All Stories

  1. One-pot three-component Synthesis, Structural characterization, Computational investigation, and anti-cancer evaluation of some novel benzo[g][1,3,5]oxadiazocine pyridine carboxamide hybrids
  2. Spectroscopic, X‐Ray Crystallographic, and Hirshfeld Surface Analyses for the Investigation of Intermolecular Interactions in Carboxamide Hydrazone Hybrids
  3. An Efficient Route to Annulated Pyrrolo[2,1‐a]Isoquinoline‐3‐Carboxamide Derivatives via Nitrogen Ylides
  4. Unreported Biginelli product with potent antifungal activity: Synthesis, DFT insights, and docking simulation analysis
  5. Recent advances on anticancer activity of benzodiazine heterocycles through kinase inhibition
  6. Synthesis of some new pyrimidine-based pyrene/benzochromene hybrids as EGFR kinase inhibitors in HCT-116 cancer cells through apoptosis
  7. Clean and Efficient Green Protocol of N,N′-Bis(2-(arylazo)-2-(aroyl)vinyl)ethane-1,2-diamines in Aqueous Medium without Catalyst: Synthesis and Photophysical Characterization
  8. Unexpected products using Biginelli reaction: Synthesis, antimicrobial potency, docking simulation, and DFT investigations of some new amidopyridines
  9. Design, assessment and antibacterial potency of novel pseudopolyrotaxanes based on cyclodextrin as drug carriers for amoxicillin and ceftriaxone
  10. Recent advances on anticancer and antimicrobial activities of directly-fluorinated five-membered heterocycles and their benzo-fused systems
  11. Recent progress in therapeutic applications of fluorinated five-membered heterocycles and their benzo-fused systems
  12. Synthesis of novel piperazine-based bis(thiazole)(1,3,4-thiadiazole) hybrids as anti-cancer agents through caspase-dependent apoptosis
  13. Synthesis and Anti-Breast Cancer Potency of Mono- and Bis-(pyrazolyl[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine) Derivatives as EGFR/CDK-2 Target Inhibitors
  14. Regioselective synthesis and computational calculation studies of some new pyrazolyl‐pyridine and bipyridine derivatives
  15. Synthesis of novel mono- and bis-pyrazolylthiazole derivatives as anti-liver cancer agents through EGFR/HER2 target inhibition
  16. Novel bis-amide-based bis-thiazoles as Anti-colorectal Cancer Agents Through Bcl-2 Inhibition: Synthesis, In Vitro, and In Vivo studies
  17. Anticancer therapeutic potential of benzofuran scaffolds
  18. Recent developments in the chemistry of 1H- and 4H-1,2,4-triazoles
  19. Microwave-assisted chemoselective synthesis and photophysical properties of 2-arylazo-biphenyl-4-carboxamides from hydrazonals
  20. Benzofuran as a promising scaffold for the synthesis of novel antimicrobial agents
  21. High-Pressure Metal-Free Catalyzed One-Pot Two-Component Synthetic Approach for New 5-Arylazopyrazolo[3,4-b]Pyridine Derivatives
  22. Transition‐metal‐catalyzed Heteroannulation Reactions in Aqueous Medium
  23. Efficient and Recyclable Solid-Supported Pd(II) Catalyst for Microwave-Assisted Suzuki Cross-Coupling in Aqueous Medium
