All Stories

  1. Practical and Efficient Synthesis of (E)-α,β-Unsaturated Amides Incorporating α-Aminophosphonates via the Horner–Wadsworth–Emmons Reaction
  2. Phospha-Michael reaction on 4H-Chromen-4-one: A Useful Application for the Synthesis of Phosphorated 4-Oxochromanes, 4-Hydroxychromanes and 4-Oxo-4H-chromenes
  3. Computer‐Aided Drug Design of (R)‐Baclofen Isoxazole and Tetrazole Derivatives: Searching for Novel GABAB Receptor Agonists
  4. Synthesis of Amino-gem-Bisphosphonate Derivatives and Their Application as Synthons for the Preparation of Biorelevant Compounds
  5. First Synthesis of All of the cis-Fused Stereoisomers of Phosphonic and Phosphinic Analogues of Octahydrocyclopenta[b]pyrrole-2-carboxylic Acid
  6. Synthesis of novel 2-alkyl and 2-aryl 4-phosphorylated oxazolines from dimethyl (±)-phosphoserinate
  7. Synthesis and Thermochemical Properties of Three 3,4-Dimethoxyaniline Imine Derivatives: Experimental and Theoretical Studies
  8. One-Pot Synthesis of Novel Tetrasubstituted α-Aminophosphonates Derived from α-Methylphosphoserine and In Vivo Evaluation as Anti-Inflammatory Agents
  9. Synthesis of Enantiopure cis- and trans-Fused Octahydroisoindole-1-Phosphonic Acids from Octahydroisoindolones
  10. Anti-Migratory Activity of Brazilin Chemodiversification on Breast Cancer Cells
  11. Organocatalysed C-2 and C-3 Functionalisation of Chromones
  12. Microwave-Assisted Hydrolysis of Ethyl Azolylacetates and Cinnamates with K2CO3: Synthesis of Potassium Carboxylates
  13. Stereodivergent Synthesis of the Four Stereoisomers of Diethyl 4-Hydroxyphosphopipecolate from Ethyl (R)-4-Cyano-3-hydroxybutanoate
  14. Stereocontrolled Synthesis of Phosphoproline Analogues Containing a trans-Fused Octahydroindole Bicyclic System
  15. A Computational Method for the Binding Mode Prediction of COX-1 and COX-2 Inhibitors: Analyzing the Union of Coxibs, Oxicams, Propionic and Acetic Acids
  16. Stereodivergent Synthesis of rac-cis- and rac-trans-4-Hydroxyphosphopipecolic Acids
  17. First Stereoselective Synthesis of Diethyl cis- and trans-(4-Hydroxy-1,2,3,4-tetrahydroquinolin-2-yl)phosphonates and Ethyl Phenylphosphinates from Quinolin-4(1H)-one
  18. Iodine(III)‐Mediated Electrophilic Chlorination and Catalytic Nitration of N‐Tosyl Anilines
  19. Diastereoselective Phosphonylation of Chiral Cyclic Imines for the Synthesis of Phosphoproline Derivatives
  20. Synthesis of 1,5‐Disubstituted Tetrazole−Indolizine Bis‐Heterocycles and Their Copper (II) Recognizing Properties
  21. An efficient synthesis of cis-4-hydroxyphosphonic and cis-4-hydroxyphosphinic analogs of pipecolic acid from cyclic enaminones
  22. Experimental and theoretical study of novel aminobenzamide–aminonaphthalimide fluorescent dyads with a FRET mechanism
  23. Discovery of Octahydroisoindolone as a Scaffold for the Selective Inhibition of Chitinase B1 from Aspergillus fumigatus: In Silico Drug Design Studies
  24. Stereocontrolled Synthesis of Enantiopure cis-Fused Octahydroisoindolones via Chiral Oxazoloisoindolone Lactams
  25. Versatile optical response of pyridylalkyl naphthalenediimides in the interaction with metal ions
  26. Synthesis of phthalimides, isoindolin-1-ones and isoindolines bearing aminobenzoic acids as a new fluorescent compounds
  27. New approaches towards the synthesis of 1,2,3,4-tetrahydro isoquinoline-3-phosphonic acid (TicP)
  28. Structural Diversity using Hyp “Customizable Units”: Proof‐of‐Concept Synthesis of Sansalvamide‐Related Antitumoral Peptides
