All Stories

  1. Film Coating of Small Molded Tablets for Pediatric Formulations with Rapid Disintegration and Bitterness-Masking Properties

    Article • Molecules, May 2025, MDPI AG

    Etsuo Yonemochi

  2. Granulation Methods and the Mechanisms for Improving Hardness of Loxoprofen Sodium Hydrate-Containing Tablets

    Article • Pharmaceutics, April 2025, MDPI AG

    Etsuo Yonemochi

  3. Evaluating Various Lactose Types as Solid Carriers for Improving Curcumin Solubility in Solid Self-Nanoemulsifying Drug Delivery Systems (S-SNEDDSs) for Oral Administration

    Article • Sci, November 2024, MDPI AG

    Etsuo Yonemochi

  4. Characterization and Crystal Structural Analysis of Novel Carvedilol Adipate and Succinate Ethanol-Solvated Salts

    Article • Molecules, October 2024, MDPI AG

    Etsuo Yonemochi

  5. Fabrication and Characterization of Pectin Films Containing Solid Lipid Nanoparticles for Buccal Delivery of Fluconazole

    Article • International Journal of Molecular Sciences, May 2024, MDPI AG

    Etsuo Yonemochi, Prof. Sontaya Limmatvapirat

  6. Crystal Polymorph Search in the NPT Ensemble via a Deposition/Sublimation Alchemical Path

    Article • Crystal Growth & Design, March 2024, American Chemical Society (ACS)

    Etsuo Yonemochi

  7. Prediction of Binding Pose and Affinity of Nelfinavir, a SARS-CoV-2 Main Protease Repositioned Drug, by Combining Docking, Molecular Dynamics, and Fragment Molecular Orbital Calculations

    Article • The Journal of Physical Chemistry, March 2024, American Chemical Society (ACS)

    Etsuo Yonemochi

  8. The Development and Characterization of Novel Ionic Liquids Based on Mono- and Dicarboxylates with Meglumine for Drug Solubilizers and Skin Permeation Enhancers

    Article • Pharmaceutics, February 2024, MDPI AG

    Etsuo Yonemochi

  9. The Effect of Cholesterol Content on the Adjuvant Activity of Nucleic-Acid-Free Lipid Nanoparticles

    Article • Pharmaceutics, January 2024, MDPI AG

    Etsuo Yonemochi

  10. Novel method for the accurate calculation of Drucker–Prager cap model parameters and reduction of experimental time and effort

    Article • Advanced Powder Technology, January 2024, Elsevier

    Etsuo Yonemochi

  11. Characterization of co-amorphous carvedilol–maleic acid system prepared by solvent evaporation

    Article • Pharmaceutical Development and Technology, April 2023, Taylor & Francis

    Etsuo Yonemochi

  12. Physicochemical Properties and Transdermal Absorption of a Flurbiprofen and Lidocaine Complex in the Non-Crystalline Form

    Article • Pharmaceutics, January 2023, MDPI AG

    Etsuo Yonemochi

  13. Swelling and Salt Formation in Ibuprofen and Tranexamic Acid-Containing Tablets during High-Temperature Storage

    Article • Crystals, October 2022, MDPI AG

    Etsuo Yonemochi

  14. Study of Orally Disintegrating Tablets Using Erythritol as an Excipient Produced by Moisture-Activated Dry Granulation (MADG)

    Article • Pharmaceuticals, August 2022, MDPI AG

    Etsuo Yonemochi

  15. Non-Effective Improvement of Absorption for Some Nanoparticle Formulations Explained by Permeability under Non-Sink Conditions

    Article • Pharmaceutics, April 2022, MDPI AG

    Etsuo Yonemochi

  16. Crystal Structures of Antiarrhythmic Drug Disopyramide and Its Salt with Phthalic Acid

    Article • Crystals, April 2021, MDPI AG

    Etsuo Yonemochi

  17. Crystal Structure of Novel Terephthalate Salt of Antiarrhythmic Drug Disopyramide

    Article • Crystals, March 2021, MDPI AG

    Etsuo Yonemochi

  18. Dose-Dependent Solubility–Permeability Interplay for Poorly Soluble Drugs under Non-Sink Conditions

    Article • Pharmaceutics, March 2021, MDPI AG

    Etsuo Yonemochi

  19. Miscibility characterization of zein/methacrylic acid copolymer composite films and plasticization effects

    Article • International Journal of Pharmaceutics, March 2021, Elsevier

    Etsuo Yonemochi

  20. Cholesteryl-Conjugated Ribonuclease A Exhibits Enzyme Activity in Aqueous Solution and Resistance to Dimethyl Sulfoxide

    Article • ACS Omega, January 2021, American Chemical Society (ACS)

    Etsuo Yonemochi

  21. Synthesis and Characterization of Cholesteryl Conjugated Lysozyme (CHLysozyme)

    Article • Molecules, August 2020, MDPI AG

    Etsuo Yonemochi

  22. Application of void forming index (VFI): Detection of the effect of physical properties of dry powder inhaler formulations on powder cohesion

    Article • International Journal of Pharmaceutics, August 2020, Elsevier

    Etsuo Yonemochi

  23. Tablet Quality-Prediction Model Using Quality Material Attributes: Toward Flexible Switching Between Batch and Continuous Granulation

    Article • Journal of Pharmaceutical Innovation, July 2020, Springer Science + Business Media

