All Stories

  1. Synthesis of novel 2-alkyl and 2-aryl 4-phosphorylated oxazolines from dimethyl (±)-phosphoserinate
  2. Synthesis and Thermochemical Properties of Three 3,4-Dimethoxyaniline Imine Derivatives: Experimental and Theoretical Studies
  3. One-Pot Synthesis of Novel Tetrasubstituted α-Aminophosphonates Derived from α-Methylphosphoserine and In Vivo Evaluation as Anti-Inflammatory Agents
  4. Synthesis of Enantiopure cis- and trans-Fused Octahydroisoindole-1-Phosphonic Acids from Octahydroisoindolones
  5. Anti-Migratory Activity of Brazilin Chemodiversification on Breast Cancer Cells
  6. Microwave-Assisted Hydrolysis of Ethyl Azolylacetates and Cinnamates with K2CO3: Synthesis of Potassium Carboxylates
  7. Stereodivergent Synthesis of the Four Stereoisomers of Diethyl 4-Hydroxyphosphopipecolate from Ethyl (R)-4-Cyano-3-hydroxybutanoate
  8. Stereocontrolled Synthesis of Phosphoproline Analogues Containing a trans-Fused Octahydroindole Bicyclic System
  9. A Computational Method for the Binding Mode Prediction of COX-1 and COX-2 Inhibitors: Analyzing the Union of Coxibs, Oxicams, Propionic and Acetic Acids
  10. Stereodivergent Synthesis of rac-cis- and rac-trans-4-Hydroxyphosphopipecolic Acids
  11. First Stereoselective Synthesis of Diethyl cis- and trans-(4-Hydroxy-1,2,3,4-tetrahydroquinolin-2-yl)phosphonates and Ethyl Phenylphosphinates from Quinolin-4(1H)-one
  12. Iodine(III)‐Mediated Electrophilic Chlorination and Catalytic Nitration of N‐Tosyl Anilines
  13. Diastereoselective Phosphonylation of Chiral Cyclic Imines for the Synthesis of Phosphoproline Derivatives
  14. Synthesis of 1,5‐Disubstituted Tetrazole−Indolizine Bis‐Heterocycles and Their Copper (II) Recognizing Properties
  15. An efficient synthesis of cis-4-hydroxyphosphonic and cis-4-hydroxyphosphinic analogs of pipecolic acid from cyclic enaminones
  16. Experimental and theoretical study of novel aminobenzamide–aminonaphthalimide fluorescent dyads with a FRET mechanism
  17. Discovery of Octahydroisoindolone as a Scaffold for the Selective Inhibition of Chitinase B1 from Aspergillus fumigatus: In Silico Drug Design Studies
  18. Stereocontrolled Synthesis of Enantiopure cis-Fused Octahydroisoindolones via Chiral Oxazoloisoindolone Lactams
  19. Versatile optical response of pyridylalkyl naphthalenediimides in the interaction with metal ions
  20. Synthesis of phthalimides, isoindolin-1-ones and isoindolines bearing aminobenzoic acids as a new fluorescent compounds
  21. New approaches towards the synthesis of 1,2,3,4-tetrahydro isoquinoline-3-phosphonic acid (TicP)
  22. Structural Diversity using Hyp “Customizable Units”: Proof‐of‐Concept Synthesis of Sansalvamide‐Related Antitumoral Peptides
  23. Practical synthesis of 3-(2-arylethylidene)isoindolin-1-ones (analogues of AKS-182) and 3-(2-arylethylidene)isobenzofuran-1(3H)-ones
  24. Synthesis, characterization and anion recognition studies of new fluorescent alkyl bis(naphthylureylbenzamide)-based receptors
  25. Stereoselective synthesis of acyclic α,α-disubstituted α-amino acids derivatives from amino acids templates
  26. Practical Synthesis of 1,2,3,4-Tetrahydroisoquinoline-1-phosphonic and -1-phosphinic Acids through Kabachnik–Fields and Aza-Pudovik Reaction
  27. Highly Diastereoselective Synthesis of Cyclic α-Aminophosphonic and α-Aminophosphinic Acids from Glycyl-l -Proline 2,5-Diketopiperazine
  28. A Straightforward Synthesis of Six‐Membered‐Ring Heterocyclic α‐Aminophosphonic Acids from N ‐Acyliminium Ions
  29. 000Synthesis of new α-aminophosphonates: Evaluation as anti-inflammatory agents and QSAR studies