  24. Regulatory Effect of Adipose-Derived Mesenchymal Stem Cells and/ or Acitretin on Adam10 Gene in Alzheimer's Disease Rat Model
  25. Inhibitory Activities of Pyrazolo-Oxazine Heterocyclic Derivatives
  26. Chemistry of Bipyrazoles: Synthesis and Applications
  27. Design and synthesis of new bis(1,2,4-triazolo[3,4-b][1,3,4]thiadiazines) and bis((quinoxalin-2-yl)phenoxy)alkanes as anti-breast cancer agents through dual PARP-1 and EGFR targets inhibition
  28. Green Protocol for the Novel Synthesis of Thiochromeno[4,3-b]pyridine and Chromeno[4,3-b]pyridine Derivatives Utilizing a High-Pressure System
  29. Novel Bis-Thiazole Derivatives: Synthesis and Potential Cytotoxic Activity Through Apoptosis With Molecular Docking Approaches
  30. Inhibitory activities of bipyrazoles: a patent review
  31. Front Cover Picture: Recent Developments in Z‐Selective Olefin Metathesis Reactions by Molybdenum, Tungsten, Ruthenium, and Vanadium Catalysts (8/2021)
  32. Recent Developments in Z‐Selective Olefin Metathesis Reactions by Molybdenum, Tungsten, Ruthenium, and Vanadium Catalysts
  33. Synthetic Routes to Bioactive Bipyrazole Derivatives
  34. Expression profiling of some Acute Myeloid Leukemia - associated markers to assess their diagnostic / prognostic potential
  35. High pressure assisted synthetic approach for novel 6,7-dihydro-5H-benzo[6,7]cyclohepta[1,2-b]pyridine and 5,6-dihydrobenzo[h]quinoline derivatives and their assessment as anticancer agents
  36. Heteroannulation Routes to Bioactive Pyrazolooxazines
  37. Inhibitory activities of indolizine derivatives: a patent review
  38. An Efficient Synthesis of Some New Coumarin Hybrids Endowed with Expected Biological Activity
  39. Synthesis and characterization of new 3,3`-bipyrazole-4,4`-dicarboxylic acid derivatives and some of their palladium(II) complexes as pre-catalyst for Suzuki coupling reaction in water
  40. Facile access to some new 3,3′‐bipyrazole‐ester derivatives utilizing bis‐hydrazonoyl chlorides
  41. An update on benzofuran inhibitors: a patent review
  42. Bis‐thiourea Derivatives and Their Utility in Synthesis of Mono‐heterocyclic, Bis‐heterocyclic, and Fused Heterocyclic Systems
  43. Facile Assembling of Novel 2,3,6,7,9-pentaazabicyclo- [3.3.1]nona-3,7-diene Derivatives under Microwave and Ultrasound Platforms
  44. Regio- and stereoselective route to bis-[3-methyl-1,1′,4′-triaryl-5-oxo-spiro-pyrazoline-4,5′-pyrazoline] derivatives via 1,3-dipolar cycloaddition under sonication
  45. Microwave promoted Heck and Suzuki coupling reactions of new 3-(5-bromobenzofuranyl)pyrazole in aqueous media
  46. Synthesis and applications of bi- and bis-triazole systems
  47. Tandem one-pot synthesis of 2-arylcinnolin-6-one derivatives from arylhydrazonopropanals and acetoacetanilides using sustainable ultrasound and microwave platforms
  48. Biological evaluation of benzosuberones
  49. Efficient direct formic acid fuel cell (DFAFC) anode of nano-sized palladium complex: High durability and activity origin
  50. Catalytic activity of some oxime-based Pd(II)-complexes in Suzuki coupling of aryl and heteroaryl bromides in water