    Etsuo Yonemochi

  24. Effect of Polymers and Storage Relative Humidity on Amorphous Rebamipide and Its Solid Dispersion Transformation: Multiple Spectra Chemometrics of Powder X-Ray Diffraction and Near-Infrared Spectroscopy

    Article • Pharmaceuticals, July 2020, MDPI AG

    Etsuo Yonemochi

  25. Prediction of the Crystal Growth Mechanism of Aspirin Using Molecular Simulations

    Article • YAKUGAKU ZASSHI, July 2020, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  26. Self‐Degradable Lipid‐Like Materials Based on “Hydrolysis accelerated by the intra‐Particle Enrichment of Reactant (HyPER)” for Messenger RNA Delivery

    Article • Advanced Functional Materials, June 2020, Wiley

    Etsuo Yonemochi

  27. Novel approach to evaluating granulation and segregation level considering the contribution of hydroxypropyl cellulose to the surface property change of granules

    Article • International Journal of Pharmaceutics, May 2020, Elsevier

    Etsuo Yonemochi

  28. Evaluation of the physical properties of dry surface-modified ibuprofen using a powder rheometer (FT4) and analysis of the influence of pharmaceutical additives on improvement of the powder flowability

    Article • International Journal of Pharmaceutics, April 2020, Elsevier

    Etsuo Yonemochi

  29. Degradation Pathway of a Taxane Derivative DS80100717 Drug Substance and Drug Product

    Article • Chemical and Pharmaceutical Bulletin, April 2020, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  30. New approach to optimizing risk management of the sticking problem using scale-independent critical material attributes and the quantitative process parameter

    Article • International Journal of Pharmaceutics, March 2020, Elsevier

    Etsuo Yonemochi

  31. Preface of the Special Issue “Pharmaceutical Crystals”

    Article • Crystals, February 2020, MDPI AG

    Etsuo Yonemochi

  32. Crystal Structural Analysis of DL-Mandelate Salt of Carvedilol and Its Correlation with Physicochemical Properties

    Article • Crystals, January 2020, MDPI AG

    Etsuo Yonemochi

  33. Structural origin of physicochemical properties differences upon dehydration and polymorphic transformation of ciprofloxacin hydrochloride revealed by structure determination from powder X-ray diffraction data

    Article • CrystEngComm, January 2020, Royal Society of Chemistry

    Etsuo Yonemochi

  34. Formulation design and evaluation of a transdermal drug delivery system containing a novel eptazocine salt with the Eudragit® E adhesive

    Article • Journal of Drug Delivery Science and Technology, December 2019, Elsevier

    Etsuo Yonemochi

  35. Examples of Clinical Formulation Design at a University and Response to Clinical Need

    Article • YAKUGAKU ZASSHI, October 2019, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  36. Importance of free water in controlling granule and tablet properties in a novel granulation method, green fluidized bed granulation (GFBG)

    Article • International Journal of Pharmaceutics, October 2019, Elsevier

    Etsuo Yonemochi

  37. A New Method for Classification of Salts and Cocrystals Using Solid-State UV Spectrophotometry

    Article • Chemical and Pharmaceutical Bulletin, September 2019, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  38. Foreword

    Article • Chemical and Pharmaceutical Bulletin, September 2019, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  39. Development of microparticles coated with poly-γ-glutamic acid to improve oral absorption of a poorly water-soluble drug

    Article • Pharmaceutical Development and Technology, June 2019, Taylor & Francis

    Etsuo Yonemochi

  40. Capturing a new hydrate polymorph of amodiaquine dihydrochloride dihydrateviaheterogeneous crystallisation

    Article • CrystEngComm, January 2019, Royal Society of Chemistry

    Etsuo Yonemochi

  41. Novel, Lean and Environment-friendly Granulation Method: Green Fluidized Bed Granulation (GFBG)

    Article • International Journal of Pharmaceutics, December 2018, Elsevier

    Etsuo Yonemochi

  42. Effect of sulfobutyl ether-β-cyclodextrin and propylene glycol alginate on the solubility of clozapine

    Article • Pharmaceutical Development and Technology, September 2018, Taylor & Francis

    Etsuo Yonemochi

  43. How Can the Researchers in University Be Involved with the Stream of Hospital Preparations from the Medical Needs to the Clinical Application?

    Article • YAKUGAKU ZASSHI, June 2018, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  44. Solubility Improvement of Benexate through Salt Formation Using Artificial Sweetener

    Article • Pharmaceutics, May 2018, MDPI AG

    Etsuo Yonemochi

  45. Improvement of tabletability desloratadine

    Article • European Journal of Pharmaceutical Sciences, January 2018, Elsevier

    Ahmad Ainurofiq, Etsuo Yonemochi

  46. Ethyl Haematommate fromStereocaulon graminosumSchaer.: Isolation and Crystal Structure

    Article • Natural Product Sciences, January 2018, The Korean Society of Pharmacognosy (KAMJE)

    Etsuo Yonemochi

  47. Simultaneous Improvement of Epalrestat Photostability and Solubility via Cocrystallization: A Case Study

    Article • Crystal Growth & Design, December 2017, American Chemical Society (ACS)

    Etsuo Yonemochi

  48. Void forming index: A new parameter for detecting microstructural transformation caused by powder agglomeration

    Article • International Journal of Pharmaceutics, October 2017, Elsevier

    Etsuo Yonemochi

  49. Enhanced dissolution and skin permeation profiles of epalrestat with β-cyclodextrin derivatives using a cogrinding method