  29. Practical synthesis of 3-(2-arylethylidene)isoindolin-1-ones (analogues of AKS-182) and 3-(2-arylethylidene)isobenzofuran-1(3H)-ones
  30. Synthesis, characterization and anion recognition studies of new fluorescent alkyl bis(naphthylureylbenzamide)-based receptors
  31. Stereoselective synthesis of acyclic α,α-disubstituted α-amino acids derivatives from amino acids templates
  32. Practical Synthesis of 1,2,3,4-Tetrahydroisoquinoline-1-phosphonic and -1-phosphinic Acids through Kabachnik–Fields and Aza-Pudovik Reaction
  33. Highly Diastereoselective Synthesis of Cyclic α-Aminophosphonic and α-Aminophosphinic Acids from Glycyl-l -Proline 2,5-Diketopiperazine
  34. A Straightforward Synthesis of Six‐Membered‐Ring Heterocyclic α‐Aminophosphonic Acids from N ‐Acyliminium Ions
  35. 000Synthesis of new α-aminophosphonates: Evaluation as anti-inflammatory agents and QSAR studies
  36. Reactions of Piperazin-2-one, Morpholin-3-one, and Thiomorpholin-3-one with Triethyl Phosphite Prompted by Phosphoryl Chloride: Scope and Limitations
  37. Synthesis and anion recognition studies of new oligomethylene bis(nitrophenylureylbenzamide) receptors
  38. An Efficient Method for the Synthesis of New Non‐Symmetrical Naphthalenediimides
  39. Efficient PhB(OH) 2 -catalyzed one-pot synthesis of 3-substituted isoindolin-1-ones and isobenzofuran-1(3 H )-ones under solvent free conditions
  40. Synthesis, biological activity and molecular modelling studies of shikimic acid derivatives as inhibitors of the shikimate dehydrogenase enzyme of Escherichia coli
  41. First and Highly Stereoselective Synthesis of Both Enantiomers of Octahydroindole-2-phosphonic Acid (OicP)
  42. First practical synthesis of novel 1-phosphonylated pyrrolo[1,2-a ]pyrazine derivatives
  43. Synthesis and anion recognition studies of new ureylbenzamide-based receptors
  44. Stereoselective Synthesis of α‐Aminophosphonic Acids through Pudovik and Kabachnik‐Fields Reaction
  45. Synthesis, antimycobacterial and cytotoxic activity of α,β-unsaturated amides and 2,4-disubstituted oxazoline derivatives
  46. ChemInform Abstract: An Update on the Stereoselective Synthesis of γ-Amino Acids
  47. An update on the stereoselective synthesis of γ-amino acids
  48. Stereoselective Synthesis of α-Amino-H-phosphinic Acids and Derivatives
  49. ChemInform Abstract: First Synthesis of (R)- and (S)-1,2,3,4-Tetrahydroisoquinoline-3-phosphonic Acid (TicP) Using a Pictet-Spengler Reaction.
  50. Practical and Efficient Synthesis of α-Aminophosphonic Acids Containing 1,2,3,4-Tetrahydroquinoline or 1,2,3,4-Tetrahydroisoquinoline Heterocycles
  51. Stereoselective Synthesis of α-Amino-C-phosphinic Acids and Derivatives
  52. ChemInform Abstract: Convenient Synthesis of Cyclic α-Aminophosphonates by Alkylation-Cyclization Reaction of Iminophosphoglycinates Using Phase-Transfer Catalysis.
  53. First Synthesis of (R)- and (S)-1,2,3,4-Tetrahydroisoquinoline-3-phosphonic Acid (TicP) Using a Pictet-Spengler Reaction
  54. Novel naphthalimide–aminobenzamide dyads asOFF/ONfluorescent supramolecular receptors in metal ion binding
  55. Practical synthesis of novel phosphonopeptides containing AibP
  56. Efficient Synthesis of β-Aryl-γ-lactams and Their Resolution with (S)-Naproxen: Preparation of (R)- and (S)-Baclofen
  57. Convenient Synthesis of Cyclic α-Aminophosphonates by Alkylation-Cyclization Reaction of Iminophosphoglycinates Using Phase-Transfer Catalysis
  58. Synthesis of Chiral 1,4,2-Oxazaphosphepines
  59. ChemInform Abstract: First Practical and Efficient Synthesis of 3-Phosphorylated β-Carboline Derivatives Using the Pictet-Spengler Reaction.
