All Stories

  1. Recent Overview on the Molecular Hybrids Integrated With Benzosuberone/Benzo[7]annulene Derivatives as Multi‐Target Therapeutics
  2. One-pot three-component Synthesis, Structural characterization, Computational investigation, and anti-cancer evaluation of some novel benzo[g][1,3,5]oxadiazocine pyridine carboxamide hybrids
  3. Spectroscopic, X‐Ray Crystallographic, and Hirshfeld Surface Analyses for the Investigation of Intermolecular Interactions in Carboxamide Hydrazone Hybrids
  4. An Efficient Route to Annulated Pyrrolo[2,1‐a]Isoquinoline‐3‐Carboxamide Derivatives via Nitrogen Ylides
  5. Unreported Biginelli product with potent antifungal activity: Synthesis, DFT insights, and docking simulation analysis
  6. Recent advances on anticancer activity of benzodiazine heterocycles through kinase inhibition
  7. Synthesis of some new pyrimidine-based pyrene/benzochromene hybrids as EGFR kinase inhibitors in HCT-116 cancer cells through apoptosis
  8. Clean and Efficient Green Protocol of N,N′-Bis(2-(arylazo)-2-(aroyl)vinyl)ethane-1,2-diamines in Aqueous Medium without Catalyst: Synthesis and Photophysical Characterization
  9. Unexpected products using Biginelli reaction: Synthesis, antimicrobial potency, docking simulation, and DFT investigations of some new amidopyridines
  10. Design, assessment and antibacterial potency of novel pseudopolyrotaxanes based on cyclodextrin as drug carriers for amoxicillin and ceftriaxone
  11. Recent advances on anticancer and antimicrobial activities of directly-fluorinated five-membered heterocycles and their benzo-fused systems
  12. Recent progress in therapeutic applications of fluorinated five-membered heterocycles and their benzo-fused systems
  13. Synthesis of novel piperazine-based bis(thiazole)(1,3,4-thiadiazole) hybrids as anti-cancer agents through caspase-dependent apoptosis
  14. Synthesis and Anti-Breast Cancer Potency of Mono- and Bis-(pyrazolyl[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine) Derivatives as EGFR/CDK-2 Target Inhibitors
  15. Regioselective synthesis and computational calculation studies of some new pyrazolyl‐pyridine and bipyridine derivatives
  16. Synthesis of novel mono- and bis-pyrazolylthiazole derivatives as anti-liver cancer agents through EGFR/HER2 target inhibition
  17. Novel bis-amide-based bis-thiazoles as Anti-colorectal Cancer Agents Through Bcl-2 Inhibition: Synthesis, In Vitro, and In Vivo studies
  18. Anticancer therapeutic potential of benzofuran scaffolds
  19. Recent developments in the chemistry of 1H- and 4H-1,2,4-triazoles
  20. Microwave-assisted chemoselective synthesis and photophysical properties of 2-arylazo-biphenyl-4-carboxamides from hydrazonals
  21. Benzofuran as a promising scaffold for the synthesis of novel antimicrobial agents
  22. High-Pressure Metal-Free Catalyzed One-Pot Two-Component Synthetic Approach for New 5-Arylazopyrazolo[3,4-b]Pyridine Derivatives
  23. Transition‐metal‐catalyzed Heteroannulation Reactions in Aqueous Medium
  24. Efficient and Recyclable Solid-Supported Pd(II) Catalyst for Microwave-Assisted Suzuki Cross-Coupling in Aqueous Medium
