5.ALPHA.-Reductase Inhibitors.

    Article • Chemical and Pharmaceutical Bulletin, January 2001, Pharmaceutical Society of Japan

    Dr Marisa Cabeza