All Stories

  1. Rapid and Efficient Radiolabeling of Short Peptides
  2. Thymidine-Inosine Dimer Building Block for Reversible Modification of Synthetic Oligonucleotides
  3. Anti-HIV and Antimicrobial Activity of 7-Hydrazino-8-hydroxyquinoline-Based Aromatic Hydrazones
  4. Synthesis of Chroman Derivatives by Group Transposition and Atom Swapping in 1‐Tetralones: Single‐Atom Editing Enabled by Oxidative Ring Contraction of Benzoxepine Silyl Ketene Acetals
  5. Redesigning methionine γ-lyase for improved stability and catalytic activity in the β-elimination reaction for the synthesis of thiosulfinates
  6. Piperazine-Substituted Pyranopyridines Exhibit Antiproliferative Activity and Act as Inhibitors of HBV Virion Production
  7. Distinct N6-Substituted Adenosine Derivatives Exhibit Receptor-Specific Anticytokinin Action by Unknown Non-competitive Mechanism
  8. Improved Synthesis of Effective 3-(Indolin-6-yl)-4-(N-pyrazole-sulfonamide)-1H-pyrrolo[2,3-b]pyridine-Based Inhibitors of NADPH Oxidase 2
  9. Revealing O-acetylhomoserine sulfhydrylase involved in direct sulfhydrylation pathway in Clostridium tetani
  10. 6-Bromoindole- and 6-Bromoindazole-Based Inhibitors of Bacterial Cystathionine γ-Lyase Containing 3-Aminothiophene-2-Carboxylate Moiety
  11. Synthesis of daidzein derivatives for targeted drug delivery
  12. Development of a New Inhibitor of Bacterial Cystathionine γ-Lyase Based on 6-Bromoindole and Aminothiophene
  13. Synthesis and Antimicrobial Activity of Thiosulfinates and Allicin Analogues
  14. Toxicity Study of the Pharmacological Pair of Encapsulated Citrobacter freundii C115H Methionine γ-Lyase/Methiin
  15. Bacterial Purine Nucleoside Phosphorylases from Mesophilic and Thermophilic Sources: Characterization of Their Interaction with Natural Nucleosides and Modified Arabinofuranoside Analogues
  16. Synthesis of Isoquinoline‐Containing 5,6‐Dicyano‐2,1,3‐Benzothiadiazoles: Unusual Heterocyclization into Dibenzo‐1,6‐Naphthyridine Framework
  17. O-Acetylhomoserine Sulfhydrylase As a Key Enzyme of Direct Sulfhydrylation in Microbial Methionine Biosynthesis (A Review)
  18. A convenient synthesis of a chlorobenzothiophenyl-indole-based inhibitor of bacterial cystathionine γ-lyase
  19. Synthesis of Spiro[imidazole‐4,3′‐pyrrolo[1,2‐a]quinolin]‐ 5‐ones via 1,3‐Dipolar Cycloaddition of Quinolinium Ylides with Arylydeneimidazol‐4‐ones
  20. Novel Hydroxamic Acids Containing Aryl-Substituted 1,2,4- or 1,3,4-Oxadiazole Backbones and an Investigation of Their Antibiotic Potentiation Activity
  21. Anticandidal Activity of In Situ Methionine γ-Lyase-Based Thiosulfinate Generation System vs. Synthetic Thiosulfinates
  22. 5-Alkyloxymethyl Derivatives of 2ʹ-Deoxyuridine Bearing 2,4-Dinitrophenyl and Dansyl Groups: Synthesis and Antibacterial Activity
  23. Examination of Diels–Alder/Tsuji–Trost Route towards Kopsia Alkaloids
  24. 5‐Substituted Uridines with Activity against Gram‐Positive Bacteria
  25. Thiosulfinates: Cytotoxic and Antitumor Activity
  26. Merging Johnson–Claisen and Aromatic Claisen [3,3]-Sigmatropic Rearrangements: Ytterbium Triflate/2,6-Di-tert-butylpyridine Catalytic System
  27. Antibacterial Conjugates of Kanamycin A with Vancomycin and Eremomycin: Biological Activity and a New MS-Fragmentation Pattern of Cbz-Protected Amines
  28. Synthesis of the Indole-Based Inhibitors of Bacterial Cystathionine γ-Lyase NL1-NL3
  29. Synthesis of Cy5-Labelled C5-Alkynyl-modified cytidine triphosphates via Sonogashira coupling for DNA labelling
  30. Synthetic Optimizations for Gram-Scale Preparation of 1-O-Methyl d-Glycero-α-d-gluco-heptoside 7-Phosphate from d-Glucose
  31. HFIP‐Mediated CH Functionalization
  32. Oligoglycol carbonate prodrugs of 5-modified 2'-deoxyuridines: synthesis and antibacterial activity
  33. Comparative analysis of the white rot fungus Trametes hirsuta 072 laccases ability to modify 17β-oestradiol in the aqueous medium
  34. Synthesis of α‐D‐Ribose 1‐Phosphate and 2‐Deoxy‐α‐D‐Ribose 1‐Phosphate Via Enzymatic Phosphorolysis of 7‐Methylguanosine and 7‐Methyldeoxyguanosine
  35. 3′-Amino modifications enhance the antifungal properties of N4-alkyl-5-methylcytidines for potential biocides
  36. Total Synthesis of Elmenols A and B and Related Rearranged Angucyclinones
  37. 1,5-Hydride-Shift-Triggered Cyclization for the Synthesis of Unsymmetric Julolidines
  38. Discovery of novel N4-alkylcytidines as promising antimicrobial agents