  25. Regulatory Effect of Adipose-Derived Mesenchymal Stem Cells and/ or Acitretin on Adam10 Gene in Alzheimer's Disease Rat Model
  26. Inhibitory Activities of Pyrazolo-Oxazine Heterocyclic Derivatives
  27. Chemistry of Bipyrazoles: Synthesis and Applications
  28. Design and synthesis of new bis(1,2,4-triazolo[3,4-b][1,3,4]thiadiazines) and bis((quinoxalin-2-yl)phenoxy)alkanes as anti-breast cancer agents through dual PARP-1 and EGFR targets inhibition
  29. Green Protocol for the Novel Synthesis of Thiochromeno[4,3-b]pyridine and Chromeno[4,3-b]pyridine Derivatives Utilizing a High-Pressure System
  30. Novel Bis-Thiazole Derivatives: Synthesis and Potential Cytotoxic Activity Through Apoptosis With Molecular Docking Approaches
  31. Inhibitory activities of bipyrazoles: a patent review
  32. Front Cover Picture: Recent Developments in Z‐Selective Olefin Metathesis Reactions by Molybdenum, Tungsten, Ruthenium, and Vanadium Catalysts (8/2021)
  33. Recent Developments in Z‐Selective Olefin Metathesis Reactions by Molybdenum, Tungsten, Ruthenium, and Vanadium Catalysts
  34. Synthetic Routes to Bioactive Bipyrazole Derivatives
  35. Expression profiling of some Acute Myeloid Leukemia - associated markers to assess their diagnostic / prognostic potential
  36. High pressure assisted synthetic approach for novel 6,7-dihydro-5H-benzo[6,7]cyclohepta[1,2-b]pyridine and 5,6-dihydrobenzo[h]quinoline derivatives and their assessment as anticancer agents
  37. Heteroannulation Routes to Bioactive Pyrazolooxazines
  38. Inhibitory activities of indolizine derivatives: a patent review
  39. An Efficient Synthesis of Some New Coumarin Hybrids Endowed with Expected Biological Activity
  40. Synthesis and characterization of new 3,3`-bipyrazole-4,4`-dicarboxylic acid derivatives and some of their palladium(II) complexes as pre-catalyst for Suzuki coupling reaction in water
  41. Facile access to some new 3,3′‐bipyrazole‐ester derivatives utilizing bis‐hydrazonoyl chlorides
  42. An update on benzofuran inhibitors: a patent review
  43. Bis‐thiourea Derivatives and Their Utility in Synthesis of Mono‐heterocyclic, Bis‐heterocyclic, and Fused Heterocyclic Systems
  44. Facile Assembling of Novel 2,3,6,7,9-pentaazabicyclo- [3.3.1]nona-3,7-diene Derivatives under Microwave and Ultrasound Platforms
  45. Regio- and stereoselective route to bis-[3-methyl-1,1′,4′-triaryl-5-oxo-spiro-pyrazoline-4,5′-pyrazoline] derivatives via 1,3-dipolar cycloaddition under sonication
  46. Microwave promoted Heck and Suzuki coupling reactions of new 3-(5-bromobenzofuranyl)pyrazole in aqueous media
  47. Synthesis and applications of bi- and bis-triazole systems
  48. Tandem one-pot synthesis of 2-arylcinnolin-6-one derivatives from arylhydrazonopropanals and acetoacetanilides using sustainable ultrasound and microwave platforms
  49. Biological evaluation of benzosuberones
  50. Efficient direct formic acid fuel cell (DFAFC) anode of nano-sized palladium complex: High durability and activity origin
