Publication
Structure–Activity Relationships for a Series of (Bis(4-fluorophenyl)methyl)sulfinyl Alkyl Alicyclic Amines at the Dopamine Transporter: Functionalizing the Terminal Nitrogen Affects Affinity, Selectivity, and Metabolic Stability
Rachel D. Slack, Therese C. Ku, Jianjing Cao, JoLynn B. Giancola, Alessandro Bonifazi, Claus J. Loland, Alexandra Gadiano, Jenny Lam, Rana Rais, Barbara S. Slusher, Mark Coggiano, Gianluigi Tanda, Amy Hauck Newman
Journal of Medicinal Chemistry, October 2019, American Chemical Society (ACS)
DOI: 10.1021/acs.jmedchem.9b01188