  51. Convenient synthesis of azolopyrimidine, azolotriazine, azinobenzimidazole and 1,3,4-thiadiazole derivatives
  52. Synthesis of Pyrazolo[1,5-a ][1,3,5]triazine, Pyrazolo[1,5-a ]pyrimidine, and Imidazo[1,2-b ]pyrazole Derivatives Based on Imidazo[2,1-b ]thiazole Moiety
  53. Synthetic Utility of Pyridinium Bromide: Synthesis and Antimicrobial Activity of Novel 2,4,6-Trisubstituted Pyridines Having Pyrazole Moiety
  54. Thiadiazole inhibitors: a patent review
  55. A Facile Access and Computational Studies of Some New 4,5'-Bipyrazole Derivatives
  56. Phytochemical investigation of Boscia angustifolia A. Rich. (Capparaceae)
  57. Synthetic routes to benzosuberone-based fused- and spiro-heterocyclic ring systems
  58. Alkoxide-Directed Hydride Addition to α,β-Unsaturated Sultones
  59. Synthetic access to some new benzothiazole-based 1,3,4-thiadiazole and 1,3-thiazole derivatives
  60. Microwave-Assisted Synthesis of Arylated Pyrrolo[2,1-a]Isoquinoline Derivatives via Sequential [3 + 2] Cycloadditions and Suzuki-Miyaura Cross-Couplings in Aqueous Medium
  61. Synthesis and antiviral activity of some new bis-1,3-thiazole derivatives
  62. Microwave-assisted synthesis of 2-acetyl-5-arylthiophenes and 4-(5-arylthiophen-2-yl)thiazoles via Suzuki coupling in water
  63. Synthesis and Reactivity of Enaminones: A Facile Synthesis of Thiophene and 1,3,4-Thiadiazole Derivatives Incorporating a Thiazole Moiety
  64. Synthesis of ethynylated biaryls and asymmetric diethynylated benzene via sequential Sonogashira and Suzuki couplings in water
  65. Chemistry and Biological Activity of Pyridotriazolopyrimidines
  66. Synthesis and Reactivity of Phenylthiourea Derivatives: An Efficient Synthesis of New Thiazole-Based Heterocycles
  67. Ultrasound-assisted regio- and stereoselective synthesis of bis-[1′,4′-diaryl-1-oxo-spiro-benzosuberane-2,5′-pyrazoline] derivatives via 1,3-dipolar cycloaddition
  68. Synthesis of Novel Indolizine, Pyrrolo[1,2-A] Quinoline, and 4,5-Dihydrothiophene Derivatives Via Nitrogen Ylides and their Antimicrobial Evaluation
  69. Synthesis and Anti-cancer Activity of 1,3,4-Thiadiazole and 1,3-Thiazole Derivatives Having 1,3,4-Oxadiazole Moiety
  70. Synthesis of 2-Phenylazonaphtho[1,8-ef][1,4]diazepines and 9-(3-Arylhydrazono)pyrrolo[1,2-a]perimidines as Antitumor Agents
  71. Synthesis of Unsymmetrical Aryl-Ethynylated Benzenes via Regiocontrolled Sonogashira Reaction of 1,3,5-Tribromobenzene
  72. Synthesis and Antimicrobial Evaluation of Some New 1,2-Bis-(2-(<i>N</i>-arylimino)-1,3-thiazolidin-3-yl)ethane Derivatives
  73. Metathesis Reactions in Domino Processes
  74. Synthesis of some new pyrazole-based 1,3-thiazoles and 1,3,4-thiadiazoles as anticancer agents
  75. Synthesis and quantum calculations of 1,3-thiazoles and 1,3,4-thiadiazole derivatives via pyridinylthioureas
  76. Benzofuran derivatives: a patent review
  77. Microwave-assisted synthesis of 5-arylbenzofuran-2-carboxylates via Suzuki coupling using 2-quinolinealdoxime-Pd(II)-complex