  51. Catalytic activity of some oxime-based Pd(II)-complexes in Suzuki coupling of aryl and heteroaryl bromides in water
  52. Convenient synthesis of azolopyrimidine, azolotriazine, azinobenzimidazole and 1,3,4-thiadiazole derivatives
  53. Synthesis of Pyrazolo[1,5-a ][1,3,5]triazine, Pyrazolo[1,5-a ]pyrimidine, and Imidazo[1,2-b ]pyrazole Derivatives Based on Imidazo[2,1-b ]thiazole Moiety
  54. Synthetic Utility of Pyridinium Bromide: Synthesis and Antimicrobial Activity of Novel 2,4,6-Trisubstituted Pyridines Having Pyrazole Moiety
  55. Thiadiazole inhibitors: a patent review
  56. A Facile Access and Computational Studies of Some New 4,5'-Bipyrazole Derivatives
  57. Phytochemical investigation of Boscia angustifolia A. Rich. (Capparaceae)
  58. Synthetic routes to benzosuberone-based fused- and spiro-heterocyclic ring systems
  59. Alkoxide-Directed Hydride Addition to α,β-Unsaturated Sultones
  60. Synthetic access to some new benzothiazole-based 1,3,4-thiadiazole and 1,3-thiazole derivatives
  61. Microwave-Assisted Synthesis of Arylated Pyrrolo[2,1-a]Isoquinoline Derivatives via Sequential [3 + 2] Cycloadditions and Suzuki-Miyaura Cross-Couplings in Aqueous Medium
  62. Synthesis and antiviral activity of some new bis-1,3-thiazole derivatives
  63. Microwave-assisted synthesis of 2-acetyl-5-arylthiophenes and 4-(5-arylthiophen-2-yl)thiazoles via Suzuki coupling in water
  64. Synthesis and Reactivity of Enaminones: A Facile Synthesis of Thiophene and 1,3,4-Thiadiazole Derivatives Incorporating a Thiazole Moiety
  65. Synthesis of ethynylated biaryls and asymmetric diethynylated benzene via sequential Sonogashira and Suzuki couplings in water
  66. Chemistry and Biological Activity of Pyridotriazolopyrimidines
  67. Synthesis and Reactivity of Phenylthiourea Derivatives: An Efficient Synthesis of New Thiazole-Based Heterocycles
  68. Ultrasound-assisted regio- and stereoselective synthesis of bis-[1′,4′-diaryl-1-oxo-spiro-benzosuberane-2,5′-pyrazoline] derivatives via 1,3-dipolar cycloaddition
  69. Synthesis of Novel Indolizine, Pyrrolo[1,2-A] Quinoline, and 4,5-Dihydrothiophene Derivatives Via Nitrogen Ylides and their Antimicrobial Evaluation
  70. Synthesis and Anti-cancer Activity of 1,3,4-Thiadiazole and 1,3-Thiazole Derivatives Having 1,3,4-Oxadiazole Moiety
  71. Synthesis of 2-Phenylazonaphtho[1,8-ef][1,4]diazepines and 9-(3-Arylhydrazono)pyrrolo[1,2-a]perimidines as Antitumor Agents
  72. Synthesis of Unsymmetrical Aryl-Ethynylated Benzenes via Regiocontrolled Sonogashira Reaction of 1,3,5-Tribromobenzene
  73. Synthesis and Antimicrobial Evaluation of Some New 1,2-Bis-(2-(<i>N</i>-arylimino)-1,3-thiazolidin-3-yl)ethane Derivatives
  74. Metathesis Reactions in Domino Processes
  75. Synthesis of some new pyrazole-based 1,3-thiazoles and 1,3,4-thiadiazoles as anticancer agents
  76. Synthesis and quantum calculations of 1,3-thiazoles and 1,3,4-thiadiazole derivatives via pyridinylthioureas
  77. Benzofuran derivatives: a patent review
  78. Microwave-assisted synthesis of 5-arylbenzofuran-2-carboxylates via Suzuki coupling using 2-quinolinealdoxime-Pd(II)-complex
