All Stories

  1. Synthesis, characterization, and anticancer activity of Schiff bases

    Article • Journal of Biomolecular Structure and Dynamics, August 2019, Taylor & Francis

    Professor saqib - ali, Sumera Zaib, Professor Jamshed Iqbal, Noor Uddin

  2. Carbonic Anhydrase Inhibitory Potential of 1,2,4-triazole-3-thione Derivatives of Flurbiprofen, Ibuprofen and 4-tert-butylbenzoic Hydrazide: Design, Synthesis, Characterization, Biochemical Evaluation, Molecular Docking and Dynamic Simulation Studies

    Article • Medicinal Chemistry, April 2019, Bentham Science Publishers

    Professor saqib - ali, Shahid Hameed, Professor Jamshed Iqbal, Sumera Zaib

  3. Identification of New Chromenone Derivatives as Cholinesterase Inhibitors and Molecular Docking Studies

    Article • Medicinal Chemistry, November 2018, Bentham Science Publishers

    Professor Jamshed Iqbal, Sumera Zaib, Jürgen Bajorath

  4. Quinolinic Carboxylic Acid Derivatives as Potential Multi-target Compounds for Neurodegeneration: Monoamine Oxidase and Cholinesterase Inhibition

    Article • Medicinal Chemistry, January 2018, Bentham Science Publishers

    Professor Jamshed Iqbal, Shahid Hameed, Sumera Zaib

  5. Synthesis, Characterization and Cholinesterase Inhibition Studies of New Arylidene Aminothiazolylethanone Derivatives

    Article • Medicinal Chemistry, October 2017, Bentham Science Publishers

    Aamer Saeed, Professor Jamshed Iqbal

  6. Synthesis, Characterization and Biological Activities of Creatinine Amides and Creatinine Schiff Bases

    Article • Medicinal Chemistry, January 2017, Bentham Science Publishers

    Professor Jamshed Iqbal, Dr Amara AM Mumtaz

  7. Biological Evaluation of Azomethine-dihydroquinazolinone Conjugates as Cancer and Cholinesterase Inhibitors

    Article • Medicinal Chemistry, January 2016, Bentham Science Publishers

    Professor Jamshed Iqbal

  8. Quinolinyl-Thienyl Chalcones as Monoamine Oxidase Inhibitors and their In Silico Modeling Studies

    Article • Medicinal Chemistry, July 2015, Bentham Science Publishers

    Professor Jamshed Iqbal

  9. Biological Evaluation of Halogenated Thioureas as Cholinesterases Inhibitors Against Alzheimer’s Disease & Molecular Modeling Studies

    Article • Letters in Drug Design & Discovery, May 2015, Bentham Science Publishers

    Professor Jamshed Iqbal, Sumera Zaib

  10. Investigation of quinoline-4-carboxylic acid as a highly potent scaffold for the development of alkaline phosphatase inhibitors: synthesis, SAR analysis and molecular modelling studies

    Article • RSC Advances, January 2015, Royal Society of Chemistry

    Shahid Hameed, Professor Jamshed Iqbal

  11. Synthesis, characterization and biological evaluation of N-(2,3-dimethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazol-4-yl)benzamides

    Article • RSC Advances, January 2015, Royal Society of Chemistry

    Aamer Saeed, Professor Jamshed Iqbal

  12. Facile and expedient access to bis-coumarin–iminothiazole hybrids by molecular hybridization approach: synthesis, molecular modelling and assessment of alkaline phosphatase inhibition, anticancer and antileishmanial potential

    Article • RSC Advances, January 2015, Royal Society of Chemistry

    Professor Jamshed Iqbal, Aamer Saeed

  13. Influence of the diversified structural variations at the imine functionality of 4-bromophenylacetic acid derived hydrazones on alkaline phosphatase inhibition: synthesis and molecular modelling studies

    Article • RSC Advances, January 2015, Royal Society of Chemistry

    Shahid Hameed, Professor Jamshed Iqbal

  14. Synthesis of chitosan-coated polyoxometalate nanoparticles against cancer and its metastasis

    Article • RSC Advances, January 2015, Royal Society of Chemistry

    Professor Jamshed Iqbal

  15. Active compounds from a diverse library of triazolothiadiazole and triazolothiadiazine scaffolds: Synthesis, crystal structure determination, cytotoxicity, cholinesterase inhibitory activity, and binding mode analysis

    Article • Bioorganic & Medicinal Chemistry, November 2014, Elsevier

    Professor Jamshed Iqbal

  16. ChemInform Abstract: A Novel Example of Double 6-exo-trig Heterocyclization: Nitrile Conversion to New Anticancer Active (HeLa Cells) Primary Amine Ionic Liquids.

