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  1. Chemical and biological insights into 3-arylphenytoins as urease inhibitors: Design, synthesis, in vitro and in silico studies

    Article • January 2026, Elsevier

    Dr. Syed Muhammad Saad

  2. In vitro and In silico Xanthine Oxidase Inhibitory Activities of 3-Aryl-2- thioxo-2,3-dihydroquinazolin-4(1H)-one Derivatives

    Article • Medicinal Chemistry, May 2023, Bentham Science Publishers

    Dr. Syed Muhammad Saad, Muhammad Iqbal Choudhary

  3. New synthetic phenylquinazoline derivatives induce apoptosis by targeting the pro-survival members of the BCL-2 family

    Article • Bioorganic & Medicinal Chemistry Letters, July 2022, Elsevier

    Dr. Syed Muhammad Saad

  4. Potential anti-acanthamoebic effects through inhibition of CYP51 by novel quinazolinones

    Article • Acta Tropica, July 2022, Elsevier

    Dr. Syed Muhammad Saad

  5. Biology‐oriented drug synthesis and evaluation of secnidazole esters as novel enzyme ınhibitors

    Article • Archiv der Pharmazie, December 2021, Wiley

    Dr. Syed Muhammad Saad, Prof. Dr Tugba Taskin-Tok

  6. An effort to find new α-amylase inhibitors as potent antidiabetics compounds based on indole-based-thiadiazole analogs

    Article • Journal of Biomolecular Structure and Dynamics, September 2021, Taylor & Francis

    Dr. Syed Muhammad Saad

  7. Antioxidant and ROS Inhibitory Activities of Heterocyclic 2-Aryl-4(3H)-quinazolinone Derivatives

    Article • Letters in Drug Design & Discovery, August 2021, Bentham Science Publishers

    Muhammad Iqbal Choudhary, Dr SHAHIDA PERVEEN, Dr. Syed Muhammad Saad

  8. Rapid Cesium Fluoride Catalyzed Synthesis of 5-Aryloxy-1-phenyl-1H-tetrazoles via Nucleophilic Aromatic Substitution

    Article • Letters in Organic Chemistry, July 2020, Bentham Science Publishers

    SHAHNAZ PERVEEN, Dr. Syed Muhammad Saad

  9. Antiamoebic activity of 3-aryl-6,7-dimethoxyquinazolin-4(3H)-one library against Acanthamoeba castellanii

    Article • Parasitology Research, June 2020, Springer Science + Business Media

    Dr. Syed Muhammad Saad

  10. Article • Pakistan Journal of Pharmaceutical Sciences, May 2020, Faculty of Pharmacy and Pharmaceutical Sciences, University of Karachi

    Dr. Syed Muhammad Saad

  11. Thymidine phosphorylase and prostrate cancer cell proliferation inhibitory activities of synthetic 4-hydroxybenzohydrazides: In vitro, kinetic, and in silico studies

    Article • PLOS One, January 2020, PLOS

    Dr. Syed Muhammad Saad

  12. Aryl Quinazolinone Derivatives as Novel Therapeutic Agents against Brain-Eating Amoebae

    Article • ACS Chemical Neuroscience, January 2020, American Chemical Society (ACS)

    Dr. Syed Muhammad Saad

  13. Facile CuCl2·2H2O catalyzed one-pot conversion of dimedone into highly functionalized indazole based N-arylhydrazinecarbothioamides

    Article • Journal of Saudi Chemical Society, January 2020, Elsevier

    Dr. Syed Muhammad Saad

  14. Novel antiacanthamoebic compounds belonging to quinazolinones

    Article • European Journal of Medicinal Chemistry, November 2019, Elsevier

    Dr. Syed Muhammad Saad

  15. Synthesis, molecular docking and xanthine oxidase inhibitory activity of 5-aryl-1H-tetrazoles

    Article • Bioorganic Chemistry, September 2018, Elsevier

    Dr. Syed Muhammad Saad

  16. Coumarin sulfonates: As potential leads for ROS inhibition

    Article • Bioorganic Chemistry, December 2016, Elsevier

    Dr. Syed Muhammad Saad

  17. Synthesis and urease inhibitory activities of benzophenone semicarbazones/thiosemicarbazones

    Article • Medicinal Chemistry Research, August 2016, Springer Science + Business Media

    Dr. Syed Muhammad Saad

  18. Synthesis, molecular docking and α-glucosidase inhibition of 5-aryl-2-(6′-nitrobenzofuran-2′-yl)-1,3,4-oxadiazoles

    Article • Bioorganic Chemistry, June 2016, Elsevier

    Dr. Syed Muhammad Saad

  19. Microwave-assisted green approach toward the unexpected synthesis of pyrazole-4-carboxylates

    Article • Journal of the Iranian Chemical Society, April 2016, Springer Science + Business Media

