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  1. Increased fibrinolysis-induced bradykinin formation in hereditary angioedema confirmed using stored plasma and biotechnological inhibitors
  2. Comparing Pathways of Bradykinin Formation in Whole Blood From Healthy Volunteers and Patients With Hereditary Angioedema Due to C1 Inhibitor Deficiency
  3. Bifunctional ligands of the bradykinin B 2 and B 1 receptors: An exercise in peptide hormone plasticity
  4. Bifunctional fusion proteins containing the sequence of the bradykinin homologue maximakinin: activities at the rat bradykinin B2 receptor
  5. D-Arg0-Bradykinin-Arg-Arg, a Latent Vasoactive Bradykinin B2 Receptor Agonist Metabolically Activated by Carboxypeptidases
  6. Editorial: Correspondence from Chirumbolo and Bjorklund
  7. Production and evaluation of parathyroid hormone receptor1 ligands with intrinsic or assembled peroxidase domains
  8. S100A9 potentiates the activation of neutrophils by the etiological agent of gout, monosodium urate crystals
  9. Species-specific pharmacology of maximakinin, an amphibian homologue of bradykinin: putative prodrug activity at the human B2receptor and peptidase resistance in rats
  10. Species-specific pharmacology of maximakinin, an amphibian homologue of bradykinin: putative prodrug activity at the human B2 receptor and peptidase resistance in rat
  11. Species-specific pharmacology of maximakinin, an amphibian homologue of bradykinin: putative prodrug activity at the human B2 receptor and peptidase resistance in rat
  12. Infrared-emitting, peptidase-resistant fluorescent ligands of the bradykinin B2 receptor: application to cytofluorometry and imaging
  13. Editorial: Improving the data reproducibility and general interest of natural product submissions
  14. Lysosomotropic cationic drugs induce cytostatic and cytotoxic effects: Role of liposolubility and autophagic flux and antagonism by cholesterol ablation
  15. Introduction: Natural product-based drug discovery in Immunopharmacology
  16. The isolated human umbilical vein as a bioassay for kinin-generating proteases: An in vitro model for therapeutic angioedema agents
  17. Biotechnological Fluorescent Ligands of the Bradykinin B1 Receptor: Protein Ligands for a Peptide Receptor
  18. In Vivo Effects of Bradykinin B2 Receptor Agonists with Varying Susceptibility to Peptidases
  19. Autophagic flux inhibition and lysosomogenesis ensuing cellular capture and retention of the cationic drug quinacrine in murine models
  20. Book review: Evidence-based validation of herbal medicine, Elsevier, Amsterdam, 2015, Edited by P. K. Mukherjee. 537 pp. ISBN: 978-0-12-800874-4
  21. Pharmacological profile of a bifunctional ligand of the formyl peptide receptor1 fused to the myc epitope
  22. Pharmacological effects of recombinant human tissue kallikrein on bradykinin B 2 receptors
  23. A tagged parathyroid hormone derivative as a carrier of antibody cargoes transported by the G protein coupled PTH1 receptor
  24. Pharmacological evidence of bradykinin regeneration from extended sequences that behave as peptidase–activated B2 receptor agonists
  25. Assessment of Cation Trapping by Cellular Acidic Compartments
  26. Vasopeptidase-activated latent ligands of the histamine receptor-1
  27. Green fluorescent protein fused to peptide agonists of two dissimilar G protein‐coupled receptors: novel ligands of the bradykinin B 2 (rhodopsin family) receptor and parathyroid hormone PTH 1 ...