  30. Reactions of Piperazin-2-one, Morpholin-3-one, and Thiomorpholin-3-one with Triethyl Phosphite Prompted by Phosphoryl Chloride: Scope and Limitations
  31. Synthesis and anion recognition studies of new oligomethylene bis(nitrophenylureylbenzamide) receptors
  32. An Efficient Method for the Synthesis of New Non‐Symmetrical Naphthalenediimides
  33. Efficient PhB(OH) 2 -catalyzed one-pot synthesis of 3-substituted isoindolin-1-ones and isobenzofuran-1(3 H )-ones under solvent free conditions
  34. Synthesis, biological activity and molecular modelling studies of shikimic acid derivatives as inhibitors of the shikimate dehydrogenase enzyme of Escherichia coli
  35. First and Highly Stereoselective Synthesis of Both Enantiomers of Octahydroindole-2-phosphonic Acid (OicP)
  36. First practical synthesis of novel 1-phosphonylated pyrrolo[1,2-a ]pyrazine derivatives
  37. Synthesis and anion recognition studies of new ureylbenzamide-based receptors
  38. Stereoselective Synthesis of α‐Aminophosphonic Acids through Pudovik and Kabachnik‐Fields Reaction
  39. Synthesis, antimycobacterial and cytotoxic activity of α,β-unsaturated amides and 2,4-disubstituted oxazoline derivatives
  40. ChemInform Abstract: An Update on the Stereoselective Synthesis of γ-Amino Acids
  41. An update on the stereoselective synthesis of γ-amino acids
  42. Stereoselective Synthesis of α-Amino-H-phosphinic Acids and Derivatives
  43. ChemInform Abstract: First Synthesis of (R)- and (S)-1,2,3,4-Tetrahydroisoquinoline-3-phosphonic Acid (TicP) Using a Pictet-Spengler Reaction.
  44. Practical and Efficient Synthesis of α-Aminophosphonic Acids Containing 1,2,3,4-Tetrahydroquinoline or 1,2,3,4-Tetrahydroisoquinoline Heterocycles
  45. Stereoselective Synthesis of α-Amino-C-phosphinic Acids and Derivatives
  46. ChemInform Abstract: Convenient Synthesis of Cyclic α-Aminophosphonates by Alkylation-Cyclization Reaction of Iminophosphoglycinates Using Phase-Transfer Catalysis.
  47. First Synthesis of (R)- and (S)-1,2,3,4-Tetrahydroisoquinoline-3-phosphonic Acid (TicP) Using a Pictet-Spengler Reaction
  48. Novel naphthalimide–aminobenzamide dyads asOFF/ONfluorescent supramolecular receptors in metal ion binding
  49. Practical synthesis of novel phosphonopeptides containing AibP
  50. Efficient Synthesis of β-Aryl-γ-lactams and Their Resolution with (S)-Naproxen: Preparation of (R)- and (S)-Baclofen
  51. Convenient Synthesis of Cyclic α-Aminophosphonates by Alkylation-Cyclization Reaction of Iminophosphoglycinates Using Phase-Transfer Catalysis
  52. Synthesis of Chiral 1,4,2-Oxazaphosphepines
  53. ChemInform Abstract: First Practical and Efficient Synthesis of 3-Phosphorylated β-Carboline Derivatives Using the Pictet-Spengler Reaction.
  54. ChemInform Abstract: Synthesis of β-Hydroxyacetamides from Unactivated Ethyl Acetates under Base-Free Conditions and Microwave Irradiation.
  55. ChemInform Abstract: An Update on the Stereoselective Synthesis of α-Aminophosphonic Acids and Derivatives
  56. Synthesis and Characterization ofm-Terphenyl (1,3-Diphenylbenzene) Compounds Containing Trifluoromethyl Groups
  57. An update on the stereoselective synthesis of α-aminophosphonic acids and derivatives
  58. First Practical and Efficient Synthesis of 3-Phosphorylated β-Carboline Derivatives Using the Pictet-Spengler Reaction
  59. Synthesis of β-hydroxyacetamides from unactivated ethyl acetates under base-free conditions and microwave irradiation
  60. ChemInform Abstract: Phenylphosphonic Acid as Efficient and Recyclable Catalyst in the Synthesis of α-Aminophosphonates under Solvent-Free Conditions.