    Article • ChemInform, September 2014, Wiley

    Professor Jamshed Iqbal, Dr George E Kostakis

  17. 2‐(Hetero(aryl)methylene)hydrazine‐1‐carbothioamides as Potent Urease Inhibitors

    Article • Chemical Biology & Drug Design, July 2014, Wiley

    Professor Jamshed Iqbal

  18. RutheniumII(η6-arene) Complexes of Thiourea Derivatives: Synthesis, Characterization and Urease Inhibition

    Article • Molecules, June 2014, MDPI AG

    Professor Jamshed Iqbal, Dr Muhammad Hanif

  19. A Facile One‐Pot Synthesis of 2‐Arylamino‐5‐Aryloxylalkyl‐1,3,4‐Oxadiazoles and Their Urease Inhibition Studies

    Article • Chemical Biology & Drug Design, June 2014, Wiley

    Professor Jamshed Iqbal

  20. New aminobenzenesulfonamide–thiourea conjugates: Synthesis and carbonic anhydrase inhibition and docking studies

    Article • European Journal of Medicinal Chemistry, May 2014, Elsevier

    Professor Jamshed Iqbal

  21. Novel structural hybrids of pyrazolobenzothiazines with benzimidazoles as cholinesterase inhibitors

    Article • European Journal of Medicinal Chemistry, May 2014, Elsevier

    Professor Jamshed Iqbal

  22. Synthesis, crystal structure and biological evaluation of some novel 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazoles and 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazines

    Article • European Journal of Medicinal Chemistry, May 2014, Elsevier

    Professor Jamshed Iqbal

  23. Synthesis, cytotoxicity and molecular modelling studies of new phenylcinnamide derivatives as potent inhibitors of cholinesterases

    Article • European Journal of Medicinal Chemistry, May 2014, Elsevier

    Professor Jamshed Iqbal

  24. ChemInform Abstract: Solution‐Phase Microwave Assisted Parallel Synthesis of N,N′‐Disubstituted Thioureas Derived from Benzoic Acid: Biological Evaluation and Molecular Docking Studies.

    Article • ChemInform, April 2014, Wiley

    Professor Jamshed Iqbal, Dr Imtiaz-ud-Din - Din

  25. Carbonic anhydrase inhibition by 1-aroyl-3-(4-aminosulfonylphenyl)thioureas

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, March 2014, Taylor & Francis

    Professor Jamshed Iqbal

  26. Design, synthesis, molecular docking studies and in vitro screening of ethyl 4-(3-benzoylthioureido) benzoates as urease inhibitors

    Article • Bioorganic Chemistry, February 2014, Elsevier

    Professor Jamshed Iqbal

  27. A novel example of double 6-exo-trig heterocyclization: nitrile conversion to new anticancer active (HeLa cells) primary amine ionic liquids

    Article • Chemical Communications, January 2014, Royal Society of Chemistry

    Professor Annie Powell, Professor Jamshed Iqbal, Dr George E Kostakis

  28. Synthesis and antiproliferative activity of (Z)-1-glycosyl-3-(5-oxo-2-thioxoimidazolidin-4-ylidene)indolin-2-ones and (Z)-3-(2-glycosylsulfanyl-4-oxo-4,5-dihydro-thiazol-5-ylidene)indolin-2-ones

