All Stories

  1. 2-Substituted-mercapto-quinazolin-4(3H)-ones as DHFR Inhibitors
  2. Synthesis, biological evaluation and molecular modeling study of 2-(1,3,4-thiadiazolyl-thio and 4-methyl-thiazolyl-thio)-quinazolin-4-ones as a new class of DHFR inhibitors
  3. Nonclassical antifolates, part 5. Benzodiazepine analogs as a new class of DHFR inhibitors: Synthesis, antitumor testing and molecular modeling study
  4. Nonclassical antifolates, part 4. 5-(2-Aminothiazol-4-yl)-4-phenyl-4H-1,2,4-triazole-3-thiols as a new class of DHFR inhibitors: Synthesis, biological evaluation and molecular modeling study
  5. Nonclassical antifolates, part 3: Synthesis, biological evaluation and molecular modeling study of some new 2-heteroarylthio-quinazolin-4-ones
  6. Novel 4(3H)-quinazolinone analogs: synthesis and anticonvulsant activity
  7. Substituted thiazoles VII. Synthesis and antitumor activity of certain 2-(substituted amino)-4-phenyl-1,3-thiazole analogs
  8. Substituted thiazoles VI. Synthesis and antitumor activity of new 2-acetamido- and 2 or 3-propanamido-thiazole analogs
  9. ChemInform Abstract: Design, Synthesis, Single-Crystal and Preliminary Antitumor Activity of Novel Arenesulfonylimidazolidin-2-ones.
  10. ChemInform Abstract: Novel 1,3,4-Heterodiazole Analogues: Synthesis and in vitro Antitumor Activity.
  11. 1-(5-Bromo-4-phenyl-1,3-thiazol-2-yl)pyrrolidin-2-one
  12. N-[4-(4-Bromophenyl)thiazol-2-yl]-4-(piperidin-1-yl)butanamide
  13. S-Phenyl 4-methoxybenzothioate
  14. Design, synthesis, single-crystal and preliminary antitumor activity of novel arenesulfonylimidazolidin-2-ones
  15. ChemInform Abstract: Synthesis and Anticonvulsant Activity of Some New Thiazolo[3,2-a][1,3]diazepine, Benzo[d]thiazolo[5,2-a][12,6]diazepine and Benzo[d]oxazolo[5,2-a][12,6]diazepine Analogues.
  16. 3-Benzyl-6-methyl-2-sulfanylidene-2,3-dihydroquinazolin-4(1H)-one
  17. Novel 1,3,4-heterodiazole analogues: Synthesis and in-vitro antitumor activity
  18. Substituted thiazoles V. Synthesis and antitumor activity of novel thiazolo[2,3-b]quinazoline and pyrido[4,3-d]thiazolo[3,2-a]pyrimidine analogues
  19. Synthesis, Antitumor and Antitubercular Evaluation of Certain New Xanthenone and Acridinone Analogs
  20. Synthesis and anticonvulsant activity of some new thiazolo[3,2-a][1,3]diazepine, benzo[d]thiazolo[5,2-a][12,6]diazepine and benzo[d]oxazolo[5,2-a][12,6]diazepine analogues
  21. Chiral Indolo[3,2-f][3]benzazecine-Type Dopamine Receptor Antagonists: Synthesis and Activity of Racemic and Enantiopure Derivatives
  22. Synthesis and biological evaluation of some novel cyclic-imides as hypoglycaemic, anti-hyperlipidemic agents
  23. Liquid chromatographic high-throughput analysis of the new ultra-short acting hypnotic ‘HIE-124’ and its metabolite in mice serum using a monolithic silica column
  24. Synthesis, antiplatelet aggregation activity, and molecular modeling study of novel substituted-piperazine analogues
  25. ChemInform Abstract: Fused Pyrimidines. Synthesis of Pyrazolo(3,4-e)(1,3,4)thiadiazolo(3,2- a)pyrimidine and Pyrazolo(4′,3′:5,6)pyrimido(2,1-b)benzothiazole Derivatives.
  26. ChemInform Abstract: 1′,2′-Secothymidines. The Preparation of 2,3′-Anhydro Derivatives and the Formation of Two Unusual Dimeric Products.
  27. ChemInform Abstract: A Facile Synthesis of β- and γ-Hydroxy Phosphonate Esters from Epoxides.
  28. ChemInform Abstract: A General and Facile Synthesis of β- and γ-Hydroxy Phosphonates from Epoxides.
  29. ChemInform Abstract: Synthesis and Biological Testing of 2,4-Disubstituted Thiazole Derivatives as Potential Antitumor Antibiotics.
