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  1. Assessment of the Physicochemical Properties and Stability for Pharmacokinetic Prediction of Pyrazinoic Acid Derivatives

    Article • Current Drug Metabolism, December 2020, Bentham Science Publishers

    Dr Joao Paulo dos Santos Fernandes , Taisa Franchin

  2. Natural Products: Key Prototypes to Drug Discovery Against Neglected Diseases Caused by Trypanosomatids

    Article • Current Medicinal Chemistry, April 2020, Bentham Science Publishers

    Dr Joao Paulo dos Santos Fernandes

  3. Targeting the Histamine H4 Receptor: Future Drugs for Inflammatory Diseases

    Article • Current Organic Chemistry, October 2018, Bentham Science Publishers

    Dr Joao Paulo dos Santos Fernandes

  4. Pyrazinoates as antiparasitic agents against Trypanosoma cruzi

    Article • Archiv der Pharmazie, October 2018, Wiley

    Dr Joao Paulo dos Santos Fernandes

  5. Antiparasitic activity of new gibbilimbol analogues and SAR analysis through efficiency and statistical methods

    Article • European Journal of Pharmaceutical Sciences, September 2018, Elsevier

    Dr Joao Paulo dos Santos Fernandes

  6. Pharmacological and SAR analysis of the LINS01 compounds at the human histamine H1 , H2 and H3 receptors

    Article • August 2018, Wiley

    Dr Joao Paulo dos Santos Fernandes

  7. QSAR Modeling of Histamine H3R Antagonists/inverse Agonists as Future Drugs for Neurodegenerative Diseases

    Article • Current Neuropharmacology, June 2018, Bentham Science Publishers

    Dr Joao Paulo dos Santos Fernandes

  8. The Importance of Medicinal Chemistry Knowledge in the Clinical Pharmacist’s Education

    Article • American Journal of Pharmaceutical Education, March 2018, American Journal of Pharmaceutical Education

    Dr Joao Paulo dos Santos Fernandes

  9. Pharmacological Characterization of 5-Substituted 1-[(2,3-dihydro-1-benzofuran-2-yl)methyl]piperazines: Novel Antagonists for the Histamine H3 and H4 Receptors with Anti-inflammatory Potential

    Article • Frontiers in Pharmacology, November 2017, Frontiers

    Dr Joao Paulo dos Santos Fernandes

  10. Evaluation of β-Aminocarboxylic Acid Derivatives in Hippocampal Excitatory Synaptic Transmission

    Article • Archiv der Pharmazie, September 2017, Wiley

    Dr Joao Paulo dos Santos Fernandes

  11. New alkenyl derivative from Piper malacophyllum and analogues: Antiparasitic activity against Trypanosoma cruzi and Leishmania infantum

    Article • Chemical Biology & Drug Design, May 2017, Wiley

    Dr Joao Paulo dos Santos Fernandes

  12. 1-[(2,3-Dihydro-1-benzofuran-2-yl) methyl]piperazines as novel anti-inflammatory compounds: Synthesis and evaluation on H3R/H4R

    Article • Chemical Biology & Drug Design, February 2017, Wiley

    Dr Joao Paulo dos Santos Fernandes , PhD Lanfranco R. P. Troncone

  13. Factorial study to assess an ultrasonic methodology for the allylation of 4-chloroaniline

    Article • Green Processing and Synthesis, January 2017, De Gruyter

    Dr Joao Paulo dos Santos Fernandes

  14. Antimycobacterial activity of pyrazinoate prodrugs in replicating and non-replicating Mycobacterium tuberculosis

    Article • Tuberculosis, July 2016, Elsevier

    Dr Joao Paulo dos Santos Fernandes

  15. Pyrazinamide and Pyrazinoic Acid Derivatives Directed to Mycobacterial Enzymes Against Tuberculosis

    Article • Current Protein and Peptide Science, March 2016, Bentham Science Publishers

    Dr Joao Paulo dos Santos Fernandes

  16. Gibbilimbol analogues as antiparasitic agents—Synthesis and biological activity against Trypanosoma cruzi and Leishmania (L.) infantum

    Article • Bioorganic & Medicinal Chemistry Letters, February 2016, Elsevier

    Dr Joao Paulo dos Santos Fernandes

  17. Factorial design study to access the “green” iodocyclization reaction of 2-allylphenols

    Article • Green Processing and Synthesis, January 2016, De Gruyter

    Dr Joao Paulo dos Santos Fernandes

  18. Histamine H4 Receptor Ligands: Future Applications and State of Art

    Article • Chemical Biology & Drug Design, October 2014, Wiley

    Dr Joao Paulo dos Santos Fernandes

  19. Synthesis and evaluation of a pyrazinoic acid prodrug in Mycobacterium tuberculosis

    Article • Saudi Pharmaceutical Journal, September 2014, Elsevier

    Dr Joao Paulo dos Santos Fernandes

  20. Estudo das relações entre estrutura e atividade de parabenos: uma aula prática

    Article • Química Nova, January 2013, FapUNIFESP (SciELO)

    Dr Joao Paulo dos Santos Fernandes

  21. Cytotoxicity evaluation ofCurcuma zedoaria(Christm.) Roscoe fluid extract used in oral hygiene products

    Article • Acta Odontologica Scandinavica, January 2012, Taylor & Francis

    Dr Joao Paulo dos Santos Fernandes

  22. Optimization of the ultrasound-assisted synthesis of allyl 1-naphthyl ether using response surface methodology

    Article • Ultrasonics Sonochemistry, March 2011, Elsevier

    Dr Joao Paulo dos Santos Fernandes

  23. Molecular modeling and QSAR studies of a set of indole and benzimidazole derivatives as H4 receptor antagonists

    Article • Journal of Molecular Modeling, July 2010, Springer Science + Business Media

    Dr Joao Paulo dos Santos Fernandes

  24. QSAR Modeling of a Set of Pyrazinoate Esters as Antituberculosis Prodrugs

    Article • Archiv der Pharmazie, January 2010, Wiley

    Dr Joao Paulo dos Santos Fernandes

  25. Simple and Efficient Access to 3-Ethoxycarbonylpyrroles, Benzofurans, and Naphthofurans

    Article • Synthesis, October 2009, Thieme Publishing Group

    Dr Joao Paulo dos Santos Fernandes

  26. Evaluation of the influence of base and alkyl bromide on synthesis of pyrazinoic acid esters through fatorial design

    Article • Química Nova, January 2009, FapUNIFESP (SciELO)

    Dr Joao Paulo dos Santos Fernandes

  27. Planejamento e sintese de compostos potencialmente ligantes dos receptores 5-HT2C e H4

    Article • Universidade de Sao Paulo Sistema Integrado de Bibliotecas - SIBiUSP

    Dr Joao Paulo dos Santos Fernandes

  28. Síntese e atividade antimicobacteriana de ésteres do ácido pirazinóico e quinolonas

    Article • Universidade de Sao Paulo Sistema Integrado de Bibliotecas - SIBiUSP

    Dr Joao Paulo dos Santos Fernandes