  78. A Facile Synthesis of Pyrido[2′,<...
  79. Synthesis and applications of bipyrazole systems
  80. Recent advances on the synthesis of azoles, azines and azepines fused to benzimidazole
  81. Synthetic Access to Azolylthiazoles
  82. Synthesis of some new azole, pyrimidine, pyran, and benzo/naphtho[b]furan derivatives incorporating thiazolo[3,2-a]benzimidazole moiety
  83. Synthetic routes to benzimidazole-based fused polyheterocycles
  84. Synthesis, anti-HSV-1, and cytotoxic activities of some new pyrazole- and isoxazole-based heterocycles
  85. Mizoroki-Heck cross-couplings of 2-acetyl-5-bromobenzofuran and aryl halides under microwave irradiation
  86. Facile Synthesis of Thiophene- and 1,3,4-Thiadiazole-Based Heterocycles
  87. Microwave-assisted C-C cross-coupling reactions of aryl and heteroaryl halides in water
  88. Facile Access to Biaryls and 2-Acetyl-5-arylbenzofurans via Suzuki Coupling in Water under Thermal and Microwave Conditions
  89. Synthesis, reactions, and biological activity of 4,5-diarylimidazole-2-thiones (Review)
  90. Microwave-assisted synthesis and in-vitro anti-tumor activity of 1,3,4-triaryl-5-N-arylpyrazole-carboxamides
  91. Use of 2-bromoacetylbenzofurans in heterocyclic synthesis (review)
  92. Microwave-Assisted Synthesis of 2-Substituted 4-Biarylyl-1,3-thiazoles by Carbon-Carbon Cross-Coupling in Water
  93. Heck and Suzuki cross-couplings of aryl and heteroaryl bromides in water using a new palladium(II)-complex
  94. A Facile Access to Some New Pyrazole, 1,3,4-Thiadiazole, and Thiophene Derivatives via β-Ketosulfones
  95. Synthesis and Antiviral Activity of New Indole-Based Heterocycles
  96. Cytotoxicity and Utility of 1-Indanone in the Synthesis of Some New Heterocycles
  97. 1H-Benzimidazole-2-acetonitriles as synthon in fused benzimidazole synthesis
  98. Utility of 2,4-Dioxoesters in the Synthesis of New Heterocycles
  99. Facile Access to Benzothiazole-Containing Pyrrolo[1,2-a]quinolines and Pyrrolo[2,1-a]isoquinolinesviaNitrogen Ylides
  100. Synthesis of bipyrazole and 1,3,4-thiadiazole derivatives
  101. Convenient synthesis and antimicrobial evaluation of some novel 2-substituted-3-methylbenzofuran derivatives
  102. New Domino Reactions with Sultones
  103. Synthesis of Some New Indolizine and Pyrrolo[1,2-a]quinoline Derivatives via Nitrogen Ylides
  104. Synthesis and Some New Indolizine and Pyrrolo[1,2-a]quinoline Derivatives via Nitrogen Ylides
  105. Facile route to novel 2-pyridone, pyrazolo[3,4-d]-1,2,3-triazine, and pyrazolo[3,4-d]- and [1,5-a]-pyrimidine derivatives
  106. Synthesis of annulated dihydroisoquinoline heterocycles via their nitrogen ylides
  107. Fused polyaza-heterocycles and 1,3,4-thiadiazolesviaa tricyano synthon
  108. Microwave-assisted Suzuki–Miyaura and Heck–Mizoroki cross-coupling reactions of aryl chlorides and bromides in water using stable benzothiazole-based palladium(II) precatalysts
  109. Regioselective Synthesis of Novel 4,4′-and 5,5′-bi-(1,2,4-triazole) Derivatives
  110. Synthesis of some new benzofuran-based thiophene, 1,3-oxathiole and 1,3,4-oxa(thia)diazole derivatives
  111. Microwave-accelerated Mizoroki-Heck and Sonogashira cross- coupling reactions in water using a heterogeneous palladium(II)-precatalyst
  112. A Convenient Access to Functionalized Pyrazole, Pyrazolyl-Azole, and Pyrazolo[3,4-d]Pyridazine Derivatives
  113. Synthesis, anticonvulsant, and anti-inflammatory evaluation of some new benzotriazole and benzofuran-based heterocycles
  114. Synthesis, Anticonvulsant, and Anti-inflammatory Activities of Some New Benzofuran-Based Heterocycles
  115. Combining enabling techniques in organic synthesis: solid-phase-assisted catalysis under microwave conditions using a stable Pd(II)-precatalyst
  116. 2-Pyridinealdoxime, a new ligand for a Pd-precatalyst: Application in solid-phase-assisted Suzuki–Miyaura reaction
