New Synthetic Routes to Triazolo-benzodiazepine Analogues: Expanding the Scope of the Bump-and-Hole Approach for Selective Bromo and Extra-Terminal (BET) Bromodomain Inhibition

• Matthias G. J. Baud, Enrique Lin-Shiao, Michael Zengerle, Cynthia Tallant, Alessio Ciulli

• Journal of Medicinal Chemistry, February 2016, American Chemical Society (ACS)
• DOI: 10.1021/acs.jmedchem.5b01135