All Stories

  1. Butadiene Sulfone-catalyzed Monobromination of Arenes with NBS as the Bromination Source: A Simple, Mild, Efficient, and Chemoselective Protocol

    Article • Letters in Organic Chemistry, February 2024, Bentham Science Publishers

    Hemant Jadhav

  2. Bioactivity predictions and virtual screening using machine learning predictive model

    Article • Journal of Biomolecular Structure and Dynamics, January 2024, Taylor & Francis

    Hemant Jadhav

  3. Investigation of antibacterial potential of Natsiatum herpeticum Buch.-Ham. ex Arn. using in silico-in vitro approach

    Article • South African Journal of Botany, January 2024, Elsevier

    Hemant Jadhav

  4. FDA approved fused-pyrimidines as potential PI3K inhibitors: a computational repurposing approach

    Article • Journal of Biomolecular Structure and Dynamics, November 2023, Taylor & Francis

    Hemant Jadhav

  5. Targeting the epigenetic reader “BET” as a therapeutic strategy for cancer

    Article • Bioorganic Chemistry, November 2023, Elsevier

    Hemant Jadhav

  6. Discovery of blood-brain barrier permeable and orally bioavailable caffeine-based amide derivatives as acetylcholinesterase inhibitors

    Article • Bioorganic Chemistry, October 2023, Elsevier

    Hemant Jadhav

  7. Progress in discovery and development of natural inhibitors of histone deacetylases (HDACs) as anti-cancer agents

    Article • Naunyn-Schmiedeberg s Archives of Pharmacology, August 2023, Springer Science + Business Media

    Hemant Jadhav

  8. Identification of Azelastine and Carvedilol as Cholinesterase Inhibitors via Structure‐Based Virtual Screening of FDA‐approved Drugs

    Article • ChemistrySelect, July 2023, Wiley

    Hemant Jadhav

  9. Editorial: Recent trends and spotlight on nucleotide-based drugs: novel targets, their design, delivery, and clinical potential

    Article • Frontiers in Pharmacology, July 2023, Frontiers

    Hemant Jadhav

  10. Nutraceuticals and network pharmacology approach for acute kidney injury: A review from the drug discovery aspect

    Article • Fitoterapia, July 2023, Elsevier

    Hemant Jadhav

  11. Methoxy-naphthyl-Linked N-Benzyl Pyridinium Styryls as Dual Cholinesterase Inhibitors: Design, Synthesis, Biological Evaluation, and Structure–Activity Relationship

    Article • ACS Omega, May 2023, American Chemical Society (ACS)

    Hemant Jadhav

  12. Design, Synthesis, and Pharmacological Evaluation of Embelin–Aryl/alkyl Amine Hybrids as Orally Bioavailable Blood–Brain Barrier Permeable Multitargeted Agents with Therapeutic Potential in Alzheimer’s Disease: Discovery of SB-1448

    Article • ACS Chemical Neuroscience, February 2023, American Chemical Society (ACS)

    Hemant Jadhav

  13. A perspective on oligonucleotide therapy: Approaches to patient customization

    Article • Frontiers in Pharmacology, October 2022, Frontiers

    Hemant Jadhav

  14. Nbs and Butadiene Sulfone Catalyzed Monobromination of Arenes: A Simple, Mild, Efficient, and Chemoselective Protocol

    Article • SSRN Electronic Journal, January 2022, Elsevier

    Hemant Jadhav

  15. Design, Synthesis and Evaluation of 2,4,6-substituted Pyrimidine Derivatives as BACE-1 Inhibitor: Plausible Lead for Alzheimer’s Disease

    Article • Medicinal Chemistry, December 2021, Bentham Science Publishers

    PRITI JAIN, Hemant Jadhav

  16. Design, Synthesis and In Vitro Evaluation of 4-Oxo-6-Substituted Phenyl- 2-Thioxo1,2,3,4-Tetrahydropyrimidine-5-Carbonitrile Derivatives as HIV Integrase Strand Transfer Inhibitors

    Article • Letters in Drug Design & Discovery, April 2021, Bentham Science Publishers

    Hemant Jadhav

  17. Glycogen Synthase Kinase 3 (GSK3): Its Role and Inhibitors

    Article • Current Topics in Medicinal Chemistry, August 2020, Bentham Science Publishers

    Hemant Jadhav

  18. Design, Synthesis and In Vitro Evaluation of 2-Oxo-N-substituted Phenyl- 2H-chromene-3-carboxamide Derivatives as HIV Integrase Strand Transfer Inhibitors

    Article • Letters in Drug Design & Discovery, April 2020, Bentham Science Publishers

    Priti Jain, Hemant Jadhav

  19. Synthesis and Evaluation of 3-(1,3-dioxoisoindolin-2-yl)-N-substituted Phenyl Benzamide Analogues as HIV Integrase Strand Transfer Inhibitors

    Article • Anti-Infective Agents, July 2019, Bentham Science Publishers

    Hemant Jadhav, Priti Jain, Arpit Patel

  20. Design, Synthesis and In vitro Evaluation of Piperazine Incorporated Novel Anticancer Agents

    Article • Letters in Drug Design & Discovery, June 2018, Bentham Science Publishers

    Hemant Jadhav, Dr Ajay Kumar

  21. Peptides, Peptidomimetics, and Carbohydrate–Peptide Conjugates as Amyloidogenic Aggregation Inhibitors for Alzheimer’s Disease

    Article • ACS Chemical Neuroscience, May 2018, American Chemical Society (ACS)

    Hemant Jadhav

  22. Quinoline, Coumarin and Other Heterocyclic Analogs Based HIV-1 Integrase Inhibitors

    Article • Current Drug Discovery Technologies, April 2018, Bentham Science Publishers