    Article • RSC Advances, January 2014, Royal Society of Chemistry

    Professor Jamshed Iqbal

  29. Synthesis and antiproliferative activity of N-glycosyl-3,3-diaryloxindoles

    Article • RSC Advances, January 2014, Royal Society of Chemistry

    Professor Jamshed Iqbal

  30. Antidiabetic potential of polyoxotungstates: in vitro and in vivo studies

    Article • Metallomics, January 2014, Oxford University Press (OUP)

    Professor Jamshed Iqbal

  31. Benzothiazolyl substituted iminothiazolidinones and benzamido-oxothiazolidines as potent and partly selective aldose reductase inhibitors

    Article • MedChemComm, January 2014, Royal Society of Chemistry

    Professor Jamshed Iqbal

  32. A capillary electrophoresis-based enzyme assay for kinetics and inhibition studies of carbonic anhydrase

    Article • Analytical Biochemistry, January 2014, Elsevier

    Professor Jamshed Iqbal

  33. Sulfa Drugs as Inhibitors of Carbonic Anhydrase: New Targets for the Old Drugs

    Article • BioMed Research International, January 2014, Hindawi Publishing Corporation

    Professor Jamshed Iqbal

  34. Cytotoxicity and enzyme inhibition studies of polyoxometalates and their chitosan nanoassemblies

    Article • Toxicology Reports, January 2014, Elsevier

    Professor Jamshed Iqbal

  35. Solution-phase microwave assisted parallel synthesis of N,N′-disubstituted thioureas derived from benzoic acid: Biological evaluation and molecular docking studies

    Article • European Journal of Medicinal Chemistry, December 2013, Elsevier

    Professor Jamshed Iqbal, Dr Imtiaz-ud-Din - Din

  36. Identification of sulfonic acids as efficient ecto-5′-nucleotidase inhibitors

    Article • European Journal of Medicinal Chemistry, December 2013, Elsevier

    Professor Jamshed Iqbal

  37. Development of a fast and efficient CE enzyme assay for the characterization and inhibition studies of α-glucosidase inhibitors

    Article • Journal of Separation Science, September 2013, Wiley

    Professor Jamshed Iqbal

  38. Therapeutic Potentials of Ecto‐Nucleoside Triphosphate Diphosphohydrolase, Ecto‐Nucleotide Pyrophosphatase/Phosphodiesterase, Ecto‐5′‐Nucleotidase, and Alkaline Phosphatase Inhibitors

    Article • Medicinal Research Reviews, September 2013, Wiley

    Professor Jamshed Iqbal

  39. Synthesis of BODIPY Derivatives Substituted with Various Bioconjugatable Linker Groups: A Construction Kit for Fluorescent Labeling of Receptor Ligands

    Article • Journal of Fluorescence, September 2013, Springer Science + Business Media

    Professor Jamshed Iqbal

  40. Identification of novel chromone based sulfonamides as highly potent and selective inhibitors of alkaline phosphatases

    Article • European Journal of Medicinal Chemistry, August 2013, Elsevier

    Professor Jamshed Iqbal, Dr George E Kostakis

  41. ChemInform Abstract: Synthesis of Functionalized Benzothiophenes and Dibenzothiophenes by Twofold Heck and Subsequent 6π‐Electrocyclization Reactions of 2,3‐Dibromothiophenes and 2,3‐Dibromobenzothiophenes.

    Article • ChemInform, June 2013, Wiley

    Professor Jamshed Iqbal

  42. ChemInform Abstract: Synthesis of 2,6‐Diaryl‐3‐(trifluoromethyl)pyridines by Regioselective Suzuki—Miyaura Reactions of 2,6‐Dichloro‐3‐(trifluoromethyl)pyridine.

    Article • ChemInform, June 2013, Wiley

    Professor Jamshed Iqbal

  43. ChemInform Abstract: Synthesis and Photophysical Properties of Tetra‐ and Pentaalkynylfluorobenzenes by Sonogashira Reactions of Novel Iodofluorobenzenes.

    Article • ChemInform, June 2013, Wiley

    Professor Jamshed Iqbal

  44. ChemInform Abstract: Synthesis of Functionalized Fluorinated Terphenyls by Site‐Selective Suzuki—Miyaura Cross‐Coupling Reactions of Dibrominated Fluorobenzenes.

