All Stories

  1. An Improved Synthesis of Glucuronide Metabolites of Hindered Phenolic Xenoestrogens

    Article • Current Organic Synthesis, November 2022, Bentham Science Publishers

    Medicinal chemist René Maltais

  2. Insight into the Mechanism of 17β-Hydroxysteroid Dehydrogenase Type 3 Inhibition by the Androsterone Derivative RM-532-105

    Article • Current Enzyme Inhibition, July 2020, Bentham Science Publishers

    Medicinal chemist René Maltais, Preyesh Stephen

  3. Parallel Solid-Phase Synthesis using a New Diethylsilylacetylenic Linker and Leading to Mestranol Derivatives with Potent Antiproliferative Activities on Multiple Cancer Cell Lines

    Article • Anti-Cancer Agents in Medicinal Chemistry, January 2019, Bentham Science Publishers

    Dr Donald Poirier, Medicinal chemist René Maltais

  4. NMR-Assisted Structure Elucidation of an Anticancer Steroid-β-Enaminone Derivative

    Article • Magnetochemistry, November 2017, MDPI AG

    Medicinal chemist René Maltais

  5. Solid-phase synthesis of libraries of ethynylated aminosteroid derivatives as potential antileukemic agents

    Article • Steroids, March 2016, Elsevier

    Medicinal chemist René Maltais

  6. A Potent Inhibitor of Steroid Sulfatase (EM-1913) Blocks Tumor Growth in Nude Mice (MCF-7 Xenograft)

    Article • Current Enzyme Inhibition, July 2015, Bentham Science Publishers

    Medicinal chemist René Maltais

  7. Development of a Simple and Efficient Solution-Phase Parallel Synthesis of Flexible Non-Steroidal Estradiol Mimics

    Article • Combinatorial Chemistry & High Throughput Screening, November 2014, Bentham Science Publishers

    Medicinal chemist René Maltais

  8. Synthesis of an Estradiol Derivative with an Adenosine-phosphate Mimic Linked at Position 16β

    Article • Current Organic Synthesis, July 2014, Bentham Science Publishers

    Medicinal chemist René Maltais

  9. Identification of a First Enzymatic Activator of a 17β-Hydroxysteroid Dehydrogenase

    Article • ACS Chemical Biology, June 2014, American Chemical Society (ACS)

    Medicinal chemist René Maltais

  10. Diversity-Oriented Synthesis of Spiro- and Fused Azacycles from Ketone Molecular Templates

    Article • European Journal of Organic Chemistry, August 2012, Wiley

    Medicinal chemist René Maltais

  11. Steroid sulfatase inhibitors: A review covering the promising 2000–2010 decade

    Article • Steroids, September 2011, Elsevier

    Medicinal chemist René Maltais

  12. Convergent stereoselective and efficient synthesis of furanic-steroid derivatives

    Article • Tetrahedron, April 2011, Elsevier

    Medicinal chemist René Maltais

  13. Solid-Phase Organic Synthesis (SPOS) of Modulators of Estrogenic and Androgenic Action

    Article • ChemInform, September 2006, Wiley

    Medicinal chemist René Maltais

  14. Steroids and Combinatorial Chemistry

    Article • ChemInform, September 2004, Wiley

    Medicinal chemist René Maltais

  15. Steroids and Combinatorial Chemistry

    Article • Journal of Combinatorial Chemistry, May 2004, American Chemical Society (ACS)

    Medicinal chemist René Maltais

  16. Solid-Phase Synthesis of Hydroxysteroid Derivatives Using the Diethylsilyloxy Linker

    Article • Journal of Combinatorial Chemistry, October 2000, American Chemical Society (ACS)

    Medicinal chemist René Maltais

  17. Efficient coupling and solid-phase synthesis of steroidal ketone derivative using polymer-bound glycerol

    Article • Tetrahedron Letters, March 2000, Elsevier

    Medicinal chemist René Maltais

  18. The Sulfamate Functional Group as a New Anchor for Solid-Phase Organic Synthesis

    Article • Organic Letters, January 2000, American Chemical Society (ACS)

    Medicinal chemist René Maltais

  19. Steroid sulfatase inhibitors

    Article • Expert Opinion on Therapeutic Patents, August 1999, Informa Healthcare

    Medicinal chemist René Maltais

  20. A solution-phase combinatorial parallel synthesis of 3β-amido-3α-hydroxy-5α-androstane-17-ones

    Article • Tetrahedron Letters, June 1998, Elsevier

    Medicinal chemist René Maltais