  117. Electrolytic Partial Fluorination of Organic Compounds. 79. Anodic Fluorination of Spiropyrazoline-5,3‘-chroman-4-ones and Thiochromanone Analogues. A Route to Aroyl Fluoride Derivatives
  118. Azoles and Azolo-Azines via 3-(3-Methylbenzofuran-2-Yl)-3-Oxopropanenitrile
  119. Regio- and stereoselective synthesis of bis-spiropyrazoline-5,3′-chroman(thiochroman)-4-one derivatives via bis-nitrilimines
  120. Synthesis of spiro-pyrazole-3,3′-thiopyrano[2,3-b]pyridines and azolo[a]pyrido[2′,3′:5,6]thiopyrano[3,4-d]pyrimidines as new ring systems with antifungal and antibacterial activities
  121. Synthesis and antimicrobial evaluation of some 1,2,4-triazole, 1,3,4-oxa(thia)diazole, and 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazine derivatives
  122. Synthesis of some new pyridazine, 1,2,4-triazine and 1,3,4-thiadiazole derivatives
  123. A Facile Access to Polysubstituted Bipyrazoles and Pyrazolylpyrimidines
  124. Electrochemical Partial Fluorination of Organic Compounds. 74. Efficient Anodic Synthesis of 2-Fluoro- and 2,3-Difluoro-2,3-dihydrobenzofuran Derivatives1
  125. Synthesis of 3,3′-bipyrazole, 5,5′-bi-1,3,4-thiadiazole and fused azole systems via bishydrazonoyl chlorides
  126. Electrolytic fluorination of organic compounds
  127. A convenient route to pyridones, pyrazolo[2,3-a]pyrimidines and pyrazolo[5,1-c]triazines incorporating antipyrine moiety
  128. Indolizines, triazolo[4,3-a]pyridines, benzimidazo[1,2-d]oxadiazoles, and pyrazolo[1,5-c]triazoles via nitrogen and sulfur ylides
  129. Synthesis of 3,3′-bi-1,2,4-Triazolo[4,5-a]- benzimidazole, 5,5′-bi-1,3,4-Thiadiazole, and Thiazolo[3,2-a]benzimidazole Derivatives
  130. Polyheterocyclic systems incorporating pyrazole, thiophene, thiazole, and thiadiazole moieties
  131. Anodic Fluorination of 3-Substituted Benzofurans. Efficient Synthesis of 2-Fluoro- and 2,3-Difluoro-2,3-dihydrobenzofuran Derivatives
  132. Simple and convenient routes to new polyheterocycles incorporating pyrazole, thiazole, thiophene, and 1,3,4-thiadiazole moieties
  133. Electrolytic Partial Fluorination of Organic Compounds. 55.1 Highly Regio- and Stereoselective Anodic Monofluorination of 2,3-Dihydrochroman-4-one and Chromone Derivatives
  134. Electrolytic Partial Fluorination of Organic Compounds. 54.1 Anodic Mono- and Trifluorination of Thiochroman-4-one Derivatives and the Factors Affecting Product Selectivity
  135. Electrolytic partial fluorination of organic compounds. Part 45: Highly regioselective anodic monofluorination of (E)-3-benzylidene-2,3-dihydrochroman-4-ones
  136. AN EFFICIENT ROUTE TOTRANS-4,5-DIHYDROTHIOPHENES AND THIAZOLES VIA NITROGEN AND SULFUR YLIDES
  137. Polyheterocyclic Ring Systems with Bridgehead Nitrogen Atoms: A Facile Route to Some Novel Azolo-1,2,4-triazine Derivatives
  138. Reactions with Hydrazonoyl Halides XXX: Synthesis of Some 2,3-Dihydro-1,3,4-Thiadiazoles and Unsymmetrical Azines Containing Benzothiazole Moiety
  139. Electrolytic partial fluorination of organic compounds. 36 . Regioselective anodic fluorination of phenylthiolated benzofuranone and benzothiazole derivatives
  140. Electrolytic Partial Fluorination of Organic Compounds. 35.1 Anodic Fluorination of 2-Pyrimidyl, 2-Pyridyl, and 2-Quinazolinonyl Sulfides
  141. Electrolytic partial fluorination of organic compounds. Part 29. Anodic mono- and difluorination of 2-benzoxazolyl sulfides
  142. Heterocyclic Synthesis via Enaminonitriles: One-pot Synthesis of Some New Pyrazole, Isoxazole, Pyrimidine, Pyrazolo[1,5-a]pyrimidine, Pyrimido[1,2-a]benzimidazole and Pyrido[1,2-a]benzimidazole Derivatives
  143. Synthesis and reactivity of cyanomethyl 2-amino-4-methylthiazolyl ketone. A facile synthesis of novel pyrazolo[5,1-c]1,2,4-triazine, 1,2,4-triazolo[5,1-c]1,2,4-triazine, 1,2,4-triazino[4,3-a]benzimidazole, pyridazine-6-imine and 6-oxopyridazinone deriv...
