All Stories

  1. Targeting STAT3 in Breast Cancer Using Innovative Natural and Synthetic Scaffolds to Trigger Apoptosis, Autophagy, and Halt Tumor Progression

    Article • Current Drug Targets, July 2026, Bentham Science Publishers

    Dr Basappa . ., Vladimir Nikolenko, Prema Venkatesh

  2. Integrative Profiling of the Ovarian Reserve using Ultrasound and MRI Data by Comparative Analysis: A Systematic Review

    Article • Current Medicinal Chemistry, March 2026, Bentham Science Publishers

    Dr Basappa . ., Vladimir Nikolenko

  3. Cyclocondensation of Sodium Azide with Methyl N(N),N'-di(tri)substituted Carbamimidothioate : A New Dimension for the Synthesis of 1,5-disubstituted Tetrazoles and Their Cytotoxicity against Human Breast Cancer Cells

    Article • Current Organic Chemistry, December 2020, Bentham Science Publishers

    Dr Basappa . .

  4. Synthesis and Biological Evaluation of Novel Thiazol-2yl-amine Derivatives as Potential Anticancer Agents

    Article • Letters in Organic Chemistry, March 2018, Bentham Science Publishers

    Chakrabhavi Dhananjaya Mohan , Dr Basappa . .

  5. Synthesis of Coumarin-benzotriazole Hybrids and Evaluation of their Anti-tubercular Activity

    Article • Letters in Organic Chemistry, December 2017, Bentham Science Publishers

    Dr Basappa . ., Chakrabhavi Dhananjaya Mohan

  6. Screening of quinoline, 1,3-benzoxazine, and 1,3-oxazine-based small molecules against isolated methionyl-tRNA synthetase and A549 and HCT116 cancer cells including an in silico binding mode analysis

    Article • Organic & Biomolecular Chemistry, January 2015, Royal Society of Chemistry

    Dr Basappa . .

  7. Synthesis, characterization and in vitro evaluation of novel enantiomerically-pure sulphonamide antimalarials

    Article • Organic & Biomolecular Chemistry, January 2015, Royal Society of Chemistry

    Dr Basappa . ., Rajesh Chandramohanadas

  8. Preparation and use of combustion derived Bi2O3 for the generation of novel heterocycles via Suzuki-Coupling Reactions: potential application as anti-cancer agents

    Article • RSC Advances, October 2014, Royal Society of Chemistry

    Dr Basappa . ., Chakrabhavi Dhananjaya Mohan

  9. A New Ibuprofen Derivative Inhibits Platelet Aggregation and ROS Mediated Platelet Apoptosis

    Article • PLOS One, September 2014, PLOS

    Dr Basappa . .

  10. Roles of glycosaminoglycans and glycanmimetics in tumor progression and metastasis

    Article • Glycoconjugate Journal, September 2014, Springer Science + Business Media

    Dr Basappa . .

  11. Novel Synthetic Biscoumarins Target Tumor Necrosis Factor-α in Hepatocellular Carcinomain Vitroandin Vivo

    Article • Journal of Biological Chemistry, September 2014, American Society for Biochemistry & Molecular Biology (ASBMB)

    Dr Basappa . ., Chakrabhavi Dhananjaya Mohan

  12. Novel Apigenin Based Small Molecule that Targets Snake Venom Metalloproteases

    Article • PLOS One, September 2014, PLOS

    Dr Basappa . .

  13. Synthesis and characterization of novel 1,2-oxazine-based small molecules that targets acetylcholinesterase

    Article • Bioorganic & Medicinal Chemistry Letters, August 2014, Elsevier

    Dr Basappa . ., Prof., Dr. Alexey Yu. Sukhorukov

  14. Novel Benzoxazine-Based Aglycones Block Glucose Uptake In Vivo by Inhibiting Glycosidases

    Article • PLOS One, July 2014, PLOS

    Dr Basappa . .

