All Stories

  1. Carbazole Derivatives as Kinase-Targeting Inhibitors for Cancer Treatment

    Article • Mini-Reviews in Medicinal Chemistry, May 2020, Bentham Science Publishers

    Fedora Grande, Pasquale Longo

  2. The Peptide ERα17p Is a GPER Inverse Agonist that Exerts Antiproliferative Effects in Breast Cancer Cells

    Article • Cells, June 2019, MDPI AG

    Fedora Grande

  3. Cryptotanshinone and tanshinone IIA from Salvia milthorrhiza Bunge (Danshen) as a new class of potential pancreatic lipase inhibitors

    Article • Natural Product Research, May 2019, Taylor & Francis

    Fedora Grande

  4. Reverse Transcriptase Inhibitors Nanosystems Designed for Drug Stability and Controlled Delivery

    Article • Pharmaceutics, April 2019, MDPI AG

    Fedora Grande

  5. CCR5/CXCR4 Dual Antagonism for the Improvement of HIV Infection Therapy

    Article • Molecules, February 2019, MDPI AG

    Fedora Grande

  6. A New Generation of Dihydropyridine Calcium Channel Blockers: Photostabilization of Liquid Formulations Using Nonionic Surfactants

    Article • Pharmaceutics, January 2019, MDPI AG

    Fedora Grande

  7. A pilot study on the nutraceutical properties of the Citrus hybrid Tacle® as a dietary source of polyphenols for supplementation in metabolic disorders

    Article • Journal of Functional Foods, January 2019, Elsevier

    Fedora Grande

  8. Benzopyrroloxazines containing a bridgehead nitrogen atom as promising scaffolds for the achievement of biologically active agents

    Article • European Journal of Medicinal Chemistry, May 2018, Elsevier

    Fedora Grande

  9. Identification by Molecular Docking ofHomoisoflavones from Leopoldia comosa as Ligands of Estrogen Receptors

    Article • Molecules, April 2018, MDPI AG

    Fedora Grande

  10. Chloro-1,4-dimethyl-9H-carbazole Derivatives Displaying Anti-HIV Activity

    Article • Molecules, January 2018, MDPI AG

    Fedora Grande

  11. New insights for the use of quercetin analogs in cancer treatment

    Article • Future Medicinal Chemistry, October 2017, Future Science

    Fedora Grande

  12. An update on small molecules targeting CXCR4 as starting points for the development of anti-cancer therapeutics

    Article • European Journal of Medicinal Chemistry, October 2017, Elsevier

    Fedora Grande

  13. Liquid crystalline microspheres for 5-fluorouracil specific release

    Article • Journal of Drug Delivery Science and Technology, October 2017, Elsevier

    Fedora Grande

  14. Identification of novel 2-(1H-indol-1-yl)-benzohydrazides CXCR4 ligands impairing breast cancer growth and motility

    Article • Future Medicinal Chemistry, February 2016, Future Science

    Fedora Grande, PhD Francesca F Aiello

  15. Dual inhibition of survivin and MAOA synergistically impairs growth of PTEN-negative prostate cancer

    Article • British Journal of Cancer, June 2015, Springer Science + Business Media

    Fedora Grande

  16. Identification of two benzopyrroloxazines acting as selective GPER antagonists in breast cancer cells and cancer-associated fibroblasts

    Article • Future Medicinal Chemistry, March 2015, Future Science

    Fedora Grande, PhD Francesca F Aiello

  17. Active manganese dioxide promoted cyclization of ortho-(1H-pyrrol-1-yl)aryl and heteroaryl carboxylic acids to 5H-pyrrolo[1,2-a][3,1]benzoxazin-5-one derivatives

