Optimization of a series of dipeptides with a P3 β-neopentyl asparagine residue as non-covalent inhibitors of the chymotrypsin-like activity of human 20S proteasome

Christopher Blackburn, Cynthia Barrett, Jonathan L. Blank, Frank J. Bruzzese, Nancy Bump, Lawrence R. Dick, Paul Fleming, Khristofer Garcia, Paul Hales, Matthew Jones, Jane X. Liu, Masayuki Nagayoshi, Darshan S. Sappal, Michael D. Sintchak, Christopher Tsu, Cindy Xia, Xiansi Zhou, Kenneth M. Gigstad
  • MedChemComm, January 2012, Royal Society of Chemistry
  • DOI: 10.1039/c2md20060k