  79. A Facile Synthesis of Pyrido[2′,<...
  80. Synthesis and applications of bipyrazole systems
  81. Recent advances on the synthesis of azoles, azines and azepines fused to benzimidazole
  82. Synthetic Access to Azolylthiazoles
  83. Synthesis of some new azole, pyrimidine, pyran, and benzo/naphtho[b]furan derivatives incorporating thiazolo[3,2-a]benzimidazole moiety
  84. Synthetic routes to benzimidazole-based fused polyheterocycles
  85. Synthesis, anti-HSV-1, and cytotoxic activities of some new pyrazole- and isoxazole-based heterocycles
  86. Mizoroki-Heck cross-couplings of 2-acetyl-5-bromobenzofuran and aryl halides under microwave irradiation
  87. Facile Synthesis of Thiophene- and 1,3,4-Thiadiazole-Based Heterocycles
  88. Microwave-assisted C-C cross-coupling reactions of aryl and heteroaryl halides in water
  89. Facile Access to Biaryls and 2-Acetyl-5-arylbenzofurans via Suzuki Coupling in Water under Thermal and Microwave Conditions
  90. Synthesis, reactions, and biological activity of 4,5-diarylimidazole-2-thiones (Review)
  91. Microwave-assisted synthesis and in-vitro anti-tumor activity of 1,3,4-triaryl-5-N-arylpyrazole-carboxamides
  92. Use of 2-bromoacetylbenzofurans in heterocyclic synthesis (review)
  93. Microwave-Assisted Synthesis of 2-Substituted 4-Biarylyl-1,3-thiazoles by Carbon-Carbon Cross-Coupling in Water
  94. Heck and Suzuki cross-couplings of aryl and heteroaryl bromides in water using a new palladium(II)-complex
  95. A Facile Access to Some New Pyrazole, 1,3,4-Thiadiazole, and Thiophene Derivatives via β-Ketosulfones
  96. Synthesis and Antiviral Activity of New Indole-Based Heterocycles
  97. Cytotoxicity and Utility of 1-Indanone in the Synthesis of Some New Heterocycles
  98. 1H-Benzimidazole-2-acetonitriles as synthon in fused benzimidazole synthesis
  99. Utility of 2,4-Dioxoesters in the Synthesis of New Heterocycles
  100. Facile Access to Benzothiazole-Containing Pyrrolo[1,2-a]quinolines and Pyrrolo[2,1-a]isoquinolinesviaNitrogen Ylides
  101. Synthesis of bipyrazole and 1,3,4-thiadiazole derivatives
  102. Convenient synthesis and antimicrobial evaluation of some novel 2-substituted-3-methylbenzofuran derivatives
  103. New Domino Reactions with Sultones
  104. Synthesis of Some New Indolizine and Pyrrolo[1,2-a]quinoline Derivatives via Nitrogen Ylides
  105. Synthesis and Some New Indolizine and Pyrrolo[1,2-a]quinoline Derivatives via Nitrogen Ylides
  106. Facile route to novel 2-pyridone, pyrazolo[3,4-d]-1,2,3-triazine, and pyrazolo[3,4-d]- and [1,5-a]-pyrimidine derivatives
  107. Synthesis of annulated dihydroisoquinoline heterocycles via their nitrogen ylides
  108. Fused polyaza-heterocycles and 1,3,4-thiadiazolesviaa tricyano synthon
  109. Microwave-assisted Suzuki–Miyaura and Heck–Mizoroki cross-coupling reactions of aryl chlorides and bromides in water using stable benzothiazole-based palladium(II) precatalysts
  110. Regioselective Synthesis of Novel 4,4′-and 5,5′-bi-(1,2,4-triazole) Derivatives
  111. Synthesis of some new benzofuran-based thiophene, 1,3-oxathiole and 1,3,4-oxa(thia)diazole derivatives
  112. Microwave-accelerated Mizoroki-Heck and Sonogashira cross- coupling reactions in water using a heterogeneous palladium(II)-precatalyst
  113. A Convenient Access to Functionalized Pyrazole, Pyrazolyl-Azole, and Pyrazolo[3,4-d]Pyridazine Derivatives
  114. Synthesis, anticonvulsant, and anti-inflammatory evaluation of some new benzotriazole and benzofuran-based heterocycles
  115. Synthesis, Anticonvulsant, and Anti-inflammatory Activities of Some New Benzofuran-Based Heterocycles
  116. Combining enabling techniques in organic synthesis: solid-phase-assisted catalysis under microwave conditions using a stable Pd(II)-precatalyst
  117. 2-Pyridinealdoxime, a new ligand for a Pd-precatalyst: Application in solid-phase-assisted Suzuki–Miyaura reaction