  60. ChemInform Abstract: Synthesis of β-Hydroxyacetamides from Unactivated Ethyl Acetates under Base-Free Conditions and Microwave Irradiation.
  61. ChemInform Abstract: An Update on the Stereoselective Synthesis of α-Aminophosphonic Acids and Derivatives
  62. Synthesis and Characterization ofm-Terphenyl (1,3-Diphenylbenzene) Compounds Containing Trifluoromethyl Groups
  63. An update on the stereoselective synthesis of α-aminophosphonic acids and derivatives
  64. First Practical and Efficient Synthesis of 3-Phosphorylated β-Carboline Derivatives Using the Pictet-Spengler Reaction
  65. Synthesis of β-hydroxyacetamides from unactivated ethyl acetates under base-free conditions and microwave irradiation
  66. ChemInform Abstract: Phenylphosphonic Acid as Efficient and Recyclable Catalyst in the Synthesis of α-Aminophosphonates under Solvent-Free Conditions.
  67. ChemInform Abstract: Synthesis of 3-Alkylideneisoindolinones and Isoindolones by a Horner-Wadsworth-Emmons Reaction.
  68. ChemInform Abstract: Diastereoselective Synthesis of Novel 5-Substituted Morpholine-3-phosphonic Acids: Further Exploitation of N-Acyliminium Intermediates.
  69. ChemInform Abstract: Practical and Efficient Synthesis of Chiral 2,4-Disubstituted Oxazolines from β-Phosphonoamides.
  70. Phenylphosphonic Acid as Efficient and Recyclable Catalyst in the Synthesis of α-Aminophosphonates under Solvent-Free Conditions
  71. Diastereoselective synthesis of novel 5-substituted morpholine-3-phosphonic acids: further exploitation of N-acyliminium intermediates
  72. Synthesis of 3-alkylideneisoindolinones and isoindolones by a Horner–Wadsworth–Emmons reaction
  73. Practical and efficient synthesis of chiral 2,4-disubstituted oxazolines from β-phosphonoamides
  74. A Novel and Highly Regioselective Synthesis of New Carbamoylcarboxylic Acids from Dianhydrides
  75. A versatile synthesis of bicyclic lactams from 1,8-naphthalaldehydic acid: an extension of Meyers’ method
  76. ChemInform Abstract: Practical and Highly Stereoselective Synthesis of 3-(Arylmethylene)isoindolin-1-ones from 2-Formylbenzoic Acid.
  77. ChemInform Abstract: Synthesis of Quaternary α-Aminophosphonic Acids
  78. ChemInform Abstract: Phenylboronic Acid as Efficient and Eco-Friendly Catalyst for the One-Pot, Three-Component Synthesis of α-Aminophosphonates under Solvent-Free Conditions.
  79. Practical and high stereoselective synthesis of 3-(arylmethylene)isoindolin-1-ones from 2-formylbenzoic acid
  80. ChemInform Abstract: Stereoselective Synthesis of α-Aminophosphonic Acid Analogues of the 20 Proteinogenic α-Amino Acids
  81. Synthesis of quaternary α-aminophosphonic acids
  82. Phenylboronic Acid as Efficient and Eco-Friendly Catalyst for the One-Pot, Three-Component Synthesis of α-Aminophosphonates under Solvent-Free Conditions
  83. ChemInform Abstract: An Easy Approach for the Synthesis of N-Substituted Isoindolin-1-ones.
  84. Stereoselective Synthesis of α-Aminophosphonic Acids Analogs of the 20 Proteinogenic α-Amino Acids
  85. An Easy Approach for the Synthesis of N-Substituted Isoindolin-1-ones
  86. Synthesis of cis- and trans-3-Aminocyclohexanols by Reduction of β-Enaminoketones
  87. Microwave-Assisted Improved Synthesis of Oxazolidin-2-ones, Oxazolidine-2-thiones and Thiazolidine-2-thione Chiral Auxiliaries
  88. Synthesis of Phosphoproline Derivatives with an Octahydroisoindole Structure
  89. One-pot three-component highly diastereoselective synthesis of isoindolin-1-one-3-phosphonates under solvent and catalyst free-conditions
  90. Stereodivergent Synthesis of Two Novel α-Aminophosphonic Acids Characterised by a cis-Fused Octahydroindole System
  91. First Total Synthesis of 5-Hydroxy-3-methyl-4-propylsulfanyl-5H-furan-2-one: A Cancer Chemopreventive Agent
  92. Reversal Diastereoselectivity in the Benzylation of Phosphonopropanoamides
  93. ChemInform Abstract: Uncatalyzed One-Pot Diastereoselective Synthesis of α-Amino Phosphonates under Solvent-Free Conditions.