  39. Synthesis and Aerobic Dehydrogenation of Indolizin-1-ol Derivatives
  40. Glycol and Phosphate Depot Forms of 4- and/or 5-Modified Nucleosides Exhibiting Antibacterial Activity
  41. Disclosing biosynthetic connections and functions of atypical angucyclinones with a fragmented C-ring
  42. Three-Component Reaction of 3,3-Difluorocyclopropenes, s-Tetrazines, and (benzo) Pyridines
  43. Construction of siloxane structures with P-Tolyl substituents at the silicon atom
  44. Direct Reductive Amination of Camphor Using Iron Pentacarbonyl as Stoichiometric Reducing Agent: Features and Limitations
  45. Imidazolone-activated donor-acceptor cyclopropanes with a peripheral stereocenter. A study on stereoselectivity of cycloaddition with aldehydes
  46. Construction of the Heterologous Laccase Producer Aspergillus nidulans lac№4 (argB–) and Its Application for the Progesterone Transformation
  47. Imidazol-5-one as an Acceptor in Donor–Acceptor Cyclopropanes: Cycloaddition with Aldehydes
  48. 5-Alkylthiomethyl Derivatives of 2'-Deoxyuridine: Synthesis and Antibacterial Activity
  49. Synthesis of water-soluble prodrugs of 5-modified 2ʹ-deoxyuridines and their antibacterial activity
  50. (3+2) Cycloaddition of N-benzylazomethine methylide with 4-arylidene-1H-imidazol-5(4H)-ones
  51. Structural isomers of cinnamic hydroxamic acids block HCV replication via different mechanisms
  52. Enzymatic Synthesis of 2-Deoxyribose 1-Phosphate and Ribose 1 Phosphate and Subsequent Preparation of Nucleosides
  53. Investigation of 5’-Norcarbocyclic Nucleoside Analogues as Antiprotozoal and Antibacterial Agents
  54. Biotransformation of progesterone by Aspergillus nidulans VKPM F-1069 (wild type)
  55. Structure-activity studies of irumamycin type macrolides from Streptomyces sp. INA-Ac-5812
  56. Novel 5-substituted derivatives of 2’-deoxy-6-azauridine with antibacterial activity
  57. Aerobic Co-/N-Hydroxysuccinimide-Catalyzed Oxidation of p-Tolylsiloxanes to p-Carboxyphenylsiloxanes: Synthesis of Functionalized Siloxanes as Promising Building Blocks for Siloxane-Based Materials
  58. Hydrazo coupling: the efficient transition-metal-free C–H functionalization of 8-hydroxyquinoline and phenol through base catalysis
  59. Novel 5′-Norcarbocyclic Pyrimidine Derivatives as Antibacterial Agents
  60. Novel 5′-Norcarbocyclic Derivatives of Bicyclic Pyrrolo- and Furano[2,3-d]Pyrimidine Nucleosides
  61. Synthesis of Cytokinins via Enzymatic Arsenolysis of Purine Nucleosides
  62. Conjugates of 17-substituted testosterone and epitestosterone with pyropheophorbide a differing in the length of linkers
  63. 4-Chloro-l-kynurenine as fluorescent amino acid in natural peptides
  64. One-step irreversible and efficient chemoenzymatic cleavage of ribose for preparation of nucleobases
  65. Biotransformation of progesterone by the ascomycete Aspergillus niger N402
  66. Aerobic Co or Cu/NHPI-catalyzed oxidation of hydride siloxanes: synthesis of siloxanols
  67. Crystallomycin revisited after 60 years: aspartocins B and C
  68. Synthesis of a New Imidazo[4′,5′:3,4]pyrazolo[5,1-c ][1,2,4]triazine-4,8-dione Heterocyclic System
  69. Modulation of Cell Death Pathways by Hepatitis C Virus Proteins in Huh7.5 Hepatoma Cells
  70. New benzophenone phosphonate derivatives
  71. New tools in nucleoside toolbox of tick-borne encephalitis virus reproduction inhibitors
  72. Selective N1-Alkylation of 1,3-Dibenzoyluracils: One-Pot Way to N1-Monosubstituted Uracil Derivatives
  73. 5-(4-alkyl-1,2,3-triazol-1-yl)methyl derivatives of 2′-deoxyuridine as inhibitors of viral and bacterial growth
  74. ONH2-functionalized Sepharose and Toyopearl resins
  75. New acyclic nucleotide antiviral agents with oxime fragment in the chain
  76. Simple oximes of 3′-O-aminothymidine inhibit HIV replication
  77. 1,3-Dipolar cycloaddition of alkenes to 3’-azido-3’-deoxythymidine as a route to 3’-deoxythymidin-3’-yl derivatives
  78. New Dinucleoside Phosphonate Derivatives as Prodrugs of 3′-Azido-3′-Deoxythymidine andβ-L-2′,3′-Dideoxy-3′-Thiacytidine: Synthesis and Anti-HIV Properties
  79. Synthesis and Anti-HIV Properties of New Carbamate Prodrugs of AZT
  80. 5′-Phosphonate Derivatives of 2′,3′-Dideoxy-3′-Thiacytidine as New Anti-HIV Prodrugs
  81. Phosphomonomorpholidates of the acyclic nucleosides bearing a double bond conjugated with the purine base
  82. New derivatives of alkyl-and aminocarbonylphosphonic acids containing 3′-azido-3′-deoxythymidine