  61. ChemInform Abstract: Synthesis of 3-Alkylideneisoindolinones and Isoindolones by a Horner-Wadsworth-Emmons Reaction.
  62. ChemInform Abstract: Diastereoselective Synthesis of Novel 5-Substituted Morpholine-3-phosphonic Acids: Further Exploitation of N-Acyliminium Intermediates.
  63. ChemInform Abstract: Practical and Efficient Synthesis of Chiral 2,4-Disubstituted Oxazolines from β-Phosphonoamides.
  64. Phenylphosphonic Acid as Efficient and Recyclable Catalyst in the Synthesis of α-Aminophosphonates under Solvent-Free Conditions
  65. Diastereoselective synthesis of novel 5-substituted morpholine-3-phosphonic acids: further exploitation of N-acyliminium intermediates
  66. Synthesis of 3-alkylideneisoindolinones and isoindolones by a Horner–Wadsworth–Emmons reaction
  67. Practical and efficient synthesis of chiral 2,4-disubstituted oxazolines from β-phosphonoamides
  68. A Novel and Highly Regioselective Synthesis of New Carbamoylcarboxylic Acids from Dianhydrides
  69. A versatile synthesis of bicyclic lactams from 1,8-naphthalaldehydic acid: an extension of Meyers’ method
  70. ChemInform Abstract: Practical and Highly Stereoselective Synthesis of 3-(Arylmethylene)isoindolin-1-ones from 2-Formylbenzoic Acid.
  71. ChemInform Abstract: Synthesis of Quaternary α-Aminophosphonic Acids
  72. ChemInform Abstract: Phenylboronic Acid as Efficient and Eco-Friendly Catalyst for the One-Pot, Three-Component Synthesis of α-Aminophosphonates under Solvent-Free Conditions.
  73. Practical and high stereoselective synthesis of 3-(arylmethylene)isoindolin-1-ones from 2-formylbenzoic acid
  74. ChemInform Abstract: Stereoselective Synthesis of α-Aminophosphonic Acid Analogues of the 20 Proteinogenic α-Amino Acids
  75. Synthesis of quaternary α-aminophosphonic acids
  76. Phenylboronic Acid as Efficient and Eco-Friendly Catalyst for the One-Pot, Three-Component Synthesis of α-Aminophosphonates under Solvent-Free Conditions
  77. ChemInform Abstract: An Easy Approach for the Synthesis of N-Substituted Isoindolin-1-ones.
  78. Stereoselective Synthesis of α-Aminophosphonic Acids Analogs of the 20 Proteinogenic α-Amino Acids
  79. An Easy Approach for the Synthesis of N-Substituted Isoindolin-1-ones
  80. Synthesis of cis- and trans-3-Aminocyclohexanols by Reduction of β-Enaminoketones
  81. Microwave-Assisted Improved Synthesis of Oxazolidin-2-ones, Oxazolidine-2-thiones and Thiazolidine-2-thione Chiral Auxiliaries
  82. Synthesis of Phosphoproline Derivatives with an Octahydroisoindole Structure
  83. One-pot three-component highly diastereoselective synthesis of isoindolin-1-one-3-phosphonates under solvent and catalyst free-conditions
  84. Stereodivergent Synthesis of Two Novel α-Aminophosphonic Acids Characterised by a cis-Fused Octahydroindole System
  85. First Total Synthesis of 5-Hydroxy-3-methyl-4-propylsulfanyl-5H-furan-2-one: A Cancer Chemopreventive Agent
  86. Reversal Diastereoselectivity in the Benzylation of Phosphonopropanoamides
  87. ChemInform Abstract: Uncatalyzed One-Pot Diastereoselective Synthesis of α-Amino Phosphonates under Solvent-Free Conditions.