    Article • ChemInform, June 2013, Wiley

    Professor Jamshed Iqbal

  45. ChemInform Abstract: Pyrrole versus Quinoline Formation in the Palladium Catalyzed Reaction of 2‐Alkynyl‐3‐bromothiophenes and 2‐Alkynyl‐3‐bromofurans with Anilines. A Combined Experimental and Computational Study.

    Article • ChemInform, May 2013, Wiley

    Professor Jamshed Iqbal

  46. Synthesis of 2,6-diaryl-3-(trifluoromethyl)pyridines by regioselective Suzuki–Miyaura reactions of 2,6-dichloro-3-(trifluoromethyl)pyridine

    Article • Tetrahedron Letters, March 2013, Elsevier

    Professor Jamshed Iqbal

  47. Synthesis of functionalized fluorinated terphenyls by site-selective Suzuki–Miyaura cross-coupling reactions of dibrominated fluorobenzenes

    Article • Journal of Fluorine Chemistry, February 2013, Elsevier

    Professor Jamshed Iqbal

  48. Advances in immobilized enzyme microbioreactors in capillary electrophoresis

    Article • The Analyst, January 2013, Royal Society of Chemistry

    Professor Jamshed Iqbal

  49. Synthesis and antiproliferative activity of selenoindirubins and selenoindirubin-N-glycosides

    Article • Organic & Biomolecular Chemistry, January 2013, Royal Society of Chemistry

    Professor Jamshed Iqbal

  50. Synthesis of N,N′-diglycosylated isoindigos

    Article • Organic & Biomolecular Chemistry, January 2013, Royal Society of Chemistry

    Professor Jamshed Iqbal

  51. Synthesis, crystal structure, enzyme inhibition, DNA protection, and antimicrobial studies of di- and triorganotin(IV) derivatives of 2-thiopheneacetic acid

    Article • Journal of Coordination Chemistry, January 2013, Taylor & Francis

    Professor Jamshed Iqbal

  52. Synthesis and photophysical properties of tetra- and pentaalkynylfluorobenzenes by Sonogashira reactions of novel iodofluorobenzenes

    Article • Tetrahedron, January 2013, Elsevier

    Professor Jamshed Iqbal

  53. Dual action spirobicycloimidazolidine-2,4-diones: Antidiabetic agents and inhibitors of aldose reductase-an enzyme involved in diabetic complications

    Article • Bioorganic & Medicinal Chemistry Letters, January 2013, Elsevier

    Professor Jamshed Iqbal

  54. Synthesis of functionalized benzothiophenes and dibenzothiophenes by twofold Heck and subsequent 6π-electrocyclization reactions of 2,3-dibromothiophenes and 2,3-dibromobenzothiophenes

    Article • Tetrahedron, January 2013, Elsevier

    Professor Jamshed Iqbal

  55. Structural, enzyme inhibition, antibacterial and DNA protection studies of organotin(IV) derivatives of thiophene-2-carboxylic acid

    Article • Journal of Organometallic Chemistry, January 2013, Elsevier

    Professor Jamshed Iqbal, Professor saqib - ali

  56. Synthesis of trifluoromethyl-substituted bi- and terphenyls by site-selective Suzuki–Miyaura reactions of various dihalogenated trifluoromethyl-benzene derivatives

    Article • Journal of Fluorine Chemistry, January 2013, Elsevier

    Professor Jamshed Iqbal

  57. Synthesis, molecular docking studies, and in vitro screening of sulfanilamide-thiourea hybrids as antimicrobial and urease inhibitors

    Article • Medicinal Chemistry Research, November 2012, Springer Science + Business Media

    Professor Jamshed Iqbal

  58. Identification of Small Molecule Sulfonic Acids as Ecto-5'-Nucleotidase Inhibitors

    Article • Medicinal Chemistry, November 2012, Bentham Science Publishers

    Professor Jamshed Iqbal

  59. Identification of Small Molecule Sulfonic Acids as Ecto-5'-Nucleotidase Inhibitors

    Article • Medicinal Chemistry, September 2012, Bentham Science Publishers

    Professor Jamshed Iqbal

  60. Pharmacological Evaluation and Docking Studies of 3-Thiadiazolyl- and Thioxo-1,2,4-triazolylcoumarin Derivatives as Cholinesterase Inhibitors