    Article • European Journal of Pharmaceutical Sciences, August 2017, Elsevier

    Etsuo Yonemochi

  50. A new solvate of epalerstat, a drug for diabetic neuropathy

    Article • Acta Crystallographica Section E Crystallographic Communications, July 2017, International Union of Crystallography

    Etsuo Yonemochi

  51. Epalrestat tetrahydrofuran monosolvate: crystal structure and phase transition

    Article • Acta Crystallographica Section E Crystallographic Communications, June 2017, International Union of Crystallography

    Etsuo Yonemochi

  52. Molecular Dynamics of Amorphous Sulfamethazine With Structurally Related Sulfonamide Impurities Evaluated Using Thermal Analysis

    Article • Journal of Pharmaceutical Sciences, April 2017, Elsevier

    Etsuo Yonemochi

  53. Mechanisms for Improved Hygroscopicity of L-Arginine Valproate Revealed by X-Ray Single Crystal Structure Analysis

    Article • Journal of Pharmaceutical Sciences, March 2017, Elsevier

    Etsuo Yonemochi

  54. Characterization of complexes between phenethylamine enantiomers and β-cyclodextrin derivatives by capillary electrophoresis-Determination of binding constants and complex mobilities

    Article • Electrophoresis, February 2017, Wiley

    Etsuo Yonemochi

  55. Solubility improvement of epalrestat by layered structure formation via cocrystallization

    Article • CrystEngComm, January 2017, Royal Society of Chemistry

    Etsuo Yonemochi

  56. Effect of Magnesium Stearate Mono- and Dihydrate Dispersibilities on Physical Properties of Tablets

    Article • Chemical and Pharmaceutical Bulletin, January 2017, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  57. The effect of structurally related impurities on crystallinity reduction of sulfamethazine by grinding

    Article • International Journal of Pharmaceutics, December 2016, Elsevier

    Etsuo Yonemochi

  58. Crystallographic Analysis of Phase Dissociation Related to Anomalous Solubility of Irsogladine Maleate

    Article • Crystal Growth & Design, October 2016, American Chemical Society (ACS)

    Etsuo Yonemochi

  59. Isostructural Multicomponent Gliclazide Crystals with Improved Solubility

    Article • Crystal Growth & Design, October 2016, American Chemical Society (ACS)

    Okky Putra, Etsuo Yonemochi

  60. Crystal Structure Determination of Dimenhydrinate after More than 60 Years: Solving Salt–Cocrystal Ambiguity via Solid-State Characterizations and Solubility Study

    Article • Crystal Growth & Design, September 2016, American Chemical Society (ACS)

    Okky Putra, Etsuo Yonemochi

  61. Drug–Drug Multicomponent Crystals as an Effective Technique to Overcome Weaknesses in Parent Drugs

    Article • Crystal Growth & Design, July 2016, American Chemical Society (ACS)

    Okky Putra, Etsuo Yonemochi

  62. The effect of water activity on granule characteristics and tablet properties produced by moisture activated dry granulation (MADG)

    Article • Powder Technology, June 2016, Elsevier

    Etsuo Yonemochi

  63. Tumor delivery of liposomal doxorubicin prepared with poly-L-glutamic acid as a drug-trapping agent

    Article • Journal of Liposome Research, May 2016, Taylor & Francis

    Etsuo Yonemochi

  64. General understanding on physical stability of pharmaceutical glasses

    Article • Asian Journal of Pharmaceutical Sciences, February 2016, Elsevier

    Etsuo Yonemochi

  65. Characterization and Quality Control of Pharmaceutical Cocrystals

    Article • Chemical and Pharmaceutical Bulletin, January 2016, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  66. siRNA delivery to lung-metastasized tumor by systemic injection with cationic liposomes

    Article • Journal of Liposome Research, September 2015, Taylor & Francis

    Etsuo Yonemochi

  67. Triboelectrification of active pharmaceutical ingredients: week acids and their salts

    Article • International Journal of Pharmaceutics, September 2015, Elsevier

    Etsuo Yonemochi

  68. Therapeutic effect for liver-metastasized tumor by sequential intravenous injection of anionic polymer and cationic lipoplex of siRNA

    Article • Journal of Drug Targeting, August 2015, Taylor & Francis

    Etsuo Yonemochi

  69. Physicochemical and crystal structure analysis of pranlukast pseudo-polymorphs II: Solvate and cocrystal

    Article • Journal of Pharmaceutical and Biomedical Analysis, July 2015, Elsevier

    Etsuo Yonemochi

  70. Zoledronic acid enhances antitumor efficacy of liposomal doxorubicin

    Article • International Journal of Oncology, May 2015, Spandidos Publications

    Etsuo Yonemochi

  71. Correlation between Glass-Forming Ability and Fragility of Pharmaceutical Compounds

    Article • The Journal of Physical Chemistry, March 2015, American Chemical Society (ACS)

    Etsuo Yonemochi

  72. Physicochemical and crystal structure analysis of pranlukast pseudo-polymorphs I: Anhydrates and hydrate

    Article • Journal of Pharmaceutical and Biomedical Analysis, March 2015, Elsevier

    Etsuo Yonemochi

  73. The importance of binder moisture content in Metformin HCL high-dose formulations prepared by moist aqueous granulation (MAG)

    Article • Results in Pharma Sciences, January 2015, Elsevier

    Etsuo Yonemochi

  74. Sequential intravenous injection of anionic polymer and cationic lipoplex of siRNA could effectively deliver siRNA to the liver