  15. Small Molecule Targeting Malaria Merozoite Surface Protein-1 (MSP-1) Prevents Host Invasion of Divergent Plasmodial Species

    Article • The Journal of Infectious Diseases, May 2014, Oxford University Press (OUP)

    Dr Basappa . ., Rajesh Chandramohanadas

  16. Synthesis and biological evaluation of tetrahydropyridinepyrazoles (‘PFPs’) as inhibitors of STAT3 phosphorylation

    Article • MedChemComm, January 2014, Royal Society of Chemistry

    Dr Basappa . .

  17. Synthesis, biological evaluation and in silico and in vitro mode-of-action analysis of novel dihydropyrimidones targeting PPAR-γ

    Article • RSC Advances, January 2014, Royal Society of Chemistry

    Dr Basappa . .

  18. Anti-cancer activity of novel dibenzo[b,f]azepine tethered isoxazoline derivatives

    Article • BMC Chemical Biology, October 2012, Springer Science + Business Media

    Dr Basappa . .

  19. Anti-Tumor Activity of a Novel HS-Mimetic-Vascular Endothelial Growth Factor Binding Small Molecule

    Article • PLOS One, August 2012, PLOS

    Dr Basappa . .

  20. Neutralization of Haemorrhagic Activity of Viper Venoms by 1-(3-Dimethylaminopropyl)-1-(4-Fluorophenyl)-3-Oxo-1,3-Dihydroisobenzofuran-5-Carbonitrile

    Article • Basic & Clinical Pharmacology & Toxicology, June 2011, Wiley

    Dr Basappa . ., Dr Santosh L Gaonkar

  21. Homology modeling and in silico screening of inhibitors for the substrate binding domain of human Siah2: implications for hypoxia-induced cancers

    Article • Journal of Molecular Modeling, March 2011, Springer Science + Business Media

    Dr Basappa . .

  22. N-[4-Cyano-3-(trifluoromethyl)phenyl]-2-methoxybenzamide

    Article • Acta Crystallographica Section E Structure Reports Online, December 2010, International Union of Crystallography

    Dr Basappa . .

  23. A small oxazine compound as an anti-tumor agent: A novel pyranoside mimetic that binds to VEGF, HB-EGF, and TNF-α

    Article • Cancer Letters, November 2010, Elsevier

    Dr Basappa . .

  24. Cheminformatics-Based Drug Design Approach for Identification of Inhibitors Targeting the Characteristic Residues of MMP-13 Hemopexin Domain

    Article • PLOS One, August 2010, PLOS

    Dr Basappa . .

  25. N-[4-Cyano-3-(trifluoromethyl)phenyl]-2-ethoxybenzamide

    Article • Acta Crystallographica Section E Structure Reports Online, June 2010, International Union of Crystallography

    Dr Basappa . .

  26. Synthesis, characterization and in vitro anti-tumor activities of novel 9-ethyl-9H-purine derivatives

    Article • Investigational New Drugs, September 2009, Springer Science + Business Media

    Dr Basappa . .

  27. Anti-tumor and anti-angiogenic activity of novel hydantoin derivatives: Inhibition of VEGF secretion in liver metastatic osteosarcoma cells

    Article • Bioorganic & Medicinal Chemistry, July 2009, Elsevier

    Dr Basappa . .

  28. Involvement of chondroitin sulfate E in the liver tumor focal formation of murine osteosarcoma cells

    Article • Glycobiology, March 2009, Oxford University Press (OUP)

    Dr Basappa . .

  29. Determination of iduronic acid and glucuronic acid in sulfated chondroitin/dermatan hybrid chains by 1H-nuclear magnetic resonance spectroscopy

    Article • Glycoconjugate Journal, March 2008, Springer Science + Business Media

    Dr Basappa . .

  30. Chondroitinase-mediated Degradation of Rare 3-O-Sulfated Glucuronic Acid in Functional Oversulfated Chondroitin Sulfate K and E

    Article • Journal of Biological Chemistry, October 2007, American Society for Biochemistry & Molecular Biology (ASBMB)

    Dr Basappa . .

