Publication
Discovery of 4-{1-[({1-[4-(trifluoromethyl)benzyl]-1H-indol-7-yl}carbonyl)amino]cyclopropyl}benzoic acid (MF-766), a highly potent and selective EP4 antagonist for treating inflammatory pain
John Colucci, Michael Boyd, Carl Berthelette, Jean-Francois Chiasson, Zhaoyin Wang, Yves Ducharme, Rick Friesen, Mark Wrona, Jean-Francois Levesque, Danielle Denis, Marie-Claude Mathieu, Rino Stocco, Alex G. Therien, Patsy Clarke, Steve Rowland, Daigen Xu, Yongxin Han
Bioorganic & Medicinal Chemistry Letters, June 2010, Elsevier
DOI: 10.1016/j.bmcl.2010.04.065