    Article • ISRN Pharmacology, August 2012, Hindawi Publishing Corporation

    Professor Jamshed Iqbal

  61. Synthesis, Urease Inhibition, Antioxidant, Antibacterial, and Molecular Docking Studies of 1,3,4-Oxadiazole Derivatives

    Article • ISRN Pharmacology, August 2012, Hindawi Publishing Corporation

    Professor Jamshed Iqbal

  62. Synthesis and Biological Evaluation of 3‐thiazolocoumarinyl Schiff‐base Derivatives as Cholinesterase Inhibitors

    Article • Chemical Biology & Drug Design, July 2012, Wiley

    Professor Jamshed Iqbal

  63. Antioxidant, Antimicrobial, and Free Radical Scavenging Potential of Aerial Parts of Periploca aphylla and Ricinus communis

    Article • ISRN Pharmacology, July 2012, Hindawi Publishing Corporation

    Professor Jamshed Iqbal

  64. Polyoxometalates as potent inhibitors for acetyl and butyrylcholinesterases and as potential drugs for the treatment of Alzheimer’s disease

    Article • Medicinal Chemistry Research, June 2012, Springer Science + Business Media

    Professor Jamshed Iqbal

  65. Synthesis, urease inhibition, antioxidant and antibacterial studies of some 4-amino-5-aryl-3H-1,2,4-triazole-3-thiones and their 3,6-disubstituted 1,2,4-triazolo[3,4-b]1,3,4-thiadiazole derivatives

    Article • Journal of the Brazilian Chemical Society, May 2012, FapUNIFESP (SciELO)

    Professor Jamshed Iqbal

  66. Benzothiazinones: A Novel Class of Adenosine Receptor Antagonists Structurally Unrelated to Xanthine and Adenine Derivatives

    Article • Journal of Medicinal Chemistry, March 2012, American Chemical Society (ACS)

    Professor Jamshed Iqbal

  67. Polyoxometalates as potent and selective inhibitors of alkaline phosphatases with profound anticancer and amoebicidal activities

    Article • Dalton Transactions, January 2012, Royal Society of Chemistry

    Professor Jamshed Iqbal

  68. Design, synthesis and molecular modelling of novel methyl[4-oxo-2-(aroylimino)-3-(substituted phenyl)thiazolidin-5-ylidene]acetates as potent and selective aldose reductase inhibitors

    Article • MedChemComm, January 2012, Royal Society of Chemistry

    Professor Jamshed Iqbal

  69. Pyrrole versus quinoline formation in the palladium catalyzed reaction of 2-alkynyl-3-bromothiophenes and 2-alkynyl-3-bromofurans with anilines. A combined experimental and computational study

    Article • Organic & Biomolecular Chemistry, January 2012, Royal Society of Chemistry

    Professor Jamshed Iqbal

  70. Synthesis, Acetylcholinesterase and Alkaline Phosphatase Inhibition of Some New 1,2,4-Triazole and 1,3,4-Thiadiazole Derivatives

    Article • Australian Journal of Chemistry, January 2012, CSIRO Publishing

    Professor Jamshed Iqbal

  71. Synthesis, biological assay in vitro and molecular docking studies of new Schiff base derivatives as potential urease inhibitors

    Article • European Journal of Medicinal Chemistry, November 2011, Elsevier

    Professor Jamshed Iqbal

  72. Identification of Potent and Selective Human Ecto-Nucleotide Pyrophosphatase/ Phosphodiesterase-3 (hNPP3) Inhibitors

    Article • The Open Enzyme Inhibition Journal, October 2011, Bentham Science Publishers

    Professor Jamshed Iqbal

  73. An enzyme immobilized microassay in capillary electrophoresis for characterization and inhibition studies of alkaline phosphatases