    Hemant Jadhav, Priti Jain

  23. Targeting non-small cell lung cancer with small-molecule EGFR tyrosine kinase inhibitors

    Article • Drug Discovery Today, March 2018, Elsevier

    Hemant Jadhav

  24. Fast Dissolving Oral Films

    Article • May 2017, Bentham Science Publishers

    Hemant Jadhav, mahaveer singh

  25. Dynamin Functions and Ligands: Classical Mechanisms Behind

    Article • Molecular Pharmacology, November 2016, American Society for Pharmacology & Experimental Therapeutics (ASPET)

    Hemant Jadhav, mahaveer singh

  26. Design, synthesis and in vitro evaluation studies of sulfonyl-amino-acetamides as small molecule BACE-1 inhibitors

    Article • Bioorganic & Medicinal Chemistry, June 2016, Elsevier

    Hemant Jadhav

  27. Design, synthesis and evaluation of acridin-9-yl hydrazide derivatives as BACE-1 inhibitors

    Article • Medicinal Chemistry Research, April 2016, Springer Science + Business Media

    Hemant Jadhav

  28. QSAR and Docking Studies of N-hydroxy Urea Derivatives as Flap Endonuclease-1 Inhibitors

    Article • Current Computer - Aided Drug Design, January 2016, Bentham Science Publishers

    Hemant Jadhav

  29. Formulation and characterization of taste masked ondansetron–magnesium aluminum silicate adsorption systems

    Article • Drug Development and Industrial Pharmacy, January 2016, Taylor & Francis

    Dr Vikas Anand Saharan, Hemant Jadhav

  30. Rational design, synthesis and in vitro evaluation of allylidene hydrazinecarboximidamide derivatives as BACE-1 inhibitors

    Article • Bioorganic & Medicinal Chemistry Letters, January 2016, Elsevier

    Hemant Jadhav

  31. Reactive Astrogliosis: Role in Alzheimer's Disease

    Article • CNS & Neurological Disorders - Drug Targets, July 2015, Bentham Science Publishers

    Hemant Jadhav

  32. Small Molecular Inhibitors for the Treatment of Rheumatoid Arthritis: Progress so Far

    Article • Mini-Reviews in Medicinal Chemistry, March 2015, Bentham Science Publishers

    Hemant Jadhav

  33. Formulation and evaluation of lipid based taste masked granules of ondansetron HCl

    Article • European Journal of Pharmaceutical Sciences, October 2014, Elsevier

    Dr Vikas Anand Saharan, Hemant Jadhav

  34. A new open source data analysis python script for QSAR study and its validation

    Article • Medicinal Chemistry Research, September 2014, Springer Science + Business Media

    Hemant Jadhav

  35. Melatonin: functions and ligands

    Article • Drug Discovery Today, September 2014, Elsevier

    Hemant Jadhav

  36. Bitterness Score and its Correlation to Drug Concentration: An Approach for Estimating Bitterness Suppression in a Marketed Product of Ofloxacin

    Article • Analytical Chemistry Letters, July 2014, Taylor & Francis

    Dr Vikas Anand Saharan, Hemant Jadhav

  37. A Proposed Methodology for In Vitro Evaluation of Bitterness in Drug Solutions and In Vitro Drug Release Samples

    Article • Journal of Pharmaceutical Innovation, April 2014, Springer Science + Business Media

    Dr Vikas Anand Saharan, Hemant Jadhav

  38. Formulation, evaluation and 32full factorial design-based optimization of ondansetron hydrochloride incorporated taste masked microspheres

    Article • Pharmaceutical Development and Technology, September 2013, Taylor & Francis

    Dr Vikas Anand Saharan, Hemant Jadhav

  39. ChemInform Abstract: Microwave-Assisted Mild, Rapid, Solventless, and Catalyst-Free Chemoselective N-tert-Butyloxycarbonylation of Amines.

    Article • ChemInform, January 2013, Wiley

    Hemant Jadhav

  40. Histamine H3 Receptor Function and Ligands: Recent Developments

    Article • Mini-Reviews in Medicinal Chemistry, January 2013, Bentham Science Publishers

    Hemant Jadhav

  41. Histamine H3 Receptor Function and Ligands: Recent Developments

    Article • Mini-Reviews in Medicinal Chemistry, December 2012, Bentham Science Publishers

    Hemant Jadhav

  42. Histamine H3 Receptor Function and Ligands: Recent Developments

    Article • Mini-Reviews in Medicinal Chemistry, December 2012, Bentham Science Publishers

    Hemant Jadhav

  43. Microwave assisted mild, rapid, solvent-less, and catalyst-free chemoselective N-tert-butyloxycarbonylation of amines

    Article • Tetrahedron Letters, October 2012, Elsevier

    Hemant Jadhav

  44. Quantitative structure activity relationship analysis of aminoimidazoles as BACE-I inhibitors

    Article • Medicinal Chemistry Research, July 2012, Springer Science + Business Media

    Hemant Jadhav

  45. Therapeutic Advances in the Treatment of Alzheimer's Disease: Present and Future

    Article • Current Drug Therapy, August 2011, Bentham Science Publishers

    Hemant Jadhav

  46. RATIONALE FOR IMMUNOMODULATORY AND ANTI-INFLAMMATORY EFFECTS OF OCIMUM SANCTUM: RADICAL SCAVENGING POTENTIAL AND EFFECT ON NITRIC OXIDE PRODUCTION

    Article • Acta Horticulturae, February 2005, International Society for Horticultural Science (ISHS)

    Hemant Jadhav

  47. Antioxidant properties of Indian medicinal plants

    Article • Phytotherapy Research, January 2002, Wiley

    Hemant Jadhav