  94. Study of the fragmentation pathway of α-aminophosphonates by chemical ionization and fast atom bombardment mass spectrometry
  95. Uncatalyzed One-Pot Diastereoselective Synthesis of α-Amino Phosphonates Under Solvent-Free Conditions
  96. ChemInform Abstract: Enantioselective Diels-Alder Reactions Catalyzed by Chiral Magnesium Lewis Acids Prepared from Hydroxysulfoxides.
  97. ChemInform Abstract: Synthesis of Aldehydes from Oxiranes Using Silica Gel as Reagent.
  98. ChemInform Abstract: Improved Large Scale Preparation of Both Enantiomers of Methyl p-Tolyl Sulfoxide from Diacetone-D-glucose.
  99. ChemInform Abstract: A Convenient Synthesis of (E)-γ-Hydroxy- and (E)-γ-Keto-. alpha.,β-Unsaturated Sulfoxides.
  100. Stereochemistry of base-induced cleavage of methoxide ion on cis- and trans-1,4-diphenylphosphorinanium salts. A different behavior with a phenyl substituent
  101. ChemInform Abstract: Conformational Preference of the Sulfinyl Group in Six-Membered Heterocycles
  102. ChemInform Abstract: Stereoselective Synthesis of GABOB, Carnitine and Statine Phosphonates Analogues.
  103. ChemInform Abstract: Palladium-Catalyzed Allylic Nucleophilic Substitution Reactions of (E)-γ-Acetoxy-α,β-unsaturated p-Tolylsulfoxides.
  104. ChemInform Abstract: Diastereoselective Reduction of β-Ketophosphonates Derived from Amino Acids. A New Entry to Enantiopure β-Hydroxy-γ-aminophosphonate Derivatives.
  105. Synthesis of syn-γ-Amino-β-hydroxyphosphonates by Reduction of β-Ketophosphonates Derived from L-Proline and L-Serine
  106. Stereoselective synthesis of GABOB, carnitine and statine phosphonates analogues
  107. ChemInform Abstract: Recent Progress on the Stereoselective Synthesis of Cyclic Quaternary α-Amino Acids.
  108. ChemInform Abstract: Stereoselective Synthesis of α-Aminophosphonic Acids and Derivatives.
  109. Recent progress on the stereoselective synthesis of cyclic quaternary α-amino acids
  110. An overview of stereoselective synthesis of α-aminophosphonic acids and derivatives
  111. Reversal of diastereoselectivity in the benzylation of the lithium enolates of phosphonopropanoamides by changing the base equivalents
  112. ChemInform Abstract: A Convenient Method for the Preparation of Chiral Phosphonoacetamides and Their Horner-Wadsworth-Emmons Reaction.
  113. A practical synthesis of syn- and anti-α,β-dihydroxyphosphinates via diastereoselective reduction of α-phosphinoyl ketones
  114. A convenient method for the preparation of chiral phosphonoacetamides and their Horner–Wadsworth–Emmons reaction
  115. Stereoselective Synthesis of γ-Amino Acids
  116. Stereoselective synthesis of γ-amino acids
  117. Preparation of dimethyl (R)- and (S)-2-(2-hydroxyphenyl)-2-hydroxyethylphosphonate derived from salicylaldehyde via resolution using (S)-methoxyphenylacetic acid (MPA)
  118. Practical and Efficient Synthesis of (E)-α,β-Unsaturated Amides Bearing (S)-α-Methylbenzylamine from 2-Phosphonamides via Horner—Wadsworth—Emmons Reaction.
  119. Practical and Efficient Synthesis of (E)-α,β-Unsaturated Amides Bearing (S)-α-Methylbenzylamine from 2-Phosphonamides via Horner-Wadsworth-Emmons Reaction
  120. Synthesis of some monocyclic analogues of mycophenolic acid via the Johnson ortho ester Claisen rearrangement
  121. Synthesis of New 1,3-Oxaphosphorinanium Salts. Stereochemistry of Hydroxide-Induced Displacement of Methoxide Ion
  122. Asymmetric Alkylation of Dimethoxyphosphoryl-N-[1-(S)-α-methylbenzyl]acetamide Enolates. Synthesis of Both Stereoisomers from the Same Source of Chirality by Changing the Equivalents of LDA.
