Discovery of a potent and highly β1 specific proteasome inhibitor from a focused library of urea-containing peptide vinyl sulfones and peptide epoxyketones

Wouter A. van der Linden, Lianne I. Willems, Tamer B. Shabaneh, Nan Li, Mark Ruben, Bogdan I. Florea, Gijs A. van der Marel, Markus Kaiser, Alexei F. Kisselev, Herman S. Overkleeft
  • Organic & Biomolecular Chemistry, January 2012, Royal Society of Chemistry
  • DOI: 10.1039/c1ob06554h