  28. High affinity capture and concentration of quinacrine in polymorphonuclear neutrophils via vacuolar ATPase-mediated ion trapping: Comparison with other peripheral blood leukocytes and implications for the distribution of cationic drugs
  29. Inhibitory effects of cytoskeleton disrupting drugs and GDP-locked Rab mutants on bradykinin B2 receptor cycling
  30. Bifunctional epitope-agonist ligands of the bradykinin B2 receptor
  31. C-C chemokine receptor-7 mediated endocytosis of antibody cargoes into intact cells
  32. NLRP3 promotes autophagy of urate crystals phagocytized by human osteoblasts
  33. An in vitro reconstitution system to address the mechanism of the vascular expression of the bradykinin B1 receptor in response to angiotensin converting enzyme inhibition
  34. N-terminal extended conjugates of the agonists and antagonists of both bradykinin receptor subtypes: Structure–activity relationship, cell imaging using ligands conjugated with fluorophores and prospect for functionally active cargoes
  35. Prolonged signalling and trafficking of the bradykinin B2 receptor stimulated with the amphibian peptide maximakinin: Insight into the endosomal inactivation of kinins
  36. Cation trapping by cellular acidic compartments: Beyond the concept of lysosomotropic drugs
  37. Met-Lys-bradykinin-Ser-Ser, a peptide produced by the neutrophil from kininogen, is metabolically activated by angiotensin converting enzyme in vascular tissue
  38. Bradykinin B2 receptor-mediated transport into intact cells: Anti-receptor antibody-based cargoes
  39. Dissociation of the vacuolar and macroautophagic cytopathology from the cytotoxicity induced by the lipophilic local anesthetic bupivacaine
  40. 5 Drugs in the kallikrein-kinin system
  41. Kinins
  42. Design of Fluorescent Bradykinin Analogs: Application to Imaging of B2 Receptor-Mediated Agonist Endocytosis and Trafficking and Angiotensin-Converting Enzyme
  43. Effect of interferon-γ on inflammatory cytokine-induced bradykinin B1 receptor expression in human vascular cells
  44. Vascular smooth muscle contractility assays for inflammatory and immunological mediators
  45. A ligand-based approach to investigate the expression and function of angiotensin converting enzyme in intact human umbilical vein endothelial cells
  46. Bradykinin forming capacity of oversulfated chondroitin sulfate contaminated heparin in vitro
  47. Guest Editorial for the Special Issue Peptide Receptors: Focus on Neuropeptides and Kinins
  48. Altered cardiac bradykinin metabolism in experimental diabetes caused by the variations of angiotensin-converting enzyme and other peptidases
  49. Vacuolar ATPase-mediated sequestration of local anesthetics in swollen macroautophagosomes
  50. Effects of inactivation-resistant agonists on the signalling, desensitization and down-regulation of bradykinin B2 receptors
  51. Vacuolar ATPase-Mediated Cellular Concentration and Retention of Quinacrine: A Model for the Distribution of Lipophilic Cationic Drugs to Autophagic Vacuoles
  52. Tumor cells expressing tissue factor influence the migration of smooth muscle cells in a catalytic activity-dependent way
  53. Intracellular sequestration of amiodarone: role of vacuolar ATPase and macroautophagic transition of the resulting vacuolar cytopathology
  54. NTPDase1 (CD39) controls nucleotide-dependent vasoconstriction in mouse
  55. Angiotensin converting enzyme inhibitor induced angio-oedema: a review of the pathophysiology and risk factors
  56. Receptor tyrosine kinases as mediators of injury-induced bradykinin B1 receptor expression in rabbit aortic smooth muscle
  57. Fluorescent Ligands of the Bradykinin B1 Receptors: Pharmacologic Characterization and Application to the Study of Agonist-Induced Receptor Translocation and Cell Surface Receptor Expression
  58. A fluorescent version of the bradykinin B2 receptor antagonist B-9430: Pharmacological characterization and use in live cell imaging
  59. Therapeutic options in inflammatory bowel disease: experimental evidence of a beneficial effect of kinin B1 receptor blockade
  60. Receptor-independent, vacuolar ATPase-mediated cellular uptake of histamine receptor-1 ligands: Possible origin of pharmacological distortions and side effects
  61. Intense pseudotransport of a cationic drug mediated by vacuolar ATPase: Procainamide-induced autophagic cell vacuolization
  62. Lack of direct interaction between enalaprilat and the kinin B1 receptors
  63. Structural modification of the highly potent peptide bradykinin B1 receptor antagonist B9958
  64. Cardiovascular expression of inflammatory signaling molecules, the kinin B1 receptor and COX2, in the rabbit: Effects of LPS, anti-inflammatory and anti-hypertensive drugs
  65. Trapping of adrenergic decongestant drugs into cellular endomembrane compartments: Toxicological and pharmacological consequences
  66. B-9972 (D-Arg-[Hyp3,Igl5,Oic7,Igl8]-bradykinin) Is an Inactivation-Resistant Agonist of the Bradykinin B2 Receptor Derived from the Peptide Antagonist B-9430 (D-Arg-[Hyp3,Igl5,D-Igl7,Oic8]-bradykinin): Pharmacologic Profile and Effective Induction of R...