  123. Preparation of phosphostatine and phosphoepistatine from L-leucine via high diastereoselective reduction of 3-amino-2-ketophosphonates
  124. Diastereoselective Reduction of Dimethyl ?-[(N-p-Toluenesulfonyl)amino]-?-ketophosphonates Derived from Amino Acids.
  125. Asymmetric alkylation of dimethoxyphosphoryl-N-[1-(S)-α-methylbenzyl]acetamide enolates. Synthesis of both stereoisomers from the same source of chirality by changing the equivalents of LDA
  126. Diastereoselective reduction of dimethyl γ-[(N-p-toluenesulfonyl)amino]-β-ketophosphonates derived from amino acids
  127. Highly diastereoselective reduction of β-ketophosphonates bearing homochiral bis(α-methylbenzyl)amine: preparation of both enantiomers of phosphogabob (GABOBP)
  128. Highly Diastereoselective Synthesis of anti-γ-N-Benzylamino-β-hydroxyphosphonates.
  129. Preparation of dimethyl (R)- and (S)-2-(2-aminophenyl)-2-hydroxyethylphosphonate from anthranilic acid
  130. Highly Diastereoselective Addition of Et2AlCN to β-Keto Amides Derived from (S)-4-Isopropyl-2-oxazolidinone.
  131. Highly diastereoselective synthesis of anti-γ-N-benzylamino-β-hydroxyphosphonates
  132. Diels–Alder reaction of optically active (E)-γ-keto-α,β-unsaturated p-tolylsulfoxides with cyclopentadiene
  133. Generation of alkoxyalkynylketenes from a bicyclic precursor. Cycloaddition chemistry with alkynes and theoretical studies regarding the formation of five- versus six-membered ring products
  134. Highly diastereoselective addition of Et2AlCN to β-keto amides derived from (S)-4-isopropyl-2-oxazolidinone
  135. Preparation of (R)- and (S)-γ-amino-β-hydroxypropylphosphonic acid from glycine
  136. Allylic strain effects on the stereochemistry of the alkylation reaction of mycophenolic acid chiral enolates
  137. Diastereoselective reduction of β-ketophosphonates derived from amino acids. A new entry to enantiopure β-hydroxy-γ-aminophosphonate derivatives
  138. Asymmetric synthesis of both diastereomers of protected S-methyl-l-cysteine and S-n-propyl-l-cysteine sulphoxides
  139. Palladium-catalyzed allylic nucleophilic substitution reactions of (E)-γ-acetoxy-α,β-unsaturated p-tolylsulfoxides
  140. ChemInform Abstract: Efficient Preparation of Enantiomerically Pure (E)-γ-Hydroxy-α,β-Unsaturated p-Tolylsulfoxides Using Lipase-Mediated Acylations.
  141. Efficient preparation of enantiomerically pure (E)-γ-hydroxy-α,β-unsaturated p-tolylsulfoxides using lipase-mediated acylations
  142. Conformational Energy of the (η5-Cyclopentadienyl) Iron(II) Dicarbonyl Group
  143. Conformational analysis of 2-(diphenylphosphinoyl)-tetrahydrothiopyran: Lack of additivity of the S-C-P anomeric effect
  144. Chapter 3 Conformational preference of the sulfinyl group in six-membered heterocycles
  145. Enantioselective Diels-Alder reactions catalyzed by chiral magnesium lewis acids prepared from hydroxysulfoxides
  146. Synthesis of Aldehydes from Oxiranes using Silica Gel as Reagent
  147. Improved Large Scale Preparation on Both Enantiomers of Methyl p-Tolyl Sulfoxide from Diacetone-D-glucose
  148. A convenient synthesis of (E)-γ-hydroxy- and (E)-γ-keto-α,β-unsaturated sulfoxides
  149. Conformational analysis of 2-halotetrahydrothiopyran S-oxides. Diminution of the anomeric effect in S(O)-C-X compared to S-C-X segments.
  150. Lack of manifestation of an anomeric effect in 2-diphenylphosphinoyl-1, 3-dioxane and 2-diphenylphosphinoyl-1, 3-oxathiane1
  151. ChemInform Abstract: Synthesis of 4-Hydroxy-4-(2-thienyl)pentamide.
  152. SYNTHESIS OF 4-HYDROXY-4-(2-THIENYL)PENTAMIDE