Publication
Discovery of novel hepatoselective HMG-CoA reductase inhibitors for treating hypercholesterolemia: A bench-to-bedside case study on tissue selective drug distribution
Jeffrey A. Pfefferkorn, John Litchfield, Richard Hutchings, Xue-Min Cheng, Scott D. Larsen, Bruce Auerbach, Mark R. Bush, Chitase Lee, Noe Erasga, Daniel M. Bowles, David C. Boyles, Gina Lu, Catherine Sekerke, Valerie Askew, Jeffrey C. Hanselman, Lisa Dillon, Zhiwu Lin, Andrew Robertson, Karl Olsen, Carine Boustany, Karen Atkinson, Theunis C. Goosen, Vaishali Sahasrabudhe, Jonathan Chupka, David B. Duignan, Bo Feng, Renato Scialis, Emi Kimoto, Yi-An Bi, Yurong Lai, Ayman El-Kattan, Rebecca Bakker-Arkema, Paul Barclay, Erick Kindt, Vu Le, Jaap W. Mandema, Mark Milad, Bradley D. Tait, Robert Kennedy, Bharat K. Trivedi, Mark Kowala
Bioorganic & Medicinal Chemistry Letters, May 2011, Elsevier
DOI: 10.1016/j.bmcl.2010.11.103