  67. Ô miroir, dis-moi comment les amines effacent les rides
  68. Does zaltoprofen antagonize the bradykinin receptors?
  69. Generation of kinins during preparation and storage of whole blood?derived platelet concentrates
  70. The antiwrinkle effect of topical concentrated 2-dimethylaminoethanol involves a vacuolar cytopathology
  71. Antagonist, partial agonist and antiproliferative actions of B-9870 (CU201) as a function of the expression and density of the bradykinin B1 and B2 receptors
  72. Bradykinin Receptors
  73. B-2 Bradykinin Receptor
  74. B-1 Bradykinin Receptor
  75. Role of Nuclear Factor-κB and Protein Kinase C Signaling in the Expression of the Kinin B1 Receptor in Human Vascular Smooth Muscle Cells
  76. The bradykinin B2 receptor antagonist icatibant (Hoe 140) blocks aminopeptidase N at micromolar concentrations: Off-target alterations of signaling mediated by the bradykinin B1 and angiotensin receptors
  77. Inhibition of human and rabbit arterial smooth muscle cell migration mediated by the kinin B 1 receptor: role of receptor density and released mediators
  78. Advances in the Development of Bradykinin Receptor Ligands
  79. Molecular identification and pharmacological profile of the bovine kinin B1 receptor
  80. A Nonpeptide Antagonist Reveals a Highly Glycosylated State of the Rabbit Kinin B1 Receptor
  81. Dual antagonists of the bradykinin B1 and B2 receptors based on a postulated common pharmacophore from existing non-peptide antagonists
  82. Discovery of a Dual-Function Peptide That Combines Aminopeptidase N Inhibition and Kinin B1Receptor Antagonism
  83. N-Substituted 4-Aminobenzamides (Procainamide Analogs): An Assessment of Multiple Cellular Effects Concerning Ion Trapping
  84. Expression of Metallopeptidases and Kinin Receptors in Swine Oropharyngeal Tissues: Effects of Angiotensin I-Converting Enzyme Inhibition and Inflammation
  85. Endogenous Aminopeptidase N Decreases the Potency of Peptide Agonists and Antagonists of the Kinin B1 Receptors in the Rabbit Aorta
  86. A possible common pharmacophore in the non-peptide antagonists of the bradykinin B1 receptor
  87. International Union of Pharmacology. XLV. Classification of the Kinin Receptor Family: from Molecular Mechanisms to Pathophysiological Consequences
  88. Studies on rabbit natural and recombinant tissue factors: intracellular retention and regulation of surface expression in cultured cells
  89. The Kallikrein-Kinin System: Current and Future Pharmacological Targets
  90. Bradykinin receptor ligands: therapeutic perspectives
  91. A Novel Nonpeptide Antagonist of the Kinin B1 Receptor: Effects at the Rabbit Receptor
  92. Massive Cell Vacuolization Induced by Organic Amines Such as Procainamide
  93. Loss of function of vascular smooth muscle cells by nitric oxide-dependent and -independent interactions with tumorigenic cells
  94. A non-peptide antagonist unusually selective for the human form of the bradykinin B2 receptor
  95. Wortmannin alters the intracellular trafficking of the bradykinin B2 receptor: role of phosphoinositide 3-kinase and Rab5
