A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced-Fit Pocket Stabilized by a Cation-π Interaction

Timothy P. C. Rooney, Panagis Filippakopoulos, Oleg Fedorov, Sarah Picaud, Wilian A. Cortopassi, Duncan A. Hay, Sarah Martin, Anthony Tumber, Catherine M. Rogers, Martin Philpott, Minghua Wang, Amber L. Thompson, Tom D. Heightman, David C. Pryde, Andrew Cook, Robert S. Paton, Susanne Müller, Stefan Knapp, Paul E. Brennan, Stuart J. Conway
  • Angewandte Chemie International Edition, May 2014, Wiley
  • DOI: 10.1002/anie.201402750

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The following have contributed to this page: Associate Prof. Robert S Paton