    Article • International Journal of Pharmaceutics, December 2014, Elsevier

    Etsuo Yonemochi

  75. Evaluation of antitumor effect of zoledronic acid entrapped in folate-linked liposome for targeting to tumor-associated macrophages

    Article • Journal of Liposome Research, September 2014, Taylor & Francis

    Etsuo Yonemochi

  76. Effects of Formulation and Process Factors on the Crystal Structure of Freeze-Dried Myo-Inositol

    Article • Journal of Pharmaceutical Sciences, August 2014, Elsevier

    Etsuo Yonemochi

  77. Studying the Morphology of Lyophilized Protein Solids Using X-ray Micro-CT: Effect of Post-freeze Annealing and Controlled Nucleation

    Article • AAPS PharmSciTech, May 2014, American Association of Pharmaceutical Scientists (AAPS)

    Etsuo Yonemochi

  78. Relationship between Crystallization Tendencies during Cooling from Melt and Isothermal Storage: Toward a General Understanding of Physical Stability of Pharmaceutical Glasses

    Article • Molecular Pharmaceutics, April 2014, American Chemical Society (ACS)

    Etsuo Yonemochi

  79. Low-Density Microparticles with Petaloid Surface Structure for Pulmonary Drug Delivery

    Article • Journal of Pharmaceutical Sciences, April 2014, Elsevier

    Etsuo Yonemochi

  80. Clarifying the mechanism of aggregation of particles in high-shear granulation based on their surface properties by using micro-spectroscopy

    Article • International Journal of Pharmaceutics, January 2014, Elsevier

    Etsuo Yonemochi

  81. In vivo siRNA delivery system for targeting to the liver by poly-l-glutamic acid-coated lipoplex

    Article • Results in Pharma Sciences, January 2014, Elsevier

    Etsuo Yonemochi

  82. Optimization of Primary Drying Condition for Pharmaceutical Lyophilization Using a Novel Simulation Program with a Predictive Model for Dry Layer Resistance

    Article • Chemical and Pharmaceutical Bulletin, January 2014, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  83. Importance of excipient wettability on tablet characteristics prepared by moisture activated dry granulation (MADG)

    Article • International Journal of Pharmaceutics, November 2013, Elsevier

    Etsuo Yonemochi

  84. Determination for dry layer resistance of sucrose under various primary drying conditions using a novel simulation program for designing pharmaceutical lyophilization cycle

    Article • International Journal of Pharmaceutics, August 2013, Elsevier

    Etsuo Yonemochi

  85. Polymorphic and pseudomorphic transformation behavior of acyclovir based on thermodynamics and crystallography

    Article • Journal of Thermal Analysis and Calorimetry, April 2013, Springer Science + Business Media

    Etsuo Yonemochi

  86. Evaluation of physicochemical properties on the blending process of pharmaceutical granules with magnesium stearate by thermal effusivity sensor

    Article • Journal of Thermal Analysis and Calorimetry, March 2013, Springer Science + Business Media

    Etsuo Yonemochi

  87. Evaluation of the crystalline and amorphous states of drug products by nanothermal analysis and Raman imaging

    Article • Journal of Pharmaceutical and Biomedical Analysis, March 2013, Elsevier

    Etsuo Yonemochi

  88. Diffusivity of amorphous drug in solid dispersion

    Article • Journal of Thermal Analysis and Calorimetry, February 2013, Springer Science + Business Media

    Etsuo Yonemochi

  89. Competition of Thermodynamic and Dynamic Factors During Formation of Multicomponent Particles via Spray Drying

    Article • Journal of Pharmaceutical Sciences, February 2013, Elsevier

    Etsuo Yonemochi

  90. Practical Approach for Measuring Heat Capacity of Pharmaceutical Crystals/Glasses by Modulated-Temperature Differential Scanning Calorimetry

    Article • Chemical and Pharmaceutical Bulletin, January 2013, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  91. Mechanism of Dehydration–Hydration Processes of Lisinopril Dihydrate Investigated by ab Initio Powder X-ray Diffraction Analysis

    Article • Crystal Growth & Design, November 2012, American Chemical Society (ACS)

    Etsuo Yonemochi

  92. Determination of Surface Free Energy and Contact Angle for Hydrolyzed Shellac

    Article • Advanced Materials Research, April 2012, Trans Tech Publications

    Limmatvapirat Sontaya, Etsuo Yonemochi, Prof. Sontaya Limmatvapirat

  93. Applying terahertz technology for nondestructive detection of crack initiation in a film-coated layer on a swelling tablet

    Article • Results in Pharma Sciences, January 2012, Elsevier

    Etsuo Yonemochi

  94. Cocrystallization and amorphization induced by drug–excipient interaction improves the physical properties of acyclovir

    Article • International Journal of Pharmaceutics, January 2012, Elsevier

    Etsuo Yonemochi

  95. Component Crystallization and Physical Collapse during Freeze-Drying of L-Arginine^|^#8211;Citric Acid Mixtures

    Article • Chemical and Pharmaceutical Bulletin, January 2012, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  96. Potential of synchrotron X-ray powder diffractometry for detection and quantification of small amounts of crystalline drug substances in pharmaceutical tablets

    Article • Journal of Pharmaceutical and Biomedical Analysis, September 2011, Elsevier

    Etsuo Yonemochi

  97. Process analytical technology applied for end-point detection of pharmaceutical blending by combining two calibration-free methods: Simultaneously monitoring specific near-infrared peak intensity and moving block standard deviation

    Article • Powder Technology, June 2011, Elsevier

    Etsuo Yonemochi

  98. Swelling kinetics of spray-dried chitosan acetate assessed by magnetic resonance imaging and their relation to drug release kinetics of chitosan matrix tablets

    Article • European Journal of Pharmaceutics and Biopharmaceutics, February 2011, Elsevier

    Limmatvapirat Sontaya, Etsuo Yonemochi, Prof. Sontaya Limmatvapirat

  99. Development of a Rapid Process Monitoring Method for Dry-Coated Tableting Process by Using Near-Infrared Spectroscopy

    Article • Chemical and Pharmaceutical Bulletin, January 2011, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  100. Do Amorphous Troglitazones Prepared from Two Diastereomer-Pairs Have the Same Molecular Mobility and Crystallization Rate at the Surface?

