All Stories

  1. Recent applications of gold-catalyzed cascade reactions in total synthesis of natural product

    Article • Tetrahedron Letters, November 2017, Elsevier

    Dr. Kenji SUGIMOTO

  2. Highly Efficient Access to Both Geometric Isomers of Silyl Enol Ethers: Sequential 1,2-Brook/Wittig Reactions

    Article • Angewandte Chemie International Edition, July 2016, Wiley

    Dr. Kenji SUGIMOTO

  3. A Macrosphelide as the Unexpected Product of a Pleurotus ostreatus Strain-Mediated Biotransformation of Halolactones Containing the gem-Dimethylcyclohexane Ring. Part 1

    Article • Molecules, June 2016, MDPI AG

    Dr. Kenji SUGIMOTO

  4. Synthesis of Substituted Pyrrolo[2,1-a]isoquinolines by Gold-Catalyzed Domino Cyclization of Alkynyl Iminoesters

    Article • Synthesis, April 2016, Thieme Publishing Group

    Dr. Kenji SUGIMOTO

  5. Synthesis of Substituted Quinolizidines via a Gold-Catalyzed Double Cyclization Cascade

    Article • Advanced Synthesis & Catalysis, January 2016, Wiley

    Dr. Kenji SUGIMOTO

  6. In vitro and in vivo antiherpetic effects of (1R,2R)-1-(5′-methylful-3′-yl)propane-1,2,3-triol

    Article • Journal of Natural Medicines, January 2016, Springer Science + Business Media

    Dr. Kenji SUGIMOTO

  7. Synthesis of Denosomin–Vitamin D3Hybrids and Evaluation of Their Anti-Alzheimer’s Disease Activities

    Article • Organic Letters, December 2015, American Chemical Society (ACS)

    Dr. Kenji SUGIMOTO

  8. Total Synthesis of (−)-Isoschizogamine

    Article • Chemistry - A European Journal, October 2015, Wiley

    Dr. Kenji SUGIMOTO

  9. Total synthesis of (−)-rhazinilam using 1,3-dipolar cycloaddition of optically active münchnone intermediate

    Article • Tetrahedron, June 2015, Elsevier

    Dr. Kenji SUGIMOTO

  10. Three-Component Domino Process for the Pyrrolizine Skeleton via [3 + 2]-Cycloaddition–Enamine Cyclization Triggered by a Gold Catalyst

    Article • Organic Letters, March 2015, American Chemical Society (ACS)

    Dr. Kenji SUGIMOTO

  11. Total Synthesis of (−)-Haouamine B Pentaacetate and Structural Revision of Haouamine B

    Article • Angewandte Chemie International Edition, October 2014, Wiley

    Dr. Kenji SUGIMOTO

  12. Autotandem Catalysis: Synthesis of Pyrroles by Gold-Catalyzed Cascade Reaction

    Article • Organic Letters, September 2014, American Chemical Society (ACS)

    Dr. Kenji SUGIMOTO

  13. Stereoselective approach to potential scaffold of A-nor B-aromatic OSW-1 analogues via [4+2] cycloaddition of o-quinodimethane

    Article • Tetrahedron, July 2014, Elsevier

    Dr. Kenji SUGIMOTO

  14. Synthesis of 8-Amino-(dihydrofuran-Fused Perhydrophenanthrene) via Copper-Mediated Amination Reaction

    Article • Heterocycles, January 2014, Japan Institute of Heterocyclic Chemistry

    Dr. Kenji SUGIMOTO

  15. Synthesis of phenylalkyl-substituted polyhydroxypiperidines as potent inhibitors for α-l-fucosidase

    Article • Tetrahedron, December 2013, Elsevier

    Dr. Kenji SUGIMOTO

  16. ChemInform Abstract: Protecting-Group-Free Total Synthesis of (-)-Rhazinilam (VII) and (-)-Rhazinicine (VIII) Using a Gold-Catalyzed Cascade Cyclization.