  144. SYNTHESIS OF 1,2,4 - TRIAZOLE, 1,2,4 - TRIAZOLO [3,4 -b] [1,3,4] THIADIAZOLE AND 1,2,4 -TRIAZOLO [3,4 -b] [1,3,4] THIADIAZINE DERIVATIVES OF 3- [5- (BENZOTHIAZOL - 2 - YL) THIENO [2,3-d] PYRIMIDINE - 4- ONE] ACETIC ACID HYDRAZIDE.
  145. Heterocyclic synthesis via enaminones: Regioselective synthesis of some novel pyrazole, isoxazole, pyrimidine, pyrido[1,2-a]benzimidazole and pyrazolo[1,5-a]-pyrimidine derivatives
  146. Synthesis and reactivity of cyanomethyl 2‐amino‐4‐methylthiazolyl ketone. A facile synthesis of novel pyrazolo[5,1‐c]1,2,4‐triazine, 1,2,4‐triazolo[5,1‐c]1,2,4‐triazine, 1,2,4‐triazino[4,3‐a]benzimidazole, pyridazine‐6‐imine and 6‐oxopyridazinone deriv...
  147. Electrolytic Partial Fluorination of Organic Compounds. 31.1 Regioselective Anodic Fluorination of 2-Quinolyl and 4-(7-Trifluoromethyl)quinolyl Sulfides and the Factors Affecting Its Optimization
  148. Heterocyclic Synthesis via Enaminonitriles: A Convenient Route to Some New Pyrazole, Isoxazole, Pyrimidine, Pyrazolo[1,5-a]pyrimidine, Pyrimido[1,2-a]benzimidazole and Pyrido[1,2-a]benzimidazole Derivatives†
  149. One-pot Synthesis of Novel Polysubstituted Pyrazole and Pyrrolo[2,1-b]benzothiazole Derivatives†
  150. Synthesis and reactivity of benzothiazol-2-ylcarbonylhydroximoyl chloride, a versatile synthon
  151. CONVENIENT SYNTHESIS OF SOME NEW 1,3,4-THIADIAZOLE AND 1,3,4-SELENADIAZOLE DERIVATIVES
  152. Facile synthesis of novel polysubstituted thiopene and 1,3,4-thiadiazole derivatives
  153. Synthesis and reactivity of 2-(benzothiazol-2-yl)-1-bromo-1,2-ethanedione-1-arylhydrazones
  154. One-pot synthesis of imidazo[1,2-b]pyrazole, imidazo[1,2-b]-1,2,4-triazole, imidazo[1,2-a]pyridine, imidazo[1,2-a]pyrimidine, imidazo[1,2-a]benzimidazole, and 1,2,4-triazolo[4,3-a]benzimidazole derivatives
  155. Synthesis and reactivity of 3-(benzothiazol-2-yl)-3-oxopropanenitrile
  156. A FACILE, ONE-POT SYNTHESIS OF NOVEL 2,2′-BI(4,5-DIHYDRO-1,3,4-SELENADIAZOLE) DERIVATIVES VIA DIHYDRAZONOYL DIHALIDES
  157. One-step synthesis of novel 2,2′-bi(4,5-dihydro-1,3,4-thiadiazole) and 2,3-disubstituted 1,4-benzothiazine derivatives
  158. Facile Syntheses of Bi-1,2,4-triazoles via hydrazonyl halides