  88. Study of the fragmentation pathway of α-aminophosphonates by chemical ionization and fast atom bombardment mass spectrometry
  89. Uncatalyzed One-Pot Diastereoselective Synthesis of α-Amino Phosphonates Under Solvent-Free Conditions
  90. ChemInform Abstract: Enantioselective Diels-Alder Reactions Catalyzed by Chiral Magnesium Lewis Acids Prepared from Hydroxysulfoxides.
  91. ChemInform Abstract: Synthesis of Aldehydes from Oxiranes Using Silica Gel as Reagent.
  92. ChemInform Abstract: Improved Large Scale Preparation of Both Enantiomers of Methyl p-Tolyl Sulfoxide from Diacetone-D-glucose.
  93. ChemInform Abstract: A Convenient Synthesis of (E)-γ-Hydroxy- and (E)-γ-Keto-. alpha.,β-Unsaturated Sulfoxides.
  94. Stereochemistry of base-induced cleavage of methoxide ion on cis- and trans-1,4-diphenylphosphorinanium salts. A different behavior with a phenyl substituent
  95. ChemInform Abstract: Conformational Preference of the Sulfinyl Group in Six-Membered Heterocycles
  96. ChemInform Abstract: Stereoselective Synthesis of GABOB, Carnitine and Statine Phosphonates Analogues.
  97. ChemInform Abstract: Palladium-Catalyzed Allylic Nucleophilic Substitution Reactions of (E)-γ-Acetoxy-α,β-unsaturated p-Tolylsulfoxides.
  98. ChemInform Abstract: Diastereoselective Reduction of β-Ketophosphonates Derived from Amino Acids. A New Entry to Enantiopure β-Hydroxy-γ-aminophosphonate Derivatives.
  99. Synthesis of syn-γ-Amino-β-hydroxyphosphonates by Reduction of β-Ketophosphonates Derived from L-Proline and L-Serine
  100. Stereoselective synthesis of GABOB, carnitine and statine phosphonates analogues
  101. ChemInform Abstract: Recent Progress on the Stereoselective Synthesis of Cyclic Quaternary α-Amino Acids.
  102. ChemInform Abstract: Stereoselective Synthesis of α-Aminophosphonic Acids and Derivatives.
  103. Recent progress on the stereoselective synthesis of cyclic quaternary α-amino acids
  104. An overview of stereoselective synthesis of α-aminophosphonic acids and derivatives
  105. Reversal of diastereoselectivity in the benzylation of the lithium enolates of phosphonopropanoamides by changing the base equivalents
  106. ChemInform Abstract: A Convenient Method for the Preparation of Chiral Phosphonoacetamides and Their Horner-Wadsworth-Emmons Reaction.
  107. A practical synthesis of syn- and anti-α,β-dihydroxyphosphinates via diastereoselective reduction of α-phosphinoyl ketones
  108. A convenient method for the preparation of chiral phosphonoacetamides and their Horner–Wadsworth–Emmons reaction
  109. Stereoselective Synthesis of γ-Amino Acids
  110. Stereoselective synthesis of γ-amino acids
  111. Preparation of dimethyl (R)- and (S)-2-(2-hydroxyphenyl)-2-hydroxyethylphosphonate derived from salicylaldehyde via resolution using (S)-methoxyphenylacetic acid (MPA)
  112. Practical and Efficient Synthesis of (E)-α,β-Unsaturated Amides Bearing (S)-α-Methylbenzylamine from 2-Phosphonamides via Horner—Wadsworth—Emmons Reaction.
  113. Practical and Efficient Synthesis of (E)-α,β-Unsaturated Amides Bearing (S)-α-Methylbenzylamine from 2-Phosphonamides via Horner-Wadsworth-Emmons Reaction
  114. Synthesis of some monocyclic analogues of mycophenolic acid via the Johnson ortho ester Claisen rearrangement
  115. Synthesis of New 1,3-Oxaphosphorinanium Salts. Stereochemistry of Hydroxide-Induced Displacement of Methoxide Ion
  116. Asymmetric Alkylation of Dimethoxyphosphoryl-N-[1-(S)-α-methylbenzyl]acetamide Enolates. Synthesis of Both Stereoisomers from the Same Source of Chirality by Changing the Equivalents of LDA.