  118. Electrolytic Partial Fluorination of Organic Compounds. 79. Anodic Fluorination of Spiropyrazoline-5,3‘-chroman-4-ones and Thiochromanone Analogues. A Route to Aroyl Fluoride Derivatives
  119. Azoles and Azolo-Azines via 3-(3-Methylbenzofuran-2-Yl)-3-Oxopropanenitrile
  120. Regio- and stereoselective synthesis of bis-spiropyrazoline-5,3′-chroman(thiochroman)-4-one derivatives via bis-nitrilimines
  121. Synthesis of spiro-pyrazole-3,3′-thiopyrano[2,3-b]pyridines and azolo[a]pyrido[2′,3′:5,6]thiopyrano[3,4-d]pyrimidines as new ring systems with antifungal and antibacterial activities
  122. Synthesis and antimicrobial evaluation of some 1,2,4-triazole, 1,3,4-oxa(thia)diazole, and 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazine derivatives
  123. Synthesis of some new pyridazine, 1,2,4-triazine and 1,3,4-thiadiazole derivatives
  124. A Facile Access to Polysubstituted Bipyrazoles and Pyrazolylpyrimidines
  125. Electrochemical Partial Fluorination of Organic Compounds. 74. Efficient Anodic Synthesis of 2-Fluoro- and 2,3-Difluoro-2,3-dihydrobenzofuran Derivatives1
  126. Synthesis of 3,3′-bipyrazole, 5,5′-bi-1,3,4-thiadiazole and fused azole systems via bishydrazonoyl chlorides
  127. Electrolytic fluorination of organic compounds
  128. A convenient route to pyridones, pyrazolo[2,3-a]pyrimidines and pyrazolo[5,1-c]triazines incorporating antipyrine moiety
  129. Indolizines, triazolo[4,3-a]pyridines, benzimidazo[1,2-d]oxadiazoles, and pyrazolo[1,5-c]triazoles via nitrogen and sulfur ylides
  130. Synthesis of 3,3′-bi-1,2,4-Triazolo[4,5-a]- benzimidazole, 5,5′-bi-1,3,4-Thiadiazole, and Thiazolo[3,2-a]benzimidazole Derivatives
  131. Polyheterocyclic systems incorporating pyrazole, thiophene, thiazole, and thiadiazole moieties
  132. Anodic Fluorination of 3-Substituted Benzofurans. Efficient Synthesis of 2-Fluoro- and 2,3-Difluoro-2,3-dihydrobenzofuran Derivatives
  133. Simple and convenient routes to new polyheterocycles incorporating pyrazole, thiazole, thiophene, and 1,3,4-thiadiazole moieties
  134. Electrolytic Partial Fluorination of Organic Compounds. 55.1 Highly Regio- and Stereoselective Anodic Monofluorination of 2,3-Dihydrochroman-4-one and Chromone Derivatives
  135. Electrolytic Partial Fluorination of Organic Compounds. 54.1 Anodic Mono- and Trifluorination of Thiochroman-4-one Derivatives and the Factors Affecting Product Selectivity
  136. Electrolytic partial fluorination of organic compounds. Part 45: Highly regioselective anodic monofluorination of (E)-3-benzylidene-2,3-dihydrochroman-4-ones
  137. AN EFFICIENT ROUTE TOTRANS-4,5-DIHYDROTHIOPHENES AND THIAZOLES VIA NITROGEN AND SULFUR YLIDES
  138. Polyheterocyclic Ring Systems with Bridgehead Nitrogen Atoms: A Facile Route to Some Novel Azolo-1,2,4-triazine Derivatives
  139. Reactions with Hydrazonoyl Halides XXX: Synthesis of Some 2,3-Dihydro-1,3,4-Thiadiazoles and Unsymmetrical Azines Containing Benzothiazole Moiety
  140. Electrolytic partial fluorination of organic compounds. 36 . Regioselective anodic fluorination of phenylthiolated benzofuranone and benzothiazole derivatives
  141. Electrolytic Partial Fluorination of Organic Compounds. 35.1 Anodic Fluorination of 2-Pyrimidyl, 2-Pyridyl, and 2-Quinazolinonyl Sulfides
  142. Electrolytic partial fluorination of organic compounds. Part 29. Anodic mono- and difluorination of 2-benzoxazolyl sulfides
  143. Heterocyclic Synthesis via Enaminonitriles: One-pot Synthesis of Some New Pyrazole, Isoxazole, Pyrimidine, Pyrazolo[1,5-a]pyrimidine, Pyrimido[1,2-a]benzimidazole and Pyrido[1,2-a]benzimidazole Derivatives
  144. Synthesis and reactivity of cyanomethyl 2-amino-4-methylthiazolyl ketone. A facile synthesis of novel pyrazolo[5,1-c]1,2,4-triazine, 1,2,4-triazolo[5,1-c]1,2,4-triazine, 1,2,4-triazino[4,3-a]benzimidazole, pyridazine-6-imine and 6-oxopyridazinone deriv...