    Article • Chemical and Pharmaceutical Bulletin, January 2011, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  101. Molecular States of p-Dimethylaminobenzonitrile Coground with β-Cyclodextrin Investigated Using Solid-State Fluorescence Spectroscopy

    Article • Chemical and Pharmaceutical Bulletin, January 2011, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  102. Study of the Pseudo-Crystalline Transformation from Form I to Form II of Thiamine Hydrochloride (Vitamin B1)

    Article • Chemical and Pharmaceutical Bulletin, January 2011, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  103. Development of a method for nondestructive NIR transmittance spectroscopic analysis of acetaminophen and caffeine anhydrate in intact bilayer tablets

    Article • Journal of Pharmaceutical and Biomedical Analysis, November 2010, Elsevier

    Etsuo Yonemochi

  104. Effects of Solute Miscibility on the Micro- and Macroscopic Structural Integrity of Freeze-Dried Solids

    Article • Journal of Pharmaceutical Sciences, November 2010, Elsevier

    Etsuo Yonemochi

  105. Investigation of the dynamic process during spray-drying to improve aerodynamic performance of inhalation particles

    Article • International Journal of Pharmaceutics, May 2010, Elsevier

    Etsuo Yonemochi

  106. Freeze-drying of proteins with glass-forming oligosaccharide-derived sugar alcohols

    Article • International Journal of Pharmaceutics, April 2010, Elsevier

    Etsuo Yonemochi

  107. Physicochemical Understanding of Polymorphism and Solid-State Dehydration/Rehydration Processes for the Pharmaceutical Material Acrinol, by Ab Initio Powder X-ray Diffraction Analysis and Other Techniques

    Article • The Journal of Physical Chemistry C, November 2009, American Chemical Society (ACS)

    Etsuo Yonemochi

  108. Prediction of the induction period of crystallization of naproxen in solid dispersion using differential scanning calorimetry

    Article • Journal of Thermal Analysis and Calorimetry, September 2009, Springer Science + Business Media

    Etsuo Yonemochi

  109. Reevaluation of solubility of tolbutamide and polymorphic transformation from Form I to unknown crystal form

    Article • International Journal of Pharmaceutics, March 2009, Elsevier

    Etsuo Yonemochi

  110. Freeze-Drying of Proteins in Glass Solids Formed by Basic Amino Acids and Dicarboxylic Acids

    Article • Chemical and Pharmaceutical Bulletin, January 2009, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  111. Solid States Fluorescence Study of p-Dimethylaminobenzonitrile by Co-grinding with Cyclodextrins

    Article • YAKUGAKU ZASSHI, January 2009, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  112. Stabilization of Protein Structure in Freeze-Dried Amorphous Organic Acid Buffer Salts

    Article • Chemical and Pharmaceutical Bulletin, January 2009, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  113. Evaluation of solid dispersions on a molecular level by the Raman mapping technique

    Article • International Journal of Pharmaceutics, September 2008, Elsevier

    Etsuo Yonemochi

  114. Development of a method for the determination of caffeine anhydrate in various designed intact tables by near-infrared spectroscopy: A comparison between reflectance and transmittance technique

    Article • Journal of Pharmaceutical and Biomedical Analysis, August 2008, Elsevier

    Etsuo Yonemochi

  115. Effect of the type of lubricant on the characteristics of orally disintegrating tablets manufactured using the phase transition of sugar alcohol

    Article • European Journal of Pharmaceutics and Biopharmaceutics, August 2008, Elsevier

    Etsuo Yonemochi

  116. Applicability of DPI formulations for novel neurokinin receptor antagonist

    Article • International Journal of Pharmaceutics, May 2008, Elsevier

    Etsuo Yonemochi

  117. Effect of grinding on the dehydration behavior of nedocromil sodium hydrates

    Article • Journal of Thermal Analysis and Calorimetry, May 2008, Springer Science + Business Media

    Etsuo Yonemochi

  118. Evaluation of dispersion state of the two racemic compounds of troglitazone in pharmaceutical granules using IR-to-THz imaging

    Article • Infrared Physics & Technology, May 2008, Elsevier

    Etsuo Yonemochi

  119. Application and Mechanism of Inhalation Profile Improvement of DPI Formulations by Mechanofusion with Magnesium Stearate

    Article • Chemical and Pharmaceutical Bulletin, January 2008, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  120. Glass-State Amorphous Salt Solids Formed by Freeze-Drying of Amines and Hydroxy Carboxylic Acids: Effect of Hydrogen-Bonding and Electrostatic Interactions

    Article • Chemical and Pharmaceutical Bulletin, January 2008, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  121. Effect of physical properties of troglitazone crystal on the molecular interaction with PVP during heating