  30. ChemInform Abstract: Synthesis, Antimicrobial and Antiviral Evaluation of Certain Thienopyrimidine Derivatives.
  31. ChemInform Abstract: Synthesis and Anticonvulsant Activity of Some 1-Substituted-2- oxopyrrolidine Derivatives.
  32. ChemInform Abstract: Synthesis of Phosphonate Isosteres of 2′-Deoxy-1′,2′-seco-nucleotides.
  33. ChemInform Abstract: 2,4-Disubstituted Thiazoles. Part 2. A Novel Class of Antitumor Agents, Synthesis and Biological Evaluation.
  34. Novel, selective sample stacking microemulsion electrokinetic capillary chromatography induced by reverse migrating pseudostationary phase for the determination of the new ultra-short acting hypnotic “HIE-124” in mice serum
  35. ChemInform Abstract: Synthesis and Antitumor Activity of 9-Anilino, Phenylhydrazino, and Sulfonamido Analogues of 2- or 4-Methoxy-6-nitroacridines.
  36. ChemInform Abstract: Synthesis and Biological Evaluation of New Cyclopenteno[b]thiophene Derivatives as Local Anesthetic and Antiarrhythmic Agents.
  37. ChemInform Abstract: Synthesis, Antitumor and Antitubercular Evaluation of Certain New Xanthenone and Acridinone Analogues.
  38. ChemInform Abstract: Synthesis and Antitumor Activity of Some New Substituted Quinolin-4-one and 1,7-Naphthyridin-4-one Analogues.
  39. ChemInform Abstract: 2,4-Disubstituted Thiazoles. Part 3. Synthesis and Antitumor Activity of Ethyl 2-Substituted-aminothiazole-4-carboxylate Analogues.
  40. ChemInform Abstract: Synthesis and Antitumor Activity of Certain New Substituted 1H-Isoindoledione Derivatives.
  41. ChemInform Abstract: Substituted Quinazolines. Part 1. Synthesis and Antitumor Activity of Certain Substituted 2-Mercapto-4(3H)-quinazolinone Analogues.
  42. Non-classical antifolates. Part 2: Synthesis, biological evaluation, and molecular modeling study of some new 2,6-substituted-quinazolin-4-ones
  43. ChemInform Abstract: Synthesis and Biological Evaluation of Some Polymethoxylated Fused Pyridine Ring Systems as Antitumor Agents.
  44. Synthesis and Biological Evaluation of Some Polymethoxylated Fused Pyridine Ring Systems as Antitumor Agents
  45. ChemInform Abstract: Substituted Quinazolines. Part 3. Synthesis, in vitro Antitumor Activity and Molecular Modeling Study of Certain 2-Thieno-4(3H)-quinazolinone Analogues.
  46. HPTLC analysis of a new ultra-short-acting thiazolodiazepine hypnotic (HIE-124) in spiked human plasma
  47. Substituted quinazolines, part 3. Synthesis, in vitro antitumor activity and molecular modeling study of certain 2-thieno-4(3H)-quinazolinone analogs☆
  48. Cytarabine
  49. Itraconazole: Comprehensive Profile
  50. ChemInform Abstract: New Ultra-Short Acting Hypnotic: Synthesis, Biological Evaluation, and Metabolic Profile of Ethyl 8-Oxo-5,6,7,8-tetrahydro-thiazolo[3,2-a][1,3]diazepin-3-carboxylate (HIE-124).
  51. Oral colon targeted delivery systems for treatment of inflammatory bowel diseases: Synthesis, in vitro and in vivo assessment
  52. ChemInform Abstract: Synthesis, Ultra-Short Acting Hypnotic Activity, and Metabolic Profile of Ethyl 8-Oxo-5,6,7,8-tetrahydro-thiazolo[3,2-a][1,3]diazepin-3-carboxylate (HIE-124).
  53. Synthesis, Ultra-Short Acting Hypnotic Activity, and Metabolic Profile of Ethyl 8-Oxo-5,6,7,8-tetrahydro-thiazolo[3,2-a] [1,3]diazepin-3-carboxylate (HIE-124)
  54. New ultra-short acting hypnotic: Synthesis, biological evaluation, and metabolic profile of ethyl 8-oxo-5,6,7,8-tetrahydro-thiazolo[3,2-a][1,3]diazepin-3-carboxylate (HIE-124)
  55. Synthesis, dihydrofolate reductase inhibition, antitumor testing, and molecular modeling study of some new 4(3H)-quinazolinone analogs
  56. Dopamine/Serotonin Receptor Ligands. 10: SAR Studies on Azecine-type Dopamine Receptor Ligands by Functional Screening at Human Cloned D1, D2L, and D5 Receptors with a Microplate Reader Based Calcium Assay Lead to a Nov...