  31. 2-(2-(2-Ethoxybenzoylamino)-4-chlorophenoxy)-N-(2-ethoxybenzoyl)benzamine inhibits EAT cell induced angiogenesis by down regulation of VEGF secretion

    Article • Bioorganic & Medicinal Chemistry Letters, May 2007, Elsevier

    Dr Basappa . .

  32. N-Substituted-2-butyl-5-chloro-3H-imidazole-4-carbaldehyde Derivatives as Anti-tumor Agents Against Ehrlich Ascites tumor Cells In Vivo

    Article • Medicinal Chemistry, May 2007, Bentham Science Publishers

    Dr Basappa . ., Dr Santosh L Gaonkar

  33. Pro-apoptotic activity of imidazole derivatives mediated by up-regulation of Bax and activation of CAD in Ehrlich Ascites Tumor cells

    Article • Investigational New Drugs, March 2007, Springer Science + Business Media

    Dr Basappa . .

  34. Conformational Studies on Five Octasaccharides Isolated from Chondroitin Sulfate Using NMR Spectroscopy and Molecular Modeling

    Article • Biochemistry, January 2007, American Chemical Society (ACS)

    Dr Basappa . .

  35. (2-Ethoxyphenyl)[4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl]methanone

    Article • Acta Crystallographica Section E Structure Reports Online, January 2007, International Union of Crystallography

    Dr Basappa . .

  36. Crystal and Molecular Structure Analysis of 1,2,4-Triazolo-N-amino-thiols

    Article • Molecular Crystals and Liquid Crystals, November 2006, Taylor & Francis

    Dr Basappa . .

  37. Synthesis, characterization, antimicrobial and single crystal X-ray crystallographic studies of some new sulfonyl, 4-chloro phenoxy benzene and dibenzoazepine substituted benzamides

    Article • European Journal of Medicinal Chemistry, November 2006, Elsevier

    Dr Basappa . ., Dr Santosh L Gaonkar

  38. Synthesis and Crystal Structure Studies of (2RS)‐3‐[(2RS)‐2‐(1‐hydroxycyclohexyl)‐2‐(4‐methoxyphenyl)ethyl] ‐2‐(pyridin‐3‐yl)thiazolidin‐4‐one.

    Article • ChemInform, September 2006, Wiley

    Dr Basappa . .

  39. Synthesis of Pharmaceutically Important Condensed Heterocyclic 4,6‐Disubstituted‐1,2,4‐triazolo‐1,3,4‐triadiazole Derivatives as Antimicrobials.

    Article • ChemInform, August 2006, Wiley

    Dr Basappa . ., Dr Doreswamy B H swamy

  40. Synthesis of New Bioactive Venlafaxine Analogues: Novel Thiazolidin‐4‐ones as Antimicrobials.

    Article • ChemInform, May 2006, Wiley

    Dr Basappa . .

  41. Synthesis and crystal structure studies of (2 RS )-3-[(2 RS )-2-(1-hydroxycyclohexyl)-2-(4-methoxyphenyl)ethyl]-2-(pyridin-3-yl)thiazolidin-4-one

    Article • Journal of Chemical Research, May 2006, SAGE Publications

    Dr Basappa . .

  42. Microwave‐Assisted Synthesis of N‐Alkylated Benzotriazole Derivatives: Antimicrobial Studies.

    Article • ChemInform, April 2006, Wiley

    Dr Basappa . .

  43. Synthesis of new bioactive venlafaxine analogs: Novel thiazolidin-4-ones as antimicrobials

    Article • Bioorganic & Medicinal Chemistry, April 2006, Elsevier

    Dr Basappa . .

  44. Synthesis of pharmaceutically important condensed heterocyclic 4,6-disubstituted-1,2,4-triazolo-1,3,4-thiadiazole derivatives as antimicrobials

    Article • European Journal of Medicinal Chemistry, April 2006, Elsevier

    Dr Basappa . .