    Dr. Syed Muhammad Saad

  20. Synthesis, α-glucosidase inhibitory, cytotoxicity and docking studies of 2-aryl-7-methylbenzimidazoles

    Article • Bioorganic Chemistry, April 2016, Elsevier

    Dr. Syed Muhammad Saad

  21. An efficient one-pot protocol for the conversion of benzaldehydes into tetrazole analogs

    Article • Tetrahedron Letters, February 2016, Elsevier

    Dr. Syed Muhammad Saad

  22. 2-Arylquinazolin-4(3H)-ones: Inhibitory Activities Against Xanthine Oxidase

    Article • Medicinal Chemistry, January 2016, Bentham Science Publishers

    Dr. Syed Muhammad Saad

  23. 4-Arylamino-6-nitroquinazolines: Synthesis and their activities against neglected disease leishmaniasis

    Article • European Journal of Medicinal Chemistry, January 2016, Elsevier

    Dr. Syed Muhammad Saad

  24. Evaluation of 2-indolcarbohydrazones as potent α-glucosidase inhibitors, in silico studies and DFT based stereochemical predictions

    Article • Bioorganic Chemistry, December 2015, Elsevier

    Dr. Syed Muhammad Saad

  25. 2-Arylquinazolin-4(3H)-ones: A new class of α-glucosidase inhibitors

    Article • Bioorganic & Medicinal Chemistry, December 2015, Elsevier

    Dr. Syed Muhammad Saad

  26. 2-Arylquinazolin-4(3H)-ones: A novel class of thymidine phosphorylase inhibitors

    Article • Bioorganic Chemistry, December 2015, Elsevier

    Dr. Syed Muhammad Saad

  27. Corrigendum to “2-Arylquinazolin-4(3H)-ones: A new class of α-glucosidase inhibitors” [Bioorg. Med. Chem. 23 (2015) 7417–7421]

    Article • Bioorganic & Medicinal Chemistry, December 2015, Elsevier

    Dr. Syed Muhammad Saad

  28. Synthesis of new oxadiazole derivatives as α-glucosidase inhibitors

    Article • Bioorganic & Medicinal Chemistry, August 2015, Elsevier

    Dr. Syed Muhammad Saad

  29. Synthesis and Biological Potential Assessment of 2-Substituted Quinazolin-4(3H)-ones as Inhibitors of Phosphodiesterase-I and Carbonic Anhydrase-II

    Article • Medicinal Chemistry, April 2015, Bentham Science Publishers

    Dr. Syed Muhammad Saad

  30. A new and facile CuCl2·2H2O-catalyzed one-pot three-component synthesis for quinazolines

    Article • Monatshefte für Chemie - Chemical Monthly, March 2015, Springer Science + Business Media

    Dr. Syed Muhammad Saad

  31. Synthesis of phenyl thiazole hydrazones and their activity against glycation of proteins

    Article • Medicinal Chemistry Research, March 2015, Springer Science + Business Media

    Dr. Syed Muhammad Saad

  32. Synthesis of triazole Schiff bases: Novel inhibitors of nucleotide pyrophosphatase/phosphodiesterase-1

    Article • Bioorganic & Medicinal Chemistry, November 2014, Elsevier

    Muhammad Saleem, Dr. Syed Muhammad Saad

  33. β-Glucuronidase Inhibitory Studies on Coumarin Derivatives

    Article • Medicinal Chemistry, October 2014, Bentham Science Publishers

    Dr. Syed Muhammad Saad

  34. Oxadiazoles and thiadiazoles: Novel α-glucosidase inhibitors

    Article • Bioorganic & Medicinal Chemistry, October 2014, Elsevier

    Dr. Syed Muhammad Saad

  35. WITHDRAWN: 2-Arylquinazolin-4(3H)-ones: A new class of α-glucosidase inhibitors

    Article • Bioorganic & Medicinal Chemistry, October 2014, Elsevier

    Dr. Syed Muhammad Saad

  36. Synthesis and β-glucuronidase inhibitory activity of 2-arylquinazolin-4(3H)-ones

    Article • Bioorganic & Medicinal Chemistry, July 2014, Elsevier

    Dr. Syed Muhammad Saad

  37. 2-{[(Dimethylamino)methylidene]amino}-5-nitrobenzonitrile

    Article • Acta Crystallographica Section E Structure Reports Online, December 2012, International Union of Crystallography

    Dr. Syed Muhammad Saad

  38. N-(2,5-Dimethoxyphenyl)-6-nitroquinazolin-4-amine

    Article • Acta Crystallographica Section E Structure Reports Online, December 2012, International Union of Crystallography

    Dr. Syed Muhammad Saad

  39. N′-(3-Chlorobenzylidene)-4-hydroxybenzohydrazide

    Article • Acta Crystallographica Section E Structure Reports Online, November 2012, International Union of Crystallography

    Dr. Syed Muhammad Saad

  40. Ethyl (E)-3-(6-methyl-4-oxo-4H-chromen-3-yl)prop-2-enoate

    Article • Acta Crystallographica Section E Structure Reports Online, September 2012, International Union of Crystallography

    Dr. Syed Muhammad Saad

  41. 6-Methyl-4-oxo-4H-chromene-3-carbaldehyde

    Article • Acta Crystallographica Section E Structure Reports Online, September 2012, International Union of Crystallography

    Dr. Syed Muhammad Saad