  57. Synthesis and in vitro Antioxidant Activity of Some New Fused Pyridine Analogues.
  58. Lewis acid-promoted transformation of 2-alkoxypyridines into 2-aminopyridines and their antibacterial activity. Part 2: Remarkably facile C–N bond formation
  59. Synthesis andIn Vitro Antioxidant Activity of some New Fused Pyridine Analogs
  60. Interaction of 2-thio-4-oxo-quinazoline Derivatives with Guinea Pig Liver Molybdenum Hydroxylases, Xanthine Oxidase and Aldehyde Oxidase
  61. Penicillamine: Physical Profile
  62. Synthesis,in vitro andin vivo Evaluation of a Delivery System for Targeting Anticancer Drugs to the Brain
  63. Substituted Quinazolines. Part 2. Synthesis and in-vitro Anticancer Evaluation of New 2-Substituted Mercapto-3H-quinazoline Analogues.
  64. Dopamine/Serotonin Receptor Ligands. Part 4. Synthesis and Pharmacology of Novel 3-Benzazecines and 3-Benzazonines as Potential 5-HT2A and Dopamine Receptor Ligands.
  65. Substituted Quinazolines, Part 2. Synthesis and In-Vitro Anticancer Evaluation of New 2-Substituted Mercapto-3H-quinazoline Analogs
  66. Dopamine/Serotonin Receptor Ligands. Part IV [1]: Synthesis and Pharmacology of Novel 3-Benzazecines and 3-Benzazonines as Potential 5-HT2A and Dopamine Receptor Ligands
  67. The in vitro antitumor assay of 5-(Z)-arylidene-4-imidazolidinones in screens of AIDS-related leukemia and lymphomas
  68. Histamine
  69. Lansoprazole
  70. Synthesis and Biological Evaluation of Certain α,β-Unsaturated Ketones and Their Corresponding Fused Pyridines as Antiviral and Cytotoxic Agents
  71. Synthesis and Antitumor Activity of Ethyl 2-Substituted-aminothiazole-4-carboxylate Analogs
  72. Synthesis and Antitumor Activity of Ethyl 2-Substituted-aminothiazole-4-carboxylate Analogs
  73. Isoxsuprine Hydrochloride
  74. SYNTHESIS, CONFORMATIONAL ANALYSIS AND ANTITUMOR TESTING OF 5-(Z)-ARYLIDENE-4-IMIDAZOLIDINONE DERIVATIVES
  75. Praziquantel
  76. Synthesis and Antitumor Activity of 9‐Anilino, Phenylhydrazino, and Sulphonamido Analogs of 2‐ or 4‐Methoxy‐6‐nitroacridines
  77. 5-Substituted-2-thiohydantoin analogs as a novel class of antitumor agents
  78. Synthesis of Phosphonate Isosteres of 2‘-Deoxy-1‘,2‘-seco-nucleotides
  79. 2,4-Disubstituted thiazoles II. A novel class of antitumor agents, synthesis and biological evaluation
  80. Synthesis and Biological Evaluation of 1‘,2‘-Seconucleo-5‘-phosphonates
  81. Synthesis, antimicrobial and antiviral evaluation of certain thienopyrimidine derivatives
  82. A general and facile synthesis of .beta.- and .gamma.-hydroxy phosphonates from epoxides
  83. A facile synthesis of β- and γ- hydroxyphosphonate esters from epoxides
  84. A Stereospecific Synthesis of Pyrimidine β-D-2′-Deoxyribonucleosides
  85. Synthesis of 1′,2′-Seco-nucleoside Analogues of AZT
  86. Spectrophotometric Determination of Isoniazid Using Ethyl 8-Quinolinoxy Acetate
  87. 1',2'-Secothymidines. The preparation of 2,3'-anhydro derivatives and the formation of two unusual dimeric products
  88. Thienobenzothiopyranones III new 4H-thieno[2,3-b][1]benzothiopyran-4-ones carrying different heterocyclic moieties of expected pharmacological interest
  89. Synthesis of substituted 4H-thieno[2,3-b][1]benzothiopyran-4-ones as possible schistosomicidal agents
  90. Triazoles and fused triazoles, III: Facile and efficient synthesis of 2,5-disubstituted-s-triazolo[3,4-b]-1,3,4-thiadiazoles
  91. Errata
  92. Synthesis of substituted 4H-thiazolo[4,5-b][1]benzothiopyran-4-ones as possible schistosomicidal agents
  93. Synthesis of certain substituted pyrimidines as potential schistosomicidal agents
  94. Synthesis of 2-substituted 4H-thieno[2,3-b][1]benzothiopyran-4-ones as potential chemotherapeutic agents
  95. Synthesis of substituted arylazothioxanthones as potential schistosomicidal agents
  96. Synthesis of certain thiaxanthones as potential schistosomicidal agents