    Article • Analytical Biochemistry, July 2011, Elsevier

    Professor Jamshed Iqbal

  74. High-sensitivity capillary electrophoresis method for monitoring purine nucleoside phosphorylase and adenosine deaminase reactions by a reversed electrode polarity switching mode

    Article • Journal of Chromatography A, July 2011, Elsevier

    Professor Jamshed Iqbal

  75. Development of Potent and Selective Inhibitors of ecto-5′-Nucleotidase Based on an Anthraquinone Scaffold

    Article • Journal of Medicinal Chemistry, February 2010, American Chemical Society (ACS)

    Professor Jamshed Iqbal

  76. Development of a microbioreactor with ecto-nucleoside triphosphate diphosphohydrolase 2 (NTPDase2) immobilized on a polyacrylamide-coated capillary at the outlet

    Article • Journal of Chromatography A, January 2010, Elsevier

    Professor Jamshed Iqbal

  77. Nucleoside-5′-monophosphates as Prodrugs of Adenosine A2A Receptor Agonists Activated by ecto-5′-Nucleotidase†Contribution to celebrate the 100th anniversary of the Division of Medicinal Chemistry of the American Chemical Society.

    Article • Journal of Medicinal Chemistry, July 2009, American Chemical Society (ACS)

    Professor Jamshed Iqbal

  78. Tether tracking and control of ROSA robotic rover

    Article • December 2008, Institute of Electrical & Electronics Engineers (IEEE)

    Professor Jamshed Iqbal

  79. A highly sensitive CE‐UV method with dynamic coating of silica‐fused capillaries for monitoring of nucleotide pyrophosphatase/phosphodiesterase reactions

    Article • Electrophoresis, August 2008, Wiley

    Professor Jamshed Iqbal

  80. Selective Nucleoside Triphosphate Diphosphohydrolase-2 (NTPDase2) Inhibitors: Nucleotide Mimetics Derived from Uridine-5′-carboxamide

    Article • Journal of Medicinal Chemistry, July 2008, American Chemical Society (ACS)

    Professor Jamshed Iqbal

  81. Structure-activity relationships of anthraquinone derivatives derived from bromaminic acid as inhibitors of ectonucleoside triphosphate diphosphohydrolases (E-NTPDases)

    Article • Purinergic Signalling, June 2008, Springer Science + Business Media

    Professor Jamshed Iqbal

  82. Capillary electrophoresis-based nanoscale assays for monitoring ecto-5′-nucleotidase activity and inhibition in preparations of recombinant enzyme and melanoma cell membranes

    Article • Analytical Biochemistry, February 2008, Elsevier

    Professor Jamshed Iqbal

  83. Polyoxometalates—a new class of potent ecto-nucleoside triphosphate diphosphohydrolase (NTPDase) inhibitors

    Article • Bioorganic & Medicinal Chemistry Letters, December 2006, Elsevier

    Professor Jamshed Iqbal

  84. Characterization of human and rodent native and recombinant adenosine A2B receptors by radioligand binding studies

    Article • Purinergic Signalling, July 2006, Springer Science + Business Media

    Professor Jamshed Iqbal

  85. Development of off‐line and on‐line capillary electrophoresis methods for the screening and characterization of adenosine kinase inhibitors and substrates

    Article • Electrophoresis, June 2006, Wiley

    Professor Jamshed Iqbal

  86. A capillary electrophoresis method for the characterization of ecto-nucleoside triphosphate diphosphohydrolases (NTPDases) and the analysis of inhibitors by in-capillary enzymatic microreaction

    Article • Purinergic Signalling, December 2005, Springer Science + Business Media

    Professor Jamshed Iqbal

  87. Novel Amino Acid Derived Natural Products from the Ascidian Atriolum robustum: Identification and Pharmacological Characterization of a Unique Adenosine Derivative (IIIa).

    Article • ChemInform, August 2004, Wiley

    Professor Jamshed Iqbal

  88. Novel Amino Acid Derived Natural Products from the Ascidian Atriolum robustum:  Identification and Pharmacological Characterization of a Unique Adenosine Derivative

    Article • Journal of Medicinal Chemistry, March 2004, American Chemical Society (ACS)

    Professor Jamshed Iqbal