  145. SYNTHESIS OF 1,2,4 - TRIAZOLE, 1,2,4 - TRIAZOLO [3,4 -b] [1,3,4] THIADIAZOLE AND 1,2,4 -TRIAZOLO [3,4 -b] [1,3,4] THIADIAZINE DERIVATIVES OF 3- [5- (BENZOTHIAZOL - 2 - YL) THIENO [2,3-d] PYRIMIDINE - 4- ONE] ACETIC ACID HYDRAZIDE.
  146. Heterocyclic synthesis via enaminones: Regioselective synthesis of some novel pyrazole, isoxazole, pyrimidine, pyrido[1,2-a]benzimidazole and pyrazolo[1,5-a]-pyrimidine derivatives
  147. Synthesis and reactivity of cyanomethyl 2‐amino‐4‐methylthiazolyl ketone. A facile synthesis of novel pyrazolo[5,1‐c]1,2,4‐triazine, 1,2,4‐triazolo[5,1‐c]1,2,4‐triazine, 1,2,4‐triazino[4,3‐a]benzimidazole, pyridazine‐6‐imine and 6‐oxopyridazinone deriv...
  148. Electrolytic Partial Fluorination of Organic Compounds. 31.1 Regioselective Anodic Fluorination of 2-Quinolyl and 4-(7-Trifluoromethyl)quinolyl Sulfides and the Factors Affecting Its Optimization
  149. Heterocyclic Synthesis via Enaminonitriles: A Convenient Route to Some New Pyrazole, Isoxazole, Pyrimidine, Pyrazolo[1,5-a]pyrimidine, Pyrimido[1,2-a]benzimidazole and Pyrido[1,2-a]benzimidazole Derivatives†
  150. One-pot Synthesis of Novel Polysubstituted Pyrazole and Pyrrolo[2,1-b]benzothiazole Derivatives†
  151. Synthesis and reactivity of benzothiazol-2-ylcarbonylhydroximoyl chloride, a versatile synthon
  152. CONVENIENT SYNTHESIS OF SOME NEW 1,3,4-THIADIAZOLE AND 1,3,4-SELENADIAZOLE DERIVATIVES
  153. Facile synthesis of novel polysubstituted thiopene and 1,3,4-thiadiazole derivatives
  154. Synthesis and reactivity of 2-(benzothiazol-2-yl)-1-bromo-1,2-ethanedione-1-arylhydrazones
  155. One-pot synthesis of imidazo[1,2-b]pyrazole, imidazo[1,2-b]-1,2,4-triazole, imidazo[1,2-a]pyridine, imidazo[1,2-a]pyrimidine, imidazo[1,2-a]benzimidazole, and 1,2,4-triazolo[4,3-a]benzimidazole derivatives
  156. Synthesis and reactivity of 3-(benzothiazol-2-yl)-3-oxopropanenitrile
  157. A FACILE, ONE-POT SYNTHESIS OF NOVEL 2,2′-BI(4,5-DIHYDRO-1,3,4-SELENADIAZOLE) DERIVATIVES VIA DIHYDRAZONOYL DIHALIDES
  158. One-step synthesis of novel 2,2′-bi(4,5-dihydro-1,3,4-thiadiazole) and 2,3-disubstituted 1,4-benzothiazine derivatives
  159. Facile Syntheses of Bi-1,2,4-triazoles via hydrazonyl halides