  117. Preparation of phosphostatine and phosphoepistatine from L-leucine via high diastereoselective reduction of 3-amino-2-ketophosphonates
  118. Diastereoselective Reduction of Dimethyl ?-[(N-p-Toluenesulfonyl)amino]-?-ketophosphonates Derived from Amino Acids.
  119. Asymmetric alkylation of dimethoxyphosphoryl-N-[1-(S)-α-methylbenzyl]acetamide enolates. Synthesis of both stereoisomers from the same source of chirality by changing the equivalents of LDA
  120. Diastereoselective reduction of dimethyl γ-[(N-p-toluenesulfonyl)amino]-β-ketophosphonates derived from amino acids
  121. Highly diastereoselective reduction of β-ketophosphonates bearing homochiral bis(α-methylbenzyl)amine: preparation of both enantiomers of phosphogabob (GABOBP)
  122. Highly Diastereoselective Synthesis of anti-γ-N-Benzylamino-β-hydroxyphosphonates.
  123. Preparation of dimethyl (R)- and (S)-2-(2-aminophenyl)-2-hydroxyethylphosphonate from anthranilic acid
  124. Highly Diastereoselective Addition of Et2AlCN to β-Keto Amides Derived from (S)-4-Isopropyl-2-oxazolidinone.
  125. Highly diastereoselective synthesis of anti-γ-N-benzylamino-β-hydroxyphosphonates
  126. Diels–Alder reaction of optically active (E)-γ-keto-α,β-unsaturated p-tolylsulfoxides with cyclopentadiene
  127. Generation of alkoxyalkynylketenes from a bicyclic precursor. Cycloaddition chemistry with alkynes and theoretical studies regarding the formation of five- versus six-membered ring products
  128. Highly diastereoselective addition of Et2AlCN to β-keto amides derived from (S)-4-isopropyl-2-oxazolidinone
  129. Preparation of (R)- and (S)-γ-amino-β-hydroxypropylphosphonic acid from glycine
  130. Allylic strain effects on the stereochemistry of the alkylation reaction of mycophenolic acid chiral enolates
  131. Diastereoselective reduction of β-ketophosphonates derived from amino acids. A new entry to enantiopure β-hydroxy-γ-aminophosphonate derivatives
  132. Asymmetric synthesis of both diastereomers of protected S-methyl-l-cysteine and S-n-propyl-l-cysteine sulphoxides
  133. Palladium-catalyzed allylic nucleophilic substitution reactions of (E)-γ-acetoxy-α,β-unsaturated p-tolylsulfoxides
  134. ChemInform Abstract: Efficient Preparation of Enantiomerically Pure (E)-γ-Hydroxy-α,β-Unsaturated p-Tolylsulfoxides Using Lipase-Mediated Acylations.
  135. Efficient preparation of enantiomerically pure (E)-γ-hydroxy-α,β-unsaturated p-tolylsulfoxides using lipase-mediated acylations
  136. Conformational Energy of the (η5-Cyclopentadienyl) Iron(II) Dicarbonyl Group
  137. Conformational analysis of 2-(diphenylphosphinoyl)-tetrahydrothiopyran: Lack of additivity of the S-C-P anomeric effect
  138. Chapter 3 Conformational preference of the sulfinyl group in six-membered heterocycles
  139. Enantioselective Diels-Alder reactions catalyzed by chiral magnesium lewis acids prepared from hydroxysulfoxides
  140. Synthesis of Aldehydes from Oxiranes using Silica Gel as Reagent
  141. Improved Large Scale Preparation on Both Enantiomers of Methyl p-Tolyl Sulfoxide from Diacetone-D-glucose
  142. A convenient synthesis of (E)-γ-hydroxy- and (E)-γ-keto-α,β-unsaturated sulfoxides
  143. Conformational analysis of 2-halotetrahydrothiopyran S-oxides. Diminution of the anomeric effect in S(O)-C-X compared to S-C-X segments.
  144. Lack of manifestation of an anomeric effect in 2-diphenylphosphinoyl-1, 3-dioxane and 2-diphenylphosphinoyl-1, 3-oxathiane1
  145. ChemInform Abstract: Synthesis of 4-Hydroxy-4-(2-thienyl)pentamide.
  146. SYNTHESIS OF 4-HYDROXY-4-(2-THIENYL)PENTAMIDE