    Article • International Journal of Pharmaceutics, May 2007, Elsevier

    Etsuo Yonemochi

  122. Application of microcalorimetry to the formulation study

    Article • Journal of Thermal Analysis and Calorimetry, August 2006, Springer Science + Business Media

    Etsuo Yonemochi

  123. Estimation of physical stability of amorphous solid dispersion using differential scanning calorimetry

    Article • Journal of Thermal Analysis and Calorimetry, August 2006, Springer Science + Business Media

    Etsuo Yonemochi

  124. Mechanism of glass ampoule breakage prevention during the freeze-drying process of sodium thiopental lyophilization products on addition of sodium chloride

    Article • Journal of Thermal Analysis and Calorimetry, August 2006, Springer Science + Business Media

    Etsuo Yonemochi

  125. Application of XRD-DSC system to the optimization of manufacturing process for the freeze-dried pharmaceuticals

    Article • Journal of Thermal Analysis and Calorimetry, August 2006, Springer Science + Business Media

    Etsuo Yonemochi

  126. Solid-state 13C NMR study of indomethacin polymorphism

    Article • International Journal of Pharmaceutics, August 2006, Elsevier

    Etsuo Yonemochi

  127. Evaluation of rapidly disintegrating tablets containing glycine and carboxymethylcellulose

    Article • International Journal of Pharmaceutics, March 2006, Elsevier

    Etsuo Yonemochi

  128. Novel Approach to DPI Carrier Lactose with Mechanofusion Process with Additives and Evaluation by IGC

    Article • Chemical and Pharmaceutical Bulletin, January 2006, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  129. Formulation design of a novel fast-disintegrating tablet

    Article • International Journal of Pharmaceutics, December 2005, Elsevier

    Etsuo Yonemochi

  130. Effects of water content in physical mixture and heating temperature on crystallinity of troglitazone-PVP K30 solid dispersions prepared by closed melting method

    Article • International Journal of Pharmaceutics, September 2005, Elsevier

    Etsuo Yonemochi

  131. Evaluation of the physical stability and local crystallization of amorphous terfenadine using XRD–DSC and micro-TA

    Article • Thermochimica Acta, July 2005, Elsevier

    Etsuo Yonemochi

  132. Investigation of optimal manufacturing process for freeze-dried formulations: Observation of frozen solutions by low temperature X-ray diffraction measurements

    Article • Thermochimica Acta, June 2005, Elsevier

    Etsuo Yonemochi

  133. Comparison of Molecular Mobility in the Glassy State Between Amorphous Indomethacin and Salicin Based on Spin-Lattice Relaxation Times

    Article • Pharmaceutical Research, May 2005, Springer Science + Business Media

    Etsuo Yonemochi

  134. Effects of sugar ester and hydroxypropyl methylcellulose on the physicochemical stability of amorphous cefditoren pivoxil in aqueous suspension

    Article • International Journal of Pharmaceutics, February 2005, Elsevier

    Etsuo Yonemochi

  135. Application of Eudragit RS to thermo-sensitive drug delivery systems

    Article • Journal of Controlled Release, January 2005, Elsevier

    Etsuo Yonemochi

  136. Development of Fast Disintegrating Compressed Tablets Using Amino Acid as Disintegratation Accelerator: Evaluation of Wetting and Disintegration of Tablet on the Basis of Surface Free Energy

    Article • Chemical and Pharmaceutical Bulletin, January 2005, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  137. Amorphous ultrafine particle preparation for improvement of bioavailability of insoluble drugs: grinding characteristics of fine grinding mills

    Article • International Journal of Mineral Processing, December 2004, Elsevier

    Etsuo Yonemochi

  138. Change in the physicochemical properties of ursodeoxycholic acid by grinding

    Article • Solid State Ionics, August 2004, Elsevier

    Etsuo Yonemochi

  139. Changes in surface properties by granulation and physicochemical stability of granulated amorphous cefditoren pivoxil with additives

    Article • International Journal of Pharmaceutics, August 2004, Elsevier

    Etsuo Yonemochi

  140. Physicochemical properties and surface free energy of ground talc

    Article • Solid State Ionics, August 2004, Elsevier

    Etsuo Yonemochi

  141. Uniformity and physical states of troglitazone in solid dispersions determined by electron probe microanalysis and microthermal analysis

    Article • International Journal of Pharmaceutics, August 2004, Elsevier

    Etsuo Yonemochi

  142. Microscopic molecular mobility of amorphous AG-041R measured by solid-state 13C NMR

    Article • International Journal of Pharmaceutics, May 2004, Elsevier

    Etsuo Yonemochi

  143. Quantitative Determination of Amorphous Nicardipine Hydrochloride in Long Acting Formula (NIC-LA®) Using Light Anhydrous Silicic Acid

    Article • Chemical and Pharmaceutical Bulletin, January 2004, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  144. Factors affecting the apparent solubility of ursodeoxycholic acid in the grinding process

    Article • International Journal of Pharmaceutics, April 2003, Elsevier

    Etsuo Yonemochi

  145. Solid-State Fluorescence Study of Naphthalene Adsorption on Porous Material

    Article • Journal of Colloid and Interface Science, April 2002, Elsevier

    Etsuo Yonemochi

  146. Application of Eudragit RS to Thermo-Sensitive Drug Delivery Systems. I. Thermo-Sensitive Drug Release from Acetaminophen Matrix Tablets Consisting of Eudragit RS/PEG 400 Blend Polymers

    Article • Chemical and Pharmaceutical Bulletin, January 2002, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  147. Estimation of Initial Dissolution Rate of Drug Substance by Thermal Analysis: Application for Carbamazepine Hydrate

    Article • Pharmaceutical Development and Technology, January 2002, Taylor & Francis

    Etsuo Yonemochi

  148. Characterization of Polymorphs of a Novel Quinolinone Derivative, TA-270 (4-Hydroxy-1-methyl-3-octyloxy-7-sinapinoylamino-2(1H)-quinolinone).