  45. Δ2-ISOXAZOLINE DERIVATIVES AS ANTIMICROBIALS

    Article • Heterocyclic Communications, February 2006, De Gruyter

    Dr Basappa . .

  46. Microwave-assisted synthesis of N-alkylated benzotriazole derivatives: Antimicrobial studies

    Article • Bioorganic & Medicinal Chemistry Letters, February 2006, Elsevier

    Dr Basappa . ., Dr Santosh L Gaonkar

  47. Synthesis and crystal structure analysis of 2-(4-methyl-2′-biphenyl)-4-amino-1,2,4-triazole-3-thiol

    Article • Structural Chemistry, February 2006, Springer Science + Business Media

    Dr Basappa . .

  48. Synthesis and Crystal Structure of 3,4,5-Trimethoxybenzaldehyde oxime monohydrate

    Article • Analytical Sciences X-ray Structure Analysis Online, January 2006, Japan Society for Analytical Chemistry

    Dr Basappa . .

  49. Crystal Structure of a Bioactive Intermediate: 1-Benzhydrylpiperazine

    Article • Analytical Sciences X-ray Structure Analysis Online, January 2006, Japan Society for Analytical Chemistry

    Dr Basappa . .

  50. Synthesis and Crystal Structure of 5-Ethyl-2-[2-(4-nitrophenoxy)ethyl]-pyridine

    Article • Analytical Sciences X-ray Structure Analysis Online, January 2006, Japan Society for Analytical Chemistry

    Dr Basappa . .

  51. Crystal Structure of 3-para tolyl-6-(4′-methyl-biphenyl-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole

    Article • Analytical Sciences X-ray Structure Analysis Online, January 2006, Japan Society for Analytical Chemistry

    Dr Basappa . .

  52. Crystal Structure of 2-Ethoxy-N-[4-(pyrimidin-2-ylsulfamoyl)-phenyl]-benzamide

    Article • Analytical Sciences X-ray Structure Analysis Online, January 2006, Japan Society for Analytical Chemistry

    Dr Basappa . .

  53. Crystal Structure of Bioactive Venlafaxine Analog: 3-(2-(1-Hydroxycyclohexyl)-2-(4-methoxyphenyl)ethyl)-2-(4-hydroxyphenyl)-thiazolidin-4-one

    Article • Analytical Sciences X-ray Structure Analysis Online, January 2006, Japan Society for Analytical Chemistry

    Dr Basappa . .

  54. Synthesis and molecular structure analysis of venlafaxine intermediate and its analog

    Article • Journal of Chemical Crystallography, December 2005, Springer Science + Business Media

    Dr Basappa . .

  55. 2-(Biphenyl-4-yl)-3-(4-methoxyphenyl)-1,3-thiazolidin-4-one

    Article • Acta Crystallographica Section E Structure Reports Online, June 2005, International Union of Crystallography

    Dr Basappa . .

  56. New cholinesterase inhibitors: synthesis and structure–activity relationship studies of 1,2‐benzisoxazole series and novel imidazolyl‐d2‐isoxazolines

    Article • Journal of Physical Organic Chemistry, May 2005, Wiley

    Dr Basappa . .

  57. Reduction of Aldehydes and Oximes to Their Corresponding Alcohols and Amines by Catalytic Hydrogenation Method.

    Article • ChemInform, April 2005, Wiley

    Dr Basappa . ., Dr Doreswamy B H swamy

  58. Synthesis and X-ray Crystal Studies of 6-(2-chlorophenyl)-3-methyl[1,2,4] triazolo[4,5-b][1,3,4]thiadiazole

    Article • Journal of Chemical Research, April 2005, SAGE Publications

    Dr Basappa . .

  59. Synthesis and characterization of novel 6-fluoro-4-piperidinyl-1,2-benzisoxazole amides and 6-fluoro-chroman-2-carboxamides: antimicrobial studies

    Article • Bioorganic & Medicinal Chemistry, April 2005, Elsevier

    Dr Basappa . .

