All Stories

  1. Efficient synthesis of 2-nitroimidazole derivatives and the bioreductive clinical candidate Evofosfamide (TH-302)
  2. The design and synthesis of 5- and 6-isoxazolylbenzimidazoles as selective inhibitors of the BET bromodomains
  3. Wavelength-orthogonal photolysis of neurotransmittersin vitro
  4. The use of phosphate bioisosteres in medicinal chemistry and chemical biology