  96. Characterization of a fluorescent conjugate of the rabbit angiotensin AT1 receptor
  97. Do angiotensin-converting enzyme inhibitors directly stimulate the kinin B1receptor?
  98. Tissue Kallikrein Actions at the Rabbit Natural or Recombinant Kinin B2 Receptors
  99. High agonist-independent clearance of rabbit kinin B1receptors in cultured cells
  100. Kinin receptors: functional aspects
  101. Contractile Effect of Anaphylatoxin C5a and of a Mimetic Peptide on the Human Umbilical Artery: Further Evidence for Leukocyte-Dependent Vasomotion
  102. Bradykinin B 2 receptor gene polymorphism is associated with altered urinary albumin/creatinine values in diabetic patients
  103. Expression of kinin B1receptor in fresh or cultured rabbit aortic smooth muscle: role of NF-κB
  104. Agonist-Induced Translocation of the Kinin B1Receptor to Caveolae-Related Rafts
  105. Effects of two novel non-peptide antagonists at the rabbit bradykinin B2 receptor
  106. Absence of ligand-induced regulation of kinin receptor expression in the rabbit
  107. Ligand-Mediated Regulation of Kinin Receptors in the Rabbit
  108. The contribution of angiotensin-converting enzyme (ACE) to the metabolism of kinins (bradykinin and des-Arg9-bradykinin) and effect of ACE inhibitors on their in vitro and in vivo metabolism
  109. The kallikrein-kininogen-kinin system: lessons from the quantification of endogenous kinins
  110. Altered frequency of a promoter polymorphism of the kinin B2 receptor gene in hypertensive African-Americans
  111. Non-competitive pharmacological antagonism at the rabbit B1 receptor
  112. In vivo protein-DNA interactions at the kinin B1 receptor gene promoter: No modification on interleukin-1 beta or lipopolysaccharide induction
  113. Antagonist-Induced Intracellular Sequestration of Rabbit Bradykinin B2 Receptor
  114. Inflammatory hyperalgesia induced by zymosan in the plantar tissue of the rat: effect of kinin receptor antagonists
  115. Cloning and preliminary pharmacological characterization of the anaphylatoxin C5a receptor in the rabbit
  116. Characterization of a polymorphism in the coding region of the human C5a anaphylatoxin receptor
  117. Kinin receptors
  118. Interleukin 8 (IL-8) Induces the Expression of Kinin B1Receptor in Human Lung Fibroblasts
  119. Altered frequency of a promoter polymorphic allele of the kinin B receptor gene in inflammatory bowel disease
  120. Down-regulation of interleukin-1β production and PGE2 accumulation by an indomethacin-phenylalanine derivative in human monocytes
  121. Human kallikrein hK2 has low kininogenase activity while prostate-specific antigen (hK3) has none
  122. The kinin B 1 receptor: an inducible G protein coupled receptor
  123. Oxidative Stress Induced Actin Reorganization Mediated by the p38 Mitogen-Activated Protein Kinase/Heat Shock Protein 27 Pathway in Vascular Endothelial Cells
  124. Kinin B1 Receptor Induction and Inflammination
  125. The kinin B1 receptor: an inducible G protein coupled receptor
  126. Evidence for vascular tone regulation by resident or infiltrating leukocytes
  127. Mechanism of the contractile effect of diaspirin-cross-linked hemoglobin in rat isolated aorta strip denuded of endothelium as revealed using an oil-immersion procedure
  128. Structure and Genomic Organization of the Human B1Receptor Gene for Kinins (BDKRB1)
  129. Mechanism of the contractile effect of diaspirin-cross-linked hemoglobin in rat isolated aorta strip denuded of endothelium as revealed using an oil-immersion procedure
  130. Regulation of kinin-induced contraction and DNA synthesis by inflammatory cytokines in the smooth muscle of the rabbit aorta
  131. Mode of action of thrombin in the rabbit aorta
  132. Kinin B1 receptors: a review
  133. Recombinant Human Hemoglobin (rHb1.1) Selectively Inhibits Vasorelaxation Elicited by Nitric Oxide Donors in Rabbit Isolated Aortic Rings
  134. Development of a binding assay for the B1 receptors for kinins
  135. Quantification of des-Arg9-bradykinin using a chemiluminescence enzyme immunoassay: application to its kinetic profile during plasma activation
  136. Inflammatory Peptides at the Beginning of Hemodialysis in Asymptomatic Patients Treated or Not with Angiotensin l-Converting Inhibitors
  137. Further analysis of the upregulation of bradykinin B1 receptors in isolated rabbit aorta by using metabolic inhibitors
  138. Recombinant Human Hemoglobin Inhibits Both Constitutive and Cytokine-Induced Nitric Oxide-Mediated Relaxation of Rabbit Isolated Aortic Rings
  139. Recombinant Human Hemoglobin Inhibits Both Constitutive and Cytokine-Induced Nitric Oxide-Mediated Relaxation of Rabbit Isolated Aortic Rings
