Publication
Optimization of a Dibenzodiazepine Hit to a Potent and Selective Allosteric PAK1 Inhibitor
Alexei S. Karpov, Payman Amiri, Cornelia Bellamacina, Marie-Helene Bellance, Werner Breitenstein, Dylan Daniel, Regis Denay, Doriano Fabbro, Cesar Fernandez, Inga Galuba, Stephanie Guerro-Lagasse, Sascha Gutmann, Linda Hinh, Wolfgang Jahnke, Julia Klopp, Albert Lai, Mika K. Lindvall, Sylvia Ma, Henrik Möbitz, Sabina Pecchi, Gabriele Rummel, Kevin Shoemaker, Joerg Trappe, Charles Voliva, Sandra W. Cowan-Jacob, Andreas L. Marzinzik
ACS Medicinal Chemistry Letters, May 2015, American Chemical Society (ACS)
DOI: 10.1021/acsmedchemlett.5b00102