  60. Synthesis and crystal structure of 5-allyl-5Hdibenzo[b,f]azepine

    Article • Journal of Chemical Crystallography, March 2005, Springer Science + Business Media

    Dr Basappa . ., Dr Doreswamy B H swamy

  61. Synthesis and X-ray structure of 3-(4-methyl phenyl)-2-(4-biphenyl)-1,3-thiazolidin-4-one

    Article • Journal of Chemical Crystallography, January 2005, Springer Science + Business Media

    Dr Basappa . .

  62. A Simple and Efficient Method for the Synthesis of 1,2‐Benzisoxazoles: A Series of Its Potent Acetylcholinesterase Inhibitors.

    Article • ChemInform, December 2004, Wiley

    Dr Basappa . .

  63. Novel δ2‐Isoxazolines as Group II Phospholipase A2 Inhibitors.

    Article • ChemInform, October 2004, Wiley

    Dr Basappa . .

  64. Simple and Efficient Method for the Synthesis of 1‐[2‐Dimethylamino‐1‐(4‐methoxy‐phenyl)‐ethyl]‐cyclohexanol Hydrochloride: (.+‐.) Venlafaxine Racemic Mixtures.

    Article • ChemInform, September 2004, Wiley

    Dr Basappa . .

  65. Novel δ2-isoxazolines as group II phospholipase A2 inhibitors

    Article • Bioorganic & Medicinal Chemistry Letters, July 2004, Elsevier

    Dr Basappa . .

  66. Simple and an efficient method for the synthesis of 1-[2-dimethylamino-1-(4-methoxy-phenyl)-ethyl]-cyclohexanol hydrochloride: (±) venlafaxine racemic mixtures

    Article • Bioorganic & Medicinal Chemistry Letters, June 2004, Elsevier

    Dr Basappa . .

  67. A Facile Route for the Syntheis of Novel γ‐Lactams.

    Article • ChemInform, December 2003, Wiley

    Dr Basappa . .

  68. Synthesis and crystal structure of 1-ethyl-3-(phenyl)-1,2,3-triazolium percholorate

    Article • Open Chemistry, December 2003, De Gruyter

    Dr Basappa . .

  69. Solution-phase synthesis of novel Δ2-isoxazoline libraries via 1,3-dipolar cycloaddition and their antifungal properties

    Article • Bioorganic & Medicinal Chemistry, October 2003, Elsevier

    Dr Basappa . .

  70. Synthesis of Novel Isoxazolidine Derivatives and Studies for Their Antifungal Properties.

    Article • ChemInform, September 2003, Wiley

    Dr Basappa . .

  71. A facile route for the synthesis of novel γ‐lactams

    Article • Journal of Heterocyclic Chemistry, July 2003, Wiley

    Dr Basappa . .

  72. SYNTHESIS AND CRYSTAL STRUCTURE OF 1-METHYL-3-(4-NITROPHENYL)-1,2,3 TRIAZOLIUM PERCHLORATE

    Article • Molecular Crystals and Liquid Crystals Science and Technology Section A Molecular Crystals and Liquid Crystals, June 2003, Taylor & Francis

    Dr Basappa . .

  73. SYNTHESIS OF NOVEL ISOXAZOLIDINES VIA 1,3-DIPOLAR CYCLOADDITION OF NITRONES TO OLEFINS

    Article • Heterocyclic Communications, April 2003, De Gruyter

    Dr Basappa . .

  74. SYNTHESIS AND CRYSTAL STRUCTURE OF 1-METHYL-3-(4-NITROPHENYL)-1,2,3 TRIAZOLIUM PERCHLORATE

    Article • Molecular Crystals and Liquid Crystals, January 2003, Taylor & Francis

    Dr Basappa . .

  75. Microwave-Assisted Synthesis and Crystal Structure of 2-Butyl-4-chloro-1H-imidazole-5-carboxaldehyde

    Article • Analytical Sciences X-ray Structure Analysis Online, January 2003, Japan Society for Analytical Chemistry

    Dr Basappa . .