All Stories

  1. Triple inhibitors of monoamine reuptake transporters: first results and outlook

    Article • Chemical Biology & Drug Design, December 2015, Wiley

    Dr Gennady B Lapa

  2. Group determination of 14-membered macrolide antibiotics and azithromycin using antibodies against common epitopes

    Article • Analytical Biochemistry, January 2015, Elsevier

    Dr Gennady B Lapa

  3. Thienoquinolines as Novel Disruptors of the PKCε/RACK2 Protein–Protein Interaction

    Article • Journal of Medicinal Chemistry, April 2014, American Chemical Society (ACS)

    Dr Gennady B Lapa

  4. Synthesis and study of antibacterial activities of antibacterial glycopeptide antibiotics conjugated with benzoxaboroles

    Article • Future Medicinal Chemistry, April 2013, Future Science

    Dr Gennady B Lapa

  5. Regioselective acylation of congeners of 3-amino-1H-pyrazolo[3,4-b]quinolines, their activity on bacterial serine/threonine protein kinases and in vitro antibacterial (including antimycobacterial) activity

    Article • Journal of Enzyme Inhibition and Medicinal Chemistry, September 2012, Taylor & Francis

    Dr Gennady B Lapa

  6. Erratum To the article "Triple Inhibitors of Monoamine Reuptake Transporters: First Results and Outlook" by G. B. Lapa, Vol. 45, No. 6, pp. 323 – 328, September, 2011

    Article • Pharmaceutical Chemistry Journal, November 2011, Springer Science + Business Media

    Dr Gennady B Lapa

  7. Molecular-biological problems of drug design and mechanism of drug action

    Article • Pharmaceutical Chemistry Journal, September 2011, Springer Science + Business Media

    Dr Gennady B Lapa

  8. ChemInform Abstract: Acid-Catalyzed Cyclocondensation of Nitriles. Part 2. New Synthesis of 3-Aminoisoquinolines, 3-Imidoylaminoisoquinolines and 3-Imino-2-azaspiro(4.5)deca-6,9-diene-8-one Derivatives.

    Article • ChemInform, August 2010, Wiley

    Dr Gennady B Lapa

  9. ChemInform Abstract: Synthesis of New Dithiacycloalkanes.

    Article • ChemInform, June 2010, Wiley

    Dr Gennady B Lapa

  10. The Synthesis and Biological Evaluation of Dopamine Transporter Inhibiting Activity of Substituted Diphenylmethoxypiperidines.

    Article • ChemInform, February 2006, Wiley

    Dr Gennady B Lapa

  11. No role of the dopamine transporter in acute ethanol effects on striatal dopamine dynamics

    Article • Synapse, January 2006, Wiley

    Dr Gennady B Lapa

  12. The synthesis and biological evaluation of dopamine transporter inhibiting activity of substituted diphenylmethoxypiperidines

    Article • Bioorganic & Medicinal Chemistry Letters, November 2005, Elsevier

    Dr Gennady B Lapa

  13. Neuropsychological Disorders Indicative of Postresuscitation Encephalopathy in Rats

    Article • The Spanish Journal of Psychology, November 2005, Cambridge University Press

    Dr Gennady B Lapa

  14. Local effects of acute ethanol on dopamine neurotransmission in the ventral striatum in C57BL/6 mice

    Article • European Journal of Pharmacology, October 2005, Elsevier

    Dr Gennady B Lapa

  15. Diphenylpyraline, a histamine H1 receptor antagonist, has psychostimulant properties

    Article • European Journal of Pharmacology, January 2005, Elsevier

    Dr Gennady B Lapa

  16. P.6.013 2-Amino-adamantane derivativeLadasten enhances ex vivo dopamine synthesis and release in rat striata

    Article • European Neuropsychopharmacology, January 2005, Elsevier

    Dr Gennady B Lapa

  17. HPLC Determination of Glaucine in Yellow Horn Poppy Grass (Glaucium flavum Crantz)

    Article • Pharmaceutical Chemistry Journal, August 2004, Springer Science + Business Media

    Dr Gennady B Lapa

  18. Enzymatic synthesis of chromogenic substrates for Glu,Asp-specific proteinases

    Article • Journal of Peptide Research, July 2001, Wiley

    Dr Gennady B Lapa

  19. Epimerization of 2-bromergocryptines

    Article • Pharmaceutical Chemistry Journal, May 2000, Springer Science + Business Media

    Dr Gennady B Lapa

  20. Fragmentation of nitro(bromo)-substituted methylpapaverinium iodides under Kost-Sagitullin reaction conditions

    Article • Pharmaceutical Chemistry Journal, July 1999, Springer Science + Business Media

    Dr Gennady B Lapa

  21. Solubility of dihydroergocristine mesylate

    Article • Pharmaceutical Chemistry Journal, October 1998, Springer Science + Business Media

    Dr Gennady B Lapa

  22. Synthesis of new dithiacycloalkanes

    Article • Chemistry of Heterocyclic Compounds, September 1997, Springer Science + Business Media

    Dr Gennady B Lapa

  23. Acid-catalyzed cyclocondensation of nitriles. Part IV. Synthesis and spasmolytic activity of 1-substituted 3-aminoisoquinolines and their derivatives

    Article • Pharmaceutical Chemistry Journal, April 1997, Springer Science + Business Media

    Dr Gennady B Lapa

  24. Acid-catalyzed cyclocondensation of nitriles. III. Synthesis of substituted 3-aminoisoquinolines and study of their cytotoxicity

    Article • Pharmaceutical Chemistry Journal, January 1996, Springer Science + Business Media

    Dr Gennady B Lapa