    Article • Chemical and Pharmaceutical Bulletin, January 2001, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  149. Interaction of Microcrystalline Cellulose and Water in Granules Prepared by a High-Shear Mixer.

    Article • Chemical and Pharmaceutical Bulletin, January 2001, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  150. Molecular Properties of Propranolol Hydrochloride Prepared as Drug-Resin Complexes

    Article • Drug Development and Industrial Pharmacy, January 2001, Taylor & Francis

    Etsuo Yonemochi, Prof. Sontaya Limmatvapirat

  151. Molecular States of 2-Naphthoic Acid in Solid Dispersions with Porous Crystalline Cellulose, as Investigated by Fluorescence Spectroscopy

    Article • Bulletin of the Chemical Society of Japan, July 2000, The Chemical Society of Japan

    Etsuo Yonemochi

  152. Quantitative correlation between initial dissolution rate and heat of fusion of drug substance

    Article • International Journal of Pharmaceutics, June 2000, Elsevier

    Etsuo Yonemochi

  153. Near IR spectroscopy to quantify the silica content and difference between silicified microcrystalline cellulose and physical mixtures of microcrystalline cellulose and silica

    Article • European Journal of Pharmaceutical Sciences, March 2000, Elsevier

    Etsuo Yonemochi

  154. Specific complexation of ursodeoxycholic acid with guest compounds induced by co-grinding

    Article • Physical Chemistry Chemical Physics, January 2000, Royal Society of Chemistry

    Limmatvapirat Sontaya, Etsuo Yonemochi, Prof. Sontaya Limmatvapirat

  155. Article • January 2000, Springer Science + Business Media

    Etsuo Yonemochi

  156. Effect of Water-Soluble Carriers on Dissolution Characteristics of Nifedipine Solid Dispersions

    Article • Drug Development and Industrial Pharmacy, January 2000, Taylor & Francis

    Etsuo Yonemochi

  157. Article • Pharmaceutical Research, January 2000, Springer Science + Business Media

    Etsuo Yonemochi

  158. Article • Pharmaceutical Research, January 2000, Springer Science + Business Media

    Etsuo Yonemochi

  159. Molecular State of Chlorpheniramine in Resinates.

    Article • Chemical and Pharmaceutical Bulletin, January 2000, Pharmaceutical Society of Japan

    Etsuo Yonemochi, Prof. Sontaya Limmatvapirat

  160. Physicochemical Properties of Ursodeoxycholic Acid Dispersed in Controlled Pore Glass

    Article • Journal of Colloid and Interface Science, August 1999, Elsevier

    Etsuo Yonemochi

  161. Water sorption and near IR spectroscopy to study the differences between microcrystalline cellulose and silicified microcrystalline cellulose before and after wet granulation

    Article • International Journal of Pharmaceutics, April 1999, Elsevier

    Etsuo Yonemochi

  162. Physicochemical properties of amorphous clarithromycin obtained by grinding and spray drying

    Article • European Journal of Pharmaceutical Sciences, March 1999, Elsevier

    Etsuo Yonemochi

  163. Article • Pharmaceutical Research, January 1999, Springer Science + Business Media

    Etsuo Yonemochi

  164. Fluorometric Studies of Pyrene Adsorption on Porous Crystalline Cellulose

    Article • Journal of Colloid and Interface Science, September 1998, Elsevier

    Etsuo Yonemochi

  165. The use of near infra-red spectroscopy to detect changes in the form of amorphous and crystalline lactose

    Article • International Journal of Pharmaceutics, June 1998, Elsevier

    Etsuo Yonemochi

  166. Structural change and complexation of strictly linear amylose induced by sealed-heating with salicylic acid

    Article • Journal of the Chemical Society Faraday Transactions, January 1998, Royal Society of Chemistry

    Limmatvapirat Sontaya, Etsuo Yonemochi

  167. Effect of Guest Species on Inclusion Compound Formation of Deoxycholic Acid by Co-Grinding.

    Article • Bulletin of the Chemical Society of Japan, January 1998, Chemical Society of Japan

    Limmatvapirat Sontaya, Etsuo Yonemochi, Prof. Sontaya Limmatvapirat

  168. Article • Journal of Inclusion Phenomena and Macrocyclic Chemistry, January 1998, Springer Science + Business Media

    Etsuo Yonemochi, Prof. Sontaya Limmatvapirat

  169. Improved dissolution of ofloxacin via solid dispersion

    Article • International Journal of Pharmaceutics, October 1997, Elsevier

    Etsuo Yonemochi

  170. A 1:1 Deoxycholic Acid–Salicylic Acid Complex

    Article • Acta Crystallographica Section C Crystal Structure Communications, June 1997, International Union of Crystallography

    Limmatvapirat Sontaya, Etsuo Yonemochi, Prof. Sontaya Limmatvapirat

  171. Enhanced Dissolution of Ursodeoxycholic Acid from the Solid Dispersion

    Article • Drug Development and Industrial Pharmacy, January 1997, Taylor & Francis

