Publication
Encoded Library Technology as a Source of Hits for the Discovery and Lead Optimization of a Potent and Selective Class of Bactericidal Direct Inhibitors of Mycobacterium tuberculosis InhA
Lourdes Encinas, Heather O’Keefe, Margarete Neu, Modesto J. Remuiñán, Amish M. Patel, Ana Guardia, Christopher P. Davie, Natalia Pérez-Macías, Hongfang Yang, Maire A. Convery, Jeff A. Messer, Esther Pérez-Herrán, Paolo A. Centrella, Daniel Álvarez-Gómez, Matthew A. Clark, Sophie Huss, Gary K. O’Donovan, Fátima Ortega-Muro, William McDowell, Pablo Castañeda, Christopher C. Arico-Muendel, Stane Pajk, Joaquín Rullás, Iñigo Angulo-Barturen, Emilio Álvarez-Ruíz, Alfonso Mendoza-Losana, Lluís Ballell Pages, Julia Castro-Pichel, Ghotas Evindar
Journal of Medicinal Chemistry, February 2014, American Chemical Society (ACS)
DOI: 10.1021/jm401326j