    Article • ChemInform, November 2013, Wiley

    Dr. Kenji SUGIMOTO

  17. Synthesis and biological evaluation of N-(2-fluorophenyl)-2β-deoxyfuconojirimycin acetamide as a potent inhibitor for α-l-fucosidases

    Article • Bioorganic & Medicinal Chemistry, November 2013, Elsevier

    Dr. Kenji SUGIMOTO

  18. Synthesis and structure–activity relationship of 2-phenyliminochromene derivatives as inhibitors for aldo–keto reductase (AKR) 1B10

    Article • Bioorganic & Medicinal Chemistry, November 2013, Elsevier

    Dr. Kenji SUGIMOTO

  19. Search for a novel SIRT1 activator: Structural modification of SRT1720 and biological evaluation

    Article • Bioorganic & Medicinal Chemistry Letters, September 2013, Elsevier

    Dr. Kenji SUGIMOTO

  20. Synthesis and antitumor activity of des-AB analogue of steroidal saponin OSW-1

    Article • Tetrahedron, September 2013, Elsevier

    Dr. Kenji SUGIMOTO

  21. Structure–activity-relationship studies on dihydrofuran-fused perhydrophenanthrenes as an anti-Alzheimer’s disease agent

    Article • Bioorganic & Medicinal Chemistry, August 2013, Elsevier

    Dr. Kenji SUGIMOTO

  22. Protecting-Group-Free Total Synthesis of (−)-Rhazinilam and (−)-Rhazinicine using a Gold-Catalyzed Cascade Cyclization

    Article • Angewandte Chemie, June 2013, Wiley

    Dr. Kenji SUGIMOTO

  23. Protecting-Group-Free Total Synthesis of (−)-Rhazinilam and (−)-Rhazinicine using a Gold-Catalyzed Cascade Cyclization

    Article • Angewandte Chemie International Edition, June 2013, Wiley

    Dr. Kenji SUGIMOTO

  24. Enantiocontrolled Total Synthesis of (−)-Mersicarpine

    Article • Chemistry - A European Journal, May 2013, Wiley

    Dr. Kenji SUGIMOTO

  25. Rational design and synthesis of 4-substituted 2-pyridin-2-ylamides with inhibitory effects on SH2 domain-containing inositol 5′-phosphatase 2 (SHIP2)

    Article • European Journal of Medicinal Chemistry, April 2013, Elsevier

    Dr. Kenji SUGIMOTO

  26. Stereoselective Total Synthesis of (-)-Batzellasides A, B, and C

    Article • European Journal of Organic Chemistry, March 2013, Wiley

    Dr. Kenji SUGIMOTO

  27. Synthesis and antitumor evaluation of arctigenin derivatives based on antiausterity strategy

    Article • European Journal of Medicinal Chemistry, February 2013, Elsevier

    Professor Suresh Awale, Dr. Kenji SUGIMOTO

  28. A novel compound, denosomin, ameliorates spinal cord injury via axonal growth associated with astrocyte-secreted vimentin

    Article • British Journal of Pharmacology, January 2013, Wiley

    Dr. Kenji SUGIMOTO

  29. Novel sequential 1,4-Brook rearrangement–Wittig reaction: new one-pot approach for silyl dienol ethers

    Article • Tetrahedron Letters, October 2012, Elsevier

    Dr. Kenji SUGIMOTO

  30. Efficient Approach to 1,2-Diazepines via Formal Diazomethylene Insertion into the C–C bond of Cyclobutenones

    Article • Organic Letters, July 2012, American Chemical Society (ACS)

    Dr. Kenji SUGIMOTO

  31. Synthesis and biological evaluation of optically active Ki16425

    Article • Bioorganic & Medicinal Chemistry Letters, July 2012, Elsevier

    Dr. Kenji SUGIMOTO

  32. Ring-Expansion Reaction of Oximes with Aluminum Reductants

    Article • Molecules, June 2012, MDPI AG

    Dr. Kenji SUGIMOTO

  33. Concise Total Synthesis of (−)-Mersicarpine

    Article • Organic Letters, May 2012, American Chemical Society (ACS)

    Dr. Kenji SUGIMOTO

  34. ChemInform Abstract: Development of Domino Reactions Based on Skeletal Rearrangement

    Article • ChemInform, March 2012, Wiley

    Dr. Kenji SUGIMOTO

  35. Design, synthesis, and biological evaluation of novel (1-thioxo-1,2,3,4-tetrahydro-β-carbolin-9-yl)acetic acids as selective inhibitors for AKR1B1

    Article • Bioorganic & Medicinal Chemistry, January 2012, Elsevier

    Dr. Kenji SUGIMOTO

  36. Synthesis of dihydrofuran-fused perhydrophenanthrenes having a phenolic hydroxyl group as a novel anti-Alzheimer’s disease agent

