Publication
A Developability-Focused Optimization Approach Allows Identification of in Vivo Fast-Acting Antimalarials: N -[3-[(Benzimidazol-2-yl)amino]propyl]amides
Leena Keurulainen, Mikko Vahermo, Margarita Puente-Felipe, Elena Sandoval-Izquierdo, Benigno Crespo-Fernández, Laura Guijarro-López, Leticia Huertas-Valentín, Laura de las Heras-Dueña, Teppo O. Leino, Antti Siiskonen, Lluís Ballell-Pages, Laura M. Sanz, Pablo Castañeda-Casado, M. Belén Jiménez-Díaz, María S. Martínez-Martínez, Sara Viera, Paula Kiuru, Félix Calderón, Jari Yli-Kauhaluoma
Journal of Medicinal Chemistry, June 2015, American Chemical Society (ACS)
DOI: 10.1021/acs.jmedchem.5b00114