Publication
Optimization and Characterization of N-Acetamide Indoles as Antimalarials That Target PfATP4
Jon Kyle Awalt, Zi Kang Ooi, Trent D. Ashton, Mahta Mansouri, Petar P. S. Calic, Qingmiao Zhou, Santhya Vasanthan, Serena Lee, Katie Loi, Kate E. Jarman, Jocelyn S. Penington, Deyun Qiu, Xinxin Zhang, Adele M. Lehane, Emma Y. Mao, Maria R. Gancheva, Danny W. Wilson, Carlo Giannangelo, Christopher A. MacRaild, Darren J. Creek, Tomas Yeo, Tanaya Sheth, David A. Fidock, Alisje Churchyard, Jake Baum, Mufuliat T. Famodimu, Michael J. Delves, Mojca Kristan, Lindsay Stewart, Colin J. Sutherland, Rachael Coyle, Hannah Jagoe, Marcus C. S. Lee, Mrittika Chowdury, Tania F. de Koning-Ward, Delphine Baud, Stephen Brand, Paul F. Jackson, Alan F. Cowman, Madeline G. Dans, Brad E. Sleebs
Journal of Medicinal Chemistry, April 2025, American Chemical Society (ACS)
DOI: 10.1021/acs.jmedchem.5c00614