    Article • Bioorganic & Medicinal Chemistry Letters, January 2012, Elsevier

    Dr. Kenji SUGIMOTO

  37. Syntheses of aza-analogues of macrosphelides via RCM strategy and their biological evaluation

    Article • Tetrahedron, October 2011, Elsevier

    Dr. Kenji SUGIMOTO

  38. Dihydroazamacrosphelides: Synthesis and Apoptosis Inducing Activities

    Article • Heterocycles, January 2011, Japan Institute of Heterocyclic Chemistry

    Dr. Kenji SUGIMOTO

  39. Development of Domino Reactions Based on Skeletal Rearrangement

    Article • YAKUGAKU ZASSHI, January 2011, Pharmaceutical Society of Japan

    Dr. Kenji SUGIMOTO

  40. Synthetic Studies toward Haouamine B: Construction of Indenotetrahydropyridone Skeleton

    Article • Synlett, December 2010, Thieme Publishing Group

    Dr. Kenji SUGIMOTO

  41. Regioselective Synthesis of Heterocycles Containing Nitrogen Neighboring an Aromatic Ring by Reductive Ring Expansion Using Diisobutylaluminum Hydride and Studies on the Reaction Mechanism

    Article • The Journal of Organic Chemistry, February 2010, American Chemical Society (ACS)

    Dr. Kenji SUGIMOTO

  42. Regiospecific Rearrangement of Hydroxylamines to Secondary Amines Using Diisobutylaluminum Hydride

    Article • Heterocycles, January 2010, Japan Institute of Heterocyclic Chemistry

    Dr. Kenji SUGIMOTO

  43. Total Synthesis of (+)-Haplophytine

    Article • Angewandte Chemie International Edition, September 2009, Wiley

    Dr. Kenji SUGIMOTO

  44. Regiospecific Synthesis of Unsubstituted Basic Skeletons of Heterocycles Containing Nitrogen Neighboring an Aromatic Ring by the Reductive Ring Expansion Reaction Using Diisobutylaluminum Hydride

    Article • Heterocycles, January 2009, Japan Institute of Heterocyclic Chemistry

    Dr. Kenji SUGIMOTO

  45. Synthesis of vinyloxazolidinones by palladium-catalyzed CO2-recycling reaction of 4-(benzylamino)-2-butenyl carbonates

    Article • Tetrahedron Letters, December 2007, Elsevier

    Dr. Kenji SUGIMOTO

  46. Palladium-Catalyzed Three-Component Coupling of Propargylic Oxiranes, Phenols and Carbon Dioxide

    Article • Synlett, March 2007, Thieme Publishing Group

    Dr. Kenji SUGIMOTO

  47. Ruthenium-Catalyzed Ring Expansion Reaction of 1-Acetylenylcyclobutanols with Methyl Vinyl Ketone.

    Article • ChemInform, December 2006, Wiley

    Dr. Kenji SUGIMOTO

  48. Ruthenium-Catalyzed Ring Expansion Reaction of 1-Acetylenylcyclobutanols with Methyl Vinyl Ketone

    Article • Synlett, August 2006, Thieme Publishing Group

    Dr. Kenji SUGIMOTO

  49. Palladium-Catalyzed Ring Expansion Reaction of (Z)-1-(1,3-Butadienyl)cyclobutanols with Aryl Iodides. Stereospecific Synthesis of (Z)-2-(3-Aryl-1-propenyl)cyclopentanones

    Article • Organic Letters, June 2004, American Chemical Society (ACS)

    Dr. Kenji SUGIMOTO

  50. Stereoselective synthesis of α-disubstituted cyclopentanones by palladium-catalyzed rearrangement of allenylcyclobutanols with aryl halides

    Article • Tetrahedron, September 2002, Elsevier

    Dr. Kenji SUGIMOTO

  51. Ruthenium-catalyzed ring expansion reaction of allenylcyclobutanols

    Article • Tetrahedron Letters, June 2001, Elsevier

    Dr. Kenji SUGIMOTO

  52. Palladium-catalyzed stereospecific ring expansion reaction of allenylcyclobutanols with aryl iodides: a novel route to the α-substituted cyclopentanones with quaternary carbon stereocenters

    Article • Tetrahedron Letters, June 2000, Elsevier

    Dr. Kenji SUGIMOTO