    Article • Tetrahedron, November 2013, Elsevier

    Fedora Grande, PhD Francesca F Aiello

  18. Stabilization of MDA-7/IL-24 for colon cancer therapy

    Article • Cancer Letters, July 2013, Elsevier

    Fedora Grande

  19. Discovery of a Novel Orally Active Small-Molecule gp130 Inhibitor for the Treatment of Ovarian Cancer

    Article • Molecular Cancer Therapeutics, March 2013, American Association for Cancer Research (AACR)

    Fedora Grande

  20. Small Molecule Inhibitors of CXCR4

    Article • Theranostics, January 2013, Ivyspring International Publisher

    Fedora Grande

  21. Design and Synthesis of 3-Carbamoylbenzoic Acid Derivatives as Inhibitors of Human Apurinic/Apyrimidinic Endonuclease 1 (APE1)

    Article • ChemMedChem, September 2012, Wiley

    PhD Francesca F Aiello , Fedora Grande

  22. Cytotoxic potential of novel 6,7-dimethoxyquinazolines

    Article • European Journal of Medicinal Chemistry, February 2012, Elsevier

    Fedora Grande

  23. Convenient synthesis of fluorazone derivatives by one-pot pyrrolation/cyclization of anthranilic acids

    Article • Tetrahedron Letters, November 2011, Elsevier

    PhD Francesca F Aiello , Fedora Grande

  24. Direct cyclization of ortho-(1H-pyrrol-1-yl)aryl and heteroaryl carboxylic acids into fused pyrrolizinones

    Article • Tetrahedron Letters, December 2010, Elsevier

    PhD Francesca F Aiello , Fedora Grande

  25. Efficient synthesis of 9H-pyrrolo[1,2-a]indol-9-one derivatives based on active manganese dioxide promoted intramolecular cyclization

    Article • Tetrahedron, January 2010, Elsevier

    PhD Francesca F Aiello , Fedora Grande

  26. Synthesis and biological evaluation of novel hydrazide based cytotoxic agents

    Article • Expert Opinion on Investigational Drugs, April 2009, Informa Healthcare

    PhD Francesca F Aiello , Fedora Grande

  27. Discovery of Novel Anticancer Compounds Based on a Quinoxalinehydrazine Pharmacophore

    Article • ChemMedChem, November 2008, Wiley

    Fedora Grande, PhD Francesca F Aiello

  28. Naphthoxazepine Inhibitors of HIV-1 Integrase: Synthesis and Biological Evaluation

    Article • ChemMedChem, June 2008, Wiley

    Fedora Grande, PhD Francesca F Aiello

  29. Small Molecules Anti-HIV Therapeutics Targeting CXCR4

    Article • Current Pharmaceutical Design, February 2008, Bentham Science Publishers

    Fedora Grande

  30. Small Molecule Inhibitors of Stat3 Signaling Pathway

    Article • Current Cancer Drug Targets, February 2007, Bentham Science Publishers

    Fedora Grande

  31. Synthesis and antitumor activities of a series of novel quinoxalinhydrazides

    Article • Bioorganic & Medicinal Chemistry, January 2007, Elsevier

    PhD Francesca F Aiello , Fedora Grande

  32. Recent advances in the design and discovery of small-molecule therapeutics targeting HER2/neu

    Article • Expert Opinion on Therapeutic Patents, January 2007, Informa Healthcare

    Fedora Grande

  33. A critical study on the application of the zero-crossing derivative spectrophotometry to the photodegradation monitoring of lacidipine

    Article • Journal of Pharmaceutical and Biomedical Analysis, September 2006, Elsevier

    Fedora Grande

  34. An approach to the stereo-controlled synthesis of polycyclic derivatives of l-4-thiazolidinecarboxylic acid active against HIV-1 integrase

    Article • European Journal of Medicinal Chemistry, August 2006, Elsevier

    Fedora Grande, PhD Francesca F Aiello

  35. Synthesis of novel thiazolothiazepine based HIV-1 integrase inhibitors

    Article • Bioorganic & Medicinal Chemistry, August 2004, Elsevier

    PhD Francesca F Aiello , Fedora Grande