  140. Epidermal growth factor-induced rapid relaxation of the isolated rabbit mesenteric artery
  141. The nonpeptide WIN 64338 is a bradykinin B2 receptor antagonist.
  142. Aminopeptidase modulation of the pharmacological responses to synthetic thrombin receptor agonists
  143. Vascular mode of action of kinin B1 receptors and development of a cellular model for the investigation of these receptors
  144. Synthetic C5a receptor agonists
  145. Synthesis and pharmacological evaluation of amide derivatives of non-steroidal anti-inflammatory drugs
  146. Dissociation of the antimicrobial activity of bacitracin USP from its renovascular effects.
  147. Effects of experimental conditions on the production of interleukin-1α and -1β by human endothelial cells cultured in vitro
  148. Synergism between the contractile effect of epidermal growth factor and that of des-Arg9-bradykinin or of α.-thrombin in rabbit aortic rings
  149. Comparison of two classes of non-peptide drugs as antagonists of neutrophil receptors for f-Met-Leu-Phe
  150. Human interleukin-1 induces a rapid relaxation of the rabbit isolated mesenteric artery
  151. Pulse exposure to protein synthesis inhibitors enhances vascular responses to des-Arg9-bradykinin: possible role of interleukin-1
  152. The interaction of 3,5-pyrazolidinedione drugs with receptors for f-Met-Leu-Phe on human neutrophil leukocytes: a study of the structure–activity relationship
  153. Long-term culture and characterization of human limbal microvascular endothelial cells
  154. Contractile effect of the chemotactic factors f-Met-Leu-Phe and C5a on the human isolated umbilical artery. Role of cyclooxygenase products and tissue macrophages
  155. Pharmacological modulation of interleukin 1 production by cultured endothelial cells from human umbilical veins
  156. Bacitracin U.S.P. contains a factor that stimulates receptors for 5-hydroxytryptamine on rabbit aortic strips
  157. Pharmacological modulation of the up-regulated responses to des-Arg9-bradykinin in vivo and in vitro
  158. Prostacyclin release induced by neurokinins in cultured human endothelial cells
  159. Small fibronectin fragments induce endothelium-dependent vascular relaxations
  160. Effect of glucocorticoids, monokines and growth factors on the spontaneously developing responses of the rabbit isolated aorta to des-Arg9-bradykinin
  161. Studies on the effects of disease-modifying antirheumatic drugs on lipoxygenase product synthesis in human neutrophils in vitro
  162. Effects of the anaphylatoxins on circulation
  163. The ability of des-Arg9-bradykinin to relax rabbit isolated mesenteric arteries is acquired during in vitro incubation
  164. Studies on the induction of pharmacological responses to des-Arg9-bradykinin in vitro and in vivo
  165. Effects of low molecular weight fibrin degradation products 6A and 6D on rabbit aorta strips
  166. Carboxypeptidase N (Kininase I) activity in blood and synovial fluid from patients with arthritis
  167. Mitogenic effect of bradykinin and of des-Arg9-bradykinin on cultured fibroblasts
  168. Anaphylatoxin C5a fails to promote prostacyclin release in cultured endothelial cells from human umbilical veins
  169. Effects of the C5a anaphylatoxin and its relationship to cyclo-oxygenase metabolites in rabbit vascular strips
  170. Selective Induction of Cardiovascular Responses to des-Arg9-Bradykinin by Bacterial Endotoxin
  171. Rapid assay of human plasma carboxypeptidase N by high-performance liquid chromatographic separation of hippuryl-lysine and its product
  172. Pharmacology of kinins: Their relevance to tissue injury and inflammation
  173. Kininases and vascular responses to kinins
  174. Pharmacological characterization of the vascular permeability enhancing effects of kinins in the rabbit skin
  175. Induction of B1-receptors for kinins in the rabbit by a bacterial lipopolysaccharide
  176. The degradation of bradykinin (BK) and of des-Arg 9 -BK in plasma
  177. Kinin receptors in experimental inflammation
  178. Cardiovascular actions of kinins in the rabbit
  179. De novo formation of vascular receptors for bradykinin
  180. The rabbit mesenteric vein: a specific bioassay for substance P