    Etsuo Yonemochi

  172. Article • Pharmaceutical Research, January 1997, Springer Science + Business Media

    Etsuo Yonemochi

  173. Time resolved fluorescent analysis for sealed heating of dimethyl-?-cyclodextrin and naphthalene system

    Article • Journal of Inclusion Phenomena and Macrocyclic Chemistry, January 1996, Springer Science + Business Media

    Etsuo Yonemochi

  174. Freeze-drying of drug-additive binary systems. IV. Effects of saccharide addition on the crystallization of cefazolin sodium in frozen aqueous solution

    Article • Pharmaceutica Acta Helvetiae, July 1995, Elsevier

    Etsuo Yonemochi

  175. Thermal Behavior of Methyl p-hydroxybenzoate in Controlled-Pore Glass Solid Dispersion

    Article • Journal of Colloid and Interface Science, July 1995, Elsevier

    Etsuo Yonemochi

  176. Dissolution studies in organic solvents for evaluating hydrogen-bond matrix of cellulose in the ground mixture

    Article • International Journal of Pharmaceutics, January 1995, Elsevier

    Etsuo Yonemochi

  177. Factors affecting the formation in the solid state of the metastable complex between naphthalene and dimethyl-?-cyclodextrin

    Article • Journal of Inclusion Phenomena and Macrocyclic Chemistry, January 1995, Springer Science + Business Media

    Etsuo Yonemochi

  178. Peculiar Peak Shifts in the IR Spectrum of Benzoic Acid Crystals by Compression with Methylated Additives.

    Article • Chemical and Pharmaceutical Bulletin, January 1995, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  179. Complex formation between naphthalene and dimethyl-β-cyclodextrin by heating in a sealed ampoule

    Article • Journal of the Chemical Society Faraday Transactions, January 1994, Royal Society of Chemistry

    Etsuo Yonemochi

  180. Article • Pharmaceutical Research, January 1994, Springer Science + Business Media

    Etsuo Yonemochi

  181. meta-Stable Complex Formation between 2,6-Di-O-methyl-,.BETA.-cyclodextrin and Naphthalene during Sealed-Heating Process.

    Article • Chemical and Pharmaceutical Bulletin, January 1994, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  182. Physicochemical Properties of Amorphous Ursodeoxycholic Acid Obtained by Grinding.

    Article • Chemical and Pharmaceutical Bulletin, January 1994, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  183. Acceleration of the addition reaction of succinic anhydride and p-nitroaniline in synthetic aluminium silicate

    Article • Advanced Powder Technology, January 1993, Brill

    Etsuo Yonemochi

  184. Molecular States of Pyrene in the Ground Mixtures with Cyclodextrins Studied by Fluorescence Spectroscopy.

    Article • NIPPON KAGAKU KAISHI, January 1993, The Chemical Society of Japan

    Etsuo Yonemochi

  185. Thermal behavior of ground mixtures of heptakis (2,6-di-O-methyl)-?-cyclodextrin and benzoic acid

    Article • Journal of Inclusion Phenomena and Macrocyclic Chemistry, January 1993, Springer Science + Business Media

    Etsuo Yonemochi

  186. Polymorphism of Tegafur: Physico-chemical Properties of Four Polymorphs.

    Article • Chemical and Pharmaceutical Bulletin, January 1993, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  187. Effect of Saccharide on the Decomposition of Cephalothin Sodium and Benzylpenicillin Potassium in Freeze-Dried Preparations.

    Article • Chemical and Pharmaceutical Bulletin, January 1992, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  188. Solubility Parameter and Dissolution Behavior of Cefalexin Powders with Different Crystallinity.

    Article • Chemical and Pharmaceutical Bulletin, January 1992, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  189. Diffusion and reaction of p-nitroaniline and succinic anhydride in controlled pore glass.

    Article • Chemical and Pharmaceutical Bulletin, January 1991, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  190. New Methods for Preparing Cyclodextrin Inclusion Compounds. IV. Enhancement of Combining Molar Ratio by Using a Ground Mixture in Heptakis-(2,6-di-O-methyl)-.BETA.-cyclodextrin and Benzoic Acid System.

    Article • Chemical and Pharmaceutical Bulletin, January 1991, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  191. Stability of aspirin in controlled pore glass solid dispersions.

    Article • Chemical and Pharmaceutical Bulletin, January 1991, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  192. Freeze-drying of drug-additive binary systems III. Crystallization of α-cyclodextrin inclusion complex in freezing process

    Article • International Journal of Pharmaceutics, June 1990, Elsevier

    Etsuo Yonemochi

  193. Effect of grinding on dehydration of crystal water of theophylline.

    Article • Chemical and Pharmaceutical Bulletin, January 1990, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  194. New methods for preparing cyclodextrin inclusion compounds. III. Preparation of heptakis-(2,6-di-O-methyl)-.BETA.-cyclodextrin-benzoic acid inclusion compound by sealed heating.

    Article • Chemical and Pharmaceutical Bulletin, January 1990, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  195. Acceleration of the addition reaction of succinic anhydride and p-nitroaniline in controlled-pore glass solid dispersions.

    Article • Chemical and Pharmaceutical Bulletin, January 1989, Pharmaceutical Society of Japan

    Etsuo Yonemochi

  196. Freeze-drying of drug-additive binary systems. II. Relationship between decarboxylation behavior and molecular states of p-aminosalicylic acid.

    Article • Chemical and Pharmaceutical Bulletin, January 1989, Pharmaceutical Society of Japan

    Etsuo Yonemochi